ym 09151-2 has been researched along with sulpiride in 24 studies
Studies (ym 09151-2) | Trials (ym 09151-2) | Recent Studies (post-2010) (ym 09151-2) | Studies (sulpiride) | Trials (sulpiride) | Recent Studies (post-2010) (sulpiride) |
---|---|---|---|---|---|
249 | 6 | 13 | 4,152 | 427 | 635 |
Protein | Taxonomy | ym 09151-2 (IC50) | sulpiride (IC50) |
---|---|---|---|
Carbonic anhydrase 1 | Homo sapiens (human) | 1.2 | |
Carbonic anhydrase 2 | Homo sapiens (human) | 0.04 | |
Alpha-2A adrenergic receptor | Homo sapiens (human) | 2.019 | |
D(2) dopamine receptor | Homo sapiens (human) | 0.0858 | |
D(3) dopamine receptor | Homo sapiens (human) | 0.2651 | |
D(2) dopamine receptor | Rattus norvegicus (Norway rat) | 0.2215 | |
Carbonic anhydrase 4 | Bos taurus (cattle) | 0.62 | |
D(2) dopamine receptor | Canis lupus familiaris (dog) | 0.2 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 7 (29.17) | 18.7374 |
1990's | 13 (54.17) | 18.2507 |
2000's | 3 (12.50) | 29.6817 |
2010's | 1 (4.17) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Kobayashi, M; Koshikawa, N; Maruyama, Y; Mori, E; Yatsushige, N | 1 |
Kobayashi, T; Shimizu, H; Toru, M | 1 |
Arai, I; Higuchi, T; Kazawa, T; Mikuni, M; Takahashi, K; Yamauchi, T | 1 |
Hatano, K; Hatazawa, J; Ido, T; Ishiwata, K; Itoh, M; Kawashima, K | 1 |
Wambebe, C | 1 |
De Vlieger, TA; Lodder, JC; Stoof, JC; Werkman, TR | 1 |
Fitten, J; Gordon, LI; Kodama, CK; Menon, MK | 1 |
Jenks, BG; Tonon, MC; Vaudry, H; Verburg-Van Kemenade, BM | 1 |
Maeno, H; Nishikori, K; Noshiro, O; Usuda, S | 1 |
Chihara, K; Fujita, T; Iwasaki, J; Kaji, H; Kodama, H; Matsumoto, S; Minamitani, N; Shirataki, K; Tamaki, N | 1 |
Inami, K; Ishiwata, K; Nozaki, T; Sasaki, T; Senda, M | 1 |
Skarsfeldt, T | 1 |
Kikuchi de Beltrán, K; Kobayashi, M; Koshikawa, N; Miwa, Y | 1 |
Farooqui, SM | 1 |
Nishi, S; Yamada, S; Yokoo, H | 1 |
Nowak, JZ; Zawilska, JB | 1 |
Kamijo, N; Nagao, T; Ono, H | 1 |
Kobayashi, M; Koshikawa, N; Noguchi, M; Tomiyama, K | 1 |
Kuribara, H | 1 |
Fang, H; Helmeste, DM; Li, M; Tang, SW | 1 |
Castelli, MP; Gessa, GL; Mocci, I; Pani, L; Sanna, AM | 1 |
Hashimoto, K; Higashi, T; Matsushita, S; Nakano, K; Takagi, R; Tanaka, Y | 1 |
Baroni, S; Betti, L; Castagna, M; Catena Dell'Osso, M; Consoli, G; Giannaccini, G; Lucacchini, A; Marazziti, D; Masala, I; Palego, L | 1 |
Dai, F; Hong, SJ; Kim, TI; Li, S; Song, JH; Won, MH; Yoo, WG | 1 |
24 other study(ies) available for ym 09151-2 and sulpiride
Article | Year |
---|---|
Role of dopamine D-1 and D-2 receptors in the ventral striatum in the turning behaviour of rats.
Topics: Animals; Apomorphine; Benzamides; Benzazepines; Corpus Striatum; Dopamine Agents; Dopamine Antagonists; Flupenthixol; Male; Methamphetamine; Microinjections; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereotyped Behavior; Sulpiride | 1990 |
[The inhibition of dopamine D1 and D2 receptors in human putamen by antipsychotic drugs].
Topics: Aged; Aged, 80 and over; Antipsychotic Agents; Benzamides; Benzazepines; Chlorpromazine; Depression, Chemical; Female; Haloperidol; Humans; In Vitro Techniques; Putamen; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Sulpiride | 1990 |
Characterization of sulpiride-displaceable 3H-YM-09151-2 binding sites in rat frontal cortex and the effects of subchronic treatment with haloperidol on cortical D-2 dopamine receptors.
