Page last updated: 2024-09-04

ym 09151-2 and 3-n-methylspiperone

ym 09151-2 has been researched along with 3-n-methylspiperone in 3 studies

Compound Research Comparison

Studies
(ym 09151-2)
Trials
(ym 09151-2)
Recent Studies (post-2010)
(ym 09151-2)
Studies
(3-n-methylspiperone)
Trials
(3-n-methylspiperone)
Recent Studies (post-2010) (3-n-methylspiperone)
24961315567

Protein Interaction Comparison

ProteinTaxonomyym 09151-2 (IC50)3-n-methylspiperone (IC50)
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0013
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.0013
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0013
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.0101
D(2) dopamine receptorRattus norvegicus (Norway rat)0.0002

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's1 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chen, J; Fu, D; Javitch, JA1
Endo, K; Hayakawa, N; Ishiwata, K; Oda, K; Ogi, N; Senda, M; Tanaka, A; Toyama, H1
Endo, K; Hayakawa, N; Ishiwata, K; Nagaoka, T; Oda, K; Ogi, N; Senda, M; Tanaka, A; Toyama, H; Umegaki, H1

Other Studies

3 other study(ies) available for ym 09151-2 and 3-n-methylspiperone

ArticleYear
Differentiating dopamine D2 ligands by their sensitivities to modification of the cysteine exposed in the binding-site crevice.
    Molecular pharmacology, 1996, Volume: 49, Issue:4

    Topics: Benzamides; Binding Sites; Cell Line; Cysteine; Humans; Mutagenesis, Site-Directed; Receptors, Dopamine D2; Spiperone; Structure-Activity Relationship

1996
Comparison of three PET dopamine D2-like receptor ligands, [11C]raclopride, [11C]nemonapride and [11C]N-methylspiperone, in rats.
    Annals of nuclear medicine, 1999, Volume: 13, Issue:3

    Topics: Animals; Benzamides; Brain; Cerebellum; Dopamine Agonists; Dopamine Antagonists; Ligands; Male; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D2; Salicylamides; Spiperone; Tissue Distribution; Tomography, Emission-Computed; Visual Cortex

1999
Positron emission tomography and ex vivo and in vitro autoradiography studies on dopamine D2-like receptor degeneration in the quinolinic acid-lesioned rat striatum: comparison of [11C]raclopride, [11C]nemonapride and [11C]N-methylspiperone.
    Nuclear medicine and biology, 2002, Volume: 29, Issue:3

    Topics: Animals; Autoradiography; Benzamides; Dopamine Antagonists; Glucose; Magnetic Resonance Imaging; Male; Neostriatum; Neurotoxins; Quinolinic Acid; Raclopride; Radiopharmaceuticals; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, GABA-A; Spiperone; Tomography, Emission-Computed

2002