Page last updated: 2024-08-16

zaleplon and gamma-aminobutyric acid

zaleplon has been researched along with gamma-aminobutyric acid in 6 studies

*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]

*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (50.00)29.6817
2010's2 (33.33)24.3611
2020's1 (16.67)2.80

Authors

AuthorsStudies
Kitazumi, K; Mori, M; Noguchi, H; Shiba, T1
Foster, AC; Grigoriadis, DE; Gross, RS; Petroski, RE; Sullivan, SK; Verge, G1
Biggio, F; Caria, S; Follesa, P; Gorini, G; Murru, L; Sanna, E1
Abd-Elrasheed, E; El-Ashmoony, MM; El-Helaly, SN; Salah, S1
Abd-Elrasheed, E; El-Ashmoony, MM; Nageeb El-Helaly, S; Salah, S1
Abosalha, AK; Donia, AA; El-Gizawy, SA; Essa, EA; Haggag, YA; Osman, EY; Tambuwala, MM1

Other Studies

6 other study(ies) available for zaleplon and gamma-aminobutyric acid

ArticleYear
Binding and neuropharmacological profile of zaleplon, a novel nonbenzodiazepine sedative/hypnotic.
    European journal of pharmacology, 2002, Jan-02, Volume: 434, Issue:1-2

    Topics: Acetamides; Animals; Benzodiazepinones; Electroencephalography; Flunitrazepam; gamma-Aminobutyric Acid; Hypnotics and Sedatives; Male; Muscimol; Pyrimidines; Rabbits; Rats; Rats, Sprague-Dawley; Sleep

2002
Characterization of the interaction of indiplon, a novel pyrazolopyrimidine sedative-hypnotic, with the GABAA receptor.
    The Journal of pharmacology and experimental therapeutics, 2004, Volume: 311, Issue:2

    Topics: Acetamides; Animals; Azides; Benzodiazepines; Binding Sites; Brain; Cell Membrane; Cerebellum; Cerebral Cortex; Chloride Channels; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; Kinetics; Male; Pyridines; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Thiophenes; Triazolam; Tritium; Zolpidem

2004
Flumazenil selectively prevents the increase in alpha(4)-subunit gene expression and an associated change in GABA(A) receptor function induced by ethanol withdrawal.
    Journal of neurochemistry, 2007, Volume: 102, Issue:3

    Topics: Acetamides; Alcohol-Induced Disorders, Nervous System; Animals; Animals, Newborn; Anticonvulsants; Cells, Cultured; Central Nervous System Depressants; Drug Interactions; Drug Tolerance; Ethanol; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; Gene Expression Regulation; Neuronal Plasticity; Patch-Clamp Techniques; Protein Subunits; Pyrimidines; Rats; Receptors, GABA-A; Substance Withdrawal Syndrome; Up-Regulation

2007
Brain Targeted Intranasal Zaleplon Nano-emulsion: In-Vitro Characterization and Assessment of Gamma Aminobutyric Acid Levels in Rabbits' Brain and Plasma at Low and High Doses.
    Current drug delivery, 2018, Volume: 15, Issue:6

    Topics: Acetamides; Administration, Intranasal; Animals; Brain; Dose-Response Relationship, Drug; Drug Carriers; Drug Delivery Systems; Emulsions; gamma-Aminobutyric Acid; Nanoparticles; Nanotechnology; Particle Size; Pyrimidines; Rabbits; Solubility; Thermodynamics

2018
Brain-targeted intranasal zaleplon solid dispersion in hydrophilic carrier system; 2
    Drug development and industrial pharmacy, 2018, Volume: 44, Issue:5

    Topics: Acetamides; Animals; Brain; Calorimetry, Differential Scanning; gamma-Aminobutyric Acid; Hydrophobic and Hydrophilic Interactions; Microscopy, Electron, Scanning; Neurotransmitter Agents; Poloxamer; Polyethylene Glycols; Pyrimidines; Rabbits; Solubility; Tablets; X-Ray Diffraction

2018
Polymeric nanoencapsulation of zaleplon into PLGA nanoparticles for enhanced pharmacokinetics and pharmacological activity.
    Biopharmaceutics & drug disposition, 2021, Volume: 42, Issue:1

    Topics: Acetamides; Animals; Anticonvulsants; Biological Availability; gamma-Aminobutyric Acid; Hypnotics and Sedatives; Male; Nanoparticles; Polylactic Acid-Polyglycolic Acid Copolymer; Pyrimidines; Rabbits; Rats

2021