yohimbine has been researched along with ici 118551 in 36 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 10 (27.78) | 18.7374 |
1990's | 13 (36.11) | 18.2507 |
2000's | 7 (19.44) | 29.6817 |
2010's | 6 (16.67) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET | 1 |
Bartoccini, F; Carminati, P; Castorina, M; Di Cesare, MA; Di Serio, S; Gallo, G; Ghirardi, O; Giorgi, F; Giorgi, L; Minetti, P; Piersanti, G; Tarzia, G; Tinti, MO | 1 |
Altenbach, RJ; Brioni, JD; Carr, TL; Chandran, P; Cowart, MD; Esbenshade, TA; Honore, P; Hsieh, GC; Lewis, LG; Liu, H; Manelli, AM; Marsh, KC; Milicic, I; Miller, TR; Strakhova, MI; Vortherms, TA; Wakefield, BD; Wetter, JM; Witte, DG | 1 |
Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K | 1 |
Colau, D; Dolusić, E; Frédérick, R; Larrieu, P; Masereel, B; Moineaux, L; Pilotte, L; Pochet, L; Stroobant, V; Van den Eynde, B; Wouters, J | 1 |
Anzini, M; Brogi, S; Butini, S; Campiani, G; Cappelli, A; Caselli, G; Castriconi, F; Gemma, S; Giordani, A; Giorgi, G; Giuliani, G; Lanza, M; Letari, O; Makovec, F; Manini, M; Mennuni, L; Valenti, S | 1 |
Belyakov, S; Dambrova, M; Kazoka, H; Kuznecovs, J; Lebedev, A; Liepinsh, E; Mishnev, A; Orlova, N; Ponomaryov, Y; Vavers, E; Veinberg, G; Vikainis, S; Vilskersts, R; Vorona, M; Zvejniece, L | 1 |
Bednarski, M; Gunia-Krzyżak, A; Marona, H; Nitek, W; Pękala, E; Powroźnik, B; Słoczyńska, K; Walczak, M; Waszkielewicz, AM; Żesławska, E | 1 |
Filipek, B; Gunia-Krzyżak, A; Marona, H; Nitek, W; Pańczyk, K; Pękala, E; Rapacz, A; Słoczyńska, K; Waszkielewicz, AM; Żelaszczyk, D; Żesławska, E | 1 |
Dandona, P; DeSouza, V; Gill, J; Jeremy, JY; Wakeling, A | 1 |
Goldberg, SR; Schindler, CW; Tella, SR | 1 |
Amstislavskaja, TG; Naumenko, EV; Osadchuk, AV | 1 |
Hyman, AL; Kadowitz, PJ; Lippton, HL | 1 |
Hyman, AL; Kadowitz, PJ | 2 |
Bos, EA; Knot, HJ; Remie, R; Zaagsma, J | 1 |
Costall, B; Naylor, RJ; Tan, CC | 1 |
Bouritius, H; Bruntink, R; Dreteler, GH; Remie, R; Scheurink, AJ; Steffens, AB; Zaagsma, J | 1 |
Göthert, M; Hentrich, F | 1 |
DiBona, GF; Jones, S; Koepke, JP | 1 |
Knudtzon, J | 1 |
De Jonge, A; Thoolen, MJ; Timmermans, PB; Van Zwieten, PA; Wilffert, B | 1 |
Nakashima, M; Vanhoutte, PM | 1 |
Benthem, L; Coppes, RP; Smit, J; Van der Leest, J; Zaagsma, J | 1 |
Abe, K; Hidaka, S; Okina, A; Tashiro, M | 1 |
Arner, P; Blaak, EE; Gafvels, ME; Lonnqvist, F; Shimizu, M | 1 |
Burrello, N; Calogero, AE; D'Agata, R; Ossino, AM; Weber, RF | 1 |
Goepel, M; Michel, MC; Rübben, H; Wittmann, A | 1 |
Dang, H; Gruber, DD; Scofield, MA; Shimozono, M; Wangemann, P | 1 |
de Haas, JR; Kockelbergh, PG; Roffel, AF; Terpstra, JS; van der Zwaag, M; Zaagsma, J | 1 |
Chen, SF; Cheng, FC; Chung, LJ; Hsueh, CM; Huang, HJ; Kuo, JS; Lin, RJ | 1 |
Castrucci, AM; de Oliveira, AR; Scarparo, AC; Visconti, MA | 1 |
Lee, TJ; Sarwinski, S; Zhang, W | 1 |
Lelieveld, H; Nieveen, M; Ponce, MC; Steffens, A; van den Thillart, G; Van Raaij, M; Vianen, G; Zaagsma, J | 1 |
Cardin, JA; Schmidt, MF | 1 |
Barrot, M; Doridot, S; Freund-Mercier, MJ; Hein, L; Petit-Demoulière, N; Tessier, LH; Yalcin, I | 1 |
36 other study(ies) available for yohimbine and ici 118551
Article | Year |
---|---|
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium | 1985 |
2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A2A adenosine receptor antagonists. Design, synthesis, and pharmacological characterization.
