Page last updated: 2024-08-20

yohimbine and mk 912

yohimbine has been researched along with mk 912 in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19902 (15.38)18.7374
1990's4 (30.77)18.2507
2000's6 (46.15)29.6817
2010's1 (7.69)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chen, R; Clineschmidt, BV; Flagg, SD; Huff, JR; Pettibone, DJ; Totaro, JA; Young, SD1
Clineschmidt, BV; Hucker, HB; Huff, JR; Lis, EV; Lotti, VJ; Pettibone, DJ; Reiss, DR; Sweeney, BM; Vacca, J1
Harrison, JK; Huang, L; Muir, JC; Okusa, MD; Rosin, DL1
Eglen, RM; Jasper, JR; Luong, LA; MacLennan, SJ; To, ZP1
Akerman, KE; Cockcroft, V; Huifang, G; Jansson, CC; Kukkonen, JP; Savola, JM; Wurster, S1
Dambrova, M; Gu, Y; Näsman, J; Schiöth, HB; Uhlén, S; Wikberg, JE; Wikberg-Matsson, A1
Bylund, DB; Gerety, ME; Happe, HK; Murrin, LC1
Arulmani, U; Centurión, D; Saxena, PR; Valdivia, LF; Villalón, CM1
Centurión, D; Gupta, S; Jiménez-Mena, LR; Lozano-Cuenca, J; MaassenVanDenBrink, A; Mehrotra, S; Muñoz-Islas, E; Sánchez-López, A; Villalón, CM1
Centurión, D; Görnemann, T; Jähnichen, S; Kleuser, B; Pertz, HH; Villalón, CM; von Wenckstern, H1
Johnson, MS; Karlsson, HK; Laurila, JM; Rantanen, MJ; Ruuskanen, JO; Scheinin, M; Xhaard, H1
Albarrán-Juárez, JA; Centurión, D; Görnemann, T; Lozano-Cuenca, J; Pertz, HH; Villalón, CM1
Centurión, D; Hofmann, RA; Jantschak, F; Pertz, HH; Popp, AM; Villalón, CM1

Other Studies

13 other study(ies) available for yohimbine and mk 912

ArticleYear
[3H]L-657,743 (MK-912): a new, high affinity, selective radioligand for brain alpha 2-adrenoceptors.
    Life sciences, 1989, Volume: 44, Issue:7

    Topics: Adrenergic alpha-Antagonists; Animals; Cerebral Cortex; Humans; In Vitro Techniques; Male; Quinolizines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine

1989
A peripherally acting alpha-2 adrenoceptor antagonist: L-659,066.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Blood-Brain Barrier; Callitrichinae; Clonidine; Decerebrate State; Dihydroxyphenylalanine; Gastrointestinal Motility; Male; Muscle Contraction; Quinolizines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Vas Deferens; Yohimbine

1988
Regulation of rat renal alpha 2 B-adrenergic receptors by potassium depletion.
    The American journal of physiology, 1994, Volume: 266, Issue:2 Pt 2

    Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Blotting, Northern; Blotting, Western; Cell Membrane; Gene Expression; Kidney; Kinetics; Male; Potassium Deficiency; Quinolizines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; RNA, Messenger; Tritium; Yohimbine

1994
Characterization of alpha 2-adrenoceptors mediating contraction of dog saphenous vein: identity with the human alpha 2A subtype.
    British journal of pharmacology, 1997, Volume: 121, Issue:8

    Topics: Animals; Cricetinae; Dogs; Female; Humans; In Vitro Techniques; Male; Norepinephrine; Phenoxybenzamine; Quinolizines; Receptors, Adrenergic, alpha-2; Saphenous Vein; Vasoconstriction; Yohimbine

1997
Different apparent modes of inhibition of alpha2A-adrenoceptor by alpha2-adrenoceptor antagonists.
    European journal of pharmacology, 1997, Sep-17, Volume: 335, Issue:1

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Humans; Idazoxan; Quinolizines; Receptors, Adrenergic, alpha-2; Tritium; Tumor Cells, Cultured; Yohimbine