Topics: Animals; Benzamides; Binding Sites; Corpus Striatum; Dopamine Antagonists; Frontal Lobe; Haloperidol; In Vitro Techniques; Ketanserin; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride | 1990 |
D2-dopamine receptor specific brain uptake of carbon-11-labeled YM-09151-2.
Topics: Animals; Antipsychotic Agents; Benzamides; Brain; Carbon Radioisotopes; Cerebellum; Corpus Striatum; Dogs; Male; Piperidines; Radionuclide Imaging; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Ritanserin; Serotonin Antagonists; Spiperone; Sulpiride | 1989 |
Influence of (-)-sulpiride and YM-09151-2 on stereotyped behavior in chicks and catalepsy in rats.
Topics: Aging; Animals; Antipsychotic Agents; Benzamides; Catalepsy; Chickens; Dextroamphetamine; Fenclonine; Haloperidol; Male; Rats; Rats, Inbred Strains; Stereoisomerism; Stereotyped Behavior; Sulpiride | 1987 |
Further pharmacological characterization of a D-2-like dopamine receptor on growth hormone producing cells in Lymnaea stagnalis.
Topics: Animals; Antipsychotic Agents; Benzamides; Electrophysiology; Growth Hormone; Lymnaea; Microelectrodes; Neurosecretory Systems; Receptors, Dopamine; Receptors, Dopamine D2; Sulpiride | 1987 |
Influence of D-1 receptor system on the D-2 receptor-mediated hypothermic response in mice.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Anti-Anxiety Agents; Apomorphine; Benzamides; Benzazepines; Dopamine; Dopamine Antagonists; Ergolines; Haloperidol; Hypothermia; Male; Mice; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride | 1988 |
Characteristics of receptors for dopamine in the pars intermedia of the amphibian Xenopus laevis.
Topics: Animals; Apomorphine; Benzamides; Domperidone; Dopamine; Drug Interactions; Ergolines; Haloperidol; Melanocyte-Stimulating Hormones; Pituitary Gland, Anterior; Quinpirole; Receptors, Dopamine; Sulpiride; Xenopus laevis | 1986 |
Neuroleptic properties of cis-N-(1-benzyl-2-methylpyrrolidin-3-yl)-5-chloro-2-methoxy-4-methylaminobenzamide (YM-09151-2) with selective antidopaminergic activity.
Topics: Animals; Antipsychotic Agents; Apomorphine; Benzamides; Chlorpropamide; Dogs; Drug Evaluation, Preclinical; Female; Haloperidol; Humans; Hypothermia; Male; Methamphetamine; Mice; Mice, Inbred ICR; Receptors, Dopamine; Stereotyped Behavior; Sulpiride; Vomiting | 1981 |
Prolactin secretion from human prolactinomas perifused in vitro: effect of TRH, prostaglandin E1, theophylline, dopamine and dopamine receptor blockers.
Topics: Adult; Alprostadil; Benzamides; Dopamine; Female; Humans; Male; Perfusion; Pituitary Neoplasms; Prolactin; Prostaglandins E; Receptors, Dopamine; Sulpiride; Theophylline; Thyrotropin-Releasing Hormone | 1984 |
Characterization of [3H]nemonapride binding to mouse brain dopamine D2 receptors assessed in vivo and ex vivo for metabolic modeling in PET studies.
Topics: Animals; Benzamides; Brain; Cerebellum; Cerebral Cortex; Chromatography, High Pressure Liquid; Cytosol; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Male; Mice; Mice, Inbred Strains; Neostriatum; Receptors, Dopamine D2; Sulpiride; Tomography, Emission-Computed | 1994 |
Comparison of the effect of substituted benzamides on midbrain dopamine neurones after treatment of rats for 21 days.
Topics: Animals; Antipsychotic Agents; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Dopamine; Dopamine D2 Receptor Antagonists; Male; Neurons; Pyrrolidines; Raclopride; Rats; Rats, Wistar; Salicylamides; Substantia Nigra; Sulpiride; Ventral Tegmental Area | 1993 |
Dorsal striatal mechanisms involved in the dopamine D2 receptor-mediated potentiation of apomorphine-induced jaw movements.
Topics: Animals; Apomorphine; Benzamides; Benzazepines; Corpus Striatum; Dopamine Agents; Dopamine D2 Receptor Antagonists; Drug Synergism; Ergolines; Jaw; Male; Motor Activity; N-Methylscopolamine; Parasympatholytics; Pyrrolidines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Scopolamine Derivatives; Sulpiride | 1994 |
Induction of adenylate cyclase sensitive dopamine D2-receptors in retinoic acid induced differentiated human neuroblastoma SHSY-5Y cells.
