Page last updated: 2024-09-04

ym 09151-2 and raclopride

ym 09151-2 has been researched along with raclopride in 27 studies

Compound Research Comparison

Studies (ym 09151-2)	Trials (ym 09151-2)	Recent Studies (post-2010) (ym 09151-2)	Studies (raclopride)	Trials (raclopride)	Recent Studies (post-2010) (raclopride)
249	6	13	1,802	132	419

Protein Interaction Comparison

Protein	Taxonomy	raclopride (IC50)
D(2) dopamine receptor	Homo sapiens (human)	0.052
D(2) dopamine receptor	Mus musculus (house mouse)	0.032
D(2) dopamine receptor	Rattus norvegicus (Norway rat)	0.0279

Research

Studies (27)

Timeframe	Studies, this research(%)	All Research%
pre-1990	1 (3.70)	18.7374
1990's	19 (70.37)	18.2507
2000's	7 (25.93)	29.6817
2010's	0 (0.00)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Civelli, O; Guan, HC; Niznik, HB; Seeman, P; Sunahara, RK; Van Tol, HH	1
Clifton, PG; Cooper, SJ; Rusk, IN	1
Hidaka, K; Nakamura, Y; Terai, M	1
Meltzer, HY; Overholser, JC; Stockmeier, CA; Sumiyoshi, T; Thompson, PA	1
Strange, PG; Vile, JM	1
Asghari, V; Buchwaldt, S; Jovanovic, V; Paterson, A; Sanyal, S; Van Tol, HH	1
Seeman, P; Van Tol, HH	1
Bigelow, LB; Carter, JM; Herman, MM; Hyde, TM; Kleinman, JE; Knable, MB; Murray, AM; Weinberger, DR	1
Skarsfeldt, T	1
Mason, SL; Reynolds, GP	1
Guan, HC; Niznik, HB; Seeman, P; Van Tol, HH	1
Fang, H; Helmeste, D; Li, M; Tang, SW	1
Hyde, TM; Knable, MB; Murray, AM	1
Creese, I; Florijn, WJ; Tarazi, FI	1
Antonelli, MC; Defagot, MC	1
Bunney, W; Fang, H; Helmeste, DM; Jones, EG; Li, M; Potkin, S; Tang, SW; Vu, R	1
Copolov, D; Hill, C; Keks, N; Marzella, PL; Singh, B	1
Kleven, MS; Koek, W; Prinssen, EP	2
Tsuchiya, K	1
Endo, K; Hayakawa, N; Ishiwata, K; Oda, K; Ogi, N; Senda, M; Tanaka, A; Toyama, H	1
Antonelli, MC; Defagot, MC; Falzone, TL; Grandy, DK; Low, MJ; Rubinstein, M	1
Endo, K; Hayakawa, N; Ishiwata, K; Nagaoka, T; Oda, K; Ogi, N; Senda, M; Tanaka, A; Toyama, H; Umegaki, H	1
Berra, R; Flores, G; Gómez, Mde J; Nadeau, R; Rousseau, G; Suárez, J	1
Ishiwata, K; Kawamura, K; Kobayashi, T; Matsuno, K	1
Lin, H; Strange, PG; Vivo, M	1
Baroni, S; Betti, L; Castagna, M; Catena Dell'Osso, M; Consoli, G; Giannaccini, G; Lucacchini, A; Marazziti, D; Masala, I; Palego, L	1

