Page last updated: 2024-09-03

zd 7288 and isoproterenol

zd 7288 has been researched along with isoproterenol in 11 studies

Compound Research Comparison

Studies
(zd 7288)
Trials
(zd 7288)
Recent Studies (post-2010)
(zd 7288)
Studies
(isoproterenol)
Trials
(isoproterenol)
Recent Studies (post-2010) (isoproterenol)
382013730,7808032,640

Protein Interaction Comparison

ProteinTaxonomyzd 7288 (IC50)isoproterenol (IC50)
Beta-2 adrenergic receptorHomo sapiens (human)0.246
Beta-1 adrenergic receptorHomo sapiens (human)0.333
Beta-2 adrenergic receptorRattus norvegicus (Norway rat)0.2125
Polyunsaturated fatty acid lipoxygenase ALOX15Oryctolagus cuniculus (rabbit)1.77
Beta-1 adrenergic receptorRattus norvegicus (Norway rat)0.2125
Beta-3 adrenergic receptorRattus norvegicus (Norway rat)0.2125
Beta-2 adrenergic receptorCanis lupus familiaris (dog)0.6667

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (18.18)18.2507
2000's2 (18.18)29.6817
2010's7 (63.64)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Maccaferri, G; McBain, CJ1
Choi, HS; Lee, CO; Noble, D; Wang, DY1
Gainullin, AA; Zefirov, AL; Zefirov, TL; Ziyatdinova, NI1
Akar, FG; Cho, HC; Jones, SP; Li, RA; Marbán, E; Tomaselli, GF; Tsang, SY; Xue, T1
Chen, PS; Joung, B; Kim, D; Lin, SF; Luk, HN; Maruyama, M; Shinohara, T1
Chen, PS; Choi, EK; Joung, B; Kim, D; Lin, SF; On, YK; Piccirillo, G; Shinohara, T; Zhang, H1
Chen, PS; Han, S; Kim, D; Lin, SF; Maruyama, M; Park, HW; Shen, MJ; Shinohara, T1
Chen, PS; Chua, SK; Han, S; Joung, B; Lin, SF; Maruyama, M; Park, HW; Shen, MJ; Shinohara, T1
Greene, D; Hoshi, N; Kang, S; Kosenko, A1
Hernández-Cascales, J; Merino, B; Quesada, I1
Brown, JT; Church, TW; Marrion, NV1

Other Studies

11 other study(ies) available for zd 7288 and isoproterenol

ArticleYear
The hyperpolarization-activated current (Ih) and its contribution to pacemaker activity in rat CA1 hippocampal stratum oriens-alveus interneurones.
    The Journal of physiology, 1996, Nov-15, Volume: 497 ( Pt 1)

    Topics: Action Potentials; Adrenergic beta-Agonists; Animals; Cardiovascular Agents; Cesium; Electrophysiology; Hippocampus; Isoproterenol; Neurons; Norepinephrine; Patch-Clamp Techniques; Pyrimidines; Rats; Rats, Sprague-Dawley

1996
Effect of isoprenaline, carbachol, and Cs+ on Na+ activity and pacemaker potential in rabbit SA node cells.
    The American journal of physiology, 1999, Volume: 276, Issue:1

    Topics: Action Potentials; Animals; Carbachol; Cardiac Pacing, Artificial; Cardiotonic Agents; Cesium; Electrophysiology; Female; Intracellular Membranes; Isoproterenol; Male; Pyrimidines; Rabbits; Sinoatrial Node; Sodium

1999
Blockade of hyperpolarization-activated channels modifies the effect of beta-adrenoceptor stimulation.
    Bulletin of experimental biology and medicine, 2002, Volume: 133, Issue:5

    Topics: Animals; Bradycardia; Cardiovascular Agents; Electrophysiology; Heart; Isoproterenol; Pyrimidines; Rats; Receptors, Adrenergic, beta; Time Factors; Vagotomy; Vagus Nerve

2002
Functional integration of electrically active cardiac derivatives from genetically engineered human embryonic stem cells with quiescent recipient ventricular cardiomyocytes: insights into the development of cell-based pacemakers.
    Circulation, 2005, Jan-04, Volume: 111, Issue:1

    Topics: Action Potentials; Adrenergic beta-Agonists; Animals; Cell Differentiation; Cell Fusion; Cells, Cultured; Defective Viruses; Electrophysiology; Female; Genes, Reporter; Genetic Vectors; Giant Cells; Green Fluorescent Proteins; Guinea Pigs; Heart; Heart Conduction System; Heart Ventricles; HIV-1; Humans; Isoproterenol; Lidocaine; Mice; Myocardial Contraction; Myocytes, Cardiac; Organ Culture Techniques; Pericardium; Pluripotent Stem Cells; Pyrimidines; Rats; Transduction, Genetic

