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zidovudine and r 82150

zidovudine has been researched along with r 82150 in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's8 (88.89)18.2507
2000's0 (0.00)29.6817
2010's1 (11.11)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bamberger, DL; Fisher, TE; Goldman, ME; Hoffman, JM; Jones, JH; Rooney, CS; Saari, WS; Smith, AM; Thomas, CM; Wai, JS1
Breslin, HJ; De Clercq, E; Diamond, CJ; Grous, PP; Ho, CY; Kukla, MJ; Miranda, M; Pauwels, R; Rodgers, JD; Sherrill, RG1
Breslin, HJ; De Clercq, E; Diamond, CJ; Grous, PP; Ho, CY; Ho, W; Kukla, MJ; Ludovici, DW; Miranda, M; Rodgers, JD1
De Clercq, E; Li, D; Liu, X; Zhan, P1
Andries, K; De Clercq, E; Debyser, Z; Pauwels, R1
Cheng, YC; Dutschman, GE; Im, GJ; Mellors, JW; Tramontano, E; Winkler, SR1
Baba, M; De Clercq, E; Debyser, Z; Desmyter, J; Pauwels, R1
Andries, K; Breslin, HJ; Desmyter, J; Heykants, J; Kukla, MJ; Pauwels, R; Raeymaeckers, A; Schols, D; Van Gelder, J; Woestenborghs, R1
Busso, M; Resnick, L1

Reviews

1 review(s) available for zidovudine and r 82150

ArticleYear
Specific HIV-1 reverse transcriptase inhibitors.
    Journal of enzyme inhibition, 1992, Volume: 6, Issue:1

    Topics: Antiviral Agents; Benzodiazepines; HIV Reverse Transcriptase; HIV-1; Imidazoles; Models, Genetic; Reverse Transcriptase Inhibitors; Thymine; Transcription, Genetic; Zidovudine

1992

Other Studies

8 other study(ies) available for zidovudine and r 82150

ArticleYear
Synthesis and evaluation of 2-pyridinone derivatives as HIV-1-specific reverse transcriptase inhibitors. 2. Analogues of 3-aminopyridin-2(1H)-one.
    Journal of medicinal chemistry, 1992, Oct-16, Volume: 35, Issue:21

    Topics: Aminopyridines; Antiviral Agents; Benzoxazoles; Cells, Cultured; HIV Reverse Transcriptase; HIV-1; Pyridones; Reverse Transcriptase Inhibitors; Structure-Activity Relationship

1992
Synthesis and anti-HIV-1 activity of 4,5,6,7-tetrahydro-5-methylimidazo[4,5,1-jk][1,4]benzodiazepin-2(1H)-on e (TIBO) derivatives. 2.
    Journal of medicinal chemistry, 1991, Volume: 34, Issue:11

    Topics: Antiviral Agents; Benzodiazepines; HIV-1; Imidazoles; Microbial Sensitivity Tests; Structure-Activity Relationship; Virus Replication

1991
Synthesis and anti-HIV-1 activity of 4,5,6,7-tetrahydro-5-methylimidazo-[4,5,1-jk][1,4]benzodiazepin- 2(1H)-one (TlBO) derivatives. 4.
    Journal of medicinal chemistry, 1995, Mar-03, Volume: 38, Issue:5

    Topics: Antiviral Agents; Benzodiazepines; Cell Line; Cytopathogenic Effect, Viral; HIV-1; Imidazoles; Structure-Activity Relationship; Virus Replication

1995
Strategies for the design of HIV-1 non-nucleoside reverse transcriptase inhibitors: lessons from the development of seven representative paradigms.
    Journal of medicinal chemistry, 2012, Apr-26, Volume: 55, Issue:8

    Topics: Anti-HIV Agents; Benzodiazepines; Binding Sites; Crystallography, X-Ray; Drug Design; HIV Reverse Transcriptase; HIV-1; Hydrogen Bonding; Imidazoles; Indoles; Nitriles; Reverse Transcriptase Inhibitors; Structure-Activity Relationship

2012
In vitro selection and molecular characterization of human immunodeficiency virus-1 resistant to non-nucleoside inhibitors of reverse transcriptase.
    Molecular pharmacology, 1992, Volume: 41, Issue:3

    Topics: Antiviral Agents; Base Sequence; Benzodiazepines; CD4-Positive T-Lymphocytes; Cloning, Molecular; Drug Resistance, Microbial; Foscarnet; Gene Expression; HeLa Cells; HIV-1; Humans; Imidazoles; Molecular Sequence Data; Nevirapine; Phosphonoacetic Acid; Polymerase Chain Reaction; Pyridines; Recombinant Proteins; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Zidovudine

1992
Common features in the interaction of tetrahydroimidazo[4,5,1-jk][1,4]benzodiazepin-2(1H)-one and -thione and 1-[(2-hydroxyethoxy)methyl]-6-(phenylthio)thymine derivatives with the human immunodeficiency virus type 1 reverse transcriptase.
    Molecular pharmacology, 1992, Volume: 41, Issue:5

    Topics: Antiviral Agents; Benzodiazepines; Dideoxynucleotides; HIV-1; Imidazoles; Kinetics; Molecular Structure; Recombinant Proteins; Reverse Transcriptase Inhibitors; Structure-Activity Relationship; Templates, Genetic; Thymidine; Thymine Nucleotides; Uracil; Zidovudine

1992
Potent and selective inhibition of HIV-1 replication in vitro by a novel series of TIBO derivatives.
    Nature, 1990, Feb-01, Volume: 343, Issue:6257

    Topics: Animals; Antiviral Agents; Benzodiazepines; CD4-Positive T-Lymphocytes; Cell Line; Cytopathogenic Effect, Viral; Didanosine; Dogs; HIV-1; HIV-2; Humans; Imidazoles; Lymphocytes; Molecular Conformation; Molecular Structure; Reverse Transcriptase Inhibitors; Virus Replication; Zidovudine

1990
Development of an assay that detects transcriptionally competent human immunodeficiency virus type one particles.
    Journal of virological methods, 1994, Volume: 47, Issue:1-2

    Topics: Antiviral Agents; Benzodiazepines; Dideoxynucleotides; DNA, Viral; Drug Resistance, Microbial; HIV Reverse Transcriptase; HIV-1; Humans; Imidazoles; Polymerase Chain Reaction; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Sensitivity and Specificity; Thymine Nucleotides; Zidovudine

1994