Other Studies

27 other study(ies) available for ym 09151-2 and raclopride

Article	Year
The cloned dopamine D2 receptor reveals different densities for dopamine receptor antagonist ligands. Implications for human brain positron emission tomography. European journal of pharmacology, 1992, Oct-01, Volume: 227, Issue:2 Topics: Antipsychotic Agents; Benzamides; Brain Chemistry; Cloning, Molecular; Dopamine D2 Receptor Antagonists; Humans; Pituitary Gland, Anterior; Raclopride; Receptors, Dopamine D2; Salicylamides; Spiperone; Tomography, Emission-Computed	1992
Effects of dopamine D1 and dopamine D2 antagonists on the free feeding and drinking patterns of rats. Behavioral neuroscience, 1991, Volume: 105, Issue:2 Topics: Animals; Antipsychotic Agents; Arousal; Benzamides; Benzazepines; Brain; Circadian Rhythm; Dopamine Antagonists; Dose-Response Relationship, Drug; Drinking Behavior; Feeding Behavior; Male; Motivation; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine D1; Receptors, Dopamine D2; Remoxipride; Salicylamides	1991
Comparison of [3H]YM-09151-2 with [3H]spiperone and [3H]raclopride for dopamine d-2 receptor binding to rat striatum. European journal of pharmacology, 1989, Dec-07, Volume: 173, Issue:2-3 Topics: Animals; Antipsychotic Agents; Benzamides; Corpus Striatum; Kinetics; Male; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Salicylamides; Spiperone	1989
Dopamine D4 receptors and effects of guanine nucleotides on [3H]raclopride binding in postmortem caudate nucleus of subjects with schizophrenia or major depression. Brain research, 1995, May-29, Volume: 681, Issue:1-2 Topics: Adult; Aged; Aged, 80 and over; Benzamides; Caudate Nucleus; Depressive Disorder; Dopamine Antagonists; Female; GTP-Binding Proteins; Guanine Nucleotides; Guanylyl Imidodiphosphate; Humans; In Vitro Techniques; Kinetics; Male; Middle Aged; Raclopride; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Salicylamides; Schizophrenia	1995
D4 receptors and schizophrenia. Journal of neurochemistry, 1995, Volume: 65, Issue:5 Topics: Benzamides; Binding, Competitive; Dopamine Antagonists; Humans; Raclopride; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Salicylamides; Schizophrenia	1995
Modulation of intracellular cyclic AMP levels by different human dopamine D4 receptor variants. Journal of neurochemistry, 1995, Volume: 65, Issue:3 Topics: Animals; Benzamides; Cell Line; CHO Cells; Clozapine; Colforsin; Cricetinae; Cyclic AMP; Dinoprostone; Dopamine; Haloperidol; HeLa Cells; Humans; Raclopride; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Proteins; Salicylamides; Spiperone; Transfection	1995
Dopamine D4-like receptor elevation in schizophrenia: cloned D2 and D4 receptors cannot be discriminated by raclopride competition against [3H]nemonapride. Journal of neurochemistry, 1995, Volume: 64, Issue:3 Topics: Animals; Benzamides; Binding, Competitive; Dopamine Antagonists; Humans; In Vitro Techniques; Raclopride; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Recombinant Proteins; Salicylamides; Schizophrenia	1995
Distribution of putative D4 dopamine receptors in postmortem striatum from patients with schizophrenia. The Journal of neuroscience : the official journal of the Society for Neuroscience, 1995, Volume: 15, Issue:3 Pt 2 Topics: Adult; Aged; Aged, 80 and over; Antipsychotic Agents; Benzamides; Corpus Striatum; Female; Humans; Male; Mental Disorders; Middle Aged; Nucleus Accumbens; Raclopride; Radioligand Assay; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Salicylamides; Schizophrenia; Suicide; Up-Regulation	1995
Comparison of the effect of substituted benzamides on midbrain dopamine neurones after treatment of rats for 21 days. European journal of pharmacology, 1993, Aug-24, Volume: 240, Issue:2-3 Topics: Animals; Antipsychotic Agents; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Dopamine; Dopamine D2 Receptor Antagonists; Male; Neurons; Pyrrolidines; Raclopride; Rats; Rats, Wistar; Salicylamides; Substantia Nigra; Sulpiride; Ventral Tegmental Area	1993
