Page last updated: 2024-09-04

ym 872 and 2-amino-5-phosphonovalerate

ym 872 has been researched along with 2-amino-5-phosphonovalerate in 5 studies

Compound Research Comparison

Studies
(ym 872)
Trials
(ym 872)
Recent Studies (post-2010)
(ym 872)
Studies
(2-amino-5-phosphonovalerate)
Trials
(2-amino-5-phosphonovalerate)
Recent Studies (post-2010) (2-amino-5-phosphonovalerate)
41054,3931539

Protein Interaction Comparison

ProteinTaxonomyym 872 (IC50)2-amino-5-phosphonovalerate (IC50)
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)0.29

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (20.00)18.2507
2000's4 (80.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Gyermek, L; Kawasaki-Yatsugi, S; Lee, C; Nishiyama, T; Yamaguchi, T2
Gyermek, L; Hanaoka, K; Kawasaki-Yatsugi, S; Lee, C; Nishiyama, T; Yamaguchi, T1
Arendt-Nielsen, L; Sumikura, H1
Nishiyama, T1

Other Studies

5 other study(ies) available for ym 872 and 2-amino-5-phosphonovalerate

ArticleYear
Analgesic interaction between intrathecal midazolam and glutamate receptor antagonists on thermal-induced pain in rats.
    Anesthesiology, 1999, Volume: 91, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Animals; Dose-Response Relationship, Drug; Drug Synergism; Excitatory Amino Acid Antagonists; GABA Modulators; Imidazoles; Injections, Spinal; Midazolam; Motor Activity; Pain; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate

1999
The analgesic interaction between intrathecal clonidine and glutamate receptor antagonists on thermal and formalin-induced pain in rats.
    Anesthesia and analgesia, 2001, Volume: 92, Issue:3

    Topics: Adrenergic alpha-Agonists; Analgesics, Non-Narcotic; Animals; Clonidine; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Imidazoles; Injections, Spinal; Pain; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Valine

2001
Synergistic analgesic effects of intrathecal midazolam and NMDA or AMPA receptor antagonists in rats.
    Canadian journal of anaesthesia = Journal canadien d'anesthesie, 2001, Volume: 48, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Adjuvants, Anesthesia; Animals; Dose-Response Relationship, Drug; Drug Synergism; Excitatory Amino Acid Antagonists; Formaldehyde; Imidazoles; Male; Midazolam; Neuroprotective Agents; Pain Measurement; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate

2001
MAC reduction after intrathecal coadministration of GABA(A) agonist and glutamate antagonist in rats.
    Journal of anesthesia, 2003, Volume: 17, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Anesthetics, Inhalation; Animals; Drug Synergism; Excitatory Amino Acid Antagonists; GABA Agonists; Imidazoles; Injections, Spinal; Male; Methyl Ethers; Muscimol; N-Methylaspartate; Pain; Pulmonary Alveoli; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Sevoflurane

2003
Interaction between a NMDA receptor antagonist, AP-5 and an AMPA receptor antagonist, YM 872 in antinociception in the spinal cord.
    Acta anaesthesiologica Scandinavica, 2008, Volume: 52, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; Acute Disease; Analgesics; Animals; Chronic Disease; Dose-Response Relationship, Drug; Drug Synergism; Excitatory Amino Acid Antagonists; Imidazoles; Male; Pain; Pain Measurement; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spinal Cord

2008