Page last updated: 2024-09-04

ym 09151-2 and sk&f-38393

ym 09151-2 has been researched along with sk&f-38393 in 14 studies

Compound Research Comparison

Studies
(ym 09151-2)
Trials
(ym 09151-2)
Recent Studies (post-2010)
(ym 09151-2)
Studies
(sk&f-38393)
Trials
(sk&f-38393)
Recent Studies (post-2010) (sk&f-38393)
2496132,01229242

Protein Interaction Comparison

ProteinTaxonomyym 09151-2 (IC50)sk&f-38393 (IC50)
Replicase polyprotein 1abSevere acute respiratory syndrome coronavirus 22.8
DRattus norvegicus (Norway rat)0.19

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19906 (42.86)18.7374
1990's5 (35.71)18.2507
2000's3 (21.43)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cody, P; Eisner, GM; Felder, RA; Jose, PA; Seikaly, MG1
Bickford-Wimer, PC; Gratton, A; Parfitt, KD1
Arnt, J; Hyttel, J1
Beaulieu, M; Felder, R; Kebabian, JW1
Fernández, M; Jantos, H; Monti, JM1
Fitten, J; Gordon, LI; Kodama, CK; Menon, MK1
Walters, JR; Weick, BG1
Agui, T; Chase, TN; Kebabian, JW1
Palacios, JM; Wiederhold, KH1
Kamijo, N; Nagao, T; Ono, H1
Deveney, AM; Waddington, JL1
Clifford, JJ; Croke, DT; Drago, J; Kinsella, A; McNamara, FN; Tighe, O; Waddington, JL1
Kinsella, A; O'Sullivan, GJ; Roth, BL; Waddington, JL1
Cools, AR; Fujita, S; Kiguchi, M; Koshikawa, N; Lee, J; Uchida, T; Waddington, JL1

Other Studies

14 other study(ies) available for ym 09151-2 and sk&f-38393

ArticleYear
Attenuated renal response to dopaminergic drugs in spontaneously hypertensive rats.
    Hypertension (Dallas, Tex. : 1979), 1990, Volume: 15, Issue:6 Pt 1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzamides; Benzazepines; Dopamine Agents; Dopamine Antagonists; Hypertension; Kidney; Male; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Dopamine; Receptors, Dopamine D1; Regression Analysis; Urodynamics

1990
Electrophysiological effects of selective D1 and D2 dopamine receptor agonists in the medial prefrontal cortex of young and aged Fischer 344 rats.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 254, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Aging; Animals; Benzamides; Benzazepines; Cerebral Cortex; Dopamine Agents; Dopamine Antagonists; Dose-Response Relationship, Drug; Electrophysiology; Male; Naphthalenes; Neurons; Rats; Rats, Inbred F344; Tetrahydronaphthalenes; Thiophenes

1990
Dopamine D-2 agonists with high and low efficacies: differentiation by behavioural techniques.
    Journal of neural transmission. General section, 1990, Volume: 80, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzamides; Drug Combinations; Male; Motor Activity; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Stereotyped Behavior

1990
D-2 dopaminergic agonists and adenosine 3',5'-monophosphate directly regulate the synthesis of alpha-melanocyte-stimulating hormone-like peptides by cultured rat melanotrophs.
    Endocrinology, 1986, Volume: 118, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Benzamides; Benzazepines; Bromocriptine; Cells, Cultured; Chemical Precipitation; Cholera Toxin; Chromatography, High Pressure Liquid; Colforsin; Cyclic AMP; Dopamine; Ergolines; Immunologic Techniques; Melanocyte-Stimulating Hormones; Pituitary Gland; Pro-Opiomelanocortin; Quinpirole; Rats; Receptors, Dopamine; Spiperone

1986
Effects of the selective dopamine D-2 receptor agonist, quinpirole on sleep and wakefulness in the rat.
    European journal of pharmacology, 1989, Oct-04, Volume: 169, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Benzamides; Dopamine Agents; Electroencephalography; Ergolines; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sleep; Sleep, REM; Wakefulness

1989
Influence of D-1 receptor system on the D-2 receptor-mediated hypothermic response in mice.
    Life sciences, 1988, Volume: 43, Issue:10

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Anti-Anxiety Agents; Apomorphine; Benzamides; Benzazepines; Dopamine; Dopamine Antagonists; Ergolines; Haloperidol; Hypothermia; Male; Mice; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride

1988
Effects of D1 and D2 dopamine receptor stimulation on the activity of substantia nigra pars reticulata neurons in 6-hydroxydopamine lesioned rats: D1/D2 coactivation induces potentiated responses.
    Brain research, 1987, Mar-10, Volume: 405, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Action Potentials; Animals; Apomorphine; Benzamides; Benzazepines; Dopamine; Dopamine Antagonists; Drug Interactions; Ergolines; Hydroxydopamines; Male; Oxidopamine; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Substantia Nigra; Time Factors

1987
Identification of D1-dopamine receptor in chicken embryo retina with [125I]SCH 23982.
    Brain research, 1988, Jun-14, Volume: 452, Issue:1-2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Benzamides; Benzazepines; Chick Embryo; Corpus Striatum; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Retina

1988
Dopamine D2 receptor agents, but not dopamine D1, modify brain glucose metabolism.
    Brain research, 1985, Feb-18, Volume: 327, Issue:1-2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Benzamides; Benzazepines; Brain; Ergolines; Glucose; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2

1985
Depression of the monosynaptic reflex by apomorphine or bromocriptine is not mediated by D1/D2 receptors.
    Neuropharmacology, 1993, Volume: 32, Issue:8

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzamides; Bromocriptine; Decerebrate State; Depression, Chemical; Dopamine Agents; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Ergolines; Male; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Reflex, Monosynaptic; Sulpiride; Synaptic Transmission

1993
Pharmacological characterization of behavioural responses to SK&F 83959 in relation to 'D1-like' dopamine receptors not linked to adenylyl cyclase.
    British journal of pharmacology, 1995, Volume: 116, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Behavior, Animal; Benzamides; Benzazepines; Binding, Competitive; Chromans; Dopamine Agonists; Dopamine Antagonists; Enzyme Induction; Isoquinolines; Male; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Spiperone; Tetrahydroisoquinolines

1995
Congenic D1A dopamine receptor mutants: ethologically based resolution of behavioural topography indicates genetic background as a determinant of knockout phenotype.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2003, Volume: 28, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Animals, Congenic; Behavior, Animal; Benzamides; Benzazepines; Dopamine Agonists; Dopamine Antagonists; Exploratory Behavior; Habituation, Psychophysiologic; Mice; Mice, Inbred C57BL; Mice, Knockout; Motor Activity; Mutation; Phenethylamines; Phenotype; Receptors, Dopamine D1; Transgenes

2003
SK&F 83822 distinguishes adenylyl cyclase from phospholipase C-coupled dopamine D1-like receptors: behavioural topography.
    European journal of pharmacology, 2004, Feb-23, Volume: 486, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Benzamides; Benzazepines; Binding, Competitive; Dopamine D2 Receptor Antagonists; Male; Mice; Mice, Inbred C57BL; Motor Activity; Radioligand Assay; Receptors, Dopamine D1; Type C Phospholipases

2004
Topographical resolution of jaw movements mediated by cyclase- vs. non-cyclase-coupled dopamine D(1)-like receptors: studies with SK&F 83822.
    European journal of pharmacology, 2006, May-24, Volume: 538, Issue:1-3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Analysis of Variance; Animals; Benzamides; Benzazepines; Dopamine Agonists; Dopamine Antagonists; Jaw; Male; Movement; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Time Factors

2006