Page last updated: 2024-09-03

zd 7288 and 6-cyano-7-nitroquinoxaline-2,3-dione

zd 7288 has been researched along with 6-cyano-7-nitroquinoxaline-2,3-dione in 15 studies

Compound Research Comparison

Studies
(zd 7288)
Trials
(zd 7288)
Recent Studies (post-2010)
(zd 7288)
Studies
(6-cyano-7-nitroquinoxaline-2,3-dione)
Trials
(6-cyano-7-nitroquinoxaline-2,3-dione)
Recent Studies (post-2010) (6-cyano-7-nitroquinoxaline-2,3-dione)
38201372,6981353

Protein Interaction Comparison

ProteinTaxonomyzd 7288 (IC50)6-cyano-7-nitroquinoxaline-2,3-dione (IC50)
Glutamate receptor 1Homo sapiens (human)1.02
Glutamate receptor 2Homo sapiens (human)1.02
Glutamate receptor 3Homo sapiens (human)1.02
Glutamate receptor 4Homo sapiens (human)1.02

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (13.33)18.2507
2000's7 (46.67)29.6817
2010's5 (33.33)24.3611
2020's1 (6.67)2.80

Authors

AuthorsStudies
Cope, DW; Crunelli, V; Hughes, SW1
Carlen, PL; Perez Velazquez, JL; Skinner, FK; Tian, GF; Wu, CP; Zhang, L; Zhang, Y1
Ross, ST; Soltesz, I1
Morris, NP; Robertson, B; Southan, AP; Stephens, GJ1
Dresse, A; Massotte, L; Renette, MF; Seutin, V1
Andreasen, M; Fernandez, N; Nedergaard, S1
Bie, B; Pan, ZZ; Peng, Y; Zhang, Y1
Bartfai, T; Behrens, M; Conti, B; Korn, H; Tabarean, IV1
Israel, JM; Oliet, SH; Poulain, DA1
Bayliss, DA; Chen, X; Kapur, J; Schwartz, LC; Shu, S; Sun, C1
Koizumi, H; Moorjani, BR; Smerin, SE; Smith, JC; Yamanishi, T; Zhang, R1
Ibáñez-Sandoval, O; Koós, T; Shah, F; Tecuapetla, F; Tepper, JM; Unal, B1
Chen, L; Chen, XY; Deng, WS; Han, XH; Hao, XM; Liu, HX; Liu, ZR; Sun, FJ; Wang, H; Xie, JX; Xu, R; Xue, Y; Yung, WH1
Arts, M; Ben-Shaul, Y; Drose, DR; Gorin, M; Hanganu-Opatz, IL; Kahan, A; Mathar, R; O'Connor, S; Spehr, M; Tsitoura, C; Watznauer, K1
Correa, AMB; Dos Santos E Alhadas, É; Kushmerick, C; Naves, LA1

Other Studies

15 other study(ies) available for zd 7288 and 6-cyano-7-nitroquinoxaline-2,3-dione

ArticleYear
Dynamic clamp study of Ih modulation of burst firing and delta oscillations in thalamocortical neurons in vitro.
    Neuroscience, 1998, Volume: 87, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Bicuculline; Cardiovascular Agents; Cats; Cerebral Cortex; Excitatory Amino Acid Antagonists; Female; GABA Antagonists; Geniculate Bodies; In Vitro Techniques; Male; Neurons; Organophosphorus Compounds; Patch-Clamp Techniques; Periodicity; Pyrimidines; Rats; Rats, Wistar; Sleep; Thalamus; Wakefulness

1998
Slow oscillations (
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1998, Nov-15, Volume: 18, Issue:22

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Adenosine; Age Factors; Animals; Benzoates; Bicuculline; Cardiovascular Agents; Cesium; Chlorides; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Gap Junctions; Glycine; Hippocampus; Interneurons; Male; Membrane Potentials; Neural Pathways; Organ Culture Techniques; Patch-Clamp Techniques; Periodicity; Pyrimidines; Rats; Rats, Wistar; Receptors, GABA-A; Synapses; Temperature; Xanthines

