Page last updated: 2024-09-03

zd 7288 and glutamic acid

zd 7288 has been researched along with glutamic acid in 12 studies

Compound Research Comparison

Studies
(zd 7288)
Trials
(zd 7288)
Recent Studies (post-2010)
(zd 7288)
Studies
(glutamic acid)
Trials
(glutamic acid)
Recent Studies (post-2010) (glutamic acid)
382013741,75745212,876

Protein Interaction Comparison

ProteinTaxonomyzd 7288 (IC50)glutamic acid (IC50)
Chain A, GLUTAMATE RECEPTOR SUBUNIT 2Rattus norvegicus (Norway rat)0.821
Chain A, Glutamate Receptor Subunit 2Rattus norvegicus (Norway rat)0.821
Chain B, Glutamate Receptor Subunit 2Rattus norvegicus (Norway rat)0.821
Metabotropic glutamate receptor 8Homo sapiens (human)0.0057
Glutamate receptor ionotropic, NMDA 2DHomo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 3BHomo sapiens (human)0.07
Glutamate receptor 1Rattus norvegicus (Norway rat)0.5885
Glutamate receptor 2Rattus norvegicus (Norway rat)0.5885
Glutamate receptor 3Rattus norvegicus (Norway rat)0.5885
Glutamate receptor 4Rattus norvegicus (Norway rat)0.5885
Glutamate receptor ionotropic, kainate 1Rattus norvegicus (Norway rat)0.38
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, kainate 2Rattus norvegicus (Norway rat)0.38
Glutamate receptor 1Homo sapiens (human)0.613
Glutamate receptor 2Homo sapiens (human)0.613
Glutamate receptor 3Homo sapiens (human)0.613
Glutamate receptor ionotropic, kainate 3Rattus norvegicus (Norway rat)0.38
Excitatory amino acid transporter 1Homo sapiens (human)207
Glutamate receptor 4Homo sapiens (human)0.613
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, kainate 4Rattus norvegicus (Norway rat)0.38
Glutamate receptor ionotropic, NMDA 1Homo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 2AHomo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 2BHomo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 2CHomo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, kainate 5Rattus norvegicus (Norway rat)0.38
Glutamate receptor ionotropic, NMDA 3AHomo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)0.1533

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's9 (75.00)29.6817
2010's3 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Finlayson, PG; Shaikh, AG2
Chiu, K; Raastad, M; Soleng, AF1
Buhl, EH; Cunningham, MO; Davies, CH; Kopell, N; Whittington, MA1
Chen, C1
Abbas, SY; Goldstein, PA; Harrison, NL; Ying, SW1
Abbas, SY; Goldstein, PA; Ying, SW1
Genlain, M; Godaux, E; Ris, L1
Fleming, R; Li, Q; Madison, RD; Swartzwelder, HS; Wilson, WA; Yan, H1
Eysel, UT; Koesling, D; Mergia, E; Mittmann, T; Neitz, A1
Chan, CS; Kiritani, T; Sheets, PL; Shepherd, GM; Surmeier, DJ; Suter, BA1
Chen, L; Mao, J; McCabe, MF; Mi, W; Shen, S; Sun, Y; Wang, S; Yang, J; Yang, L; You, Z; Zhang, S1

Other Studies

12 other study(ies) available for zd 7288 and glutamic acid

ArticleYear
Hyperpolarization-activated (I(h)) conductances affect brainstem auditory neuron excitability.
    Hearing research, 2003, Volume: 183, Issue:1-2

    Topics: Acoustic Stimulation; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Auditory Perception; Brain Stem; Cochlear Nerve; Dose-Response Relationship, Drug; Electrophysiology; Evoked Potentials, Auditory, Brain Stem; Excitatory Amino Acid Agonists; Glutamic Acid; Ion Channels; Male; Neurons; Olivary Nucleus; Pyrimidines; Rats; Rats, Long-Evans; Time Factors

2003
Unmyelinated axons in the rat hippocampus hyperpolarize and activate an H current when spike frequency exceeds 1 Hz.
    The Journal of physiology, 2003, Oct-15, Volume: 552, Issue:Pt 2

    Topics: Action Potentials; Animals; Axons; Cesium; Electric Stimulation; Electrophysiology; Female; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; Hydrogen; In Vitro Techniques; Ion Channels; Male; Myelin Sheath; Nerve Fibers; Neural Conduction; Pyrimidines; Rats; Receptors, Presynaptic; Synapses

2003
Gamma oscillations induced by kainate receptor activation in the entorhinal cortex in vitro.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2003, Oct-29, Volume: 23, Issue:30

    Topics: Action Potentials; Animals; Biological Clocks; Electroencephalography; Entorhinal Cortex; Excitatory Amino Acid Agonists; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; In Vitro Techniques; Interneurons; Pyramidal Cells; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, Kainic Acid; Theta Rhythm

2003
ZD7288 inhibits postsynaptic glutamate receptor-mediated responses at hippocampal perforant path-granule cell synapses.
    The European journal of neuroscience, 2004, Volume: 19, Issue:3

    Topics: Analysis of Variance; Animals; Cardiotonic Agents; Cesium; Electric Conductivity; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Hippocampus; In Vitro Techniques; Long-Term Potentiation; Male; Mice; Mice, Inbred C57BL; Neurons; Patch-Clamp Techniques; Perforant Pathway; Pyrimidines; Quinoxalines; Receptors, Glutamate; Synapses; Time Factors

