Page last updated: 2024-09-04

ym 09151-2 and sulpiride

ym 09151-2 has been researched along with sulpiride in 24 studies

Compound Research Comparison

Studies
(ym 09151-2)
Trials
(ym 09151-2)
Recent Studies (post-2010)
(ym 09151-2)
Studies
(sulpiride)
Trials
(sulpiride)
Recent Studies (post-2010) (sulpiride)
2496134,152427635

Protein Interaction Comparison

ProteinTaxonomyym 09151-2 (IC50)sulpiride (IC50)
Carbonic anhydrase 1Homo sapiens (human)1.2
Carbonic anhydrase 2Homo sapiens (human)0.04
Alpha-2A adrenergic receptorHomo sapiens (human)2.019
D(2) dopamine receptorHomo sapiens (human)0.0858
D(3) dopamine receptorHomo sapiens (human)0.2651
D(2) dopamine receptorRattus norvegicus (Norway rat)0.2215
Carbonic anhydrase 4Bos taurus (cattle)0.62
D(2) dopamine receptorCanis lupus familiaris (dog)0.2

Research

Studies (24)

TimeframeStudies, this research(%)All Research%
pre-19907 (29.17)18.7374
1990's13 (54.17)18.2507
2000's3 (12.50)29.6817
2010's1 (4.17)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kobayashi, M; Koshikawa, N; Maruyama, Y; Mori, E; Yatsushige, N1
Kobayashi, T; Shimizu, H; Toru, M1
Arai, I; Higuchi, T; Kazawa, T; Mikuni, M; Takahashi, K; Yamauchi, T1
Hatano, K; Hatazawa, J; Ido, T; Ishiwata, K; Itoh, M; Kawashima, K1
Wambebe, C1
De Vlieger, TA; Lodder, JC; Stoof, JC; Werkman, TR1
Fitten, J; Gordon, LI; Kodama, CK; Menon, MK1
Jenks, BG; Tonon, MC; Vaudry, H; Verburg-Van Kemenade, BM1
Maeno, H; Nishikori, K; Noshiro, O; Usuda, S1
Chihara, K; Fujita, T; Iwasaki, J; Kaji, H; Kodama, H; Matsumoto, S; Minamitani, N; Shirataki, K; Tamaki, N1
Inami, K; Ishiwata, K; Nozaki, T; Sasaki, T; Senda, M1
Skarsfeldt, T1
Kikuchi de Beltrán, K; Kobayashi, M; Koshikawa, N; Miwa, Y1
Farooqui, SM1
Nishi, S; Yamada, S; Yokoo, H1
Nowak, JZ; Zawilska, JB1
Kamijo, N; Nagao, T; Ono, H1
Kobayashi, M; Koshikawa, N; Noguchi, M; Tomiyama, K1
Kuribara, H1
Fang, H; Helmeste, DM; Li, M; Tang, SW1
Castelli, MP; Gessa, GL; Mocci, I; Pani, L; Sanna, AM1
Hashimoto, K; Higashi, T; Matsushita, S; Nakano, K; Takagi, R; Tanaka, Y1
Baroni, S; Betti, L; Castagna, M; Catena Dell'Osso, M; Consoli, G; Giannaccini, G; Lucacchini, A; Marazziti, D; Masala, I; Palego, L1
Dai, F; Hong, SJ; Kim, TI; Li, S; Song, JH; Won, MH; Yoo, WG1

Other Studies

24 other study(ies) available for ym 09151-2 and sulpiride

ArticleYear
Role of dopamine D-1 and D-2 receptors in the ventral striatum in the turning behaviour of rats.
    European journal of pharmacology, 1990, Mar-20, Volume: 178, Issue:2

    Topics: Animals; Apomorphine; Benzamides; Benzazepines; Corpus Striatum; Dopamine Agents; Dopamine Antagonists; Flupenthixol; Male; Methamphetamine; Microinjections; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereotyped Behavior; Sulpiride