Are striatal dopamine D4 receptors increased in schizophrenia? Journal of neurochemistry, 1994, Volume: 63, Issue:4 Topics: Aged; Animals; Antipsychotic Agents; Benzamides; Binding, Competitive; Corpus Striatum; Dopamine D2 Receptor Antagonists; Humans; Kinetics; Pyrrolidines; Raclopride; Receptors, Dopamine; Receptors, Dopamine D4; Reference Values; Salicylamides; Schizophrenia	1994
Low density of dopamine D4 receptors in Parkinson's, schizophrenia, and control brain striata. Synapse (New York, N.Y.), 1993, Volume: 14, Issue:4 Topics: Animals; Benzamides; Corpus Striatum; Dopamine D2 Receptor Antagonists; Humans; In Vitro Techniques; Kinetics; Parkinson Disease; Pituitary Gland, Anterior; Pyrrolidines; Raclopride; Rats; Receptors, Dopamine; Receptors, Dopamine D4; Salicylamides; Schizophrenia; Spiperone; Swine; Tomography, Emission-Computed	1993
Brain sigma receptors labelled by [3H]nemonapride. European journal of pharmacology, 1996, Apr-22, Volume: 301, Issue:1-3 Topics: Animals; Benzamides; Binding, Competitive; Brain Chemistry; Cattle; Dopamine Antagonists; Humans; In Vitro Techniques; Raclopride; Rats; Receptors, Dopamine D2; Receptors, Dopamine D4; Receptors, sigma; Salicylamides	1996
Distribution of dopamine D1-D4 receptor subtypes in human dorsal vagal complex. Synapse (New York, N.Y.), 1996, Volume: 24, Issue:3 Topics: Adolescent; Adult; Aged; Autoradiography; Benzamides; Benzazepines; Dopamine Antagonists; Humans; Ligands; Male; Medulla Oblongata; Middle Aged; Pyrrolidines; Raclopride; Receptors, Dopamine; Salicylamides; Vagus Nerve	1996
Dopamine receptor subtypes: differential regulation after 8 months treatment with antipsychotic drugs. The Journal of pharmacology and experimental therapeutics, 1997, Volume: 280, Issue:2 Topics: Animals; Antipsychotic Agents; Benzamides; Benzazepines; Brain; Clozapine; Corpus Striatum; Haloperidol; Iodine Radioisotopes; Male; Organ Specificity; Raclopride; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Serotonin; Salicylamides; Spiperone; Tetrahydronaphthalenes; Time Factors; Tritium; Up-Regulation	1997
Autoradiographic localization of the putative D4 dopamine receptor in rat brain. Neurochemical research, 1997, Volume: 22, Issue:4 Topics: Animals; Autoradiography; Benzamides; Brain Chemistry; Dopamine Antagonists; Kinetics; Male; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D4; Salicylamides; Tritium	1997
Differential labeling of dopamine and sigma sites by [3H]nemonapride and [3H]raclopride in postmortem human brains. Brain research, 1997, Aug-08, Volume: 765, Issue:1 Topics: Adult; Aged; Benzamides; Brain Chemistry; Dopamine Antagonists; Humans; In Vitro Techniques; Kinetics; Male; Middle Aged; Raclopride; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Receptors, sigma; Salicylamides; Schizophrenia	1997
The binding of both [3H]nemonapride and [3H]raclopride is increased in schizophrenia. Biological psychiatry, 1997, Oct-15, Volume: 42, Issue:8 Topics: Adult; Aged; Antipsychotic Agents; Autoradiography; Benzamides; Caudate Nucleus; Cerebral Cortex; Female; Humans; Male; Middle Aged; Putamen; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Dopamine D4; Reference Values; Salicylamides; Schizophrenia	1997
The cataleptogenic effects of the neuroleptic nemonapride are attenuated by its 5-HT1A receptor agonist properties. European journal of pharmacology, 1998, Sep-04, Volume: 356, Issue:2-3 Topics: Animals; Antipsychotic Agents; Benzamides; Catalepsy; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Haloperidol; Male; Piperazines; Pyridines; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Salicylamides; Serotonin Antagonists; Serotonin Receptor Agonists	1998
