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yohimbine and gamma-aminobutyric acid

yohimbine has been researched along with gamma-aminobutyric acid in 58 studies

Research

Studies (58)

TimeframeStudies, this research(%)All Research%
pre-199015 (25.86)18.7374
1990's14 (24.14)18.2507
2000's17 (29.31)29.6817
2010's12 (20.69)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andrews, PR; Craik, DJ; Martin, JL1
Axe, FU; Bembenek, SD; Butler, CR; Coles, F; Dunford, PJ; Edwards, JP; Fourie, AM; Grice, CA; Karlsson, L; Lundeen, K; Riley, JP; Savall, BM; Tays, KL; Wei, J; Williams, KN; Xue, X1
Altenbach, RJ; Brioni, JD; Carr, TL; Chandran, P; Cowart, MD; Esbenshade, TA; Honore, P; Hsieh, GC; Lewis, LG; Liu, H; Manelli, AM; Marsh, KC; Milicic, I; Miller, TR; Strakhova, MI; Vortherms, TA; Wakefield, BD; Wetter, JM; Witte, DG1
Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K1
Carmody, LC; Dandapani, S; Donckele, E; Feng, Y; Fernandez, C; Germain, AR; Gupta, PB; Lander, ES; Morgan, B; Munoz, B; Nag, PP; Palmer, M; Perez, JR; Schreiber, SL; Verplank, L1
Anzini, M; Brogi, S; Butini, S; Campiani, G; Cappelli, A; Caselli, G; Castriconi, F; Gemma, S; Giordani, A; Giorgi, G; Giuliani, G; Lanza, M; Letari, O; Makovec, F; Manini, M; Mennuni, L; Valenti, S1
Belyakov, S; Dambrova, M; Kazoka, H; Kuznecovs, J; Lebedev, A; Liepinsh, E; Mishnev, A; Orlova, N; Ponomaryov, Y; Vavers, E; Veinberg, G; Vikainis, S; Vilskersts, R; Vorona, M; Zvejniece, L1
Bednarski, M; Gunia-Krzyżak, A; Marona, H; Nitek, W; Pękala, E; Powroźnik, B; Słoczyńska, K; Walczak, M; Waszkielewicz, AM; Żesławska, E1
Filipek, B; Gunia-Krzyżak, A; Marona, H; Nitek, W; Pańczyk, K; Pękala, E; Rapacz, A; Słoczyńska, K; Waszkielewicz, AM; Żelaszczyk, D; Żesławska, E1
Fu, SX; Wang, LF; Zhang, SS1
Corbett, R; Dunn, RW1
Coupland, N; Glue, P; Nutt, DJ1
Hamada, T; Hamahashi, T; Itoh, T; Kamisaki, Y; Maeda, K1
Callaway, JK; King, RG1
Benzi, G; Curti, D; Dagani, F; Marzatico, F; Pastoris, O; Villa, RF1
Malinowska, B; Molderings, G; Schlicker, E; Schneider, D1
Aldegunde, MA; Míguez, I1
Pittaluga, A; Raiteri, M; Torelli, R1
Hamahashi, T; Itoh, T; Kamisaki, Y; Okada, CM1
Arnerić, SP; Tingley, FD1
Baba, S; Takeda, T; Tanaka, C; Taniyama, K1
Harris, RA; Peris, J; Zahniser, NR1
Maura, G; Pittaluga, A; Raiteri, M; Ulivi, M1
Limberger, N; Späth, L; Starke, K1
Iwai, S; Shirakawa, J; Tanaka, C; Taniyama, K1
Miñano, FJ; Sancibrián, M; Serrano, JS1
Arbilla, S; Langer, SZ; Maurin, Y1
Curet, O; Dennis, T; Nishikawa, T; Scatton, B1
Pittaluga, A; Raiteri, M1
Otto, S; Plotsky, PM; Sutton, S1
Baumann, N; Chauvel, P; Maurin, Y; Puech, A; Simon, P1
Starke, K; Weitzell, R1
Antonelli, T; Beani, L; Bianchi, C; Carla, V; Moroni, F; Tanganelli, S1
Allen, AM; Guyenet, PG1
Ehrenström, F; Söderpalm, A; Söderpalm, B1
Baumann, PA; Bittiger, H; Feldtrauer, JJ; Fröstl, W; Waldmeier, PC; Wicki, P1
Holmberg, M; Kurose, H; Miettinen, R; Scheinin, M1
Ciranna, L; Li Volsi, G; Licata, F; Santangelo, F1
Arseneau, LM; Beverly, JL; Beverly, MF; de Vries, MG1
Gordienko, DV; Krivobok, GK; Pankrat'ev, DV; Talalaenko, AN; Zinkovich, II1
Hirota, K; Ishihara, H; Kubota, T; Kushikata, T; Matsuki, A; Yoshida, H1
Goncharenko, NV; Pankrat'ev, DV; Talalaenko, AN1
Eriksson, KS; Haas, HL; Kuramasu, A; Selbach, O; Stevens, DR1
Atnip, LM; Chen, SR; Li, DP; Pan, HL1
Honda, M; Kasuya, N; Ono, H; Shimizu, S; Takasu, K; Tanabe, M1
Alachkar, A; Brotchie, J; Jones, OT1
Duncan, B; Evenden, J; Ko, T1
Honda, M; Ono, H; Takasu, K; Tanabe, M1
Ono, H; Takasu, K; Takeuchi, Y; Tanabe, M1
Bronzi, D; Di Mauro, M; Li Volsi, G; Licata, F; Lombardo, P; Santangelo, F1
Ayuse, T; Ishitobi, S; Miyamoto, T; Oi, K; Toda, K; Yoshida, H1
Barrot, M; Doridot, S; Freund-Mercier, MJ; Hein, L; Petit-Demoulière, N; Tessier, LH; Yalcin, I1
Abrams, JK; Hale, MW; Johnson, PL; Lowry, CA; Shekhar, A; Westerman, AM1
Cannella, N; Ciccocioppo, R; Cippitelli, A; de Guglielmo, G; Gerra, G; Kallupi, M; Massi, M; Somaini, L; Stopponi, S1
Billiras, R; Bouchez, G; Boulanger, R; Gobert, A; Millan, MJ; Rivet, JM1
Ciccocioppo, R; Cippitelli, A; de Guglielmo, G; Gerra, G; Kallupi, M; Li, H; Somaini, L; Stopponi, S; Ubaldi, M1
Ishola, IO; Olayemi, SO; Umeh, EA; Yemitan, OK1
Mendelowitz, D; Sharp, DB; Wang, X1

