Page last updated: 2024-09-03

zd 7288 and capsaicin

zd 7288 has been researched along with capsaicin in 3 studies

Compound Research Comparison

Studies
(zd 7288)
Trials
(zd 7288)
Recent Studies (post-2010)
(zd 7288)
Studies
(capsaicin)
Trials
(capsaicin)
Recent Studies (post-2010) (capsaicin)
382013711,2386613,410

Protein Interaction Comparison

ProteinTaxonomyzd 7288 (IC50)capsaicin (IC50)
Transient receptor potential cation channel subfamily V member 1Rattus norvegicus (Norway rat)0.019
Lysine-specific histone demethylase 1AHomo sapiens (human)0.6
Bile salt export pumpHomo sapiens (human)10
Cytochrome P450 1A2Homo sapiens (human)3
Prostaglandin G/H synthase 1Homo sapiens (human)2.6755
Transient receptor potential cation channel subfamily V member 1Homo sapiens (human)0.008

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (66.67)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bates, SA; Benham, CD; Cairns, W; Davies, CH; Gill, CH; Hill, K; Larkman, PM; Murdock, PR; Owen, D; Powell, AJ; Randall, A; Strijbos, PJ; Yusaf, SP1
Chancellor, MB; de Groat, WC; Hayashi, Y; Masuda, N; Matsuyoshi, H; Yoshimura, N1
Eslamizade, MJ; Hosseinmardi, N; Janahmadi, M; Meftahi, GH; Mehdizadeh, M; Mousavi, SM; Saffarzadeh, F1

Other Studies

3 other study(ies) available for zd 7288 and capsaicin

ArticleYear
Characterization of the human HCN1 channel and its inhibition by capsazepine.
    British journal of pharmacology, 2004, Volume: 143, Issue:3

    Topics: Animals; Benzazepines; Capsaicin; Cell Line; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Cyclic Nucleotide-Gated Cation Channels; Dose-Response Relationship, Drug; Electric Stimulation; Humans; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Ion Channels; Membrane Potentials; Patch-Clamp Techniques; Potassium; Potassium Channels; Pyrimidines; Time Factors; Transfection

2004
Characterization of hyperpolarization-activated current (Ih) in dorsal root ganglion neurons innervating rat urinary bladder.
    Brain research, 2006, Jun-22, Volume: 1096, Issue:1

    Topics: Action Potentials; Afferent Pathways; Animals; Capsaicin; Electrophysiology; Female; Ganglia, Spinal; In Vitro Techniques; Kinetics; Membrane Potentials; Neurons; Patch-Clamp Techniques; Potassium Channels; Pyrimidines; Rats; Rats, Sprague-Dawley; Reflex; Urinary Bladder; Urination

2006
Alterations in CA1 pyramidal neuronal intrinsic excitability mediated by Ih channel currents in a rat model of amyloid beta pathology.
    Neuroscience, 2015, Oct-01, Volume: 305

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Animals; Avoidance Learning; CA1 Region, Hippocampal; Capsaicin; Disease Models, Animal; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; In Vitro Techniques; Male; Memory Disorders; Nerve Net; Neurons; Patch-Clamp Techniques; Pyrimidines; Rats; Rats, Wistar; Sensory System Agents; TRPV Cation Channels

2015