Compounds > zacopride
Page last updated: 2024-09-02

zacopride and gr 113808

zacopride has been researched along with gr 113808 in 8 studies

Compound Research Comparison

Studies
(zacopride)		Trials
(zacopride)		Recent Studies (post-2010)
(zacopride)		Studies
(gr 113808)		Trials
(gr 113808)		Recent Studies (post-2010) (gr 113808)
180416165135

Protein Interaction Comparison

ProteinTaxonomyzacopride (IC50)gr 113808 (IC50)
5-hydroxytryptamine receptor 4Homo sapiens (human)0.0002

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's8 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bockaert, J; Claeysen, S; Dumuis, A; Journot, L; Sebben, M1
Bockaert, J; Claeysen, S; Dumuis, A; Faye, P; Lemaire, S; Sebben, M1
Blondel, O; Dahmoune, Y; Fischmeister, R; Gastineau, M; Langlois, M1
Contesse, V; Delarue, C; Hamel, C; Lefebvre, H; Vaudry, H1
Ansanay, H; Bockaert, J; Dumuis, A; Miller, R; Rondé, P1
Bunce, KT; Gale, JD; Grossman, CJ; Humphrey, PP; Oxford, AW; Whitehead, JW1
Contesse, V; Delarue, C; Dumuis, A; Hamel, C; Lefebvre, H; Vaudry, H1
Alcalde, AI; Rodríguez-Yoldi, MC; Rodríguez-Yoldi, MJ; Salvador, MT1

Other Studies

8 other study(ies) available for zacopride and gr 113808

ArticleYear
Cloning, expression and pharmacology of the mouse 5-HT(4L) receptor.
    FEBS letters, 1996, Nov-25, Volume: 398, Issue:1

    Topics: Age Factors; Amino Acid Sequence; Animals; Animals, Newborn; Base Sequence; Binding Sites; Brain; Brain Chemistry; Cloning, Molecular; Inferior Colliculi; Mice; Molecular Sequence Data; Rats; Rats, Inbred Strains; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin Antagonists; Serotonin Receptor Agonists; Species Specificity; Transfection

1996
Cloning and expression of human 5-HT4S receptors. Effect of receptor density on their coupling to adenylyl cyclase.
    Neuroreport, 1997, Oct-20, Volume: 8, Issue:15

    Topics: Adenylyl Cyclases; Amino Acid Sequence; Animals; Benzamides; Brain Chemistry; Cloning, Molecular; Cyclic AMP; Humans; LLC-PK1 Cells; Membranes; Mice; Molecular Sequence Data; Myocardium; Polymerase Chain Reaction; Radioligand Assay; Rats; Receptors, Serotonin; Species Specificity; Swine

1997
Cloning, expression, and pharmacology of four human 5-hydroxytryptamine 4 receptor isoforms produced by alternative splicing in the carboxyl terminus.
    Journal of neurochemistry, 1998, Volume: 70, Issue:6

    Topics: Alternative Splicing; Amino Acid Sequence; Animals; Cloning, Molecular; COS Cells; Cyclic AMP; DNA, Complementary; Humans; Molecular Sequence Data; Organ Specificity; Polymerase Chain Reaction; Radioligand Assay; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; RNA, Messenger; Serotonin Antagonists; Serotonin Receptor Agonists

1998
Effect of a series of 5-HT4 receptor agonists and antagonists on steroid secretion by the adrenal gland in vitro.
    European journal of pharmacology, 1994, Nov-14, Volume: 265, Issue:1-2

    Topics: Adrenal Glands; Aldosterone; Animals; Benzamides; Benzimidazoles; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Corticosterone; Dose-Response Relationship, Drug; Indoles; Male; Radioligand Assay; Ranidae; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Stereoisomerism; Structure-Activity Relationship; Sulfonamides; Tropisetron

1994
Homologous desensitization of 5-hydroxytryptamine4 receptors in rat esophagus: functional and second messenger studies.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 272, Issue:3

    Topics: 4-Aminobenzoic Acid; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cyclic AMP; Esophagus; In Vitro Techniques; Indoles; Muscle Relaxation; Muscle, Smooth; para-Aminobenzoates; Rats; Receptors, Serotonin; Serotonin; Signal Transduction; Sulfonamides; Time Factors

1995
GR113808: a novel, selective antagonist with high affinity at the 5-HT4 receptor.
    British journal of pharmacology, 1994, Volume: 111, Issue:1

    Topics: 5-Methoxytryptamine; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Colon; Dose-Response Relationship, Drug; Esophagus; Female; Guinea Pigs; Hemodynamics; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Rabbits; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sincalide; Sulfonamides

1994
Activation of 5-hydroxytryptamine4 receptors causes calcium influx in adrenocortical cells: involvement of calcium in 5-hydroxytryptamine-induced steroid secretion.
    Molecular pharmacology, 1996, Volume: 49, Issue:3

    Topics: Adrenal Cortex; Adrenal Cortex Hormones; Animals; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Calcium; Cells, Cultured; Cyclic AMP; Indoles; Male; Rana ridibunda; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Signal Transduction; Sulfonamides

1996
5-HT receptor subtypes involved in the serotonin-induced inhibition of L-leucine absorption in rabbit jejunum.
    Life sciences, 1997, Volume: 61, Issue:3

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Indoles; Intestinal Absorption; Jejunum; Leucine; Male; Ondansetron; Rabbits; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides

1997