Topics: Adenylyl Cyclases; Amino Acid Sequence; Base Sequence; Benzamides; Cell Differentiation; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Ergolines; Humans; Molecular Sequence Data; Neuroblastoma; Neurons; Quinpirole; Receptors, Dopamine D2; RNA, Messenger; Second Messenger Systems; Sulpiride; Tretinoin; Tumor Cells, Cultured | 1994 |
Effects of benzamide derivatives on dopamine release from striatal slices of rats.
Topics: Amisulpride; Animals; Benzamides; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Male; Pyrrolidines; Rats; Rats, Wistar; Sulpiride | 1993 |
Dopamine receptor regulating serotonin N-acetyltransferase activity in chick retina represents a D4-like subtype: pharmacological characterization.
Topics: Animals; Arylamine N-Acetyltransferase; Benzamides; Benzazepines; Chickens; Circadian Rhythm; Clozapine; Dopamine; Dopamine Antagonists; Ergolines; Ketanserin; Male; Quinpirole; Receptors, Dopamine; Retina; Spiperone; Sulpiride | 1994 |
Depression of the monosynaptic reflex by apomorphine or bromocriptine is not mediated by D1/D2 receptors.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzamides; Bromocriptine; Decerebrate State; Depression, Chemical; Dopamine Agents; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Ergolines; Male; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Reflex, Monosynaptic; Sulpiride; Synaptic Transmission | 1993 |
YM-09151-2 but not l-sulpiride induces transient dopamine release in rat striatum via a tetrodotoxin-insensitive mechanism.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Benzamides; Calcium; Cerebrospinal Fluid; Corpus Striatum; Dopamine; Dopamine D2 Receptor Antagonists; Homovanillic Acid; Injections; Isotonic Solutions; Male; Nomifensine; Rats; Ringer's Solution; Sulpiride; Tetrodotoxin | 1993 |
Effects of sulpiride and nemonapride, benzamide derivatives having distinct potencies of antagonistic action on dopamine D2 receptors, on sensitization to methamphetamine in mice.
Topics: Animals; Benzamides; Central Nervous System Stimulants; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Male; Methamphetamine; Mice; Motor Activity; Sulpiride; Time Factors | 1996 |
Multiple [3H]-nemonapride binding sites in calf brain.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adrenergic alpha-Antagonists; Animals; Anticonvulsants; Benzamides; Binding, Competitive; Brain; Cattle; Cerebellum; Cerebral Cortex; Corpus Striatum; Dioxanes; Dopamine Agonists; Dopamine Antagonists; Guanidines; Haloperidol; In Vitro Techniques; Isotope Labeling; Narcotic Antagonists; Pentazocine; Piperidines; Propylamines; Pyrrolidines; Receptors, Dopamine D2; Receptors, sigma; Sulpiride; Tritium | 1997 |
(-)S amisulpride binds with high affinity to cloned dopamine D(3) and D(2) receptors.
Topics: Amisulpride; Animals; Benzamides; Binding, Competitive; Cell Line; DNA, Recombinant; Dopamine Antagonists; Dose-Response Relationship, Drug; Humans; Radioligand Assay; Rats; Receptors, Dopamine D2; Receptors, Dopamine D3; Spiperone; Stereoisomerism; Sulpiride; Tritium | 2001 |
Dopamine released by dendritic cells polarizes Th2 differentiation.
Topics: Benzamides; Cell Communication; Cell Differentiation; Cells, Cultured; Colchicine; Colforsin; Cyclic AMP; Dendritic Cells; Dopamine; Dopamine D2 Receptor Antagonists; Humans; Lymphocyte Activation; Lymphocyte Culture Test, Mixed; Receptors, Dopamine D1; Receptors, Dopamine D2; Secretory Vesicles; Sulpiride; Th1 Cells; Th2 Cells | 2009 |
[(3)H]-YM-09151-2 binding sites in human brain postmortem.
Topics: Aged; Benzamides; Binding Sites; Brain Chemistry; Data Interpretation, Statistical; Dopamine Antagonists; Female; Hippocampus; Humans; In Vitro Techniques; Kinetics; Male; Middle Aged; Neostriatum; Postmortem Changes; Prefrontal Cortex; Propylamines; Raclopride; Receptors, Dopamine D4; Receptors, sigma; Sulpiride | 2009 |
Chemotactic migration of newly excysted juvenile Clonorchis sinensis is suppressed by neuro-antagonists.
Topics: Animals; Benzamides; Biphenyl Compounds; Chemotaxis; Cholic Acid; Clonorchis sinensis; Dopamine; Dopamine Uptake Inhibitors; Excitatory Amino Acid Agents; Fasciola hepatica; Fluorenes; FMRFamide; Neuropeptide Y; Neurotransmitter Agents; Peptide YY; Piperazines; Serotonin Agents; Spiro Compounds; Sulpiride | 2019 |