Page last updated: 2024-09-03

zami 1327 and propranolol

zami 1327 has been researched along with propranolol in 4 studies

Compound Research Comparison

Studies
(zami 1327)
Trials
(zami 1327)
Recent Studies (post-2010)
(zami 1327)
Studies
(propranolol)
Trials
(propranolol)
Recent Studies (post-2010) (propranolol)
70033,3103,4063,218

Protein Interaction Comparison

ProteinTaxonomyzami 1327 (IC50)propranolol (IC50)
Beta-1 adrenergic receptor Cavia porcellus (domestic guinea pig)0.0347
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.0288
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)2.294
Cytochrome P450 1A2Homo sapiens (human)4
Beta-2 adrenergic receptorHomo sapiens (human)0.0114
Beta-1 adrenergic receptorHomo sapiens (human)0.0575
5-hydroxytryptamine receptor 1AHomo sapiens (human)3.9811
Beta-2 adrenergic receptorRattus norvegicus (Norway rat)0.012
Cytochrome P450 2D6Homo sapiens (human)2.9706
Beta-3 adrenergic receptorHomo sapiens (human)0.0493
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.0288
Beta-1 adrenergic receptorRattus norvegicus (Norway rat)0.012
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.0288
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0827
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.0288
Beta-3 adrenergic receptorRattus norvegicus (Norway rat)0.012
5-hydroxytryptamine receptor 2AHomo sapiens (human)1.466
5-hydroxytryptamine receptor 2CHomo sapiens (human)2.294
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.0288
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.243
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.0288
Sodium-dependent serotonin transporterHomo sapiens (human)0.38
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.342
5-hydroxytryptamine receptor 6Homo sapiens (human)3.065
Beta-2 adrenergic receptorCanis lupus familiaris (dog)0.017
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.0288
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.0288
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)2.828
Sodium channel protein type 5 subunit alphaHomo sapiens (human)2.1
Sodium/bile acid cotransporterHomo sapiens (human)5.5
Beta-2 adrenergic receptorCavia porcellus (domestic guinea pig)0.0288
GABA theta subunitRattus norvegicus (Norway rat)0.0288
Sigma non-opioid intracellular receptor 1Homo sapiens (human)2.87
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.0288

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19904 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Braga, G; Mazzocchi, C; Mazzoleni, G; Presta, M; Ragnotti, G; Riboni, L; Ziliani, S1
Fishbein, L; Jackson, CD1
Presta, M; Ragnotti, G; Riboni, L1
Braga, M; Calovini, D; Mazzocchi, C; Mazzoleni, G; Presta, M; Ragnotti, G; Zavanella, T; Ziliani, S1

Reviews

1 review(s) available for zami 1327 and propranolol

ArticleYear
A toxicological review of beta-adrenergic blockers.
    Fundamental and applied toxicology : official journal of the Society of Toxicology, 1986, Volume: 6, Issue:3

    Topics: Acebutolol; Adrenergic beta-Antagonists; Alprenolol; Animals; Atenolol; Cocarcinogenesis; Ethanolamines; Female; Kinetics; Labetalol; Lethal Dose 50; Male; Metoprolol; Mice; Mutagens; Nadolol; Neoplasms, Experimental; Oxprenolol; Pindolol; Practolol; Propanolamines; Propranolol; Rats; Sotalol; Timolol

1986

Other Studies

3 other study(ies) available for zami 1327 and propranolol

ArticleYear
Inhibition of DNA and RNA synthesis in rat liver nuclei by oncogenic and non-oncogenic beta-blockers.
    Toxicologic pathology, 1985, Volume: 13, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Atenolol; Carcinogens; Cell Nucleus; DNA; DNA-Directed RNA Polymerases; Female; In Vitro Techniques; Liver; Male; Nucleic Acid Synthesis Inhibitors; Propanolamines; Propranolol; Rats; RNA; Sex Factors

1985
Inhibition in vitro of yeast DNA polymerase I activity by beta-blockers.
    Bioscience reports, 1982, Volume: 2, Issue:1

    Topics: Adrenergic beta-Antagonists; Atenolol; Carcinogens; Cell-Free System; DNA Polymerase I; Nucleic Acid Synthesis Inhibitors; Propanolamines; Propranolol; Saccharomyces cerevisiae; Structure-Activity Relationship

1982
Thyroid and chemical hepatocarcinogenesis: further insights from the hepatocarcinogen ZAMI 1305.
    Toxicologic pathology, 1984, Volume: 12, Issue:1

    Topics: Animals; Carcinogens; Female; Hyperplasia; Liver Neoplasms, Experimental; Male; Organ Size; Propanolamines; Propranolol; Rats; Rats, Inbred Strains; Sex Factors; Thyroid Gland; Thyroidectomy; Triiodothyronine

1984