Page last updated: 2024-09-03

y 27632 and ucn 1028 c

y 27632 has been researched along with ucn 1028 c in 8 studies

Compound Research Comparison

Studies
(y 27632)
Trials
(y 27632)
Recent Studies (post-2010)
(y 27632)
Studies
(ucn 1028 c)
Trials
(ucn 1028 c)
Recent Studies (post-2010) (ucn 1028 c)
1,9243891984260

Protein Interaction Comparison

ProteinTaxonomyy 27632 (IC50)ucn 1028 c (IC50)
Dipeptidyl peptidase 4Rattus norvegicus (Norway rat)1.1
Catenin beta-1Homo sapiens (human)10
Tyrosine-protein kinase SYKHomo sapiens (human)1.1

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (62.50)29.6817
2010's3 (37.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Doi, M; Kawasaki, S; Kimura, S; Koji, T; Nishikawa, Y; Ogawa, A; Sasaki, K; Watanabe, M1
Bitar, KN; Patil, SB1
Koide, M; Nakayama, K; Obara, K; Uchino, M; Yamanaka, A1
Ahn, DS; Cho, YE; Choi, SK; Kim, YH; Lee, YH; Morgan, KG; Ryu, SK1
Ding, H; Huang, J; Isotani, E; Kamm, KE; Mizuno, Y; Stull, JT1
Heaps, CL; Parker, JL; Robles, JC; Sturek, M1
Maxwell, PJ; Rattan, S; Singh, J1
Rattan, S; Singh, J1

Other Studies

8 other study(ies) available for y 27632 and ucn 1028 c

ArticleYear
The role of rho and rho-dependent kinase in serotonin-induced contraction observed in bovine middle cerebral artery.
    The Tohoku journal of experimental medicine, 2003, Volume: 201, Issue:4

    Topics: ADP Ribose Transferases; Amides; Animals; Azepines; Bacterial Proteins; Bacterial Toxins; Botulinum Toxins; Brain; Calcium-Calmodulin-Dependent Protein Kinases; Cattle; Cerebral Arteries; Cytotoxins; Dose-Response Relationship, Drug; Enterotoxins; Enzyme Inhibitors; Indoles; Intracellular Signaling Peptides and Proteins; Middle Cerebral Artery; Myosin-Light-Chain Kinase; Naphthalenes; Potassium; Protein Kinase C; Protein Serine-Threonine Kinases; Pyridines; rho GTP-Binding Proteins; rho-Associated Kinases; Serotonin; Sulfonamides; Time Factors

2003
RhoA- and PKC-alpha-mediated phosphorylation of MYPT and its association with HSP27 in colonic smooth muscle cells.
    American journal of physiology. Gastrointestinal and liver physiology, 2006, Volume: 290, Issue:1

    Topics: Acetylcholine; Amides; Animals; Cells, Cultured; Colon; Enzyme Activation; Enzyme Inhibitors; Gene Expression Regulation; Heat-Shock Proteins; Intracellular Signaling Peptides and Proteins; Muscle, Smooth; Myosin Light Chains; Myosin-Light-Chain Phosphatase; Naphthalenes; Phosphorylation; Protein Kinase C-alpha; Protein Serine-Threonine Kinases; Protein Transport; Pyridines; Rabbits; rho-Associated Kinases; rhoA GTP-Binding Protein; Signal Transduction

2006
Stretch-induced triphosphorylation of myosin light chain and myogenic tone in canine basilar artery.
    European journal of pharmacology, 2006, Mar-18, Volume: 534, Issue:1-3

    Topics: Amides; Animals; Azepines; Basilar Artery; Calcium; Calcium Channel Blockers; Dogs; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Muscle Contraction; Muscle, Smooth, Vascular; Myosin Light Chains; Myosin-Light-Chain Kinase; Naphthalenes; Nicardipine; Phosphorylation; Protein Kinase C; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Pyridines; Reflex, Stretch; rho-Associated Kinases; Time Factors

2006
Augmented sphingosylphosphorylcholine-induced Ca2+-sensitization of mesenteric artery contraction in spontaneously hypertensive rat.
    Naunyn-Schmiedeberg's archives of pharmacology, 2006, Volume: 373, Issue:1

    Topics: Amides; Animals; Calcium; Flavonoids; Hypertension; Mesenteric Arteries; Mitogen-Activated Protein Kinases; Myosin Light Chains; Naphthalenes; Phosphorylation; Phosphorylcholine; Protein Kinase C; Pyridines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; rho-Associated Kinases; Sphingosine; Vasoconstriction

2006
Myosin light chain kinase activation and calcium sensitization in smooth muscle in vivo.
    American journal of physiology. Cell physiology, 2008, Volume: 295, Issue:2

    Topics: Amides; Animals; Calcium; Calcium Signaling; Calmodulin; Carbachol; Intracellular Signaling Peptides and Proteins; Isometric Contraction; Mice; Mice, Transgenic; Muscle Contraction; Muscle Proteins; Muscle, Smooth; Myosin Light Chains; Myosin-Light-Chain Kinase; Myosin-Light-Chain Phosphatase; Naphthalenes; Phosphoproteins; Phosphorylation; Potassium Chloride; Protein Kinase C; Protein Kinase Inhibitors; Pyridines; rho-Associated Kinases; Urinary Bladder

2008
Ca2+ sensitization and PKC contribute to exercise training-enhanced contractility in porcine collateral-dependent coronary arteries.
    American journal of physiology. Heart and circulatory physiology, 2011, Volume: 300, Issue:4

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amides; Animals; Calcium; Collateral Circulation; Coronary Vessels; Endothelin-1; Enzyme Inhibitors; Female; Muscle Contraction; Naphthalenes; Phorbol 12,13-Dibutyrate; Physical Conditioning, Animal; Protein Kinase C; Pyridines; rho-Associated Kinases; Swine; Vasodilator Agents

2011
Immunocytochemical evidence for PDBu-induced activation of RhoA/ROCK in human internal anal sphincter smooth muscle cells.
    American journal of physiology. Gastrointestinal and liver physiology, 2011, Volume: 301, Issue:2

    Topics: ADP Ribose Transferases; Amides; Anal Canal; Botulinum Toxins; Cells, Cultured; Fluorescent Antibody Technique; Humans; Muscle Contraction; Myocytes, Smooth Muscle; Myosin-Light-Chain Phosphatase; Naphthalenes; Phorbol 12,13-Dibutyrate; Protein Kinase C-alpha; Pyridines; rho-Associated Kinases; rhoA GTP-Binding Protein; Signal Transduction

2011
Role of PKC and RhoA/ROCK pathways in the spontaneous phasic activity in the rectal smooth muscle.
    American journal of physiology. Gastrointestinal and liver physiology, 2013, Apr-15, Volume: 304, Issue:8

    Topics: Amides; Animals; Carcinogens; Enzyme Inhibitors; Fecal Incontinence; Indoles; Maleimides; Muscle Contraction; Muscle, Smooth; Naphthalenes; Phorbol 12,13-Dibutyrate; Phosphorylation; Protein Kinase C; Pyridines; Rats; Rats, Sprague-Dawley; Rectum; rho-Associated Kinases; rhoA GTP-Binding Protein; Signal Transduction

2013