Page last updated: 2024-09-02

zacopride and indazoles

zacopride has been researched along with indazoles in 12 studies

Compound Research Comparison

Studies
(zacopride)
Trials
(zacopride)
Recent Studies (post-2010)
(zacopride)
Studies
(indazoles)
Trials
(indazoles)
Recent Studies (post-2010) (indazoles)
1804165,6095503,265

Protein Interaction Comparison

ProteinTaxonomyzacopride (IC50)indazoles (IC50)
Chain A, Cell Division Protein Kinase 2Homo sapiens (human)185
Chain A, CELL DIVISION PROTEIN KINASE 2Homo sapiens (human)185
Chain A, Cell Division Protein Kinase 2Homo sapiens (human)185
Chain A, CELL DIVISION PROTEIN KINASE 2Homo sapiens (human)185
Chain A, CELL DIVISION PROTEIN KINASE 2Homo sapiens (human)185
Chain A, CELL DIVISION PROTEIN KINASE 2Homo sapiens (human)185
Chain A, CELL DIVISION PROTEIN KINASE 2Homo sapiens (human)185
Chain A, CELL DIVISION PROTEIN KINASE 2Homo sapiens (human)185
Chain A, CELL DIVISION PROTEIN KINASE 2Homo sapiens (human)185
Chain A, CELL DIVISION PROTEIN KINASE 2Homo sapiens (human)185
Chain A, CELL DIVISION PROTEIN KINASE 2Homo sapiens (human)185
Chain A, CELL DIVISION PROTEIN KINASE 2Homo sapiens (human)185
Chain A, CELL DIVISION PROTEIN KINASE 2Homo sapiens (human)185
Chain A, Cell Division Protein Kinase 2Homo sapiens (human)185

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19902 (16.67)18.7374
1990's8 (66.67)18.2507
2000's1 (8.33)29.6817
2010's1 (8.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barnes, NM; Cheng, CH; Costall, B; Ge, J; Kelly, ME; Naylor, RJ1
Andrews, PL; Bhandari, P1
Gandara, DR; Hesketh, PJ1
Barnes, NM; Costall, B; Kelly, ME; Naylor, RJ; Onaivi, ES1
Costall, B; Domeney, AM; Naylor, RJ1
King, GL1
File, SE; Johnston, AL1
Barnes, NM; Costall, B; Naylor, RJ; Tattersall, FD1
Barnes, JM; Barnes, NM1
Barrett, JE; Critchett, D; Hu, W; Sokol, PT; Solomon, AJ; Toral, J; Ziai, MR1
Berry, N; McBride, WJ; McKinzie, DL; Melendez, RI; Murphy, JM; Rodd-Henricks, ZA1
Bell, RL; Bracken, AL; Deehan, GA; Ding, ZM; Hauser, SR; McBride, WJ; Rodd, ZA; Toalston, JE; Truitt, WA1

Other Studies

12 other study(ies) available for zacopride and indazoles

ArticleYear
Profiles of interaction of R(+)/S(-)-zacopride and anxiolytic agents in a mouse model.
    European journal of pharmacology, 1992, Jul-21, Volume: 218, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Antiemetics; Behavior, Animal; Benzamides; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlordiazepoxide; Fenclonine; Granisetron; Indazoles; Male; Mice; Neurotransmitter Agents; Ondansetron; Receptors, Cholecystokinin; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Stereoisomerism

1992
Preliminary evidence for the involvement of the putative 5-HT4 receptor in zacopride- and copper sulphate-induced vomiting in the ferret.
    European journal of pharmacology, 1991, Nov-12, Volume: 204, Issue:3

    Topics: Analysis of Variance; Animals; Antiemetics; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Copper; Copper Sulfate; Female; Ferrets; Granisetron; Imidazoles; Indazoles; Indoles; Loperamide; Male; Ondansetron; Receptors, Serotonin; Serotonin Antagonists; Tropisetron; Vomiting

1991
Serotonin antagonists: a new class of antiemetic agents.
    Journal of the National Cancer Institute, 1991, May-01, Volume: 83, Issue:9

    Topics: Antiemetics; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Granisetron; Humans; Imidazoles; Indazoles; Indoles; Metoclopramide; Ondansetron; Quinolizines; Receptors, Serotonin; Serotonin Antagonists; Tropanes; Tropisetron; Vomiting