2004
Excitability of auditory brainstem neurons, in vivo, is increased by cyclic-AMP.
    Hearing research, 2005, Volume: 201, Issue:1-2

    Topics: Acoustic Stimulation; Adenylyl Cyclases; Analysis of Variance; Animals; Auditory Perception; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Electrophysiology; Excitatory Amino Acid Agonists; Glutamic Acid; Ion Channels; Male; Neurons; Olivary Nucleus; Pyrimidines; Rats; Rats, Long-Evans

2005
Propofol block of I(h) contributes to the suppression of neuronal excitability and rhythmic burst firing in thalamocortical neurons.
    The European journal of neuroscience, 2006, Volume: 23, Issue:2

    Topics: Action Potentials; Analysis of Variance; Animals; Bicuculline; Cell Count; Cyclic AMP; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Free Radical Scavengers; GABA Antagonists; Gene Expression; Glutamic Acid; Green Fluorescent Proteins; Humans; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Immunohistochemistry; In Vitro Techniques; Ion Channels; Membrane Potentials; Mice; Mice, Inbred C57BL; Microscopy, Confocal; Neural Inhibition; Neurons; Patch-Clamp Techniques; Periodicity; Potassium Channels; Propofol; Pyrimidines; Thalamus; Transfection

2006
Compartmental distribution of hyperpolarization-activated cyclic-nucleotide-gated channel 2 and hyperpolarization-activated cyclic-nucleotide-gated channel 4 in thalamic reticular and thalamocortical relay neurons.
    Neuroscience, 2006, Sep-15, Volume: 141, Issue:4

    Topics: Animals; Cell Count; Cyclic Nucleotide-Gated Cation Channels; Diagnostic Imaging; Dose-Response Relationship, Radiation; Electric Stimulation; Glutamic Acid; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Immunohistochemistry; In Vitro Techniques; Ion Channels; Membrane Potentials; Mice; Mice, Inbred C57BL; Microscopy, Confocal; Neurons; Parvalbumins; Patch-Clamp Techniques; Potassium Channels; Pyrimidines; Synaptophysin; Thalamus

2006
Involvement of hyperpolarization-activated cation channels in synaptic modulation.
    Neuroreport, 2007, Aug-06, Volume: 18, Issue:12

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic Nucleotide-Gated Cation Channels; Excitatory Postsynaptic Potentials; Glutamic Acid; Hippocampus; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Neural Pathways; Neurons; Phosphodiesterase Inhibitors; Potassium; Potassium Channel Blockers; Potassium Channels; Presynaptic Terminals; Pyrimidines; Rats; Rats, Wistar; Synaptic Membranes; Synaptic Transmission

2007
Developmental sensitivity of hippocampal interneurons to ethanol: involvement of the hyperpolarization-activated current, Ih.
    Journal of neurophysiology, 2009, Volume: 101, Issue:1

    Topics: Action Potentials; Aging; Animals; Central Nervous System Depressants; Cesium; Chlorides; Cyclic Nucleotide-Gated Cation Channels; Data Interpretation, Statistical; Electrophysiology; Ethanol; GABA Antagonists; Glutamic Acid; Hippocampus; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Interneurons; Male; Patch-Clamp Techniques; Potassium Channels; Pyramidal Cells; Pyrimidines; Rats; Rats, Sprague-Dawley

2009
Presynaptic nitric oxide/cGMP facilitates glutamate release via hyperpolarization-activated cyclic nucleotide-gated channels in the hippocampus.
    The European journal of neuroscience, 2011, Volume: 33, Issue:9

    Topics: Animals; Benzazepines; Cyclic GMP; Cyclic Nucleotide-Gated Cation Channels; Glutamic Acid; Guanylate Cyclase; Hippocampus; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Mice; Mice, Inbred C57BL; Mice, Knockout; Nitric Oxide; Potassium Channels; Presynaptic Terminals; Protein Isoforms; Pyrimidines; Receptors, Cytoplasmic and Nuclear; Signal Transduction; Soluble Guanylyl Cyclase; Synaptic Transmission

2011
Corticospinal-specific HCN expression in mouse motor cortex: I(h)-dependent synaptic integration as a candidate microcircuit mechanism involved in motor control.
    Journal of neurophysiology, 2011, Volume: 106, Issue:5

    Topics: Action Potentials; Adrenergic Agonists; Animals; Corpus Callosum; Cyclic Nucleotide-Gated Cation Channels; Dendrites; Efferent Pathways; Evoked Potentials, Motor; Excitatory Postsynaptic Potentials; Female; Glutamic Acid; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Male; Membrane Proteins; Mice; Mice, Inbred C57BL; Motor Cortex; Organ Culture Techniques; Potassium Channels; Pyramidal Cells; Pyramidal Tracts; Pyrimidines; Receptors, Adrenergic; RNA, Messenger; Synapses

2011
Neuropeptide S modulates the amygdaloidal HCN activities (Ih) in rats: Implication in chronic pain.
    Neuropharmacology, 2016, Volume: 105

    Topics: Amygdala; Animals; Chronic Pain; gamma-Aminobutyric Acid; Glutamic Acid; Hyperalgesia; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Interneurons; Male; MAP Kinase Signaling System; Neuropeptides; Patch-Clamp Techniques; Potassium Channels; Pyramidal Cells; Pyrimidines; Rats; Rats, Sprague-Dawley; Tachykinins

2016