Topics: Adenine; Adenosine A2 Receptor Antagonists; Animals; Cell Line; Cricetinae; Cricetulus; Drug Design; Humans; Imidazoles; Male; Models, Molecular; Motor Activity; Purines; Radioligand Assay; Rats; Rats, Inbred F344; Structure-Activity Relationship; Triazoles | 2005 |
cis-4-(Piperazin-1-yl)-5,6,7a,8,9,10,11,11a-octahydrobenzofuro[2,3-h]quinazolin-2-amine (A-987306), a new histamine H4R antagonist that blocks pain responses against carrageenan-induced hyperalgesia.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzofurans; Carrageenan; Disease Models, Animal; Drug Design; Drug Evaluation, Preclinical; Humans; Hyperalgesia; Ligands; Mice; Molecular Structure; Pain; Peritonitis; Quinazolines; Rats; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Stereoisomerism; Structure-Activity Relationship | 2008 |
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship | 2010 |
Tryptophan 2,3-dioxygenase (TDO) inhibitors. 3-(2-(pyridyl)ethenyl)indoles as potential anticancer immunomodulators.
Topics: Animals; Antineoplastic Agents; Biological Availability; Cell Line; Drug Design; Enzyme Inhibitors; Humans; Immunologic Factors; Indoles; Kinetics; Mice; Neoplasms; Structure-Activity Relationship; Tryptophan Oxygenase | 2011 |
Synthesis and structure-activity relationship studies in serotonin 5-HT(1A) receptor agonists based on fused pyrrolidone scaffolds.
Topics: Animals; Area Under Curve; Humans; Intestinal Absorption; Ligands; Male; Metabolic Clearance Rate; Models, Chemical; Models, Molecular; Molecular Structure; Protein Binding; Protein Structure, Tertiary; Pyrrolidinones; Radioligand Assay; Receptor, Serotonin, 5-HT1A; Receptors, Serotonin, 5-HT3; Serotonin 5-HT1 Receptor Agonists; Structure-Activity Relationship | 2013 |
Synthesis and biological evaluation of 2-(5-methyl-4-phenyl-2-oxopyrrolidin-1-yl)-acetamide stereoisomers as novel positive allosteric modulators of sigma-1 receptor.
Topics: Acetamides; Allosteric Regulation; Animals; Rats; Rats, Wistar; Receptors, sigma; Sigma-1 Receptor; Stereoisomerism; Structure-Activity Relationship | 2013 |
Design, physico-chemical properties and biological evaluation of some new N-[(phenoxy)alkyl]- and N-{2-[2-(phenoxy)ethoxy]ethyl}aminoalkanols as anticonvulsant agents.
