Page last updated: 2024-09-03

zd 7288 and sr 95531

zd 7288 has been researched along with sr 95531 in 3 studies

Compound Research Comparison

Studies
(zd 7288)
Trials
(zd 7288)
Recent Studies (post-2010)
(zd 7288)
Studies
(sr 95531)
Trials
(sr 95531)
Recent Studies (post-2010) (sr 95531)
38201376100209

Protein Interaction Comparison

ProteinTaxonomyzd 7288 (IC50)sr 95531 (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit alpha-1Homo sapiens (human)0.2763
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit gamma-2Homo sapiens (human)0.2763
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit beta-2Homo sapiens (human)0.2763
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.24
GABA theta subunitRattus norvegicus (Norway rat)0.24
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.24

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (66.67)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hashimoto, K; Kita, H1
Blethyn, KL; Cope, DW; Crunelli, V; Hughes, SW; Tóth, TI1
Bayliss, DA; Chen, X; Kapur, J; Schwartz, LC; Shu, S; Sun, C1

Other Studies

3 other study(ies) available for zd 7288 and sr 95531

ArticleYear
Slow oscillatory activity of rat globus pallidus neurons in vitro.
    The European journal of neuroscience, 2006, Volume: 23, Issue:2

    Topics: Action Potentials; Anesthetics, Local; Animals; Animals, Newborn; Biological Clocks; Cadmium Chloride; Calcium; Calcium Channel Blockers; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Antagonists; Globus Pallidus; In Vitro Techniques; Neurons; Patch-Clamp Techniques; Piperazines; Pyridazines; Pyrimidines; Quinoxalines; Rats; Rats, Sprague-Dawley; Tetrodotoxin; Time Factors

2006
Neuronal basis of the slow (<1 Hz) oscillation in neurons of the nucleus reticularis thalami in vitro.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2006, Mar-01, Volume: 26, Issue:9

    Topics: Action Potentials; Animals; Apamin; Cadmium; Cats; Computer Simulation; Cycloleucine; Dose-Response Relationship, Radiation; Drug Interactions; Electric Capacitance; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Antagonists; In Vitro Techniques; Intralaminar Thalamic Nuclei; Models, Neurological; Neural Pathways; Neurons; Neuroprotective Agents; Nickel; Organophosphorus Compounds; Periodicity; Pyridazines; Pyrimidines; Sodium Channel Blockers; Tetrodotoxin; Time Factors

2006
Homeostatic regulation of synaptic excitability: tonic GABA(A) receptor currents replace I(h) in cortical pyramidal neurons of HCN1 knock-out mice.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Feb-17, Volume: 30, Issue:7

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Anti-Anxiety Agents; Bicuculline; Cerebral Cortex; Cyclic Nucleotide-Gated Cation Channels; Desoxycorticosterone; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; GABA Agents; Homeostasis; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Male; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Knockout; Models, Neurological; Patch-Clamp Techniques; Potassium Channels; Protein Subunits; Pyramidal Cells; Pyridazines; Pyrimidines; Receptors, GABA-A; Sodium Channel Blockers; Synapses; Tetrodotoxin; Up-Regulation; Valine

2010