Page last updated: 2024-09-04

ym 872 and lofepramine hydrochloride

ym 872 has been researched along with lofepramine hydrochloride in 3 studies

Compound Research Comparison

Studies
(ym 872)
Trials
(ym 872)
Recent Studies (post-2010)
(ym 872)
Studies
(lofepramine hydrochloride)
Trials
(lofepramine hydrochloride)
Recent Studies (post-2010) (lofepramine hydrochloride)
41051701

Protein Interaction Comparison

ProteinTaxonomyym 872 (IC50)lofepramine hydrochloride (IC50)
Integrin beta-3Homo sapiens (human)0.35
Integrin alpha-IIbHomo sapiens (human)0.35
Glutamate receptor 1Rattus norvegicus (Norway rat)0.3371
Glutamate receptor 2Rattus norvegicus (Norway rat)0.3371
Glutamate receptor 3Rattus norvegicus (Norway rat)0.3371
Glutamate receptor 4Rattus norvegicus (Norway rat)0.3371
Glutamate receptor ionotropic, kainate 1Rattus norvegicus (Norway rat)0.28
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)10
Glutamate receptor ionotropic, kainate 2Rattus norvegicus (Norway rat)0.28
Glutamate receptor ionotropic, kainate 3Rattus norvegicus (Norway rat)0.28
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)10
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)10
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)10
Glutamate receptor ionotropic, kainate 4Rattus norvegicus (Norway rat)0.28
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)10
Glutamate receptor ionotropic, kainate 5Rattus norvegicus (Norway rat)0.28
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)10
P2Y purinoceptor 12Homo sapiens (human)0.35
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)10

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (66.67)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ando, N; Anraku, T; Asano, J; Shiga, F; Takano, Y; Uchiki, H1
Anraku, T; Asano, J; Hori, W; Shiga, F; Takano, Y; Uno, T1
Carcache, D; Kalkman, HO; Koller, M; Mattes, H1

Other Studies

3 other study(ies) available for ym 872 and lofepramine hydrochloride

ArticleYear
Synthesis and AMPA receptor antagonistic activity of a novel class of quinoxalinecarboxylic acid with a substituted phenyl group at the C-7 position.
    Bioorganic & medicinal chemistry letters, 2003, Oct-20, Volume: 13, Issue:20

    Topics: Animals; Quinoxalines; Rats; Receptors, AMPA

2003
Synthesis and AMPA receptor antagonistic activity of a novel 7-imidazolyl-6-trifluoromethyl quinoxalinecarboxylic acid with a substituted phenyl group and improved its good physicochemical properties by introduced CF3 group.
    Bioorganic & medicinal chemistry letters, 2004, Oct-18, Volume: 14, Issue:20

    Topics: Animals; Brain Ischemia; Disease Models, Animal; Imidazoles; In Vitro Techniques; Infusions, Intravenous; Neuroprotective Agents; Quinoxalines; Rats; Receptors, AMPA; Solubility; Structure-Activity Relationship

2004
alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) antagonists: from bench to bedside.
    Journal of medicinal chemistry, 2010, Aug-12, Volume: 53, Issue:15

    Topics: Analgesics; Animals; Anticonvulsants; Antipsychotic Agents; Clinical Trials as Topic; Drug Evaluation, Preclinical; Humans; Neuroprotective Agents; Protein Subunits; Receptors, AMPA

2010