[Effects of methamphetamine on responsiveness to conditioned fear stress]. [Hokkaido igaku zasshi] The Hokkaido journal of medical science, 1999, Volume: 74, Issue:1 Topics: Animals; Benzamides; Benzazepines; Brain Chemistry; Central Nervous System Stimulants; Conditioning, Psychological; Corpus Striatum; Dizocilpine Maleate; Dopamine; Dopamine Antagonists; Excitatory Amino Acid Antagonists; Fear; Fluoxetine; Homovanillic Acid; Male; Methamphetamine; Nalidixic Acid; Naphthyridines; Raclopride; Rats; Rats, Wistar; Salicylamides; Selective Serotonin Reuptake Inhibitors; Stress, Psychological	1999
Comparison of three PET dopamine D2-like receptor ligands, [11C]raclopride, [11C]nemonapride and [11C]N-methylspiperone, in rats. Annals of nuclear medicine, 1999, Volume: 13, Issue:3 Topics: Animals; Benzamides; Brain; Cerebellum; Dopamine Agonists; Dopamine Antagonists; Ligands; Male; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D2; Salicylamides; Spiperone; Tissue Distribution; Tomography, Emission-Computed; Visual Cortex	1999
Quantitative analysis of the dopamine D4 receptor in the mouse brain. Journal of neuroscience research, 2000, Jan-15, Volume: 59, Issue:2 Topics: Animals; Autoradiography; Benzamides; Binding Sites; Brain Chemistry; Dopamine Antagonists; Female; Ligands; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Quantitative Trait, Heritable; Raclopride; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D4; Synaptosomes; Tritium	2000
Effects of WAY 100635 on antipsychotic-induced catalepsy in 5-HT depleted animals: a role for tonic activation of 5-HT(1A) receptors. European journal of pharmacology, 2000, Apr-28, Volume: 395, Issue:2 Topics: Animals; Antipsychotic Agents; Benzamides; Catalepsy; Dose-Response Relationship, Drug; Drug Interactions; Male; Piperazines; Pyridines; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists	2000
Positron emission tomography and ex vivo and in vitro autoradiography studies on dopamine D2-like receptor degeneration in the quinolinic acid-lesioned rat striatum: comparison of [11C]raclopride, [11C]nemonapride and [11C]N-methylspiperone. Nuclear medicine and biology, 2002, Volume: 29, Issue:3 Topics: Animals; Autoradiography; Benzamides; Dopamine Antagonists; Glucose; Magnetic Resonance Imaging; Male; Neostriatum; Neurotoxins; Quinolinic Acid; Raclopride; Radiopharmaceuticals; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, GABA-A; Spiperone; Tomography, Emission-Computed	2002
Functional and autoradiographic characterization of dopamine D2-like receptors in the guinea pig heart. Canadian journal of physiology and pharmacology, 2002, Volume: 80, Issue:6 Topics: Adenylyl Cyclases; Animals; Autoradiography; Benzamides; Blood Pressure; Blotting, Western; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Electrophysiology; Guinea Pigs; Heart Rate; In Vitro Techniques; Kinetics; Male; Membranes; Myocardium; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Dopamine D4; Tetrahydronaphthalenes	2002
Sigma1 and dopamine D2 receptor occupancy in the mouse brain after a single administration of haloperidol and two dopamine D2-like receptor ligands. Nuclear medicine and biology, 2003, Volume: 30, Issue:4 Topics: Animals; Benzamides; Brain; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Drug Interactions; Haloperidol; Injections, Intraperitoneal; Ligands; Male; Mice; Nootropic Agents; Piperazines; Raclopride; Receptors, Dopamine D2; Receptors, sigma	2003
Investigation of cooperativity in the binding of ligands to the D(2) dopamine receptor. Molecular pharmacology, 2006, Volume: 69, Issue:1 Topics: Animals; Benzamides; Cell Line; Dopamine Antagonists; Ligands; Protein Binding; Raclopride; Radioligand Assay; Receptors, Dopamine D2; Spiperone	2006
[(3)H]-YM-09151-2 binding sites in human brain postmortem. Neurochemistry international, 2009, Volume: 55, Issue:7 Topics: Aged; Benzamides; Binding Sites; Brain Chemistry; Data Interpretation, Statistical; Dopamine Antagonists; Female; Hippocampus; Humans; In Vitro Techniques; Kinetics; Male; Middle Aged; Neostriatum; Postmortem Changes; Prefrontal Cortex; Propylamines; Raclopride; Receptors, Dopamine D4; Receptors, sigma; Sulpiride	2009