Page last updated: 2024-09-03

zd 7288 and h 89

zd 7288 has been researched along with h 89 in 5 studies

Compound Research Comparison

Studies
(zd 7288)
Trials
(zd 7288)
Recent Studies (post-2010)
(zd 7288)
Studies
(h 89)
Trials
(h 89)
Recent Studies (post-2010) (h 89)
38201371,6190409

Protein Interaction Comparison

ProteinTaxonomyzd 7288 (IC50)h 89 (IC50)
Rho-associated protein kinase 2Homo sapiens (human)1.9504
Ribosomal protein S6 kinase alpha-5Homo sapiens (human)0.12
cAMP-dependent protein kinase catalytic subunit alphaBos taurus (cattle)0.073
cAMP-dependent protein kinase catalytic subunit alpha Mus musculus (house mouse)0.381
cAMP-dependent protein kinase catalytic subunit alphaHomo sapiens (human)0.6365
cAMP-dependent protein kinase catalytic subunit gammaHomo sapiens (human)0.6365
cAMP-dependent protein kinase catalytic subunit betaHomo sapiens (human)0.6365
Ribosomal protein S6 kinase beta-1Homo sapiens (human)0.08
RAC-alpha serine/threonine-protein kinaseHomo sapiens (human)1.9886
RAC-beta serine/threonine-protein kinaseHomo sapiens (human)0.5417
Rho-associated protein kinase 2Rattus norvegicus (Norway rat)0.27
RAC-gamma serine/threonine-protein kinaseHomo sapiens (human)0.3207

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (80.00)29.6817
2010's1 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Aghajanian, GK; Jolas, T; Nestler, EJ1
Mellor, J; Nicoll, RA; Schmitz, D1
Bie, B; Pan, ZZ; Peng, Y; Zhang, Y1
Cadiou, H; Mason, A; McNaughton, PA; Momin, A1
Hernández-Cascales, J; Merino, B; Quesada, I1

Other Studies

5 other study(ies) available for zd 7288 and h 89

ArticleYear
Chronic morphine increases GABA tone on serotonergic neurons of the dorsal raphe nucleus: association with an up-regulation of the cyclic AMP pathway.
    Neuroscience, 2000, Volume: 95, Issue:2

    Topics: Adenylyl Cyclases; Analgesics, Opioid; Animals; Cardiovascular Agents; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Electrophysiology; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enzyme Inhibitors; Excitatory Amino Acid Agonists; gamma-Aminobutyric Acid; In Vitro Techniques; Interneurons; Isoquinolines; Male; Membrane Potentials; Morphine; N-Methylaspartate; Neural Inhibition; Periaqueductal Gray; Phenylephrine; Pyrimidines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Serotonin; Substance Withdrawal Syndrome; Sulfonamides; Sympathomimetics; Tetrazoles; Tetrodotoxin; Thionucleotides

2000
Mediation of hippocampal mossy fiber long-term potentiation by presynaptic Ih channels.
    Science (New York, N.Y.), 2002, Jan-04, Volume: 295, Issue:5552

    Topics: Adenylyl Cyclases; Animals; Benzazepines; Calcium; Cesium; Chlorides; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclic Nucleotide-Gated Cation Channels; Dentate Gyrus; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; In Vitro Techniques; Ion Channels; Isoquinolines; Long-Term Potentiation; Membrane Potentials; Membrane Proteins; Models, Neurological; Mossy Fibers, Hippocampal; Nerve Tissue Proteins; Patch-Clamp Techniques; Potassium; Potassium Channels; Presynaptic Terminals; Pyramidal Cells; Pyrimidines; Rats; Rats, Sprague-Dawley; Sulfonamides; Synaptic Transmission

2002
cAMP-mediated mechanisms for pain sensitization during opioid withdrawal.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Apr-13, Volume: 25, Issue:15

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Animals; Animals, Newborn; Behavior, Animal; Blotting, Western; Colforsin; Cyclic AMP; Dose-Response Relationship, Radiation; Drug Administration Schedule; Drug Interactions; Electric Stimulation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Gene Expression Regulation; Imines; In Vitro Techniques; Isoquinolines; Male; Membrane Potentials; Microinjections; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Opioid-Related Disorders; Oxidoreductases; Pain; Pain Measurement; Patch-Clamp Techniques; Pyrimidines; Raphe Nuclei; Rats; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sulfonamides

2005
Role of the hyperpolarization-activated current Ih in somatosensory neurons.
    The Journal of physiology, 2008, Dec-15, Volume: 586, Issue:24

    Topics: Action Potentials; Animals; Animals, Newborn; Cell Size; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic Nucleotide-Gated Cation Channels; Dinoprostone; Electric Stimulation; Ganglia, Spinal; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Isoquinolines; Menthol; Mice; Mice, Inbred Strains; Mice, Knockout; Potassium Channel Blockers; Potassium Channels; Protein Kinase Inhibitors; Pyrimidines; Rats; Rats, Wistar; Sensory Receptor Cells; Sulfonamides; TRPM Cation Channels

2008
Glucagon Increases Beating Rate but Not Contractility in Rat Right Atrium. Comparison with Isoproterenol.
    PloS one, 2015, Volume: 10, Issue:7

    Topics: Animals; Atrial Function, Right; Calcium Signaling; Carbazoles; Cyclic AMP-Dependent Protein Kinases; Glucagon; Heart Atria; Heart Rate; Isoproterenol; Isoquinolines; Male; Myocardial Contraction; Myocardium; Phosphodiesterase 3 Inhibitors; Phosphodiesterase 4 Inhibitors; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Sulfonamides

2015
chemdatabank.com