1990
[The inhibition of dopamine D1 and D2 receptors in human putamen by antipsychotic drugs].
    Yakubutsu, seishin, kodo = Japanese journal of psychopharmacology, 1990, Volume: 10, Issue:2

    Topics: Aged; Aged, 80 and over; Antipsychotic Agents; Benzamides; Benzazepines; Chlorpromazine; Depression, Chemical; Female; Haloperidol; Humans; In Vitro Techniques; Putamen; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Sulpiride

1990
Characterization of sulpiride-displaceable 3H-YM-09151-2 binding sites in rat frontal cortex and the effects of subchronic treatment with haloperidol on cortical D-2 dopamine receptors.
    Life sciences, 1990, Volume: 47, Issue:6

    Topics: Animals; Benzamides; Binding Sites; Corpus Striatum; Dopamine Antagonists; Frontal Lobe; Haloperidol; In Vitro Techniques; Ketanserin; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride

1990
D2-dopamine receptor specific brain uptake of carbon-11-labeled YM-09151-2.
    Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 1989, Volume: 30, Issue:4

    Topics: Animals; Antipsychotic Agents; Benzamides; Brain; Carbon Radioisotopes; Cerebellum; Corpus Striatum; Dogs; Male; Piperidines; Radionuclide Imaging; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Ritanserin; Serotonin Antagonists; Spiperone; Sulpiride

1989
Influence of (-)-sulpiride and YM-09151-2 on stereotyped behavior in chicks and catalepsy in rats.
    Japanese journal of pharmacology, 1987, Volume: 43, Issue:2

    Topics: Aging; Animals; Antipsychotic Agents; Benzamides; Catalepsy; Chickens; Dextroamphetamine; Fenclonine; Haloperidol; Male; Rats; Rats, Inbred Strains; Stereoisomerism; Stereotyped Behavior; Sulpiride

1987
Further pharmacological characterization of a D-2-like dopamine receptor on growth hormone producing cells in Lymnaea stagnalis.
    European journal of pharmacology, 1987, Jul-09, Volume: 139, Issue:2

    Topics: Animals; Antipsychotic Agents; Benzamides; Electrophysiology; Growth Hormone; Lymnaea; Microelectrodes; Neurosecretory Systems; Receptors, Dopamine; Receptors, Dopamine D2; Sulpiride

1987
Influence of D-1 receptor system on the D-2 receptor-mediated hypothermic response in mice.
    Life sciences, 1988, Volume: 43, Issue:10

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Anti-Anxiety Agents; Apomorphine; Benzamides; Benzazepines; Dopamine; Dopamine Antagonists; Ergolines; Haloperidol; Hypothermia; Male; Mice; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride

1988
Characteristics of receptors for dopamine in the pars intermedia of the amphibian Xenopus laevis.
    Neuroendocrinology, 1986, Volume: 44, Issue:4

    Topics: Animals; Apomorphine; Benzamides; Domperidone; Dopamine; Drug Interactions; Ergolines; Haloperidol; Melanocyte-Stimulating Hormones; Pituitary Gland, Anterior; Quinpirole; Receptors, Dopamine; Sulpiride; Xenopus laevis

1986
Neuroleptic properties of cis-N-(1-benzyl-2-methylpyrrolidin-3-yl)-5-chloro-2-methoxy-4-methylaminobenzamide (YM-09151-2) with selective antidopaminergic activity.
    Psychopharmacology, 1981, Volume: 73, Issue:2

    Topics: Animals; Antipsychotic Agents; Apomorphine; Benzamides; Chlorpropamide; Dogs; Drug Evaluation, Preclinical; Female; Haloperidol; Humans; Hypothermia; Male; Methamphetamine; Mice; Mice, Inbred ICR; Receptors, Dopamine; Stereotyped Behavior; Sulpiride; Vomiting