Reviews

1 review(s) available for yohimbine and gamma-aminobutyric acid

ArticleYear
Challenge tests: assessment of the noradrenergic and GABA systems in depression and anxiety disorders.
    Molecular aspects of medicine, 1992, Volume: 13, Issue:3

    Topics: Anxiety; Clonidine; Depression; gamma-Aminobutyric Acid; Growth Hormone; Humans; Hydrocortisone; Norepinephrine; Receptors, Neurotransmitter; Yohimbine

1992

Other Studies

57 other study(ies) available for yohimbine and gamma-aminobutyric acid

ArticleYear
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Identification of a potent, selective, and orally active leukotriene a4 hydrolase inhibitor with anti-inflammatory activity.
    Journal of medicinal chemistry, 2008, Jul-24, Volume: 51, Issue:14

    Topics: Administration, Oral; Animals; Anti-Inflammatory Agents; Catalysis; Dogs; Drug Evaluation, Preclinical; Enzyme Inhibitors; Epoxide Hydrolases; Humans; Magnetic Resonance Spectroscopy; Mice; Structure-Activity Relationship

2008
cis-4-(Piperazin-1-yl)-5,6,7a,8,9,10,11,11a-octahydrobenzofuro[2,3-h]quinazolin-2-amine (A-987306), a new histamine H4R antagonist that blocks pain responses against carrageenan-induced hyperalgesia.
    Journal of medicinal chemistry, 2008, Nov-27, Volume: 51, Issue:22

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzofurans; Carrageenan; Disease Models, Animal; Drug Design; Drug Evaluation, Preclinical; Humans; Hyperalgesia; Ligands; Mice; Molecular Structure; Pain; Peritonitis; Quinazolines; Rats; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Stereoisomerism; Structure-Activity Relationship

2008
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
    Bioorganic & medicinal chemistry, 2010, Nov-01, Volume: 18, Issue:21

    Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship

2010
Cinnamides as selective small-molecule inhibitors of a cellular model of breast cancer stem cells.
    Bioorganic & medicinal chemistry letters, 2013, Mar-15, Volume: 23, Issue:6

    Topics: Amides; Breast Neoplasms; Cell Line, Tumor; Drug Screening Assays, Antitumor; Female; Humans; Neoplastic Stem Cells; Small Molecule Libraries; Structure-Activity Relationship

2013
Synthesis and structure-activity relationship studies in serotonin 5-HT(1A) receptor agonists based on fused pyrrolidone scaffolds.
    European journal of medicinal chemistry, 2013, Volume: 63

