Page last updated: 2024-09-02

zacopride and spiperone

zacopride has been researched along with spiperone in 3 studies

Compound Research Comparison

Studies
(zacopride)
Trials
(zacopride)
Recent Studies (post-2010)
(zacopride)
Studies
(spiperone)
Trials
(spiperone)
Recent Studies (post-2010) (spiperone)
1804162,9441385

Protein Interaction Comparison

ProteinTaxonomyzacopride (IC50)spiperone (IC50)
Bile salt export pumpHomo sapiens (human)10
D(2) dopamine receptorHomo sapiens (human)0.0008
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.097
D(4) dopamine receptorHomo sapiens (human)0.0005
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.097
Histamine H1 receptorCavia porcellus (domestic guinea pig)0.097
D(3) dopamine receptorHomo sapiens (human)0.0635
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.097
D(2) dopamine receptorRattus norvegicus (Norway rat)0.0001
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.955

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's1 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Glennon, RA1
Ashby, CR; Edwards, E; Wang, RY1
Bockaert, J; Dumuis, A; Sebben, M1

Reviews

1 review(s) available for zacopride and spiperone

ArticleYear
Higher-end serotonin receptors: 5-HT(5), 5-HT(6), and 5-HT(7).
    Journal of medicinal chemistry, 2003, Jul-03, Volume: 46, Issue:14

    Topics: Animals; Humans; Ligands; Receptors, Serotonin; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists

2003

Other Studies

2 other study(ies) available for zacopride and spiperone

ArticleYear
Action of serotonin in the medial prefrontal cortex: mediation by serotonin3-like receptors.
    Synapse (New York, N.Y.), 1992, Volume: 10, Issue:1

    Topics: Analysis of Variance; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Frontal Lobe; Indoles; Injections, Intravenous; Iontophoresis; Male; Metergoline; Pindolol; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Spiperone; Tropisetron

1992
Pharmacological characterization of 5-hydroxytryptamine4(5-HT4) receptors positively coupled to adenylate cyclase in adult guinea pig hippocampal membranes: effect of substituted benzamide derivatives.
    Molecular pharmacology, 1990, Volume: 37, Issue:3

    Topics: Adenylyl Cyclases; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Enzyme Activation; Guinea Pigs; Hippocampus; In Vitro Techniques; Indoles; Male; Receptors, Serotonin; Serotonin; Signal Transduction; Spiperone; Structure-Activity Relationship; Tropisetron

1990