1998
Selective depolarization of interneurons in the early posttraumatic dentate gyrus: involvement of the Na(+)/K(+)-ATPase.
    Journal of neurophysiology, 2000, Volume: 83, Issue:5

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Benzoates; Bicuculline; Brain Injuries; Dentate Gyrus; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; Glycine; In Vitro Techniques; Interneurons; Membrane Potentials; Patch-Clamp Techniques; Pyrimidines; Rats; Rats, Wistar; Sodium-Potassium-Exchanging ATPase; Strophanthidin; Tetrodotoxin; Wounds, Nonpenetrating

2000
Hyperpolarization-activated currents in presynaptic terminals of mouse cerebellar basket cells.
    The Journal of physiology, 2000, Jul-01, Volume: 526 Pt 1

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Cardiovascular Agents; Cells, Cultured; Cerebellum; Cesium; Cyclic Nucleotide-Gated Cation Channels; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Interneurons; Ion Channels; Male; Membrane Potentials; Mice; Nerve Tissue Proteins; Neural Inhibition; Patch-Clamp Techniques; Potassium Channels; Presynaptic Terminals; Purkinje Cells; Pyrimidines; Receptors, AMPA

2000
Evidence for a modulatory role of Ih on the firing of a subgroup of midbrain dopamine neurons.
    Neuroreport, 2001, Feb-12, Volume: 12, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Biological Clocks; Calcium; Calcium Channels; Cardiovascular Agents; Cations; Cesium; Dizocilpine Maleate; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Electrophysiology; Excitatory Amino Acid Antagonists; GABA Antagonists; Male; Mesencephalon; Neurons; Organ Culture Techniques; Organophosphorus Compounds; Pyrimidines; Rats; Rats, Wistar; Sulpiride

2001
Influence of the hyperpolarization-activated cation current, I(h), on the electrotonic properties of the distal apical dendrites of hippocampal CA1 pyramidal neurones.
    Brain research, 2002, Mar-15, Volume: 930, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Barium Compounds; Cesium; Chlorides; Dendrites; Electromagnetic Fields; Electrophysiology; Excitatory Amino Acid Antagonists; Hippocampus; Ion Channels; Male; Pyramidal Cells; Pyrimidines; Rats; Rats, Wistar

2002
cAMP-mediated mechanisms for pain sensitization during opioid withdrawal.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Apr-13, Volume: 25, Issue:15

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Animals; Animals, Newborn; Behavior, Animal; Blotting, Western; Colforsin; Cyclic AMP; Dose-Response Relationship, Radiation; Drug Administration Schedule; Drug Interactions; Electric Stimulation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Gene Expression Regulation; Imines; In Vitro Techniques; Isoquinolines; Male; Membrane Potentials; Microinjections; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Opioid-Related Disorders; Oxidoreductases; Pain; Pain Measurement; Patch-Clamp Techniques; Pyrimidines; Raphe Nuclei; Rats; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sulfonamides

2005
Electrophysiological properties and thermosensitivity of mouse preoptic and anterior hypothalamic neurons in culture.
    Neuroscience, 2005, Volume: 135, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Bicuculline; Calcium Channel Blockers; Cells, Cultured; Electric Impedance; Electric Stimulation; Embryo, Mammalian; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Hypothalamus, Anterior; Immunohistochemistry; Isoenzymes; Membrane Potentials; Mice; Microtubule-Associated Proteins; Muscimol; Neural Inhibition; Neurons; Nimodipine; Patch-Clamp Techniques; Pyrimidines; Receptors, AMPA; Sodium; Sodium Channel Blockers; Temperature; Tetrodotoxin; Valine

2005
Oxytocin-induced postinhibitory rebound firing facilitates bursting activity in oxytocin neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2008, Jan-09, Volume: 28, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Antagonists; Female; GABA Antagonists; gamma-Aminobutyric Acid; Hypothalamus; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Neural Inhibition; Neurons; Nickel; Ornipressin; Oxytocin; Picrotoxin; Pyrimidines; Rats; Rats, Wistar; Time Factors; Up-Regulation