    Topics: Animals; Area Under Curve; Humans; Intestinal Absorption; Ligands; Male; Metabolic Clearance Rate; Models, Chemical; Models, Molecular; Molecular Structure; Protein Binding; Protein Structure, Tertiary; Pyrrolidinones; Radioligand Assay; Receptor, Serotonin, 5-HT1A; Receptors, Serotonin, 5-HT3; Serotonin 5-HT1 Receptor Agonists; Structure-Activity Relationship

2013
Synthesis and biological evaluation of 2-(5-methyl-4-phenyl-2-oxopyrrolidin-1-yl)-acetamide stereoisomers as novel positive allosteric modulators of sigma-1 receptor.
    Bioorganic & medicinal chemistry, 2013, May-15, Volume: 21, Issue:10

    Topics: Acetamides; Allosteric Regulation; Animals; Rats; Rats, Wistar; Receptors, sigma; Sigma-1 Receptor; Stereoisomerism; Structure-Activity Relationship

2013
Design, physico-chemical properties and biological evaluation of some new N-[(phenoxy)alkyl]- and N-{2-[2-(phenoxy)ethoxy]ethyl}aminoalkanols as anticonvulsant agents.
    Bioorganic & medicinal chemistry, 2016, Apr-15, Volume: 24, Issue:8

    Topics: Amino Alcohols; Animals; Anticonvulsants; Chemistry, Physical; Dose-Response Relationship, Drug; Drug Design; Epilepsy; Male; Mice; Microsomes, Liver; Molecular Structure; Pilocarpine

2016
Structure-anticonvulsant activity studies in the group of (E)-N-cinnamoyl aminoalkanols derivatives monosubstituted in phenyl ring with 4-Cl, 4-CH
    Bioorganic & medicinal chemistry, 2017, 01-15, Volume: 25, Issue:2

    Topics: Amino Alcohols; Animals; Anticonvulsants; Crystallography, X-Ray; Disease Models, Animal; Dose-Response Relationship, Drug; Electroshock; Mice; Models, Molecular; Molecular Structure; Rats; Seizures; Structure-Activity Relationship

2017
[An analysis of the discrepancy between the effects of central and peripheral alpha-adrenoceptor stimulations (author's transl)].
    Yao xue xue bao = Acta pharmaceutica Sinica, 1979, Volume: 14, Issue:9

    Topics: Animals; Clonidine; gamma-Aminobutyric Acid; Hypotension; Picrotoxin; Rabbits; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Yohimbine

1979
Yohimbine-induced seizures involve NMDA and GABAergic transmission.
    Neuropharmacology, 1992, Volume: 31, Issue:4

    Topics: Animals; Bicuculline; Carbolines; Convulsants; Dioxanes; gamma-Aminobutyric Acid; Idazoxan; Male; Mice; Mice, Inbred Strains; N-Methylaspartate; Receptors, Adrenergic, alpha; Receptors, GABA-A; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Seizures; Synaptic Transmission; Yohimbine

1992
Presynaptic inhibition by clonidine of neurotransmitter amino acid release in various brain regions.
    European journal of pharmacology, 1992, Jun-24, Volume: 217, Issue:1

    Topics: Adrenergic alpha-Antagonists; Amino Acids; Animals; Aspartic Acid; Brain; Calcium; Clonidine; Evoked Potentials; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Male; Nerve Endings; Neurotransmitter Agents; Potassium; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Synaptosomes; Yohimbine

1992
Effects of inhaled alpha 2-adrenoceptor and GABAB receptor agonists on citric acid-induced cough and tidal volume changes in guinea pigs.
    European journal of pharmacology, 1992, Sep-22, Volume: 220, Issue:2-3

    Topics: Acetylcholine; Administration, Inhalation; Adrenergic alpha-Agonists; Animals; Atropine; Azepines; Baclofen; Citrates; Citric Acid; Cough; gamma-Aminobutyric Acid; Guinea Pigs; Male; Receptors, GABA-A; Respiration; Tidal Volume; Xylazine; Yohimbine

1992
Sequential damage in mitochondrial complexes by peroxidative stress.
    Neurochemical research, 1991, Volume: 16, Issue:12

    Topics: Almitrine; Animals; Cyclohexanones; Cytochrome c Group; Electron Transport; Electron Transport Complex IV; gamma-Aminobutyric Acid; Glutathione; Male; Mitochondria; NADH Dehydrogenase; Oxidation-Reduction; Pantothenic Acid; Prosencephalon; Rats; Rats, Inbred Strains; Succinate Dehydrogenase; Yohimbine

