Page last updated: 2024-09-03

zd 7288 and propofol

zd 7288 has been researched along with propofol in 3 studies

Compound Research Comparison

Studies
(zd 7288)
Trials
(zd 7288)
Recent Studies (post-2010)
(zd 7288)
Studies
(propofol)
Trials
(propofol)
Recent Studies (post-2010) (propofol)
382013716,8275,1886,805

Protein Interaction Comparison

ProteinTaxonomyzd 7288 (IC50)propofol (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)8.1667
Aldo-keto reductase family 1 member B1Rattus norvegicus (Norway rat)9.393
Polyunsaturated fatty acid lipoxygenase ALOX15Oryctolagus cuniculus (rabbit)7.596
Gamma-aminobutyric acid receptor subunit alpha-1Homo sapiens (human)8
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)8.1667
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)8.1667
Gamma-aminobutyric acid receptor subunit gamma-2Homo sapiens (human)8
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)8.1667
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)8.1667
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)8.1667
Prostaglandin G/H synthase 1Homo sapiens (human)3.832
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)8.1667
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)8.1667
Sodium-dependent noradrenaline transporter Homo sapiens (human)9.393
Sodium- and chloride-dependent GABA transporter 1Rattus norvegicus (Norway rat)8.3
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)8.1667
Gamma-aminobutyric acid receptor subunit beta-3Homo sapiens (human)8
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)8.1667
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)8.1667
Sodium- and chloride-dependent GABA transporter 2Rattus norvegicus (Norway rat)8.3
Sodium- and chloride-dependent GABA transporter 3Rattus norvegicus (Norway rat)8.3
5-hydroxytryptamine receptor 2BHomo sapiens (human)5.499
Sodium- and chloride-dependent betaine transporterRattus norvegicus (Norway rat)8.3
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)8.1667
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)8.1667
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)8.1667
GABA theta subunitRattus norvegicus (Norway rat)8.1667
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)8.1667

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bayliss, DA; Chen, X; Shu, S1
Abbas, SY; Goldstein, PA; Harrison, NL; Ying, SW1
Liu, YC; Wang, YJ; Wu, PY; Wu, SN1

Other Studies

3 other study(ies) available for zd 7288 and propofol

ArticleYear
Suppression of ih contributes to propofol-induced inhibition of mouse cortical pyramidal neurons.
    Journal of neurophysiology, 2005, Volume: 94, Issue:6

    Topics: Animals; Animals, Newborn; Anticonvulsants; Bicuculline; Cerebral Cortex; Cyclic Nucleotide-Gated Cation Channels; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Female; GABA Antagonists; Glycine Agents; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; In Vitro Techniques; Ion Channel Gating; Ion Channels; Lysine; Male; Membrane Potentials; Mice; Neural Inhibition; Neural Pathways; Oocytes; Patch-Clamp Techniques; Potassium Channels; Propofol; Pyramidal Cells; Pyrimidines; Rats; Strychnine; Thalamus; Time Factors; Xenopus

2005
Propofol block of I(h) contributes to the suppression of neuronal excitability and rhythmic burst firing in thalamocortical neurons.
    The European journal of neuroscience, 2006, Volume: 23, Issue:2

    Topics: Action Potentials; Analysis of Variance; Animals; Bicuculline; Cell Count; Cyclic AMP; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Free Radical Scavengers; GABA Antagonists; Gene Expression; Glutamic Acid; Green Fluorescent Proteins; Humans; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Immunohistochemistry; In Vitro Techniques; Ion Channels; Membrane Potentials; Mice; Mice, Inbred C57BL; Microscopy, Confocal; Neural Inhibition; Neurons; Patch-Clamp Techniques; Periodicity; Potassium Channels; Propofol; Pyrimidines; Thalamus; Transfection

2006
Tramadol-induced block of hyperpolarization-activated cation current in rat pituitary lactotrophs.
    Naunyn-Schmiedeberg's archives of pharmacology, 2009, Volume: 379, Issue:2

    Topics: Action Potentials; Analgesics, Opioid; Animals; Cations; Cell Line; Cesium; Chlorides; Cyclic AMP; Cyclic Nucleotide-Gated Cation Channels; Dideoxyadenosine; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Lactotrophs; Patch-Clamp Techniques; Potassium Channels; Propofol; Pyrimidines; Rats; Thionucleotides; Tramadol

2009