Page last updated: 2024-09-03

zd 7288 and carbachol

zd 7288 has been researched along with carbachol in 8 studies

Compound Research Comparison

Studies
(zd 7288)
Trials
(zd 7288)
Recent Studies (post-2010)
(zd 7288)
Studies
(carbachol)
Trials
(carbachol)
Recent Studies (post-2010) (carbachol)
382013713,91881968

Protein Interaction Comparison

ProteinTaxonomyzd 7288 (IC50)carbachol (IC50)
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.7849
Muscarinic acetylcholine receptor M4Homo sapiens (human)2.0626
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)3.4134
Muscarinic acetylcholine receptor M3Rattus norvegicus (Norway rat)2.9961
Muscarinic acetylcholine receptor M4Rattus norvegicus (Norway rat)2.535
Muscarinic acetylcholine receptor M5Rattus norvegicus (Norway rat)2.9961
Muscarinic acetylcholine receptor M2Rattus norvegicus (Norway rat)2.6638
Muscarinic acetylcholine receptor M1Homo sapiens (human)4.849
Muscarinic acetylcholine receptor M3Homo sapiens (human)4.99

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (25.00)18.2507
2000's2 (25.00)29.6817
2010's4 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Choi, HS; Lee, CO; Noble, D; Wang, DY1
Choate, JK; Paterson, DJ; Sears, CE1
Bulters, DO; Cobb, SR; Davies, CH; Gill, CH; Larkman, PM; Oliver, L1
Basheer, R; Brown, RE; McCarley, RW; Thakkar, MM; Winston, S1
Hasselmo, ME; Heys, JG1
Chapman, CA; Sparks, DW2
Brown, RE; McKenna, JT; Yang, C1

Other Studies

8 other study(ies) available for zd 7288 and carbachol

ArticleYear
Effect of isoprenaline, carbachol, and Cs+ on Na+ activity and pacemaker potential in rabbit SA node cells.
    The American journal of physiology, 1999, Volume: 276, Issue:1

    Topics: Action Potentials; Animals; Carbachol; Cardiac Pacing, Artificial; Cardiotonic Agents; Cesium; Electrophysiology; Female; Intracellular Membranes; Isoproterenol; Male; Pyrimidines; Rabbits; Sinoatrial Node; Sodium

1999
NO-cGMP pathway accentuates the decrease in heart rate caused by cardiac vagal nerve stimulation.
    Journal of applied physiology (Bethesda, Md. : 1985), 1999, Volume: 86, Issue:2

    Topics: Animals; Blood Pressure; Carbachol; Cardiovascular Agents; Cyclic GMP; Electric Stimulation; Guinea Pigs; Heart; Heart Rate; In Vitro Techniques; Male; Molsidomine; Nitric Oxide; Nitroprusside; Pyrimidines; Rabbits; Vagus Nerve; Vasodilator Agents

1999
Activation of Ih is necessary for patterning of mGluR and mAChR induced network activity in the hippocampal CA3 region.
    Neuropharmacology, 2003, Volume: 44, Issue:3

    Topics: Animals; Carbachol; Cardiotonic Agents; Cholinergic Agonists; Cycloleucine; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; Hippocampus; In Vitro Techniques; Nerve Net; Patch-Clamp Techniques; Pyramidal Cells; Pyrimidines; Quinoxalines; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Receptors, Muscarinic; Synaptic Transmission; Theta Rhythm

2003
Electrophysiological characterization of neurons in the dorsolateral pontine rapid-eye-movement sleep induction zone of the rat: Intrinsic membrane properties and responses to carbachol and orexins.
    Neuroscience, 2006, Volume: 143, Issue:3

    Topics: Anesthetics, Local; Animals; Animals, Newborn; Carbachol; Cardiotonic Agents; Cholinergic Agonists; Dose-Response Relationship, Radiation; Electric Stimulation; Immunohistochemistry; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Membrane Potentials; Neural Inhibition; Neurons; Neuropeptides; Neurotransmitter Agents; Orexins; Patch-Clamp Techniques; Pons; Pyrimidines; Rats; Rats, Sprague-Dawley; Sleep, REM; Tetrodotoxin; Tyrosine 3-Monooxygenase

2006
Neuromodulation of I(h) in layer II medial entorhinal cortex stellate cells: a voltage-clamp study.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2012, Jun-27, Volume: 32, Issue:26

    Topics: Animals; Animals, Newborn; Anthracenes; Atropine; Biophysical Phenomena; Carbachol; Cardiotonic Agents; Cholinergic Antagonists; Colforsin; Cyclic AMP; Cyclic Nucleotide-Gated Cation Channels; Electric Stimulation; Entorhinal Cortex; Female; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; In Vitro Techniques; Male; Membrane Potentials; Neurons; Neurotransmitter Agents; Patch-Clamp Techniques; Potassium Channels; Pyrimidines; Rats; Rats, Long-Evans; Sodium Channel Blockers; Tetrodotoxin; Time Factors

2012
Cholinergic receptor activation induces a relative facilitation of synaptic responses in the entorhinal cortex during theta- and gamma-frequency stimulation of parasubicular inputs.
    Neuroscience, 2013, Jan-29, Volume: 230

    Topics: Acetylcholine; Animals; Anthracenes; Brain Waves; Carbachol; Cholinergic Agents; Cholinergic Agonists; Dose-Response Relationship, Drug; Electric Stimulation; Electroencephalography; Entorhinal Cortex; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; Hippocampus; In Vitro Techniques; Neural Pathways; Phosphinic Acids; Propanolamines; Pyrimidines; Rats; Rats, Long-Evans; Receptors, Cholinergic; Synapses; Valine

2013
Contribution of Ih to the relative facilitation of synaptic responses induced by carbachol in the entorhinal cortex during repetitive stimulation of the parasubiculum.
    Neuroscience, 2014, Oct-10, Volume: 278

    Topics: Acetylcholine; Action Potentials; Animals; Carbachol; Cholinergic Agonists; Electric Stimulation; Entorhinal Cortex; Excitatory Postsynaptic Potentials; Hippocampus; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Male; Neural Pathways; Potassium Channels; Pyrimidines; Rats; Rats, Long-Evans; Receptors, N-Methyl-D-Aspartate; Valine

2014
Intrinsic membrane properties and cholinergic modulation of mouse basal forebrain glutamatergic neurons in vitro.
    Neuroscience, 2017, 06-03, Volume: 352

    Topics: Action Potentials; Animals; Animals, Genetically Modified; Animals, Newborn; Basal Forebrain; Benzamides; Calcium Channel Blockers; Carbachol; Cholinergic Agents; Electric Stimulation; Glutamates; Luminescent Proteins; Lysine; Mice; Neurons; Patch-Clamp Techniques; Piperidines; Pyrimidines; Red Fluorescent Protein; Sodium Channel Blockers; Tetrodotoxin; Vesicular Glutamate Transport Protein 2

2017