Page last updated: 2024-09-04

ym 09151-2 and quinpirole

ym 09151-2 has been researched along with quinpirole in 19 studies

Compound Research Comparison

Studies
(ym 09151-2)
Trials
(ym 09151-2)
Recent Studies (post-2010)
(ym 09151-2)
Studies
(quinpirole)
Trials
(quinpirole)
Recent Studies (post-2010) (quinpirole)
2496132,2130367

Protein Interaction Comparison

ProteinTaxonomyym 09151-2 (IC50)quinpirole (IC50)
D(2) dopamine receptorRattus norvegicus (Norway rat)0.1

Research

Studies (19)

TimeframeStudies, this research(%)All Research%
pre-19907 (36.84)18.7374
1990's9 (47.37)18.2507
2000's3 (15.79)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cohen, AI; Harmon, S; O'Malley, KL; Todd, RD1
Clark, D; Exner, M; Furmidge, LJ1
Carey, RM; Chevalier, RL; Felder, RA; Howell, NL; Peach, MJ; Siragy, HM1
Beaulieu, M; Felder, R; Kebabian, JW1
Fernández, M; Jantos, H; Monti, JM1
Fitten, J; Gordon, LI; Kodama, CK; Menon, MK1
Walters, JR; Weick, BG1
Brücke, T; Chiueh, CC; Cohen, RM; Kung, HF; McLellan, CA; Singhaniyom, W; Tsai, YF1
Palacios, JM; Wiederhold, KH1
Jenks, BG; Tonon, MC; Vaudry, H; Verburg-Van Kemenade, BM1
Kikuchi de Beltrán, K; Kobayashi, M; Koshikawa, N; Miwa, Y1
Farooqui, SM1
Nowak, JZ; Zawilska, JB1
Kamijo, N; Nagao, T; Ono, H1
Alberts, GL; Im, WB; Pregenzer, JF1
Badia, A; Clos, MV; García-Sanz, A; Vivas, NM1
Finlay, HE; Martin, LP; Stellar, JR; Waszczak, BL; Zahr, N1
Platt, DM; Rodefer, JS; Rowlett, JK; Spealman, RD1
Cools, AR; Fujita, S; Kiguchi, M; Koshikawa, N; Lee, J; Uchida, T; Waddington, JL1

Other Studies

19 other study(ies) available for ym 09151-2 and quinpirole

ArticleYear
Photoreceptors of mouse retinas possess D4 receptors coupled to adenylate cyclase.
    Proceedings of the National Academy of Sciences of the United States of America, 1992, Dec-15, Volume: 89, Issue:24

    Topics: Adenylyl Cyclases; Animals; Base Sequence; Benzamides; Clozapine; Cyclic AMP; Ergolines; Gene Expression; In Situ Hybridization; Mice; Mice, Inbred C57BL; Mice, Mutant Strains; Molecular Sequence Data; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Quinpirole; Receptors, Dopamine; Retina; RNA, Messenger; Spiperone

1992
Role of dopamine D1 and D2 receptors in mediating the d-amphetamine discriminative cue.
    European journal of pharmacology, 1991, Sep-17, Volume: 202, Issue:2

    Topics: Animals; Antipsychotic Agents; Benzamides; Benzazepines; Cues; Dextroamphetamine; Discrimination, Psychological; Dopamine; Dopamine Agents; Dopamine Antagonists; Dose-Response Relationship, Drug; Ergolines; Male; Motor Activity; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Reinforcement Schedule

1991
Evidence that dopamine-2 mechanisms control renal function.
    The American journal of physiology, 1990, Volume: 259, Issue:5 Pt 2

    Topics: Animals; Antipsychotic Agents; Benzamides; Dogs; Dopamine Agents; Ergolines; Female; Hemodynamics; Injections; Kidney; Nephrectomy; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Renal Circulation

1990
D-2 dopaminergic agonists and adenosine 3',5'-monophosphate directly regulate the synthesis of alpha-melanocyte-stimulating hormone-like peptides by cultured rat melanotrophs.
    Endocrinology, 1986, Volume: 118, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Benzamides; Benzazepines; Bromocriptine; Cells, Cultured; Chemical Precipitation; Cholera Toxin; Chromatography, High Pressure Liquid; Colforsin; Cyclic AMP; Dopamine; Ergolines; Immunologic Techniques; Melanocyte-Stimulating Hormones; Pituitary Gland; Pro-Opiomelanocortin; Quinpirole; Rats; Receptors, Dopamine; Spiperone

1986
Effects of the selective dopamine D-2 receptor agonist, quinpirole on sleep and wakefulness in the rat.
    European journal of pharmacology, 1989, Oct-04, Volume: 169, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Benzamides; Dopamine Agents; Electroencephalography; Ergolines; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sleep; Sleep, REM; Wakefulness

1989
Influence of D-1 receptor system on the D-2 receptor-mediated hypothermic response in mice.
    Life sciences, 1988, Volume: 43, Issue:10

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Anti-Anxiety Agents; Apomorphine; Benzamides; Benzazepines; Dopamine; Dopamine Antagonists; Ergolines; Haloperidol; Hypothermia; Male; Mice; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride

1988
Effects of D1 and D2 dopamine receptor stimulation on the activity of substantia nigra pars reticulata neurons in 6-hydroxydopamine lesioned rats: D1/D2 coactivation induces potentiated responses.
    Brain research, 1987, Mar-10, Volume: 405, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Action Potentials; Animals; Apomorphine; Benzamides; Benzazepines; Dopamine; Dopamine Antagonists; Drug Interactions; Ergolines; Hydroxydopamines; Male; Oxidopamine; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Substantia Nigra; Time Factors