1981
Prolactin secretion from human prolactinomas perifused in vitro: effect of TRH, prostaglandin E1, theophylline, dopamine and dopamine receptor blockers.
    Acta endocrinologica, 1984, Volume: 105, Issue:1

    Topics: Adult; Alprostadil; Benzamides; Dopamine; Female; Humans; Male; Perfusion; Pituitary Neoplasms; Prolactin; Prostaglandins E; Receptors, Dopamine; Sulpiride; Theophylline; Thyrotropin-Releasing Hormone

1984
Characterization of [3H]nemonapride binding to mouse brain dopamine D2 receptors assessed in vivo and ex vivo for metabolic modeling in PET studies.
    Journal of neural transmission. General section, 1994, Volume: 97, Issue:2

    Topics: Animals; Benzamides; Brain; Cerebellum; Cerebral Cortex; Chromatography, High Pressure Liquid; Cytosol; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Male; Mice; Mice, Inbred Strains; Neostriatum; Receptors, Dopamine D2; Sulpiride; Tomography, Emission-Computed

1994
Comparison of the effect of substituted benzamides on midbrain dopamine neurones after treatment of rats for 21 days.
    European journal of pharmacology, 1993, Aug-24, Volume: 240, Issue:2-3

    Topics: Animals; Antipsychotic Agents; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Dopamine; Dopamine D2 Receptor Antagonists; Male; Neurons; Pyrrolidines; Raclopride; Rats; Rats, Wistar; Salicylamides; Substantia Nigra; Sulpiride; Ventral Tegmental Area

1993
Dorsal striatal mechanisms involved in the dopamine D2 receptor-mediated potentiation of apomorphine-induced jaw movements.
    European journal of pharmacology, 1994, Jan-24, Volume: 252, Issue:1

    Topics: Animals; Apomorphine; Benzamides; Benzazepines; Corpus Striatum; Dopamine Agents; Dopamine D2 Receptor Antagonists; Drug Synergism; Ergolines; Jaw; Male; Motor Activity; N-Methylscopolamine; Parasympatholytics; Pyrrolidines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Scopolamine Derivatives; Sulpiride

1994
Induction of adenylate cyclase sensitive dopamine D2-receptors in retinoic acid induced differentiated human neuroblastoma SHSY-5Y cells.
    Life sciences, 1994, Volume: 55, Issue:24

    Topics: Adenylyl Cyclases; Amino Acid Sequence; Base Sequence; Benzamides; Cell Differentiation; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Ergolines; Humans; Molecular Sequence Data; Neuroblastoma; Neurons; Quinpirole; Receptors, Dopamine D2; RNA, Messenger; Second Messenger Systems; Sulpiride; Tretinoin; Tumor Cells, Cultured

1994
Effects of benzamide derivatives on dopamine release from striatal slices of rats.
    The Kurume medical journal, 1993, Volume: 40, Issue:4

    Topics: Amisulpride; Animals; Benzamides; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Male; Pyrrolidines; Rats; Rats, Wistar; Sulpiride

1993
Dopamine receptor regulating serotonin N-acetyltransferase activity in chick retina represents a D4-like subtype: pharmacological characterization.
    Neurochemistry international, 1994, Volume: 24, Issue:3

    Topics: Animals; Arylamine N-Acetyltransferase; Benzamides; Benzazepines; Chickens; Circadian Rhythm; Clozapine; Dopamine; Dopamine Antagonists; Ergolines; Ketanserin; Male; Quinpirole; Receptors, Dopamine; Retina; Spiperone; Sulpiride

1994
Depression of the monosynaptic reflex by apomorphine or bromocriptine is not mediated by D1/D2 receptors.
    Neuropharmacology, 1993, Volume: 32, Issue:8

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzamides; Bromocriptine; Decerebrate State; Depression, Chemical; Dopamine Agents; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Ergolines; Male; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Reflex, Monosynaptic; Sulpiride; Synaptic Transmission

