Page last updated: 2024-09-03

zd 7288 and n-methylaspartate

zd 7288 has been researched along with n-methylaspartate in 3 studies

Compound Research Comparison

Studies
(zd 7288)
Trials
(zd 7288)
Recent Studies (post-2010)
(zd 7288)
Studies
(n-methylaspartate)
Trials
(n-methylaspartate)
Recent Studies (post-2010) (n-methylaspartate)
382013710,408591,902

Protein Interaction Comparison

ProteinTaxonomyzd 7288 (IC50)n-methylaspartate (IC50)
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)5.175
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)5.175
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)5.175
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)5.175
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)5.175
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)5.175
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)5.175

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (66.67)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Aghajanian, GK; Jolas, T; Nestler, EJ1
Feuerstein, TJ; Klar, M; Surges, R1
Cheng, Z; Fu, G; Guo, L; He, W; Lu, Q; Xu, X1

Other Studies

3 other study(ies) available for zd 7288 and n-methylaspartate

ArticleYear
Chronic morphine increases GABA tone on serotonergic neurons of the dorsal raphe nucleus: association with an up-regulation of the cyclic AMP pathway.
    Neuroscience, 2000, Volume: 95, Issue:2

    Topics: Adenylyl Cyclases; Analgesics, Opioid; Animals; Cardiovascular Agents; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Electrophysiology; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enzyme Inhibitors; Excitatory Amino Acid Agonists; gamma-Aminobutyric Acid; In Vitro Techniques; Interneurons; Isoquinolines; Male; Membrane Potentials; Morphine; N-Methylaspartate; Neural Inhibition; Periaqueductal Gray; Phenylephrine; Pyrimidines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Serotonin; Substance Withdrawal Syndrome; Sulfonamides; Sympathomimetics; Tetrazoles; Tetrodotoxin; Thionucleotides

2000
Ih channels as modulators of presynaptic terminal function: ZD7288 increases NMDA-evoked [3H]-noradrenaline release in rat neocortex slices.
    Naunyn-Schmiedeberg's archives of pharmacology, 2003, Volume: 367, Issue:4

    Topics: Animals; Cations; Dose-Response Relationship, Drug; In Vitro Techniques; Ion Channels; N-Methylaspartate; Neocortex; Neurons; Norepinephrine; Potassium; Presynaptic Terminals; Pyrimidines; Rats; Rats, Wistar; Tetrodotoxin; Time Factors

2003
ZD7288-induced suppression of long-term potentiation was attenuated by exogenous NMDA at the Schaffer collateral-CA1 synapse in the rat in vivo.
    European journal of pharmacology, 2010, Apr-10, Volume: 631, Issue:1-3

    Topics: Animals; CA1 Region, Hippocampal; Cyclic Nucleotide-Gated Cation Channels; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Postsynaptic Potentials; Injections, Intraventricular; Long-Term Potentiation; Male; Membrane Transport Modulators; N-Methylaspartate; Neurons; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Synapses; Synaptic Transmission; Time Factors

2010