Page last updated: 2024-09-03

ym 022 and histamine

ym 022 has been researched along with histamine in 14 studies

Compound Research Comparison

Studies
(ym 022)
Trials
(ym 022)
Recent Studies (post-2010)
(ym 022)
Studies
(histamine)
Trials
(histamine)
Recent Studies (post-2010) (histamine)
651837,7181,3723,457

Protein Interaction Comparison

ProteinTaxonomyym 022 (IC50)histamine (IC50)
Histamine H1 receptorRattus norvegicus (Norway rat)0.1585
Histamine H1 receptorHomo sapiens (human)0.1585

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's10 (71.43)18.2507
2000's4 (28.57)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Akuzawa, S; Ito, H; Kamato, T; Kobayashi-Uchida, A; Nagakura, Y; Nishida, A; Shishido, T; Takinami, Y; Yamano, M; Yuki, H1
Akuzawa, S; Ito, H; Kamato, T; Katuyama, Y; Kobayashi, A; Miyata, K; Nishida, A; Tsutsumi, R; Yamano, M; Yuki, H1
Akuzawa, S; Miyata, K; Nishida, A; Takemoto, Y; Uchida-Kobayashi, A1
Ding, XQ; Håkanson, R1
Akuzawa, S; Ito, H; Miyake, A; Miyata, K; Nishida, A; Takemoto, Y; Takinami, Y; Yuki, H1
Ding, XQ; Håkanson, R; Lindström, E2
Ding, XQ; Håkanson, R; Kitano, M1
Ding, XQ; Håkanson, R; Kitano, M; Lindström, E; Norlén, P1
Ding, XQ; Håkanson, R; Lindström, E; Norlén, P1
Björkqvist, M; Chen, D; Ding, XQ; Håkanson, R; Kitano, M; Norlén, P; Zhao, CM1
Håkanson, R; Kitano, M; Norlén, P1
Aihara, T; Chen, D; Fujishita, T; Furutani, K; Kanatani, K; Matsui, M; Nakamura, E; Okabe, S; Taketo, MM1
Imatake, K; Matsui, T; Moriyama, M1

Reviews

1 review(s) available for ym 022 and histamine

ArticleYear
CCK2 receptor antagonists: pharmacological tools to study the gastrin-ECL cell-parietal cell axis.
    Regulatory peptides, 1999, Mar-17, Volume: 80, Issue:1-2

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Chromogranin A; Gastric Acid; Gastric Mucosa; Gastrins; Histamine; Histidine Decarboxylase; Hormone Antagonists; Humans; Indoles; Pancreatic Hormones; Parietal Cells, Gastric; Phenylurea Compounds; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Stomach

1999

Other Studies

13 other study(ies) available for ym 022 and histamine

ArticleYear
Gastrin receptor antagonist YM022 prevents hypersecretion after long-term acid suppression.
    The American journal of physiology, 1995, Volume: 269, Issue:5 Pt 1

    Topics: Animals; Benzodiazepines; Cell Count; Enterochromaffin Cells; Famotidine; Female; Gastric Acid; Gastric Mucosa; Gastrins; Histamine; Histidine Decarboxylase; Omeprazole; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Time Factors

1995
Pharmacological profile of (R)-1-[2,3-dihydro-1-(2'-methylphenacyl)-2-oxo- 5-phenyl-1H-1,4-benzodiazepin-3-yl]-3-(3-methylphenyl)urea (YM022), a new potent and selective gastrin/cholecystokinin-B receptor antagonist, in vitro and in vivo.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 269, Issue:2

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Bethanechol; Bethanechol Compounds; Gastric Acid; Gastric Mucosa; Histamine; In Vitro Techniques; Indoles; Male; Meglumine; Pentagastrin; Phenylurea Compounds; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Sincalide

1994
Comparative evaluation of the role of endogenous gastrin in basal acid secretion in conscious rats provided with chronic fistula and pylorus ligation.
    Japanese journal of pharmacology, 1996, Volume: 71, Issue:3

    Topics: Animals; Atropine; Benzodiazepines; Chronic Disease; Famotidine; Gastric Acid; Gastric Fistula; Gastrins; Histamine; Ligation; Male; Parasympathetic Nervous System; Pylorus; Rats; Rats, Sprague-Dawley

1996
Effect of cholecystokinin-B/gastrin receptor blockade on gastric acid secretion in conscious rats.
    Pharmacology & toxicology, 1996, Volume: 79, Issue:6

    Topics: Animals; Anti-Ulcer Agents; Benzodiazepines; Dose-Response Relationship, Drug; Gastric Acid; Gastric Mucosa; Gastrins; Histamine; Hormone Antagonists; Male; Phenylurea Compounds; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Vagus Nerve