1987
Blockade of in vivo binding of 125I-labeled 3-iodobenzamide (IBZM) to dopamine receptors by D2 antagonist and agonist.
    Brain research, 1988, Jun-21, Volume: 453, Issue:1-2

    Topics: Animals; Autoradiography; Benzamides; Binding, Competitive; Caudate Nucleus; Dopamine; Ergolines; Mice; Mice, Inbred C57BL; Nucleus Accumbens; Olfactory Bulb; Pyrrolidines; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Septal Nuclei

1988
Dopamine D2 receptor agents, but not dopamine D1, modify brain glucose metabolism.
    Brain research, 1985, Feb-18, Volume: 327, Issue:1-2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Benzamides; Benzazepines; Brain; Ergolines; Glucose; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2

1985
Characteristics of receptors for dopamine in the pars intermedia of the amphibian Xenopus laevis.
    Neuroendocrinology, 1986, Volume: 44, Issue:4

    Topics: Animals; Apomorphine; Benzamides; Domperidone; Dopamine; Drug Interactions; Ergolines; Haloperidol; Melanocyte-Stimulating Hormones; Pituitary Gland, Anterior; Quinpirole; Receptors, Dopamine; Sulpiride; Xenopus laevis

1986
Dorsal striatal mechanisms involved in the dopamine D2 receptor-mediated potentiation of apomorphine-induced jaw movements.
    European journal of pharmacology, 1994, Jan-24, Volume: 252, Issue:1

    Topics: Animals; Apomorphine; Benzamides; Benzazepines; Corpus Striatum; Dopamine Agents; Dopamine D2 Receptor Antagonists; Drug Synergism; Ergolines; Jaw; Male; Motor Activity; N-Methylscopolamine; Parasympatholytics; Pyrrolidines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Scopolamine Derivatives; Sulpiride

1994
Induction of adenylate cyclase sensitive dopamine D2-receptors in retinoic acid induced differentiated human neuroblastoma SHSY-5Y cells.
    Life sciences, 1994, Volume: 55, Issue:24

    Topics: Adenylyl Cyclases; Amino Acid Sequence; Base Sequence; Benzamides; Cell Differentiation; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Ergolines; Humans; Molecular Sequence Data; Neuroblastoma; Neurons; Quinpirole; Receptors, Dopamine D2; RNA, Messenger; Second Messenger Systems; Sulpiride; Tretinoin; Tumor Cells, Cultured

1994
Dopamine receptor regulating serotonin N-acetyltransferase activity in chick retina represents a D4-like subtype: pharmacological characterization.
    Neurochemistry international, 1994, Volume: 24, Issue:3

    Topics: Animals; Arylamine N-Acetyltransferase; Benzamides; Benzazepines; Chickens; Circadian Rhythm; Clozapine; Dopamine; Dopamine Antagonists; Ergolines; Ketanserin; Male; Quinpirole; Receptors, Dopamine; Retina; Spiperone; Sulpiride

1994
Depression of the monosynaptic reflex by apomorphine or bromocriptine is not mediated by D1/D2 receptors.
    Neuropharmacology, 1993, Volume: 32, Issue:8

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzamides; Bromocriptine; Decerebrate State; Depression, Chemical; Dopamine Agents; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Ergolines; Male; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Reflex, Monosynaptic; Sulpiride; Synaptic Transmission

1993
Agonist-induced [35S]GTPgammaS binding in the membranes of Spodoptera frugiperda insect cells expressing the human D3 dopamine receptor.
    Neuroscience letters, 1997, Apr-25, Volume: 226, Issue:2

    Topics: Animals; Benzamides; Cell Line; Cell Membrane; Dopamine Agonists; Dopamine Antagonists; Ethylmaleimide; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Kinetics; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Recombinant Fusion Proteins; Spodoptera; Sulfur Radioisotopes; Transfection

1997
D2 dopamine receptors and modulation of spontaneous acetylcholine (ACh) release from rat striatal synaptosomes.
    British journal of pharmacology, 1997, Volume: 122, Issue:2

    Topics: Acetylcholine; Animals; Benzamides; CHO Cells; Cricetinae; Dopamine Agonists; Humans; Male; Neostriatum; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Presynaptic; Synaptosomes; Tetrahydronaphthalenes

1997
Effects of individual and concurrent stimulation of striatal D1 and D2 dopamine receptors on electrophysiological and behavioral output from rat basal ganglia.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 300, Issue:3

    Topics: Animals; Apomorphine; Basal Ganglia; Behavior, Animal; Benzamides; Benzazepines; Dopamine Agonists; Dopamine Antagonists; Electrophysiology; Extracellular Space; Male; Membrane Potentials; Microinjections; Quinpirole; Rats; Receptors, Dopamine D1; Receptors, Dopamine D2; Substantia Nigra

2002
Suppression of cocaine- and food-maintained behavior by the D2-like receptor partial agonist terguride in squirrel monkeys.
    Psychopharmacology, 2003, Volume: 166, Issue:3

    Topics: Animals; Behavior, Animal; Benzamides; Cocaine; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Food; Injections, Intravenous; Lisuride; Male; Motor Activity; Muscle Rigidity; Quinpirole; Receptors, Dopamine D2; Reinforcement Schedule; Reward; Saimiri

2003
Topographical resolution of jaw movements mediated by cyclase- vs. non-cyclase-coupled dopamine D(1)-like receptors: studies with SK&F 83822.
    European journal of pharmacology, 2006, May-24, Volume: 538, Issue:1-3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Analysis of Variance; Animals; Benzamides; Benzazepines; Dopamine Agonists; Dopamine Antagonists; Jaw; Male; Movement; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Time Factors

2006