Page last updated: 2024-09-05

zm 241385 and isoalloxazine

zm 241385 has been researched along with isoalloxazine in 6 studies

Compound Research Comparison

Studies
(zm 241385)
Trials
(zm 241385)
Recent Studies (post-2010)
(zm 241385)
Studies
(isoalloxazine)
Trials
(isoalloxazine)
Recent Studies (post-2010) (isoalloxazine)
4013124194060

Protein Interaction Comparison

ProteinTaxonomyzm 241385 (IC50)isoalloxazine (IC50)
Female germline-specific tumor suppressor gld-1Caenorhabditis elegans1.471

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's6 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ahern, DG; Jacobson, KA; Ji, X; Kim, YC; Linden, J1
Bartoccini, F; Carminati, P; Castorina, M; Di Cesare, MA; Di Serio, S; Gallo, G; Ghirardi, O; Giorgi, F; Giorgi, L; Minetti, P; Piersanti, G; Tarzia, G; Tinti, MO1
Hong, KW; Shin, HK; Shin, YW1
Brodmann, M; Lischnig, U; Lueger, A; Pilger, E; Stark, G1
Hamano, R; Iwagaki, H; Kanke, T; Liu, K; Nishibori, M; Sendo, T; Takahashi, HK; Tanaka, N; Yoshino, T1
Miriel, VA; Rivers, RJ; Thengchaisri, N1

Other Studies

6 other study(ies) available for zm 241385 and isoalloxazine

ArticleYear
[3H]MRS 1754, a selective antagonist radioligand for A(2B) adenosine receptors.
    Biochemical pharmacology, 2001, Mar-15, Volume: 61, Issue:6

    Topics: Acetamides; Cells, Cultured; Humans; Purinergic P1 Receptor Antagonists; Purines; Radioligand Assay; Radiopharmaceuticals; Receptor, Adenosine A2B; Tritium

2001
2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A2A adenosine receptor antagonists. Design, synthesis, and pharmacological characterization.
    Journal of medicinal chemistry, 2005, Nov-03, Volume: 48, Issue:22

    Topics: Adenine; Adenosine A2 Receptor Antagonists; Animals; Cell Line; Cricetinae; Cricetulus; Drug Design; Humans; Imidazoles; Male; Models, Molecular; Motor Activity; Purines; Radioligand Assay; Rats; Rats, Inbred F344; Structure-Activity Relationship; Triazoles

2005
Role of adenosine A(2B) receptors in vasodilation of rat pial artery and cerebral blood flow autoregulation.
    American journal of physiology. Heart and circulatory physiology, 2000, Volume: 278, Issue:2

    Topics: Animals; Arteries; Cerebrovascular Circulation; Cyclic AMP; Cyclic GMP; Enzyme Inhibitors; Flavins; Homeostasis; Male; NG-Nitroarginine Methyl Ester; Nitrates; Nitrites; Pia Mater; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2B; Receptors, Purinergic P1; Thionucleotides; Triazines; Triazoles; Vasodilation

2000
The effect of caffeine on peripheral vascular resistance in isolated perfused guinea pig hind limbs.
    Journal of cardiovascular pharmacology, 2003, Volume: 42, Issue:4

    Topics: Adenosine; Animals; Caffeine; Dose-Response Relationship, Drug; Female; Flavins; Guinea Pigs; Hindlimb; Hypoxia; Iliac Artery; Iloprost; Male; Nitrogen; Norepinephrine; Perfusion; Triazines; Triazoles; Vascular Resistance; Vasoconstriction; Vasodilation

2003
Stimulation of adenosine A2A receptor inhibits LPS-induced expression of intercellular adhesion molecule 1 and production of TNF-alpha in human peripheral blood mononuclear cells.
    Shock (Augusta, Ga.), 2008, Volume: 29, Issue:2

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adenosine A3 Receptor Agonists; Adenosine A3 Receptor Antagonists; CD40 Antigens; Cells, Cultured; Cyclic AMP; Enzyme-Linked Immunosorbent Assay; Flavins; Flow Cytometry; Humans; Intercellular Adhesion Molecule-1; Leukocytes, Mononuclear; Lipopolysaccharide Receptors; Lipopolysaccharides; Receptor, Adenosine A2A; Triazines; Triazoles; Tumor Necrosis Factor-alpha; Xanthines

2008
Multiple receptor subtypes and multiple mechanisms of dilation are involved in vascular network dilation caused by adenosine.
    Microvascular research, 2009, Volume: 77, Issue:3

    Topics: Adenosine; Animals; Arterioles; Cricetinae; Drug Antagonism; Endothelium, Vascular; Flavins; Mesocricetus; Methacholine Chloride; Nitroprusside; Purinergic P1 Receptor Antagonists; Quinazolines; Receptors, Purinergic P1; Triazines; Triazoles; Vasodilation; Vasodilator Agents

2009