Page last updated: 2024-09-03

zd 7288 and 8-bromo cyclic adenosine monophosphate

zd 7288 has been researched along with 8-bromo cyclic adenosine monophosphate in 17 studies

Compound Research Comparison

Studies
(zd 7288)
Trials
(zd 7288)
Recent Studies (post-2010)
(zd 7288)
Studies
(8-bromo cyclic adenosine monophosphate)
Trials
(8-bromo cyclic adenosine monophosphate)
Recent Studies (post-2010) (8-bromo cyclic adenosine monophosphate)
38201373,7075198

Protein Interaction Comparison

ProteinTaxonomyzd 7288 (IC50)8-bromo cyclic adenosine monophosphate (IC50)
cAMP-specific 3',5'-cyclic phosphodiesterase 4AHomo sapiens (human)7.7
cAMP-specific 3',5'-cyclic phosphodiesterase 4BHomo sapiens (human)7.7
cAMP-specific 3',5'-cyclic phosphodiesterase 4CHomo sapiens (human)7.7
cAMP-specific 3',5'-cyclic phosphodiesterase 4DHomo sapiens (human)7.7

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's11 (64.71)29.6817
2010's6 (35.29)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Beaumont, V; Zucker, RS1
Eder, C; Heinemann, U; Richter, H1
Herring, N; Paterson, DJ; Rigg, L; Terrar, DA1
Pan, ZZ1
Fyffe, RE; Morris, NP; Robertson, B1
Bie, B; Pan, ZZ; Peng, Y; Zhang, Y1
Ache, BW; Bobkov, Y; Gisselmann, G; Hatt, H; Marx, T; Neuhaus, EM; Wetzel, CH1
Baram, TZ; Rho, JM; Simeone, TA1
Abrahamczik, C; Budde, T; Caputi, L; Kanyshkova, T; Munsch, T; Pape, HC; Staak, R1
Rateau, Y; Ropert, N1
Fakler, B; Fleischmann, BK; Klöcker, N; Roeper, J; Weisser-Thomas, J; Wenzel, D; Zolles, G1
Chen, F; Chen, X; Hu, Z; Li, B; Li, Y; Xia, J; Xiong, Y; Yan, J; Ye, J; Zhou, Z1
Carloni, P; Cherubini, E; Giorgetti, A; Griguoli, M; Maul, A; Nguyen, C1
Holt, JR; Horwitz, GC; Jones, SM; Risner-Janiczek, JR1
Gonzalez-Iglesias, AE; Kretschmannova, K; Kucka, M; Stojilkovic, SS1
Chen, L; Chen, XY; Deng, WS; Han, XH; Hao, XM; Liu, HX; Liu, ZR; Sun, FJ; Wang, H; Xie, JX; Xu, R; Xue, Y; Yung, WH1
Altman, MT; Arnsten, AFT; Crimins, JL; Mazer, JA; Paspalas, CD; Wang, M; Yang, ST1

Other Studies

17 other study(ies) available for zd 7288 and 8-bromo cyclic adenosine monophosphate

ArticleYear
Enhancement of synaptic transmission by cyclic AMP modulation of presynaptic Ih channels.
    Nature neuroscience, 2000, Volume: 3, Issue:2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Action Potentials; Animals; Astacoidea; Axons; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclic Nucleotide-Gated Cation Channels; Electric Stimulation; Enzyme Inhibitors; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; In Vitro Techniques; Ion Channels; Muscles; Neuromuscular Junction; Phosphodiesterase Inhibitors; Potassium Channels; Presynaptic Terminals; Purinergic P1 Receptor Antagonists; Pyrimidines; Serotonin; Synaptic Transmission; Theophylline

2000
Hyperpolarization-activated cation currents in stellate and pyramidal neurons of rat entorhinal cortex.
    Neuroscience letters, 2000, Mar-03, Volume: 281, Issue:1

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Cations; Cesium; Dose-Response Relationship, Drug; Electrophysiology; Entorhinal Cortex; Ion Channels; Membrane Potentials; Neurons; Patch-Clamp Techniques; Potassium; Pyramidal Cells; Pyrimidines; Rats; Rats, Wistar; Sodium; Stellate Ganglion

2000
NO-cGMP pathway increases the hyperpolarisation-activated current, I(f), and heart rate during adrenergic stimulation.
    Cardiovascular research, 2001, Volume: 52, Issue:3

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; 8-Bromo Cyclic Adenosine Monophosphate; Adenine; Animals; Calcium Channel Blockers; Cesium; Chlorides; Cyclic GMP; Cyclic Nucleotide Phosphodiesterases, Type 2; Female; Guanylate Cyclase; Guinea Pigs; Heart Rate; Ion Channels; Nitric Oxide; Nitric Oxide Donors; Nitroprusside; Norepinephrine; Patch-Clamp Techniques; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Pyrimidines; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sinoatrial Node; Stimulation, Chemical