1996
YM022, a potent and selective gastrin/CCK-B receptor antagonist, inhibits peptone meal-induced gastric acid secretion in Heidenhain pouch dogs.
    Digestive diseases and sciences, 1997, Volume: 42, Issue:4

    Topics: Animals; Atropine; Benzodiazepines; Benzodiazepinones; Devazepide; Dogs; Dose-Response Relationship, Drug; Eating; Famotidine; Gastric Acid; Histamine; Histamine H2 Antagonists; Hormone Antagonists; Male; Methacholine Chloride; Muscarinic Antagonists; Pentagastrin; Peptones; Phenylurea Compounds; Receptors, Cholecystokinin; Sincalide; Stomach

1997
Cholecystokinin-B/gastrin receptor blockade suppresses the activity of rat stomach ECL cells.
    Pharmacology & toxicology, 1997, Volume: 81, Issue:1

    Topics: Animals; Anti-Ulcer Agents; Benzodiazepines; Chromogranin A; Chromogranins; Enterochromaffin Cells; Gastric Mucosa; Gastrins; Histamine; Histidine Decarboxylase; Hormone Antagonists; Male; Omeprazole; Pancreatic Hormones; Phenylurea Compounds; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; RNA, Messenger; RNA, Ribosomal, 18S; Stomach

1997
Time-course of deactivation of rat stomach ECL cells following cholecystokinin B/gastrin receptor blockade.
    British journal of pharmacology, 1997, Volume: 122, Issue:1

    Topics: Animals; Anti-Ulcer Agents; Benzodiazepines; Body Weight; Chromogranin A; Enterochromaffin Cells; Gastric Mucosa; Gastrins; Histamine; Hormone Antagonists; Male; Pancreatic Hormones; Phenylurea Compounds; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; RNA, Messenger; Stomach; Time Factors

1997
Sustained cholecystokinin-B/gastrin receptor blockade does not impair basal or histamine-stimulated acid secretion in chronic gastric fistula rats.
    Pharmacology & toxicology, 1998, Volume: 82, Issue:4

    Topics: Animals; Benzodiazepines; Cholecystokinin; Gastric Acid; Gastric Fistula; Gastrins; Histamine; Hormone Antagonists; Male; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin

1998
Reversibility of cholecystokinin-B/gastrin receptor blockade: a study of the gastrin-ECL cell axis in the rat.
    Pharmacology & toxicology, 1999, Volume: 84, Issue:4

    Topics: Animals; Benzodiazepines; Chromogranin A; Chromogranins; Gastric Mucosa; Gastrins; Histamine; Histidine Decarboxylase; Male; Pancreatic Hormones; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; RNA, Messenger

1999
Effect of cholecystokinin-2 receptor blockade on rat stomach ECL cells. A histochemical, electron-microscopic and chemical study.
    Cell and tissue research, 2000, Volume: 299, Issue:1

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Chromogranin A; Cytoplasmic Granules; Gastrins; Histamine; Histidine Decarboxylase; Hormone Antagonists; Immunohistochemistry; Male; Microscopy, Electron; Omeprazole; Pancreatic Hormones; Parietal Cells, Gastric; Phenylurea Compounds; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Time Factors

2000
Gastric submucosal microdialysis: a method to study gastrin- and food-evoked mobilization of ECL-cell histamine in conscious rats.
    Regulatory peptides, 2000, Jan-29, Volume: 86, Issue:1-3

    Topics: Animals; Benzodiazepines; Chromogranin A; Enterochromaffin-like Cells; Enzyme Inhibitors; Fluorescent Antibody Technique; Food; Gastric Mucosa; Gastrins; Histamine; Hormone Antagonists; Male; Methylhistidines; Microdialysis; Pancreatic Hormones; Rats; Rats, Sprague-Dawley; Time Factors; Vagotomy, Proximal Gastric

2000
Impaired gastric secretion and lack of trophic responses to hypergastrinemia in M3 muscarinic receptor knockout mice.
    Gastroenterology, 2003, Volume: 125, Issue:6

    Topics: Animals; Benzodiazepines; Calcium; Cell Division; Enterochromaffin Cells; Female; Gastric Acid; Gastric Mucosa; Gastrins; Histamine; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Receptor, Muscarinic M3

2003
The effect and mechanism of action of capsaicin on gastric acid output.
    Journal of gastroenterology, 2009, Volume: 44, Issue:5

    Topics: Animals; Benzodiazepines; Bethanechol; Calcitonin Gene-Related Peptide; Capsaicin; Dose-Response Relationship, Drug; Famotidine; Gastric Acid; Gastrins; Histamine; Histamine H2 Antagonists; Hormone Antagonists; In Vitro Techniques; Male; Muscarinic Agonists; Rats; Rats, Wistar; Somatostatin; Stomach; Vagus Nerve

2009