Page last updated: 2024-09-03

ym 12617 and clonidine

ym 12617 has been researched along with clonidine in 5 studies

Compound Research Comparison

Studies
(ym 12617)
Trials
(ym 12617)
Recent Studies (post-2010)
(ym 12617)
Studies
(clonidine)
Trials
(clonidine)
Recent Studies (post-2010) (clonidine)
322613,6922,0441,394

Protein Interaction Comparison

ProteinTaxonomyym 12617 (IC50)clonidine (IC50)
Alpha-2A adrenergic receptorHomo sapiens (human)0.101
Alpha-2B adrenergic receptorHomo sapiens (human)0.0353
Alpha-2C adrenergic receptorHomo sapiens (human)0.0115
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)5.365
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.0173
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.0173
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.0173
Alpha-1D adrenergic receptorHomo sapiens (human)1.21
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)5.365
Alpha-2A adrenergic receptorBos taurus (cattle)0.002
NischarinRattus norvegicus (Norway rat)0.3662

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19903 (60.00)18.7374
1990's2 (40.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Abe, M; Ikeda, T; Matsumoto, M; Saito, H; Togashi, H; Yoshioka, M1
Akimoto, Y; Fujiwara, M; Kurahashi, K; Sono, K1
Honda, K; Miyata-Osawa, A; Shiono, K; Takenaka, T; Terai, M1
Fujii, K; Kuriyama, H1
Guarneri, L; Leonardi, A; Poggesi, E; Simonazzi, I; Taddei, C; Testa, R1

Other Studies

5 other study(ies) available for ym 12617 and clonidine

ArticleYear
Central sympathoinhibitory action of a new type of alpha-1 adrenoceptor antagonist, YM-617, in rats.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Clonidine; Electrophysiology; Heart Rate; Injections, Intravenous; Male; Rats; Rats, Inbred Strains; RNA; Sulfonamides; Sympathetic Nervous System

1990
Effects of specific alpha-adrenoceptive agents on extraneuronal uptake (uptake2) of isoproterenol in perfused rat heart.
    Life sciences, 1989, Volume: 44, Issue:14

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Guanabenz; Isoproterenol; Male; Methoxamine; Myocardium; Neurons; Phenylephrine; Prazosin; Quinazolines; Rats; Rats, Inbred Strains; Sulfonamides; Tropolone

1989
Studies on YM-12617: a selective and potent antagonist of postsynaptic alpha 1-adrenoceptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 328, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Aorta; Blood Pressure; Brain; Brimonidine Tartrate; Clonidine; Dioxanes; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Muscle Contraction; Phenylephrine; Pulmonary Artery; Quinoxalines; Rabbits; Rats; Receptors, Adrenergic, alpha; Sulfonamides; Tritium; Vas Deferens

1985
Effects of YM-12617, an alpha adrenoceptor blocking agent, on electrical and mechanical properties of the guinea-pig mesenteric and pulmonary arteries.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Membrane Potentials; Mesenteric Arteries; Muscle, Smooth, Vascular; Norepinephrine; Pulmonary Artery; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Sulfonamides; Vasoconstriction

1985
Mediation of noradrenaline-induced contractions of rat aorta by the alpha 1B-adrenoceptor subtype.
    British journal of pharmacology, 1995, Volume: 114, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Binding, Competitive; Clonidine; Computer Simulation; Hippocampus; In Vitro Techniques; Liver; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phentolamine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Regression Analysis; Spiperone; Stereoisomerism; Sulfonamides

1995
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