Page last updated: 2024-08-24

ziprasidone and raclopride

ziprasidone has been researched along with raclopride in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (50.00)18.2507
2000's2 (25.00)29.6817
2010's2 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Audinot, V; Chaput, C; Conte, C; Gavaudan, S; Millan, MJ; Newman-Tancredi, A; Touzard, M; Verrièle, L1
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K1
Bench, CJ; Cuddigan, M; Dolan, RJ; Frackowiak, RS; Grasby, PM; Gunn, K; Lammertsma, AA; Osman, S; Turton, DJ; Warrington, SJ1
Bench, CJ; Brooks, DJ; Frackowiak, RS; Gunn, K; Hume, SP; Lammertsma, AA; Osman, S1
Bench, CJ; Boyce, M; Brannick, LY; Dolan, RJ; Frackowiak, RS; Grasby, PM; Gunn, KP; Lammertsma, AA; Warrington, SJ1
Kapur, S; Mamo, D; Mann, S; Papatheodorou, G; Remington, G; Shammi, CM; Therrien, F1
Bartenstein, P; Boy, C; Bröcheler, A; Buchholz, HG; Cumming, P; Fellows, C; Gründer, G; Hiemke, C; Janouschek, H; Landvogt, C; Rösch, F; Schäfer, W; Spreckelmeyer, K; Vernaleken, I; Veselinovic, T; Wong, DF1
Borlido, C; Caravaggio, F; Deluca, V; Graff-Guerrero, A; Ismail, Z; Mamo, D; Mulsant, B; Pollock, B; Remington, G; Suzuki, T; Uchida, H1

Trials

5 trial(s) available for ziprasidone and raclopride

ArticleYear
Dose dependent occupancy of central dopamine D2 receptors by the novel neuroleptic CP-88,059-01: a study using positron emission tomography and 11C-raclopride.
    Psychopharmacology, 1993, Volume: 112, Issue:2-3

    Topics: Adult; Brain; Cerebrovascular Circulation; Dopamine Antagonists; Dose-Response Relationship, Drug; Humans; Image Processing, Computer-Assisted; Male; Neostriatum; Piperazines; Prolactin; Raclopride; Receptors, Dopamine D2; Salicylamides; Spiro Compounds; Thiazoles; Tomography, Emission-Computed

1993
The time course of binding to striatal dopamine D2 receptors by the neuroleptic ziprasidone (CP-88,059-01) determined by positron emission tomography.
    Psychopharmacology, 1996, Volume: 124, Issue:1-2

    Topics: Adult; Antipsychotic Agents; Corpus Striatum; Humans; Male; Piperazines; Prolactin; Raclopride; Receptors, Dopamine D2; Salicylamides; Thiazoles; Time Factors; Tomography, Emission-Computed

1996
A PET study of dopamine D2 and serotonin 5-HT2 receptor occupancy in patients with schizophrenia treated with therapeutic doses of ziprasidone.
    The American journal of psychiatry, 2004, Volume: 161, Issue:5

    Topics: Adult; Antipsychotic Agents; Brain; Corpus Striatum; Drug Administration Schedule; Female; Humans; Male; Piperazines; Psychotic Disorders; Pyrimidinones; Raclopride; Receptors, Dopamine D2; Receptors, Serotonin, 5-HT2; Schizophrenia; Thiazoles; Tomography, Emission-Computed

2004
Striatal and extrastriatal D2/D3-receptor-binding properties of ziprasidone: a positron emission tomography study with [18F]Fallypride and [11C]raclopride (D2/D3-receptor occupancy of ziprasidone).
    Journal of clinical psychopharmacology, 2008, Volume: 28, Issue:6

    Topics: Adult; Antipsychotic Agents; Basal Ganglia; Benzamides; Binding, Competitive; Carbon Radioisotopes; Dopamine Antagonists; Dose-Response Relationship, Drug; Female; Fluorine Radioisotopes; Humans; Male; Piperazines; Positron-Emission Tomography; Pyrrolidines; Raclopride; Radiopharmaceuticals; Receptors, Dopamine D2; Receptors, Dopamine D3; Schizophrenia; Thiazoles; Time Factors; Young Adult

2008
Dopamine D₂/₃ occupancy of ziprasidone across a day: a within-subject PET study.
    Psychopharmacology, 2013, Volume: 228, Issue:1

    Topics: Adult; Antipsychotic Agents; Brain; Case-Control Studies; Dopamine Antagonists; Female; Half-Life; Humans; Male; Middle Aged; Piperazines; Positron-Emission Tomography; Prolactin; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D3; Schizophrenia; Thiazoles; Time Factors; Young Adult

2013

Other Studies

3 other study(ies) available for ziprasidone and raclopride

ArticleYear
Agonist and antagonist actions of antipsychotic agents at 5-HT1A receptors: a [35S]GTPgammaS binding study.
    European journal of pharmacology, 1998, Aug-21, Volume: 355, Issue:2-3

    Topics: Animals; Antipsychotic Agents; CHO Cells; Cricetinae; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Agents; Sulfur Radioisotopes

1998
QSAR-based permeability model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2011, Apr-15, Volume: 19, Issue:8

    Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2011
Comparison of methods for analysis of clinical [11C]raclopride studies.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 1996, Volume: 16, Issue:1

    Topics: Adult; Antipsychotic Agents; Body Fluid Compartments; Brain; Carbon Radioisotopes; Cerebellum; Corpus Striatum; Dopamine Antagonists; Dose-Response Relationship, Drug; Humans; Male; Models, Biological; Nonlinear Dynamics; Piperazines; Raclopride; Receptors, Dopamine D2; Reference Values; Regression Analysis; Salicylamides; Thiazoles; Tissue Distribution; Tomography, Emission-Computed

1996