Topics: Amino Alcohols; Animals; Anticonvulsants; Chemistry, Physical; Dose-Response Relationship, Drug; Drug Design; Epilepsy; Male; Mice; Microsomes, Liver; Molecular Structure; Pilocarpine | 2016 |
Structure-anticonvulsant activity studies in the group of (E)-N-cinnamoyl aminoalkanols derivatives monosubstituted in phenyl ring with 4-Cl, 4-CH
Topics: Amino Alcohols; Animals; Anticonvulsants; Crystallography, X-Ray; Disease Models, Animal; Dose-Response Relationship, Drug; Electroshock; Mice; Models, Molecular; Molecular Structure; Rats; Seizures; Structure-Activity Relationship | 2017 |
Differential changes in alpha- and beta-adrenoceptor linked [45Ca2+] uptake in platelets from patients with anorexia nervosa.
Topics: Adolescent; Adrenergic beta-Antagonists; Adult; Anorexia Nervosa; Atenolol; Blood Platelets; Bucladesine; Calcium; Calcium Radioisotopes; Epinephrine; Female; Humans; In Vitro Techniques; Isoproterenol; Kinetics; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta; Reference Values; Yohimbine | 1992 |
Adrenoceptor mechanisms in the cardiovascular effects of cocaine in conscious squirrel monkeys.
Topics: Adrenergic beta-Antagonists; Animals; Atenolol; Blood Pressure; Cocaine; Heart Rate; Labetalol; Male; Phentolamine; Prazosin; Propanolamines; Propranolol; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Saimiri; Yohimbine | 1992 |
The role of the adrenoceptors in the activation of the hypothalamic-pituitary-testicular complex of mice induced by the presence of a female.
Topics: Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Female; Hypothalamo-Hypophyseal System; Male; Metoprolol; Mice; Mice, Inbred CBA; Phentolamine; Prazosin; Propanolamines; Propranolol; Radioimmunoassay; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Sexual Behavior, Animal; Testis; Testosterone; Yohimbine | 1991 |
Analysis of pulmonary vascular responses in cats to sympathetic nerve stimulation under elevated tone conditions. Evidence that neuronally released norepinephrine acts on alpha 1-, alpha 2-, and beta 2-adrenoceptors.
Topics: Adrenergic beta-Antagonists; Animals; Blood Pressure; Cats; Electric Stimulation; Female; Lung; Male; Norepinephrine; Prazosin; Propanolamines; Propranolol; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Sympathetic Nervous System; Yohimbine | 1990 |
Analysis of responses to sympathetic nerve stimulation in the feline pulmonary vascular bed.
Topics: Adrenergic beta-Antagonists; Animals; Cats; Electric Stimulation; Lung; Norepinephrine; Prazosin; Propanolamines; Propranolol; Pulmonary Circulation; Sympathetic Nervous System; Tyramine; Vascular Resistance; Yohimbine | 1989 |
Characterization of presynaptic beta-adrenoceptors facilitating endogenous noradrenaline release in the portal vein of permanently cannulated, freely moving rats.
Topics: Animals; Catheterization; Drug Synergism; Fenoterol; Imidazoles; Male; Norepinephrine; Portal Vein; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Yohimbine | 1988 |
Mechanism of action of apomorphine on rat gastric secretion.
Topics: Adrenergic beta-Antagonists; Animals; Antipsychotic Agents; Apomorphine; Atenolol; Drug Interactions; Gastric Acid; Gastric Mucosa; Male; Prazosin; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Time Factors; Yohimbine | 1985 |
Enhancement of alpha- and beta-adrenoceptor responses by elevations in vascular tone in pulmonary circulation.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-Antagonists; Animals; Brimonidine Tartrate; Cats; Female; Male; Muscle Tonus; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Prazosin; Propanolamines; Pulmonary Circulation; Quinoxalines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Yohimbine | 1986 |
Adrenal and sympathetic catecholamines in exercising rats.
Topics: Adrenal Medulla; Animals; Cardiac Catheterization; Epinephrine; Fenoterol; Male; Norepinephrine; Physical Conditioning, Animal; Propanolamines; Rats; Rats, Inbred Strains; Sympathetic Nervous System; Yohimbine | 1989 |
Identification of presynaptic beta 2-adrenoceptors on the sympathetic nerve fibres of the human pulmonary artery.