1991
Ketotifen and its analogues reduce aversive responding in the rodent.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 37, Issue:4

    Topics: Animals; Avoidance Learning; Behavior, Animal; Benzamides; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cocaine; Diazepam; Ethanol; Exploratory Behavior; Granisetron; Indazoles; Ketotifen; Male; Mice; Mice, Inbred Strains; Nicotine; Radioligand Assay; Rats; Rats, Inbred Strains; Serotonin Antagonists; Social Behavior

1990
5-HT3 receptor antagonists attenuate dopamine-induced hyperactivity in the rat.
    Neuroreport, 1990, Volume: 1, Issue:1

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Dopamine; Dopamine Antagonists; Female; Granisetron; Indazoles; Indoles; Injections; Motor Activity; Nucleus Accumbens; Rats; Rats, Inbred Strains; Serotonin Antagonists; Tropisetron

1990
Emesis and defecations induced by the 5-hydroxytryptamine (5-HT3) receptor antagonist zacopride in the ferret.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:3

    Topics: Administration, Oral; Animals; Antiemetics; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Defecation; Dose-Response Relationship, Drug; Ferrets; Granisetron; Indazoles; Injections, Intravenous; Male; Metoclopramide; Pyrazoles; Serotonin; Serotonin Antagonists; Vagotomy; Vomiting

1990
Lack of effects of 5HT3 receptor antagonists in the social interaction and elevated plus-maze tests of anxiety in the rat.
    Psychopharmacology, 1989, Volume: 99, Issue:2

    Topics: Animals; Anxiety; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlordiazepoxide; Granisetron; Imidazoles; Indazoles; Male; Motor Activity; Ondansetron; Rats; Serotonin Antagonists; Social Behavior

1989
Identification of 5-HT3 recognition sites in the ferret area postrema.
    The Journal of pharmacy and pharmacology, 1988, Volume: 40, Issue:8

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carnivora; Cerebral Ventricles; Female; Ferrets; Granisetron; In Vitro Techniques; Indazoles; Radioligand Assay; Receptors, Serotonin; Serotonin Antagonists

1988
Differential binding characteristics of agonists at 5-HT3 receptor recognition sites in NG108-15 neuroblastoma-glioma cells labelled by [3H]-(S)-zacopride and [3H]granisetron.
    Biochemical pharmacology, 1993, May-25, Volume: 45, Issue:10

    Topics: Animals; Benzamides; Biguanides; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Glioma; Granisetron; Indazoles; Kinetics; Neuroblastoma; Ondansetron; Quipazine; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tritium

1993
5-HT3 receptor-independent inhibition of the depolarization-induced 86Rb efflux from human neuroblastoma cells, TE671, by ondansetron.
    The Journal of pharmacy and pharmacology, 1995, Volume: 47, Issue:7

    Topics: Anti-Anxiety Agents; Benzamides; Benzofurans; Biguanides; Bridged Bicyclo Compounds, Heterocyclic; Humans; Hypoglycemic Agents; Indazoles; Indoles; Neuroblastoma; Neurotoxins; Ondansetron; Potassium Channels; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Rubidium Radioisotopes; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship; Tropanes; Tropisetron; Tumor Cells, Cultured

1995
Effects of serotonin-3 receptor antagonists on the intracranial self-administration of ethanol within the ventral tegmental area of Wistar rats.
    Psychopharmacology, 2003, Volume: 165, Issue:3

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Central Nervous System Depressants; Drug Interactions; Ethanol; Female; Indazoles; Indoles; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Self Administration; Serotonin Antagonists; Stereoisomerism; Tropanes; Tropisetron; Ventral Tegmental Area

2003
Selective breeding for high alcohol preference increases the sensitivity of the posterior VTA to the reinforcing effects of nicotine.
    Addiction biology, 2014, Volume: 19, Issue:5

    Topics: Alcohol Drinking; Analysis of Variance; Animals; Benzamides; Breeding; Bridged Bicyclo Compounds, Heterocyclic; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Combinations; Female; Indazoles; Nicotine; Nicotinic Agonists; Rats, Wistar; Receptors, Serotonin, 5-HT3; Reinforcement, Psychology; Self Administration; Serotonin 5-HT3 Receptor Antagonists; Tropanes; Ventral Tegmental Area

2014