1991
Noradrenaline release in the rat vena cava is inhibited by gamma-aminobutyric acid via GABAB receptors but not affected by histamine.
    British journal of pharmacology, 1991, Volume: 104, Issue:2

    Topics: Animals; Baclofen; Bicuculline; Corticosterone; Desipramine; Electric Stimulation; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Histamine; In Vitro Techniques; Male; Muscimol; Norepinephrine; Organophosphorus Compounds; Rats; Rats, Inbred Strains; Receptors, GABA-A; Vena Cava, Inferior; Yohimbine

1991
Effect of gamma-aminobutyric acid on corticosterone secretion: involvement of the noradrenergic system.
    Life sciences, 1990, Volume: 46, Issue:12

    Topics: 1-Propanol; Adrenocorticotropic Hormone; Animals; Brain; Corticosterone; gamma-Aminobutyric Acid; Hydroxyindoleacetic Acid; Hypothalamus; Injections, Intraventricular; Male; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Serotonin; Yohimbine

1990
Clonidine differentially modulates the release of endogenous GABA in various rat brain areas.
    Pharmacological research, 1991, Volume: 24, Issue:2

    Topics: Animals; Brain Chemistry; Cerebellum; Cerebral Cortex; Clonidine; gamma-Aminobutyric Acid; Hippocampus; Imidazoles; In Vitro Techniques; Male; Medulla Oblongata; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains; Synaptosomes; Yohimbine

1991
Clonidine inhibition of potassium-evoked release of glutamate and aspartate from rat cortical synaptosomes.
    Brain research, 1991, Dec-24, Volume: 568, Issue:1-2

    Topics: Analysis of Variance; Animals; Aspartic Acid; Cerebral Cortex; Clonidine; Dioxanes; gamma-Aminobutyric Acid; Glutamates; Idazoxan; Kinetics; Male; Potassium; Potassium Chloride; Rats; Rats, Inbred Strains; Synaptosomes; Yohimbine

1991
Evidence for clonidine presynaptically modulating amino acid release in the rostral ventral medulla: role in hypertension.
    Brain research, 1990, Dec-24, Volume: 537, Issue:1-2

    Topics: Amino Acids; Animals; Aspartic Acid; Clonidine; Female; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Hypertension; In Vitro Techniques; Medulla Oblongata; Neurotransmitter Agents; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Synapses; Synaptic Transmission; Synaptosomes; Yohimbine

1990
Putative mechanisms involved in excitatory and inhibitory effects of somatostatin on intestinal motility.
    The American journal of physiology, 1989, Volume: 257, Issue:4 Pt 1

    Topics: Acetylcholine; Animals; Bicuculline; Electric Stimulation; Female; gamma-Aminobutyric Acid; Gastrointestinal Motility; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Naloxone; Somatostatin; Theophylline; Yohimbine

1989
Modulation of gamma-[3H]aminobutyric acid release from rat cortical slices by alpha 2-adrenoceptors.
    Neuroscience letters, 1987, Oct-05, Volume: 80, Issue:3

    Topics: Animals; Calcium; Clonidine; gamma-Aminobutyric Acid; Guanabenz; In Vitro Techniques; Male; Norepinephrine; Occipital Lobe; Parietal Lobe; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine

1987
Enhancement of endogenous GABA release from rat synaptosomal preparations is mediated by alpha 2-adrenoceptors pharmacologically different from alpha 2-autoreceptors.
    European journal of pharmacology, 1988, Nov-15, Volume: 157, Issue:1

    Topics: Animals; Clonidine; gamma-Aminobutyric Acid; Hippocampus; Male; Mianserin; Norepinephrine; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Synaptosomes; Yohimbine

1988
A search for receptors modulating the release of gamma-[3H]aminobutyric acid in rabbit caudate nucleus slices.
    Journal of neurochemistry, 1986, Volume: 46, Issue:4

    Topics: Acetylcholine; Adenylyl Cyclases; Animals; Carbachol; Caudate Nucleus; Dopamine; Electric Stimulation; Female; gamma-Aminobutyric Acid; Hexamethonium; Hexamethonium Compounds; Male; Methiothepin; Rabbits; Receptors, Cell Surface; Receptors, Cholinergic; Receptors, Dopamine; Receptors, Serotonin; Serotonin; Tritium; Yohimbine

1986
Regulation of [3H]GABA release from strips of guinea pig urinary bladder.
    The American journal of physiology, 1988, Volume: 255, Issue:6 Pt 2