Topics: Cocaine; Corticosterone; Dose-Response Relationship, Drug; Electric Stimulation; Ethanolamines; Humans; Isoproterenol; Mathematics; Nerve Fibers; Norepinephrine; Procaterol; Propanolamines; Pulmonary Artery; Receptors, Adrenergic, beta; Sympathetic Nervous System; Yohimbine | 1985 |
Alpha 2-adrenoceptors in amygdala control renal sympathetic nerve activity and renal function in conscious spontaneously hypertensive rats.
Topics: Amygdala; Animals; Blood Pressure; Consciousness; Guanabenz; Hypertension; Kidney; Male; Propanolamines; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha; Stress, Physiological; Sympathetic Nervous System; Yohimbine | 1987 |
Adrenergic effects on plasma levels of glucagon, insulin, glucose and free fatty acids in rabbits--influences of selective blocking drugs.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Blood Glucose; Epinephrine; Fatty Acids, Nonesterified; Female; Glucagon; Insulin; Isoproterenol; Metoprolol; Prazosin; Propanolamines; Rabbits; Yohimbine | 1984 |
Heterogeneity of the interaction between alpha 1- and alpha 2-adrenoceptor agonists with their respective receptors in the vascular system of the pithed rat.
Topics: Adrenergic alpha-Agonists; Animals; Azepines; Blood Pressure; Cocaine; Dopamine; Electric Stimulation; Emetics; Ethanolamines; Hemodynamics; Male; Naphthols; Prazosin; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tetrahydronaphthalenes; Yohimbine | 1984 |
Isoproterenol causes hyperpolarization through opening of ATP-sensitive potassium channels in vascular smooth muscle of the canine saphenous vein.
Topics: Animals; Atenolol; Charybdotoxin; Colforsin; Dogs; Female; Glyburide; Ion Channel Gating; Isoproterenol; Male; Membrane Potentials; Muscle, Smooth, Vascular; Ouabain; Potassium Channels; Propanolamines; Receptors, Adrenergic, beta; Saphenous Vein; Scorpion Venoms; Yohimbine | 1995 |
Co-released adrenaline markedly facilitates noradrenaline overflow through prejunctional beta 2-adrenoceptors during swimming exercise.
Topics: Adrenergic beta-Antagonists; Animals; Cocaine; Drug Synergism; Epinephrine; Male; Norepinephrine; Physical Conditioning, Animal; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta-2; Swimming; Sympathetic Nervous System; Yohimbine | 1995 |
The effects of tyramine on salivary flow rate and protein secretion by rat submandibular glands.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Isoelectric Focusing; Male; Metoprolol; Phenoxybenzamine; Prazosin; Propanolamines; Propranolol; Protease Inhibitors; Rats; Rats, Sprague-Dawley; Saliva; Salivary Proteins and Peptides; Salivation; Secretory Rate; Serine Endopeptidases; Stimulation, Chemical; Submandibular Gland; Tyramine; Yohimbine | 1993 |
Agonist and antagonist properties of beta 3-adrenoceptors in human omental and mouse 3T3-L1 adipocytes.
Topics: Adipose Tissue; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Humans; Isoproterenol; Lipolysis; Mice; Omentum; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Yohimbine | 1996 |
Interaction between prolactin and catecholamines on hypothalamic GnRH release in vitro.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Atenolol; Corticotropin-Releasing Hormone; Depression, Chemical; Dose-Response Relationship, Drug; Gonadotropin-Releasing Hormone; Hypothalamus; Male; Organ Culture Techniques; Phentolamine; Prazosin; Prolactin; Propanolamines; Propranolol; Rats; Rats, Sprague-Dawley; Yohimbine | 1996 |
Comparison of adrenoceptor subtype expression in porcine and human bladder and prostate.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Female; Humans; Imidazoles; Isoquinolines; Male; Oxymetazoline; Piperazines; Prazosin; Propanolamines; Prostate; Radioligand Assay; Receptors, Adrenergic; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta; Swine; Urinary Bladder; Yohimbine | 1997 |
Alpha1A-adrenergic receptors mediate vasoconstriction of the isolated spiral modiolar artery in vitro.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Arteries; Cochlea; Dose-Response Relationship, Drug; Enzyme Inhibitors; Gerbillinae; Nitric Oxide Synthase; Nitroarginine; Norepinephrine; Piperazines; Polymerase Chain Reaction; Prazosin; Propanolamines; Receptors, Adrenergic, alpha-1; RNA; Vasoconstriction; Yohimbine | 1998 |
Facilitatory beta2-adrenoceptors on cholinergic and adrenergic nerve endings of the guinea pig trachea.
