Compounds > ym 09151-2
Page last updated: 2024-09-04

ym 09151-2 and ketanserin

ym 09151-2 has been researched along with ketanserin in 7 studies

Compound Research Comparison

Studies
(ym 09151-2)		Trials
(ym 09151-2)		Recent Studies (post-2010)
(ym 09151-2)		Studies
(ketanserin)		Trials
(ketanserin)		Recent Studies (post-2010) (ketanserin)
2496133,094335283

Protein Interaction Comparison

ProteinTaxonomyym 09151-2 (IC50)ketanserin (IC50)
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0016
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.0021
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.015
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.015
5-hydroxytryptamine receptor 1DHomo sapiens (human)0.265
5-hydroxytryptamine receptor 1BHomo sapiens (human)6.5
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.0184
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.0027
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0016
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.29
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.015
D(2) dopamine receptorRattus norvegicus (Norway rat)1.8
Synaptic vesicular amine transporterHomo sapiens (human)0.18
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.001

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19902 (28.57)18.7374
1990's5 (71.43)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Arai, I; Higuchi, T; Kazawa, T; Mikuni, M; Takahashi, K; Yamauchi, T1
Buchman, O; Grigoriadis, DE; Niznik, HB; Pri-Bar, I; Seeman, P1
Arnt, J; Bach-Lauritsen, T; Hyttel, J1
Kido, H; Mori, H; Sakamoto, H; Shiba, K; Sumiyoshi, T; Suzuki, K; Urasaki, K; Yamaguchi, N; Yokogawa, K1
Mori, H; Sakamoto, H; Shiba, K; Sumiyoshi, T; Suzuki, K; Yamaguchi, N; Yokogawa, K1
Nowak, JZ; Zawilska, JB1
Hatanaka, K; Hidaka, K; Matsumoto, M; Noda-Saita, K; Ohmori, J; Okada, M; Yamaguchi, T1

Other Studies

7 other study(ies) available for ym 09151-2 and ketanserin

ArticleYear
Characterization of sulpiride-displaceable 3H-YM-09151-2 binding sites in rat frontal cortex and the effects of subchronic treatment with haloperidol on cortical D-2 dopamine receptors.
    Life sciences, 1990, Volume: 47, Issue:6

    Topics: Animals; Benzamides; Binding Sites; Corpus Striatum; Dopamine Antagonists; Frontal Lobe; Haloperidol; In Vitro Techniques; Ketanserin; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride

1990
Dopamine D2 receptors selectively labeled by a benzamide neuroleptic: [3H]-YM-09151-2.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 329, Issue:4

    Topics: Animals; Antipsychotic Agents; Benzamides; Binding, Competitive; Corpus Striatum; Dogs; Guanylyl Imidodiphosphate; Ketanserin; Kinetics; Piperidines; Receptors, Dopamine; Sodium; Spiperone; Substrate Specificity; Tetrahydronaphthalenes

1985
Further studies of the mechanism behind scopolamine-induced reversal of antistereotypic and cataleptogenic effects of neuroleptics in rats.
    Acta pharmacologica et toxicologica, 1986, Volume: 59, Issue:4

    Topics: Animals; Antipsychotic Agents; Behavior, Animal; Benzamides; Benzazepines; Catalepsy; Dopamine Antagonists; Droperidol; In Vitro Techniques; Ketanserin; Male; Prazosin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Scopolamine; Stereotyped Behavior

1986
In vivo dopamine-D2 and serotonin-5-HT2 receptor binding study of risperidone and haloperidol.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 47, Issue:3

    Topics: Animals; Antipsychotic Agents; Benzamides; Brain; Cerebellum; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Haloperidol; In Vitro Techniques; Isoxazoles; Ketanserin; Ligands; Male; Neostriatum; Piperidines; Prefrontal Cortex; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Serotonin; Risperidone

1994
Atypicality of several antipsychotics on the basis of in vivo dopamine-D2 and serotonin-5HT2 receptor occupancy.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1995, Volume: 12, Issue:1

    Topics: Animals; Antipsychotic Agents; Benzamides; Benzazepines; Brain; Dibenzazepines; Dopamine D2 Receptor Antagonists; Ketanserin; Male; Pimozide; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Serotonin; Serotonin Antagonists; Tranquilizing Agents

1995
Dopamine receptor regulating serotonin N-acetyltransferase activity in chick retina represents a D4-like subtype: pharmacological characterization.
    Neurochemistry international, 1994, Volume: 24, Issue:3

    Topics: Animals; Arylamine N-Acetyltransferase; Benzamides; Benzazepines; Chickens; Circadian Rhythm; Clozapine; Dopamine; Dopamine Antagonists; Ergolines; Ketanserin; Male; Quinpirole; Receptors, Dopamine; Retina; Spiperone; Sulpiride

1994
Dopamine D4-like binding sites labeled by [3H]nemonapride include substantial serotonin 5-HT2A receptors in primate cerebral cortex.
    Biochemical and biophysical research communications, 1999, Feb-16, Volume: 255, Issue:2

    Topics: Animals; Anisoles; Benzamides; Binding Sites; Cerebral Cortex; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Humans; Ketanserin; Ligands; Macaca fascicularis; Pindolol; Piperazines; Propylamines; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine D2; Receptors, Dopamine D4; Receptors, Serotonin; Sulfonamides; Tritium

1999