2005
Induction of atrial ectopic beats with calcium release inhibition: Local hierarchy of automaticity in the right atrium.
    Heart rhythm, 2010, Volume: 7, Issue:1

    Topics: Adrenergic beta-Agonists; Animals; Atrial Premature Complexes; Calcium; Calcium Channels, L-Type; Cardiotonic Agents; Dogs; Heart Atria; Heart Conduction System; Heart Rate; Isoproterenol; Membrane Potentials; Pyrimidines; Risk Assessment; Risk Factors; Ryanodine; Sarcoplasmic Reticulum; Sinoatrial Node; Time Factors

2010
Tachybradycardia in the isolated canine right atrium induced by chronic sympathetic stimulation and pacemaker current inhibition.
    American journal of physiology. Heart and circulatory physiology, 2010, Volume: 299, Issue:3

    Topics: Analysis of Variance; Animals; Bradycardia; Calcium; Cardiotonic Agents; Dogs; Heart Atria; Isoproterenol; Membrane Potentials; Pyrimidines; Ryanodine; Tachycardia

2010
Ca2+ clock malfunction in a canine model of pacing-induced heart failure.
    American journal of physiology. Heart and circulatory physiology, 2010, Volume: 299, Issue:6

    Topics: Adrenergic beta-Agonists; Animals; Caffeine; Calcium Signaling; Cardiac Pacing, Artificial; Circadian Clocks; Disease Models, Animal; Dogs; Electrophysiologic Techniques, Cardiac; Heart Failure; Heart Rate; Isoproterenol; Membrane Potentials; Perfusion; Pyrimidines; Sarcoplasmic Reticulum; Sinoatrial Node; Time Factors

2010
Selective sinoatrial node optical mapping and the mechanism of sinus rate acceleration.
    Circulation journal : official journal of the Japanese Circulation Society, 2012, Volume: 76, Issue:2

    Topics: Animals; Biological Clocks; Calcium; Cardiotonic Agents; Dogs; Heart Atria; Heart Rate; Hyperkalemia; Isoproterenol; Isotonic Solutions; Male; Membrane Potentials; Perfusion; Potassium; Pyrimidines; Ryanodine; Sarcoplasmic Reticulum; Sinoatrial Node; Sympathetic Nervous System; Tachycardia, Sinus

2012
Adrenergic regulation of HCN4 channel requires protein association with β2-adrenergic receptor.
    The Journal of biological chemistry, 2012, Jul-06, Volume: 287, Issue:28

    Topics: Adrenergic beta-Agonists; Amino Acid Sequence; Animals; Animals, Newborn; Cells, Cultured; Cyclic Nucleotide-Gated Cation Channels; HEK293 Cells; HeLa Cells; Humans; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Immunoblotting; Ion Channel Gating; Isoproterenol; Membrane Potentials; Molecular Sequence Data; Multiprotein Complexes; Muscle Proteins; Myocytes, Cardiac; Patch-Clamp Techniques; Peptides; Potassium Channels; Protein Binding; Protein Isoforms; Pyrimidines; Rats; Receptors, Adrenergic, beta-2; Sequence Homology, Amino Acid; Sinoatrial Node

2012
Glucagon Increases Beating Rate but Not Contractility in Rat Right Atrium. Comparison with Isoproterenol.
    PloS one, 2015, Volume: 10, Issue:7

    Topics: Animals; Atrial Function, Right; Calcium Signaling; Carbazoles; Cyclic AMP-Dependent Protein Kinases; Glucagon; Heart Atria; Heart Rate; Isoproterenol; Isoquinolines; Male; Myocardial Contraction; Myocardium; Phosphodiesterase 3 Inhibitors; Phosphodiesterase 4 Inhibitors; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Sulfonamides

2015
β
    Journal of neurophysiology, 2019, 03-01, Volume: 121, Issue:3

    Topics: Adrenergic beta-Agonists; Animals; CA1 Region, Hippocampal; Cyclic AMP; Ethanolamines; Isoproterenol; Male; Membrane Potentials; Potassium Channel Blockers; Pyramidal Cells; Pyrimidines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Small-Conductance Calcium-Activated Potassium Channels; Tetrahydronaphthalenes

2019