2001
Kappa-opioid receptor-mediated enhancement of the hyperpolarization-activated current (I(h)) through mobilization of intracellular calcium in rat nucleus raphe magnus.
    The Journal of physiology, 2003, May-01, Volume: 548, Issue:Pt 3

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Animals, Newborn; Barium Compounds; Benzeneacetamides; Caffeine; Calcium Signaling; Chlorides; Egtazic Acid; G Protein-Coupled Inwardly-Rectifying Potassium Channels; Kinetics; Male; Membrane Potentials; Neurons; Potassium Channels; Potassium Channels, Inwardly Rectifying; Pyrimidines; Pyrrolidines; Raphe Nuclei; Rats; Rats, Wistar; Receptors, Opioid, kappa

2003
Characterisation of hyperpolarization-activated currents (I(h)) in the medial septum/diagonal band complex in the mouse.
    Brain research, 2004, Apr-23, Volume: 1006, Issue:1

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Animals, Newborn; Cyclic Nucleotide-Gated Cation Channels; Electric Stimulation; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Immunohistochemistry; In Vitro Techniques; Ion Channel Gating; Ion Channels; Male; Membrane Potentials; Mice; Muscarine; Muscarinic Agonists; Neurons; Parvalbumins; Patch-Clamp Techniques; Potassium Channels; Pyrimidines; Septal Nuclei

2004
cAMP-mediated mechanisms for pain sensitization during opioid withdrawal.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Apr-13, Volume: 25, Issue:15

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Animals; Animals, Newborn; Behavior, Animal; Blotting, Western; Colforsin; Cyclic AMP; Dose-Response Relationship, Radiation; Drug Administration Schedule; Drug Interactions; Electric Stimulation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Gene Expression Regulation; Imines; In Vitro Techniques; Isoquinolines; Male; Membrane Potentials; Microinjections; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Opioid-Related Disorders; Oxidoreductases; Pain; Pain Measurement; Patch-Clamp Techniques; Pyrimidines; Raphe Nuclei; Rats; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sulfonamides

2005
Molecular and functional characterization of an I(h)-channel from lobster olfactory receptor neurons.
    The European journal of neuroscience, 2005, Volume: 21, Issue:6

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Amino Acid Sequence; Animals; Cell Line; Cells, Cultured; Cloning, Molecular; Cyclic Nucleotide-Gated Cation Channels; Dose-Response Relationship, Drug; Humans; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Ion Channels; Membrane Potentials; Molecular Sequence Data; Olfactory Receptor Neurons; Palinuridae; Potassium Channels; Pyrimidines

2005
Single channel properties of hyperpolarization-activated cation currents in acutely dissociated rat hippocampal neurones.
    The Journal of physiology, 2005, Oct-15, Volume: 568, Issue:Pt 2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Animals, Newborn; Cesium; Chlorides; Cyclic Nucleotide-Gated Cation Channels; Hippocampus; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; In Vitro Techniques; Ion Channel Gating; Ion Channels; Male; Membrane Potentials; Nerve Tissue Proteins; Potassium; Potassium Channels; Pyramidal Cells; Pyrimidines; Rats; Rats, Sprague-Dawley

2005
Impaired regulation of thalamic pacemaker channels through an imbalance of subunit expression in absence epilepsy.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Oct-26, Volume: 25, Issue:43

    Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Action Potentials; Adenine; Animals; Blotting, Northern; Cerebral Cortex; Cesium; Chlorides; Cyclic Nucleotide-Gated Cation Channels; Disease Models, Animal; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Electroencephalography; Enzyme Inhibitors; Epilepsy, Absence; Female; Gene Expression Regulation; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Immunohistochemistry; In Situ Hybridization; In Vitro Techniques; Ion Channels; Male; Membrane Potentials; Microinjections; Neurons; Patch-Clamp Techniques; Potassium Channels; Protein Isoforms; Pyrimidines; Rats; Rats, Mutant Strains; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thalamus

2005
Expression of a functional hyperpolarization-activated current (Ih) in the mouse nucleus reticularis thalami.
    Journal of neurophysiology, 2006, Volume: 95, Issue:5

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Animals, Newborn; Barium; Cesium; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Electric Stimulation; Gene Expression; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; In Vitro Techniques; Ion Channels; Membrane Potentials; Mice; Midline Thalamic Nuclei; Neurons; Patch-Clamp Techniques; Potassium; Potassium Channels; Pyrimidines; Sodium; Sodium Channel Blockers; Tetrodotoxin; Time Factors

2006
Pacemaking by HCN channels requires interaction with phosphoinositides.
    Neuron, 2006, Dec-21, Volume: 52, Issue:6