    Topics: Acetylcholine; Animals; Atropine; Baclofen; Bicuculline; Clonazepam; Clonidine; Female; gamma-Aminobutyric Acid; Guinea Pigs; Hexamethonium; Hexamethonium Compounds; In Vitro Techniques; Male; Muscimol; Pentobarbital; Phenylephrine; Pirenzepine; Potassium; Prazosin; Tritium; Urinary Bladder; Yohimbine

1988
GABA-induced hypothermia in rats: involvement of serotonergic and cholinergic mechanisms.
    General pharmacology, 1986, Volume: 17, Issue:3

    Topics: Acetylcholine; Animals; Body Temperature; Clomipramine; Drug Interactions; Female; Fenclonine; GABA Antagonists; gamma-Aminobutyric Acid; Parasympatholytics; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Yohimbine

1986
Inhibition by yohimbine of the calcium-dependent evoked release of [3H]GABA in rat and mouse brain slices in vitro.
    European journal of pharmacology, 1985, Apr-23, Volume: 111, Issue:1

    Topics: Animals; Brain; Brain Stem; Calcium; Cerebral Cortex; Electric Stimulation; Female; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Mice; Norepinephrine; Potassium; Rats; Receptors, Adrenergic, alpha; Secretory Rate; Stereoisomerism; Yohimbine

1985
Further evidence for, and nature of, the facilitatory GABAergic influence on central noradrenergic transmission.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 331, Issue:2-3

    Topics: Afferent Pathways; Animals; Central Nervous System; Cerebral Cortex; Clonidine; gamma-Aminobutyric Acid; Hypothalamus; Ibotenic Acid; Methoxyhydroxyphenylglycol; Muscimol; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin; Spinal Cord; Synaptic Transmission; Yohimbine

1985
GABAergic nerve terminals in rat hippocampus possess alpha 2-adrenoceptors regulating GABA release.
    Neuroscience letters, 1987, May-19, Volume: 76, Issue:3

    Topics: Animals; gamma-Aminobutyric Acid; Hippocampus; Male; Nerve Endings; Norepinephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Synaptosomes; Yohimbine

1987
Neurotransmitter modulation of corticotropin releasing factor secretion into the hypophysial-portal circulation.
    Life sciences, 1987, Sep-07, Volume: 41, Issue:10

    Topics: Acetylcholine; Animals; Bicuculline; Cerebral Ventricles; Corticotropin-Releasing Hormone; Epinephrine; gamma-Aminobutyric Acid; Hypothalamo-Hypophyseal System; Injections, Intraventricular; Male; Neurons; Paraventricular Hypothalamic Nucleus; Pempidine; Propranolol; Rats; Rats, Inbred Strains; Scopolamine; Yohimbine

1987
[Biochemical and pharmacological approach to the functional disorders observed in demyelination mutants (GABAergic and noradrenergic systems)].
    Comptes rendus des seances de la Societe de biologie et de ses filiales, 1980, Volume: 174, Issue:4

    Topics: Animals; Central Nervous System; Demyelinating Diseases; gamma-Aminobutyric Acid; Membrane Proteins; Mice; Mice, Quaking; Norepinephrine; Receptors, Adrenergic, alpha; Receptors, Neurotransmitter; Yohimbine

1980
gamma-Aminobutyric acid and postganglionic sympathetic transmission in the pulmonary artery of the rabbit.
    Journal of autonomic pharmacology, 1980, Volume: 1, Issue:1

    Topics: Animals; Autonomic Fibers, Postganglionic; Cocaine; Drug Interactions; Electric Stimulation; gamma-Aminobutyric Acid; In Vitro Techniques; Muscle, Smooth, Vascular; Potassium; Pulmonary Artery; Rabbits; Sympathetic Nervous System; Synaptic Transmission; Yohimbine

1980
Modulation of cortical acetylcholine and gamma-aminobutyric acid release in freely moving guinea pigs: effects of clonidine and other adrenergic drugs.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 227, Issue:2

    Topics: Acetylcholine; Animals; Cerebral Cortex; Clonidine; Female; gamma-Aminobutyric Acid; Guinea Pigs; Male; Norepinephrine; Prazosin; Receptors, Adrenergic, alpha; Sympathomimetics; Yohimbine

1983
Alpha 2-adrenoceptor-mediated inhibition of bulbospinal barosensitive cells of rat rostral medulla.
    The American journal of physiology, 1993, Volume: 265, Issue:5 Pt 2

    Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Evoked Potentials; gamma-Aminobutyric Acid; Idazoxan; Injections, Intravenous; Iontophoresis; Male; Medulla Oblongata; Neurons; Nordefrin; Pressoreceptors; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Spinal Cord; Yohimbine