1993
YM-09151-2 but not l-sulpiride induces transient dopamine release in rat striatum via a tetrodotoxin-insensitive mechanism.
    Journal of neurochemistry, 1993, Volume: 60, Issue:5

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Benzamides; Calcium; Cerebrospinal Fluid; Corpus Striatum; Dopamine; Dopamine D2 Receptor Antagonists; Homovanillic Acid; Injections; Isotonic Solutions; Male; Nomifensine; Rats; Ringer's Solution; Sulpiride; Tetrodotoxin

1993
Effects of sulpiride and nemonapride, benzamide derivatives having distinct potencies of antagonistic action on dopamine D2 receptors, on sensitization to methamphetamine in mice.
    The Journal of pharmacy and pharmacology, 1996, Volume: 48, Issue:3

    Topics: Animals; Benzamides; Central Nervous System Stimulants; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Male; Methamphetamine; Mice; Motor Activity; Sulpiride; Time Factors

1996
Multiple [3H]-nemonapride binding sites in calf brain.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adrenergic alpha-Antagonists; Animals; Anticonvulsants; Benzamides; Binding, Competitive; Brain; Cattle; Cerebellum; Cerebral Cortex; Corpus Striatum; Dioxanes; Dopamine Agonists; Dopamine Antagonists; Guanidines; Haloperidol; In Vitro Techniques; Isotope Labeling; Narcotic Antagonists; Pentazocine; Piperidines; Propylamines; Pyrrolidines; Receptors, Dopamine D2; Receptors, sigma; Sulpiride; Tritium

1997
(-)S amisulpride binds with high affinity to cloned dopamine D(3) and D(2) receptors.
    European journal of pharmacology, 2001, Dec-07, Volume: 432, Issue:2-3

    Topics: Amisulpride; Animals; Benzamides; Binding, Competitive; Cell Line; DNA, Recombinant; Dopamine Antagonists; Dose-Response Relationship, Drug; Humans; Radioligand Assay; Rats; Receptors, Dopamine D2; Receptors, Dopamine D3; Spiperone; Stereoisomerism; Sulpiride; Tritium

2001
Dopamine released by dendritic cells polarizes Th2 differentiation.
    International immunology, 2009, Volume: 21, Issue:6

    Topics: Benzamides; Cell Communication; Cell Differentiation; Cells, Cultured; Colchicine; Colforsin; Cyclic AMP; Dendritic Cells; Dopamine; Dopamine D2 Receptor Antagonists; Humans; Lymphocyte Activation; Lymphocyte Culture Test, Mixed; Receptors, Dopamine D1; Receptors, Dopamine D2; Secretory Vesicles; Sulpiride; Th1 Cells; Th2 Cells

2009
[(3)H]-YM-09151-2 binding sites in human brain postmortem.
    Neurochemistry international, 2009, Volume: 55, Issue:7

    Topics: Aged; Benzamides; Binding Sites; Brain Chemistry; Data Interpretation, Statistical; Dopamine Antagonists; Female; Hippocampus; Humans; In Vitro Techniques; Kinetics; Male; Middle Aged; Neostriatum; Postmortem Changes; Prefrontal Cortex; Propylamines; Raclopride; Receptors, Dopamine D4; Receptors, sigma; Sulpiride

2009
Chemotactic migration of newly excysted juvenile Clonorchis sinensis is suppressed by neuro-antagonists.
    PLoS neglected tropical diseases, 2019, Volume: 13, Issue:8

    Topics: Animals; Benzamides; Biphenyl Compounds; Chemotaxis; Cholic Acid; Clonorchis sinensis; Dopamine; Dopamine Uptake Inhibitors; Excitatory Amino Acid Agents; Fasciola hepatica; Fluorenes; FMRFamide; Neuropeptide Y; Neurotransmitter Agents; Peptide YY; Piperazines; Serotonin Agents; Spiro Compounds; Sulpiride

2019