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Androstadienes; Animals; Biological Clocks; Brain; Cyclic Nucleotide-Gated Cation Channels; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Embryo, Mammalian; Embryo, Nonmammalian; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; In Vitro Techniques; Ion Channel Gating; Ion Channels; Male; Membrane Potentials; Mice; Mice, Inbred C57BL; Mutation; Myocytes, Cardiac; Neurons; Oocytes; Patch-Clamp Techniques; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositols; Phosphodiesterase Inhibitors; Potassium Channels; Pyrimidines; Wortmannin; Xenopus

2006
The modulation of orexin A on HCN currents of pyramidal neurons in mouse prelimbic cortex.
    Cerebral cortex (New York, N.Y. : 1991), 2010, Volume: 20, Issue:7

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Animals, Newborn; Benzoxazoles; Biophysics; Cerebral Cortex; Cyclic Nucleotide-Gated Cation Channels; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Membrane Potentials; Mice; Mice, Inbred Strains; Naphthyridines; Neuropeptides; Neurotransmitter Agents; Orexin Receptors; Orexins; Patch-Clamp Techniques; Pyramidal Cells; Pyrimidines; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Sodium Channel Blockers; Tetrodotoxin; Urea

2010
Nicotine blocks the hyperpolarization-activated current Ih and severely impairs the oscillatory behavior of oriens-lacunosum moleculare interneurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Aug-11, Volume: 30, Issue:32

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Analysis of Variance; Animals; Biological Clocks; Cardiovascular Agents; Colforsin; Cyclic Nucleotide-Gated Cation Channels; Dihydro-beta-Erythroidine; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Antagonists; Female; gamma-Aminobutyric Acid; Green Fluorescent Proteins; Hippocampus; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; In Vitro Techniques; Interneurons; Male; Mecamylamine; Mice; Mice, Transgenic; Models, Biological; Models, Molecular; Neural Inhibition; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Patch-Clamp Techniques; Potassium Channels; Pyrimidines; Somatostatin

2010
HCN channels expressed in the inner ear are necessary for normal balance function.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Nov-16, Volume: 31, Issue:46

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Age Factors; Animals; Animals, Newborn; Benzazepines; Cyclic Nucleotide-Gated Cation Channels; Ear, Inner; Electric Stimulation; Female; Forkhead Transcription Factors; Gene Expression Regulation, Developmental; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Male; Membrane Potentials; Mice; Mice, Knockout; Motion; Nerve Tissue Proteins; Neurofilament Proteins; Patch-Clamp Techniques; Piperidines; Postural Balance; Potassium Channels; Pyrimidines; RNA, Messenger; Rotarod Performance Test; Saccule and Utricle; Vestibular Evoked Myogenic Potentials

2011
The expression and role of hyperpolarization-activated and cyclic nucleotide-gated channels in endocrine anterior pituitary cells.
    Molecular endocrinology (Baltimore, Md.), 2012, Volume: 26, Issue:1

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Action Potentials; Adenylyl Cyclases; Animals; Cell Membrane; Cells, Cultured; Cesium; Cyclic GMP; Cyclic Nucleotide-Gated Cation Channels; Endocrine Cells; Female; Gonadotrophs; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Lactotrophs; Membrane Potentials; Phosphatidylinositol 4,5-Diphosphate; Pituitary Gland, Anterior; Potassium Channels; Pyrimidines; Rats; Rats, Sprague-Dawley; RNA, Messenger; Signal Transduction; Somatotrophs; Thyrotrophs; Type C Phospholipases

2012
Hyperpolarization-activated cyclic nucleotide-gated (HCN) channels regulate firing of globus pallidus neurons in vivo.
    Molecular and cellular neurosciences, 2015, Volume: 68

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; 8-Bromo Cyclic Adenosine Monophosphate; Action Potentials; Animals; Cardiotonic Agents; Cesium; Chlorides; Excitatory Amino Acid Antagonists; Globus Pallidus; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Male; Mice; Mice, Inbred C57BL; Neurons; Posture; Pyrimidines; Rats; Rats, Wistar; Subthalamic Nucleus; Valine; Wakefulness

2015
Core Differences in Synaptic Signaling Between Primary Visual and Dorsolateral Prefrontal Cortex.
    Cerebral cortex (New York, N.Y. : 1991), 2018, 04-01, Volume: 28, Issue:4

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Cardiovascular Agents; Cyclic Nucleotide Phosphodiesterases, Type 4; Dendritic Spines; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Macaca mulatta; Membrane Potentials; Microscopy, Immunoelectron; Nerve Net; Neurons; Photic Stimulation; Prefrontal Cortex; Pyrimidines; Signal Transduction; Synapses; Visual Cortex

2018