1993
The yohimbine-induced anticonflict effect in the rat, Part II. Neurochemical findings.
    Journal of neural transmission. General section, 1995, Volume: 100, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Animals; Behavior, Animal; Cerebral Cortex; Chlorides; Conflict, Psychological; Dihydroxyphenylalanine; Enzyme Inhibitors; gamma-Aminobutyric Acid; Hippocampus; Hydrazines; Hydroxyindoleacetic Acid; Male; Norepinephrine; Oxidopamine; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Reserpine; Serotonin; Yohimbine

1995
Effects of the putative P-type calcium channel blocker, R,R-(-)-daurisoline on neurotransmitter release.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:6

    Topics: Acetylcholine; Alkaloids; Animals; Benzylisoquinolines; Binding, Competitive; Brain; Calcium Channel Blockers; Dopamine; gamma-Aminobutyric Acid; Glutamic Acid; Isotope Labeling; Lethal Dose 50; Male; Norepinephrine; omega-Conotoxin GVIA; Peptides; Radioligand Assay; Rats; Receptors, Adrenergic, alpha; Receptors, Muscarinic; Receptors, Opioid, mu; Receptors, Serotonin; Serotonin; Stereoisomerism; Synaptic Transmission; Yohimbine

1995
Adrenergic alpha2C-receptors reside in rat striatal GABAergic projection neurons: comparison of radioligand binding and immunohistochemistry.
    Neuroscience, 1999, Volume: 93, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Antibodies; Autoradiography; Binding, Competitive; Brain Chemistry; Calbindin 1; Calbindin 2; Calbindins; Corpus Striatum; gamma-Aminobutyric Acid; Idazoxan; Immunohistochemistry; Male; Neurons; Norepinephrine; Parvalbumins; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; S100 Calcium Binding Protein G; Tissue Fixation; Tritium; Yohimbine

1999
Neurotransmitter-mediated control of neuronal firing in the red nucleus of the rat: reciprocal modulation between noradrenaline and GABA.
    Experimental neurology, 2000, Volume: 163, Issue:1

    Topics: Action Potentials; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bicuculline; Clonidine; Drug Synergism; GABA Antagonists; gamma-Aminobutyric Acid; Iontophoresis; Isoproterenol; Male; Neurons; Neurotransmitter Agents; Nipecotic Acids; Norepinephrine; Rats; Rats, Wistar; Red Nucleus; Timolol; Yohimbine

2000
Norepinephrine mediates glucoprivic-induced increase in GABA in the ventromedial hypothalamus of rats.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2000, Volume: 279, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Antimetabolites; Blood Glucose; Brain Chemistry; Deoxyglucose; gamma-Aminobutyric Acid; Male; Microdialysis; Norepinephrine; Rats; Rats, Sprague-Dawley; Timolol; Ventromedial Hypothalamic Nucleus; Yohimbine

2000
The role of neurochemical mechanisms of ventromedial hypothalamus in various models of anxiety in rats.
    Bulletin of experimental biology and medicine, 2001, Volume: 131, Issue:1

    Topics: Adrenergic Agents; Animals; Anxiety; Apomorphine; Avoidance Learning; Disease Models, Animal; Dopamine; Dopamine Agents; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Hypothalamus, Middle; Male; Memantine; Microinjections; Neurotransmitter Agents; Phenylephrine; Picrotoxin; Rats; Serotonin; Sulpiride; Yohimbine

2001
Alpha-2 adrenoceptor activity affects propofol-induced sleep time.
    Anesthesia and analgesia, 2002, Volume: 94, Issue:5

    Topics: Anesthetics, Intravenous; Animals; Clonidine; gamma-Aminobutyric Acid; Male; Norepinephrine; Prefrontal Cortex; Propofol; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Sleep; Yohimbine

2002
Neurochemical characteristics of the ventromedial hypothalamus in mediating the antiaversive effects of anxiolytics in different models of anxiety.
    Neuroscience and behavioral physiology, 2003, Volume: 33, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Anti-Anxiety Agents; Anticonvulsants; Anxiety; Apomorphine; Avoidance Learning; Biguanides; Brain Chemistry; Chlordiazepoxide; Clonidine; Disease Models, Animal; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Droperidol; Drug Interactions; GABA Agents; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Glutamic Acid; Male; Memantine; Mephenytoin; Microinjections; Pentylenetetrazole; Phentolamine; Picrotoxin; Piperazines; Propranolol; Pyrimidines; Rats; Serotonin; Sulpiride; Ventromedial Hypothalamic Nucleus; Yohimbine

