Page last updated: 2024-09-02

zacopride and ritanserin

zacopride has been researched along with ritanserin in 6 studies

Compound Research Comparison

Studies
(zacopride)
Trials
(zacopride)
Recent Studies (post-2010)
(zacopride)
Studies
(ritanserin)
Trials
(ritanserin)
Recent Studies (post-2010) (ritanserin)
1804167357571

Protein Interaction Comparison

ProteinTaxonomyzacopride (IC50)ritanserin (IC50)
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0012
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.001
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.047
Diacylglycerol kinase alphaHomo sapiens (human)9
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.047
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.0025
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.0025
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0012
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.0025
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.047
D(2) dopamine receptorRattus norvegicus (Norway rat)0.012

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (83.33)18.2507
2000's1 (16.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Glennon, RA1
Barnes, NM; Cheng, CH; Costall, B; Ge, J; Kelly, ME; Naylor, RJ1
Ashby, CR; Edwards, E; Wang, RY1
Kucharik, RF; Moyer, JA; White, SM1
Alcalde, AI; Rodríguez-Yoldi, MC; Rodríguez-Yoldi, MJ; Salvador, MT1
Beleta, J; Bernabeu, E; Bou, J; Cortijo, J; Domènech, T; Fernández, AG; Martí-Cabrera, M; Morcillo, EJ; Palacios, JM1

Reviews

1 review(s) available for zacopride and ritanserin

ArticleYear
Higher-end serotonin receptors: 5-HT(5), 5-HT(6), and 5-HT(7).
    Journal of medicinal chemistry, 2003, Jul-03, Volume: 46, Issue:14

    Topics: Animals; Humans; Ligands; Receptors, Serotonin; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists

2003

Other Studies

5 other study(ies) available for zacopride and ritanserin

ArticleYear
Profiles of interaction of R(+)/S(-)-zacopride and anxiolytic agents in a mouse model.
    European journal of pharmacology, 1992, Jul-21, Volume: 218, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Antiemetics; Behavior, Animal; Benzamides; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlordiazepoxide; Fenclonine; Granisetron; Indazoles; Male; Mice; Neurotransmitter Agents; Ondansetron; Receptors, Cholecystokinin; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Stereoisomerism

1992
Action of serotonin in the medial prefrontal cortex: mediation by serotonin3-like receptors.
    Synapse (New York, N.Y.), 1992, Volume: 10, Issue:1

    Topics: Analysis of Variance; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Frontal Lobe; Indoles; Injections, Intravenous; Iontophoresis; Male; Metergoline; Pindolol; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Spiperone; Tropisetron

1992
Effects of serotonergic agents on isolation-induced aggression.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 39, Issue:3

    Topics: Aggression; Animals; Anti-Anxiety Agents; Benzamides; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Desipramine; Haloperidol; Male; Mice; Postural Balance; Ritanserin; Serotonin; Serotonin Antagonists; Social Isolation

1991
5-HT receptor subtypes involved in the serotonin-induced inhibition of L-leucine absorption in rabbit jejunum.
    Life sciences, 1997, Volume: 61, Issue:3

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Indoles; Intestinal Absorption; Jejunum; Leucine; Male; Ondansetron; Rabbits; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides

1997
Characterization of 5-HT receptors on human pulmonary artery and vein: functional and binding studies.
    British journal of pharmacology, 1997, Volume: 122, Issue:7

    Topics: Abortifacient Agents, Nonsteroidal; Adult; Aged; Benzamides; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Dinoprost; Dioxanes; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Humans; Male; Middle Aged; Oxadiazoles; Piperazines; Piperidines; Pulmonary Artery; Pulmonary Veins; Pyridines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Sumatriptan; Vasoconstrictor Agents

1997