2008
Homeostatic regulation of synaptic excitability: tonic GABA(A) receptor currents replace I(h) in cortical pyramidal neurons of HCN1 knock-out mice.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Feb-17, Volume: 30, Issue:7

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Anti-Anxiety Agents; Bicuculline; Cerebral Cortex; Cyclic Nucleotide-Gated Cation Channels; Desoxycorticosterone; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; GABA Agents; Homeostasis; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Male; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Knockout; Models, Neurological; Patch-Clamp Techniques; Potassium Channels; Protein Subunits; Pyramidal Cells; Pyridazines; Pyrimidines; Receptors, GABA-A; Sodium Channel Blockers; Synapses; Tetrodotoxin; Up-Regulation; Valine

2010
TASK channels contribute to the K+-dominated leak current regulating respiratory rhythm generation in vitro.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Mar-24, Volume: 30, Issue:12

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Biophysical Phenomena; Cadmium Chloride; Electric Stimulation; Excitatory Amino Acid Antagonists; Hydrogen-Ion Concentration; In Vitro Techniques; Membrane Potentials; Models, Neurological; Nerve Tissue Proteins; Neural Inhibition; Neurons; Patch-Clamp Techniques; Periodicity; Potassium; Potassium Channel Blockers; Potassium Channels, Tandem Pore Domain; Pyrimidines; Rats; Rats, Sprague-Dawley; Respiratory Center; Sodium Channel Blockers; Tetraethylammonium; Tetrodotoxin

2010
Electrophysiological and morphological characteristics and synaptic connectivity of tyrosine hydroxylase-expressing neurons in adult mouse striatum.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, May-19, Volume: 30, Issue:20

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Analysis of Variance; Animals; Anti-Inflammatory Agents; Bicuculline; Calcium Channel Blockers; Cardiovascular Agents; Cell Count; Colchicine; Corpus Striatum; Electric Stimulation; Excitatory Amino Acid Antagonists; Flufenamic Acid; GABA Antagonists; Green Fluorescent Proteins; In Vitro Techniques; Lysine; Mice; Mice, Transgenic; Neural Pathways; Neurons; Nimodipine; Patch-Clamp Techniques; Pyrimidines; Synapses; Synaptic Transmission; Time Factors; Tubulin Modulators; Tyrosine 3-Monooxygenase; Vesicular Monoamine Transport Proteins

2010
Hyperpolarization-activated cyclic nucleotide-gated (HCN) channels regulate firing of globus pallidus neurons in vivo.
    Molecular and cellular neurosciences, 2015, Volume: 68

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; 8-Bromo Cyclic Adenosine Monophosphate; Action Potentials; Animals; Cardiotonic Agents; Cesium; Chlorides; Excitatory Amino Acid Antagonists; Globus Pallidus; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Male; Mice; Mice, Inbred C57BL; Neurons; Posture; Pyrimidines; Rats; Rats, Wistar; Subthalamic Nucleus; Valine; Wakefulness

2015
Interdependent Conductances Drive Infraslow Intrinsic Rhythmogenesis in a Subset of Accessory Olfactory Bulb Projection Neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2016, Mar-16, Volume: 36, Issue:11

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Calcium; Calcium Channel Blockers; Cardiovascular Agents; Excitatory Amino Acid Antagonists; Group II Phospholipases A2; In Vitro Techniques; Mice; Mice, Inbred C57BL; Models, Neurological; Neurons; Olfactory Bulb; Olfactory Pathways; omega-Agatoxin IVA; Periodicity; Pyrimidines; Spider Venoms; Valine

2016
Mechanisms and functional impact of Group I metabotropic glutamate receptor modulation of excitability in mouse MNTB neurons.
    Synapse (New York, N.Y.), 2020, Volume: 74, Issue:3

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Amiloride; Animals; Dizocilpine Maleate; Excitatory Amino Acid Agents; Female; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Male; Methoxyhydroxyphenylglycol; Mice; Mice, Inbred C57BL; Neurons; Potassium Channel Blockers; Potassium Channels, Inwardly Rectifying; Pyrimidines; Receptors, Metabotropic Glutamate; Sodium Channel Blockers; Synaptic Potentials; Tetrodotoxin; Trapezoid Body

2020