2003
Alpha 2-adrenergic receptor-mediated presynaptic inhibition of GABAergic IPSPs in rat histaminergic neurons.
    Neuropharmacology, 2004, Volume: 46, Issue:7

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Female; gamma-Aminobutyric Acid; Histamine; Male; Neural Inhibition; Neurons; Norepinephrine; Presynaptic Terminals; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Synaptic Transmission; Yohimbine

2004
Regulation of synaptic inputs to paraventricular-spinal output neurons by alpha2 adrenergic receptors.
    Journal of neurophysiology, 2005, Volume: 93, Issue:1

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Afferent Pathways; Animals; Bicuculline; Brain Stem; Clonidine; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Fluorescent Antibody Technique; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Neural Inhibition; Neurons; Paraventricular Hypothalamic Nucleus; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Spinal Cord; Synapses; Synaptophysin; Time Factors; Yohimbine

2005
Role of descending noradrenergic system and spinal alpha2-adrenergic receptors in the effects of gabapentin on thermal and mechanical nociception after partial nerve injury in the mouse.
    British journal of pharmacology, 2005, Volume: 144, Issue:5

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Amines; Analgesics; Animals; Cyclohexanecarboxylic Acids; Foot; Gabapentin; gamma-Aminobutyric Acid; Hindlimb; Hot Temperature; Hyperalgesia; Male; Mice; Mice, Inbred Strains; Motor Activity; Pain Measurement; Prazosin; Receptors, Adrenergic, alpha-2; Sciatic Nerve; Touch; Yohimbine

2005
alpha2-Adrenoceptor-mediated modulation of the release of GABA and noradrenaline in the rat substantia nigra pars reticulata.
    Neuroscience letters, 2006, Mar-06, Volume: 395, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Male; Nipecotic Acids; Norepinephrine; Organ Culture Techniques; Rats; Receptors, Adrenergic, alpha-2; Substantia Nigra; Yohimbine

2006
A comparison of the effects of psychotomimetics and anxiolytics on punished and unpunished responding maintained by fixed interval schedules of food reinforcement in the rat.
    Behavioural pharmacology, 2006, Volume: 17, Issue:1

    Topics: Amphetamines; Animals; Anti-Anxiety Agents; Appetitive Behavior; Association Learning; Benzimidazoles; Chlordiazepoxide; Conditioning, Operant; Dextroamphetamine; Dizocilpine Maleate; Electroshock; gamma-Aminobutyric Acid; Hallucinogens; Oximes; Pregabalin; Punishment; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Reinforcement Schedule; Yohimbine

2006
Spinal alpha(2)-adrenergic and muscarinic receptors and the NO release cascade mediate supraspinally produced effectiveness of gabapentin at decreasing mechanical hypersensitivity in mice after partial nerve injury.
    British journal of pharmacology, 2006, Volume: 148, Issue:2

    Topics: Adrenergic alpha-2 Receptor Antagonists; Amines; Analgesics; Animals; Atropine; Cholinesterases; Cyclohexanecarboxylic Acids; Enzyme Activation; Gabapentin; gamma-Aminobutyric Acid; Hot Temperature; Hyperalgesia; Idazoxan; Injections, Intraventricular; Male; Mice; Muscarinic Antagonists; Narcotic Antagonists; Neostigmine; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; omega-N-Methylarginine; Receptors, Adrenergic, alpha-2; Receptors, Muscarinic; Sciatic Nerve; Spinal Cord; Touch; Yohimbine

2006
Pregabalin, S-(+)-3-isobutylgaba, activates the descending noradrenergic system to alleviate neuropathic pain in the mouse partial sciatic nerve ligation model.
    Neuropharmacology, 2007, Volume: 53, Issue:7

    Topics: Adrenergic Agents; Afferent Pathways; Analgesics; Animals; Behavior, Animal; Brain Stem; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Routes; gamma-Aminobutyric Acid; Hyperalgesia; Locomotion; Male; Methoxyhydroxyphenylglycol; Mice; Norepinephrine; Oxidopamine; Pain Measurement; Pregabalin; Sciatic Neuropathy; Spinal Cord; Time Factors; Yohimbine

2007
Noradrenaline modulates neuronal responses to GABA in vestibular nuclei.
    Neuroscience, 2008, Jun-02, Volume: 153, Issue:4

    Topics: Action Potentials; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Clonidine; Dose-Response Relationship, Drug; Drug Interactions; gamma-Aminobutyric Acid; Iontophoresis; Isoproterenol; Neural Inhibition; Neurons; Norepinephrine; Rats; Rats, Wistar; Timolol; Vestibular Nuclei; Yohimbine