Topics: Acetylcholine; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adrenergic Fibers; Animals; Atropine; Cholinergic Fibers; Electric Stimulation; Female; Fenoterol; Guinea Pigs; In Vitro Techniques; Male; Muscarinic Antagonists; Nerve Endings; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta; Trachea; Yohimbine | 1999 |
Involvement of catecholamines in recall of the conditioned NK cell response.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Amygdala; Animals; Atenolol; Brain Chemistry; Catecholamines; Cerebellum; Cerebral Cortex; Chromatography, High Pressure Liquid; Conditioning, Classical; Corpus Striatum; Dopamine; Dopamine Antagonists; Epinephrine; Female; Immunologic Memory; Killer Cells, Natural; Lymphocyte Activation; Mental Recall; Mice; Mice, Inbred BALB C; Norepinephrine; Oxathiins; Propanolamines; Salicylamides; Spleen; Yohimbine | 1999 |
Adrenoceptors in normal and malignant human melanocytes.
Topics: Adrenergic alpha-Antagonists; Binding, Competitive; Cells, Cultured; Dose-Response Relationship, Drug; Humans; Idazoxan; Melanocytes; Metoprolol; Oxathiins; Propanolamines; Propranolol; Receptors, Adrenergic; Tumor Cells, Cultured; Yohimbine | 2000 |
Presynaptic beta(2)-adrenoceptors mediate nicotine-induced NOergic neurogenic dilation in porcine basilar arteries.
Topics: Adrenergic beta-Antagonists; Animals; Basilar Artery; Butoxamine; Endothelium, Vascular; Female; In Vitro Techniques; Male; Models, Cardiovascular; Muscle, Smooth, Vascular; Nicotine; Nitric Oxide; Prazosin; Propanolamines; Receptors, Adrenergic, beta-2; Swine; Vasodilation; Yohimbine | 2000 |
Differential role of adrenoceptors in control of plasma glucose and fatty acids in carp, Cyprinus carpio (L.).
Topics: Adrenergic Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atenolol; Blood Glucose; Carps; Clonidine; Epinephrine; Fatty Acids, Nonesterified; Isoproterenol; Lactic Acid; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta; Yohimbine | 2001 |
Noradrenergic inputs mediate state dependence of auditory responses in the avian song system.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adrenergic Fibers; Animals; Arousal; Auditory Perception; Clonidine; Dose-Response Relationship, Drug; Finches; Guanabenz; Idazoxan; Imidazoles; Isoproterenol; Male; Norepinephrine; Oxathiins; Phenylephrine; Propanolamines; Prosencephalon; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta-2; Vocalization, Animal; Yohimbine | 2004 |
Beta2-adrenoceptors are essential for desipramine, venlafaxine or reboxetine action in neuropathic pain.
Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Amines; Animals; Anticonvulsants; Antidepressive Agents; Cyclohexanecarboxylic Acids; Cyclohexanols; Desipramine; Gabapentin; gamma-Aminobutyric Acid; Male; Mice; Mice, Transgenic; Morpholines; Pain; Pain Threshold; Propanolamines; Reboxetine; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta-2; Sciatic Nerve; Venlafaxine Hydrochloride; Yohimbine | 2009 |