Page last updated: 2024-09-05

zm 241385 and cocaine

zm 241385 has been researched along with cocaine in 2 studies

Compound Research Comparison

Studies
(zm 241385)
Trials
(zm 241385)
Recent Studies (post-2010)
(zm 241385)
Studies
(cocaine)
Trials
(cocaine)
Recent Studies (post-2010) (cocaine)
401312432,4611,0969,400

Protein Interaction Comparison

ProteinTaxonomyzm 241385 (IC50)cocaine (IC50)
Amyloid-beta precursor proteinHomo sapiens (human)0.338
Fatty acid-binding protein, heartHomo sapiens (human)0.367
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0855
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.0855
DRattus norvegicus (Norway rat)5.7544
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)5.7544
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)5.7544
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)5.7544
Sodium-dependent noradrenaline transporter Homo sapiens (human)1.2861
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)0.4321
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0855
Sodium-dependent serotonin transporterHomo sapiens (human)0.5442
Sodium-dependent serotonin transporterRattus norvegicus (Norway rat)0.8885
Sodium-dependent dopamine transporter Homo sapiens (human)0.3796
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)5.541
Sodium-dependent dopamine transporterMus musculus (house mouse)0.2
Sigma non-opioid intracellular receptor 1Homo sapiens (human)1.05
TransporterRattus norvegicus (Norway rat)3.2277

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Agnati, L; Filip, M; Franco, R; Fuxe, K; LluĂ­s, C; Marcellino, D; Navarro, G; Roberts, DC1
Brown, RM; Duncan, JR; Lawrence, AJ; Ledent, C; Stagnitti, MR1

Other Studies

2 other study(ies) available for zm 241385 and cocaine

ArticleYear
Increase in A2A receptors in the nucleus accumbens after extended cocaine self-administration and its disappearance after cocaine withdrawal.
    Brain research, 2007, Apr-27, Volume: 1143

    Topics: Animals; Behavior, Animal; Binding, Competitive; Cocaine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Male; Nucleus Accumbens; Raclopride; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2A; Reinforcement Schedule; Self Administration; Substance Withdrawal Syndrome; Time Factors; Triazines; Triazoles; Tritium

2007
mGlu5 and adenosine A2A receptor interactions regulate the conditioned effects of cocaine.
    The international journal of neuropsychopharmacology, 2012, Volume: 15, Issue:7

    Topics: Analysis of Variance; Animals; Autoradiography; Brain; Cocaine; Conditioning, Operant; Dopamine Uptake Inhibitors; Drug Interactions; Excitatory Amino Acid Antagonists; Iodine Isotopes; Locomotion; Male; Mice; Mice, Knockout; Protein Binding; Pyridines; Radionuclide Imaging; Receptor, Adenosine A2A; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Thiazoles; Time Factors; Triazines; Triazoles

2012