2008
Effects of midazolam on acquisition and extinction of conditioned taste aversion memory in rats.
    Neuroscience letters, 2009, Feb-06, Volume: 450, Issue:3

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Avoidance Learning; Brain; Conditioning, Psychological; Extinction, Psychological; GABA Modulators; gamma-Aminobutyric Acid; Male; Memory; Midazolam; Neural Inhibition; Norepinephrine; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Synaptic Transmission; Yohimbine

2009
Beta2-adrenoceptors are essential for desipramine, venlafaxine or reboxetine action in neuropathic pain.
    Neurobiology of disease, 2009, Volume: 33, Issue:3

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Amines; Animals; Anticonvulsants; Antidepressive Agents; Cyclohexanecarboxylic Acids; Cyclohexanols; Desipramine; Gabapentin; gamma-Aminobutyric Acid; Male; Mice; Mice, Transgenic; Morpholines; Pain; Pain Threshold; Propanolamines; Reboxetine; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta-2; Sciatic Nerve; Venlafaxine Hydrochloride; Yohimbine

2009
Multiple anxiogenic drugs recruit a parvalbumin-containing subpopulation of GABAergic interneurons in the basolateral amygdala.
    Progress in neuro-psychopharmacology & biological psychiatry, 2010, Oct-01, Volume: 34, Issue:7

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Brain; Caffeine; Carbolines; Cell Count; gamma-Aminobutyric Acid; Gene Expression Regulation; Interneurons; Male; Parvalbumins; Piperazines; Proto-Oncogene Proteins c-fos; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Time Factors; Yohimbine

2010
Pregabalin reduces alcohol drinking and relapse to alcohol seeking in the rat.
    Psychopharmacology, 2012, Volume: 220, Issue:1

    Topics: Alcohol Drinking; Animals; Anticonvulsants; Conditioning, Operant; Dose-Response Relationship, Drug; Drug-Seeking Behavior; Ethanol; gamma-Aminobutyric Acid; Male; Pregabalin; Rats; Secondary Prevention; Selection, Genetic; Self Administration; Yohimbine

2012
Quantification of extracellular levels of corticosterone in the basolateral amygdaloid complex of freely-moving rats: a dialysis study of circadian variation and stress-induced modulation.
    Brain research, 2012, May-03, Volume: 1452

    Topics: Amygdala; Animals; Carbolines; Circadian Rhythm; Corticosterone; Dopamine; gamma-Aminobutyric Acid; Microdialysis; Norepinephrine; Rats; Serotonin; Stress, Psychological; Yohimbine

2012
Pregabalin reduces cocaine self-administration and relapse to cocaine seeking in the rat.
    Addiction biology, 2013, Volume: 18, Issue:4

    Topics: Adrenergic alpha-2 Receptor Antagonists; Analysis of Variance; Animals; Anticonvulsants; Cocaine; Cocaine-Related Disorders; Cues; Discrimination Learning; Drug-Seeking Behavior; Feeding Behavior; gamma-Aminobutyric Acid; Humans; Male; Pregabalin; Rats; Rats, Wistar; Reinforcement, Psychology; Secondary Prevention; Self Administration; Stress, Physiological; Yohimbine

2013
Antidepressant and anxiolytic effects of the methanol root extract of Capparis thonningii: involvement of monoaminergic, cholinergic and GABAergic systems.
    Drug research, 2015, Volume: 65, Issue:4

    Topics: Adrenergic Antagonists; Animals; Anti-Anxiety Agents; Antidepressive Agents; Atropine; Behavior, Animal; Biogenic Monoamines; Capparis; Cholinergic Agents; Cholinergic Neurons; Cyproheptadine; Dopamine Antagonists; Female; Flumazenil; GABA Agents; gamma-Aminobutyric Acid; Immobility Response, Tonic; Male; Metergoline; Methanol; Mice; Muscarinic Antagonists; Plant Extracts; Plant Roots; Prazosin; Serotonin Antagonists; Sulpiride; Yohimbine

2015
Dexmedetomidine decreases inhibitory but not excitatory neurotransmission to cardiac vagal neurons in the nucleus ambiguus.
    Brain research, 2014, Jul-29, Volume: 1574

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Dexmedetomidine; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Glutamic Acid; Glycine; Heart; Medulla Oblongata; Neurons; Patch-Clamp Techniques; Rats, Sprague-Dawley; Tissue Culture Techniques; Vagus Nerve; Yohimbine

2014