Page last updated: 2024-09-03

zd 7288 and baclofen

zd 7288 has been researched along with baclofen in 4 studies

Compound Research Comparison

Studies
(zd 7288)
Trials
(zd 7288)
Recent Studies (post-2010)
(zd 7288)
Studies
(baclofen)
Trials
(baclofen)
Recent Studies (post-2010) (baclofen)
38201376,0173721,535

Protein Interaction Comparison

ProteinTaxonomyzd 7288 (IC50)baclofen (IC50)
Gamma-aminobutyric acid type B receptor subunit 2Homo sapiens (human)0.05
Gamma-aminobutyric acid type B receptor subunit 2Rattus norvegicus (Norway rat)0.2762
Gamma-aminobutyric acid type B receptor subunit 1Homo sapiens (human)0.05
Gamma-aminobutyric acid type B receptor subunit 1Rattus norvegicus (Norway rat)0.2762

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (25.00)18.2507
2000's2 (50.00)29.6817
2010's1 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lupica, CR; Svoboda, KR1
Kelly, MJ; Reyes-Vazquez, C; Ronnekleiv, OK; Wagner, EJ1
Lisman, JE; Otmakhova, NA1
Cao, JL; Deisseroth, K; Ding, HL; Guo, XY; Han, MH; Koo, JW; Li, C; Liu, D; Liu, H; Liu, MJ; Mouzon, E; Nestler, EJ; Qian, YL; Wang, L; Wang, XY; Yang, JX; Zachariou, V; Zhang, H; Zhang, S1

Other Studies

4 other study(ies) available for zd 7288 and baclofen

ArticleYear
Opioid inhibition of hippocampal interneurons via modulation of potassium and hyperpolarization-activated cation (Ih) currents.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1998, Sep-15, Volume: 18, Issue:18

    Topics: Analgesics; Analgesics, Opioid; Animals; Baclofen; Barium; Cardiovascular Agents; Cations; Cell Size; Cells, Cultured; Cesium; Electrophysiology; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; GABA Agonists; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Hippocampus; Interneurons; Male; Membrane Potentials; Potassium; Potassium Channels; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Receptors, Opioid, mu

1998
The role of intrinsic and agonist-activated conductances in determining the firing patterns of preoptic area neurons in the guinea pig.
    Brain research, 2000, Oct-06, Volume: 879, Issue:1-2

    Topics: 4-Aminopyridine; Action Potentials; Animals; Baclofen; Barium Compounds; Cesium; Chlorides; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Excitatory Amino Acid Agonists; Female; Guinea Pigs; In Vitro Techniques; Membrane Potentials; Neurons; Nickel; Ovariectomy; Patch-Clamp Techniques; Potassium Channels; Preoptic Area; Pyrimidines; Reaction Time; Tetrodotoxin

2000
Contribution of Ih and GABAB to synaptically induced afterhyperpolarizations in CA1: a brake on the NMDA response.
    Journal of neurophysiology, 2004, Volume: 92, Issue:4

    Topics: Animals; Baclofen; Calcium; Electrophysiology; Excitatory Postsynaptic Potentials; GABA Antagonists; Hippocampus; In Vitro Techniques; Ion Channels; Patch-Clamp Techniques; Perforant Pathway; Picrotoxin; Potassium Channel Blockers; Potassium Channels; Pyrimidines; Rats; Rats, Long-Evans; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Synapses

2004
Brain-Derived Neurotrophic Factor in the Mesolimbic Reward Circuitry Mediates Nociception in Chronic Neuropathic Pain.
    Biological psychiatry, 2017, Oct-15, Volume: 82, Issue:8

    Topics: Animals; Baclofen; Benzazepines; Brain-Derived Neurotrophic Factor; Cardiotonic Agents; Disease Models, Animal; Dopaminergic Neurons; Functional Laterality; GABA-B Receptor Agonists; Limbic System; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Neural Inhibition; Neuralgia; Nociception; Pain Threshold; Proto-Oncogene Proteins c-fos; Pyrimidines; Reward

2017