zacopride has been researched along with bemesetron in 10 studies
| Studies (zacopride) | Trials (zacopride) | Recent Studies (post-2010) (zacopride) | Studies (bemesetron) | Trials (bemesetron) | Recent Studies (post-2010) (bemesetron) |
|---|---|---|---|---|---|
| 180 | 4 | 16 | 254 | 3 | 25 |
| Protein | Taxonomy | zacopride (IC50) | bemesetron (IC50) |
|---|---|---|---|
| 5-hydroxytryptamine receptor 3E | Homo sapiens (human) | 0.0093 | |
| 5-hydroxytryptamine receptor 3B | Homo sapiens (human) | 0.0093 | |
| 5-hydroxytryptamine receptor 3A | Rattus norvegicus (Norway rat) | 0.097 | |
| 5-hydroxytryptamine receptor 3A | Homo sapiens (human) | 0.0928 | |
| 5-hydroxytryptamine receptor 3D | Homo sapiens (human) | 0.0093 | |
| 5-hydroxytryptamine receptor 3C | Homo sapiens (human) | 0.0093 | |
| 5-hydroxytryptamine receptor 3B | Rattus norvegicus (Norway rat) | 0.097 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 1 (10.00) | 18.7374 |
| 1990's | 9 (90.00) | 18.2507 |
| 2000's | 0 (0.00) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Airey, JE; Campbell, HF; Golec, S; Klein, S; Powers, M; Rodriguez, W; Schnapper, M; Studt, W; Woodward, R; Youssefyeh, RD | 1 |
| Bradley, G; Coleman, J; Rhodes, KF; Taylor, A; Ward, TJ; White, JC | 1 |
| Bloomquist, W; Cohen, ML; Reid, LR; Robertson, DW; Schenck, K; Wong, DT | 1 |
| Adrien, J; Franc, B; Haj-Dahmane, S; Hamon, M; Jolas, T; Lanfumey, L; Tissier, MH | 1 |
| Hitzemann, R; Svingos, AL | 1 |
| Barrett, JE; Grant, KA | 1 |
| Gandara, DR; Hesketh, PJ | 1 |
| Lucot, JB | 1 |
| Barrett, JE; Critchett, D; Hu, W; Sokol, PT; Solomon, AJ; Toral, J; Ziai, MR | 1 |
| Saederup, E; Squires, RF | 1 |
10 other study(ies) available for zacopride and bemesetron
| Article | Year |
|---|---|
Development of high-affinity 5-HT3 receptor antagonists. 2. Two novel tricyclic benzamides.
Topics: Amides; Animals; Antiemetics; Benzamides; Benzofurans; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Cisplatin; Dogs; Ferrets; Guinea Pigs; Ileum; Molecular Structure; Muscle Contraction; Rats; Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Vomiting; X-Ray Diffraction | 1992 |
Novel antagonists of the 5-HT3 receptor. Synthesis and structure-activity relationships of (2-alkoxybenzoyl)ureas.
Topics: Animals; Benzoates; In Vitro Techniques; Magnetic Resonance Spectroscopy; Male; Rats; Rats, Inbred Strains; Serotonin Antagonists; Structure-Activity Relationship; Urea; Vagus Nerve; X-Ray Diffraction | 1992 |
Synthesis and biochemical evaluation of tritium-labeled 1-methyl-N-(8-methyl-8-azabicyclo[3.2.1]oct-3-yl)-1H-indazole-3-carboxa mide, a useful radioligand for 5HT3 receptors.
Topics: Animals; Cell Membrane; Cerebral Cortex; Guinea Pigs; Heart Rate; Ileum; Indazoles; Male; Methylation; Myocardium; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Tritium; Tropanes | 1990 |
Central action of 5-HT3 receptor ligands in the regulation of sleep-wakefulness and raphe neuronal activity in the rat.
Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Electrophysiology; Indoles; Male; Neurons; Ondansetron; Propranolol; Pyrimidines; Raphe Nuclei; Rats; Rats, Wistar; Receptors, Serotonin; Reference Values; Serotonin; Serotonin Antagonists; Sleep; Time Factors; Tropanes; Tropisetron; Wakefulness | 1992 |
5-HT3 receptor antagonists block cocaine-induced locomotion via a PCPA-sensitive mechanism.
Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cocaine; Dose-Response Relationship, Drug; Fenclonine; Indoles; Male; Motor Activity; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Tropanes; Tropisetron | 1992 |
Blockade of the discriminative stimulus effects of ethanol with 5-HT3 receptor antagonists.
Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Columbidae; Conditioning, Operant; Discrimination, Psychological; Dose-Response Relationship, Drug; Ethanol; Haloperidol; Indoles; Ketanserin; Male; Serotonin Antagonists; Tropanes; Tropisetron | 1991 |
Serotonin antagonists: a new class of antiemetic agents.
Topics: Antiemetics; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Granisetron; Humans; Imidazoles; Indazoles; Indoles; Metoclopramide; Ondansetron; Quinolizines; Receptors, Serotonin; Serotonin Antagonists; Tropanes; Tropisetron; Vomiting | 1991 |
Blockade of 5-hydroxytryptamine3 receptors prevents cisplatin-induced but not motion- or xylazine-induced emesis in the cat.
Topics: Animals; Antiemetics; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cats; Cisplatin; Indoles; Motion Sickness; Receptors, Serotonin; Serotonin Antagonists; Thiazines; Tropanes; Tropisetron; Vomiting; Xylazine | 1989 |
5-HT3 receptor-independent inhibition of the depolarization-induced 86Rb efflux from human neuroblastoma cells, TE671, by ondansetron.
Topics: Anti-Anxiety Agents; Benzamides; Benzofurans; Biguanides; Bridged Bicyclo Compounds, Heterocyclic; Humans; Hypoglycemic Agents; Indazoles; Indoles; Neuroblastoma; Neurotoxins; Ondansetron; Potassium Channels; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Rubidium Radioisotopes; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship; Tropanes; Tropisetron; Tumor Cells, Cultured | 1995 |
Clozapine's antipsychotic effects do not depend on blockade of 5-HT3 receptors.
Topics: Animals; Antipsychotic Agents; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Clozapine; Drug Interactions; Female; GABA Antagonists; gamma-Aminobutyric Acid; Male; Ondansetron; Quinacrine; Quipazine; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Sulfur Radioisotopes; Tropanes | 1999 |