1997
[3H]RS79948-197 binding to human, rat, guinea pig and pig alpha2A-, alpha2B- and alpha2C-adrenoceptors. Comparison with MK912, RX821002, rauwolscine and yohimbine.
    European journal of pharmacology, 1998, Feb-05, Volume: 343, Issue:1

    Topics: Adrenergic Agents; Animals; Guinea Pigs; Humans; Idazoxan; Isoquinolines; Naphthyridines; Quinolizines; Rats; Receptors, Adrenergic, alpha-2; Swine; Yohimbine

1998
Inverse agonism at alpha(2)-adrenoceptors in native tissue.
    European journal of pharmacology, 2000, Jun-16, Volume: 398, Issue:2

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Brain; Dose-Response Relationship, Drug; Guanosine Triphosphate; Idazoxan; Kinetics; Protein Binding; Quinolizines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Tritium; Yohimbine

2000
5-HT1B receptors, alpha2A/2C- and, to a lesser extent, alpha1-adrenoceptors mediate the external carotid vasoconstriction to ergotamine in vagosympathectomised dogs.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:1

    Topics: Animals; Biphenyl Compounds; Blood Pressure; Carotid Artery, External; Dogs; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Therapy, Combination; Ergotamine; Hypotension; Imidazoles; Indoles; Injections, Intravenous; Isoindoles; Male; Piperazines; Piperidones; Prazosin; Quinolizines; Receptor, Serotonin, 5-HT1B; Receptors, Adrenergic, alpha; Regional Blood Flow; Spiro Compounds; Sympathectomy; Vagotomy; Vasoconstriction; Yohimbine

2004
Clonidine inhibits the canine external carotid vasodilatation to capsaicin by alpha2A/2C-adrenoceptors.
    European journal of pharmacology, 2006, Aug-14, Volume: 543, Issue:1-3

    Topics: Acetylcholine; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Flow Velocity; Blood Pressure; Calcitonin Gene-Related Peptide; Capsaicin; Carotid Artery, External; Clonidine; Dogs; Dose-Response Relationship, Drug; Heart Rate; Imidazoles; Indoles; Isoindoles; Male; Phenylephrine; Quinolizines; Receptors, Adrenergic, alpha-2; Reproducibility of Results; Vasodilation; Yohimbine

2006
Characterization of the postjunctional alpha 2C-adrenoceptor mediating vasoconstriction to UK14304 in porcine pulmonary veins.
    British journal of pharmacology, 2007, Volume: 151, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Gene Expression; Imidazoles; In Vitro Techniques; Indoles; Isoindoles; Isoquinolines; Neuromuscular Junction; Norepinephrine; Piperazines; Prazosin; Pulmonary Veins; Quinolizines; Quinoxalines; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Swine; Vasoconstriction; Yohimbine

2007
The second extracellular loop of alpha2A-adrenoceptors contributes to the binding of yohimbine analogues.
    British journal of pharmacology, 2007, Volume: 151, Issue:8

    Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; CHO Cells; Cricetinae; Cricetulus; Humans; Isoquinolines; Ligands; Mice; Models, Molecular; Mutation; Naphthyridines; Quinolizines; Receptors, Adrenergic, alpha-2; Species Specificity; Yohimbine

2007
Pharmacological profile of the clonidine-induced inhibition of vasodepressor sensory outflow in pithed rats: correlation with alpha(2A/2C)-adrenoceptors.
    British journal of pharmacology, 2008, Volume: 154, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Blood Vessels; Calcitonin Gene-Related Peptide; Clonidine; Decerebrate State; Electric Stimulation; Heart Rate; Imidazoles; In Vitro Techniques; Isoindoles; Male; Neurons, Afferent; Quinolizines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Yohimbine

2008
Postjunctional α2C-adrenoceptors mediate vasoconstriction in rat tail artery: influence of precontraction and temperature on vasoreactivity.
    Naunyn-Schmiedeberg's archives of pharmacology, 2010, Volume: 382, Issue:5-6

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Antagonists; Animals; Arteries; Brimonidine Tartrate; Dioxanes; Imidazoles; In Vitro Techniques; Isoindoles; Isoquinolines; Male; Mice; Mice, Inbred C57BL; Piperazines; Prazosin; Quinolizines; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Serotonin; Tail; Temperature; Vasoconstriction; Yohimbine

2010
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