Page last updated: 2024-09-03

y 27632 and tetrodotoxin

y 27632 has been researched along with tetrodotoxin in 7 studies

Compound Research Comparison

Studies
(y 27632)
Trials
(y 27632)
Recent Studies (post-2010)
(y 27632)
Studies
(tetrodotoxin)
Trials
(tetrodotoxin)
Recent Studies (post-2010) (tetrodotoxin)
1,924389112,992111,477

Protein Interaction Comparison

ProteinTaxonomyy 27632 (IC50)tetrodotoxin (IC50)
Sodium channel protein type 9 subunit alphaHomo sapiens (human)0.0186

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's7 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Aoki, K; Kuzumaki, N; Narita, M; Suzuki, T; Takagi, M1
Büyükafsar, K; Levent, A1
Andersson, KE; Arner, A; Ekman, M1
De Godoy, MA; Patel, CA; Rattan, S1
Honda, M; Ishikawa, T; Nakayama, K; Suzuki, M1
Endo, M; Hatanaka, Y; Hirai, S; Ohnami, S; Uesaka, N; Yamamoto, N; Yamashita, T1
Dhaese, I; Lefebvre, RA1

Other Studies

7 other study(ies) available for y 27632 and tetrodotoxin

ArticleYear
Implication of Rho-associated kinase in the elevation of extracellular dopamine levels and its related behaviors induced by methamphetamine in rats.
    Journal of neurochemistry, 2003, Volume: 86, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Amides; Animals; Behavior, Animal; Central Nervous System Stimulants; Dopamine; Dopamine Uptake Inhibitors; Drug Administration Routes; Enzyme Inhibitors; Extracellular Space; Homovanillic Acid; Intracellular Signaling Peptides and Proteins; Male; Methamphetamine; Microdialysis; Morphine; Narcotics; Nucleus Accumbens; Protein Serine-Threonine Kinases; Pyridines; Rats; Rats, Sprague-Dawley; rho-Associated Kinases; Signal Transduction; Tetrodotoxin

2003
Expression of Rho-kinase (ROCK-1 and ROCK-2) and its substantial role in the contractile activity of the sheep ureter.
    British journal of pharmacology, 2004, Volume: 143, Issue:3

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amides; Animals; Aorta; Atropine; Blotting, Western; Calcium Channel Blockers; Carbachol; Dose-Response Relationship, Drug; Electric Stimulation; Enzyme Inhibitors; Guanethidine; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Muscle Contraction; Muscle, Smooth; Nitric Oxide Synthase; Nitroarginine; Phenylephrine; Potassium Chloride; Protein Serine-Threonine Kinases; Pyridines; rho-Associated Kinases; Sheep; Tetrodotoxin; Ureter; Vasoconstrictor Agents; Vasodilator Agents

2004
Developmental regulation of nerve and receptor mediated contractions of mammalian urinary bladder smooth muscle.
    European journal of pharmacology, 2006, Feb-17, Volume: 532, Issue:1-2

    Topics: Adenosine Triphosphate; Age Factors; Amides; Animals; Animals, Newborn; Carbachol; Cholinergic Agonists; Cholinergic Fibers; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Electric Stimulation; Female; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Muscarinic Antagonists; Muscle Contraction; Muscle Relaxants, Central; Muscle, Smooth; Nifedipine; Pyridines; Receptors, Muscarinic; Scopolamine; Tetrodotoxin; Urinary Bladder; Vasodilator Agents

2006
Rho kinase as a novel molecular therapeutic target for hypertensive internal anal sphincter.
    Gastroenterology, 2006, Volume: 131, Issue:1

    Topics: Amides; Anal Canal; Animals; Disease Models, Animal; Enzyme Inhibitors; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Muscle Hypertonia; Muscle Relaxation; Muscle, Smooth; Protein Serine-Threonine Kinases; Pyridines; Rats; Rats, Sprague-Dawley; rho-Associated Kinases; Tetrodotoxin; Treatment Outcome

2006
Role of alpha2C-adrenoceptors in the reduction of skin blood flow induced by local cooling in mice.
    British journal of pharmacology, 2007, Volume: 152, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adrenalectomy; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Amides; Anesthetics, Local; Animals; Blood Pressure; Blood Vessels; Body Temperature Regulation; Clonidine; Cold Temperature; Heart Rate; Intracellular Signaling Peptides and Proteins; Isoquinolines; Laser-Doppler Flowmetry; Male; Mice; Naphthyridines; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Pyridines; Quinolizines; Receptors, Adrenergic, alpha-2; Reflex; Regional Blood Flow; rho-Associated Kinases; Skin; Skin Temperature; Sympathetic Nervous System; Tetrodotoxin; Vasoconstriction

2007
Role of RhoA in activity-dependent cortical axon branching.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2008, Sep-10, Volume: 28, Issue:37

    Topics: Amides; Animals; Animals, Newborn; Axons; Bacterial Proteins; Electroporation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Gene Expression Regulation; Humans; Luminescent Proteins; Lysophospholipids; Microscopy, Confocal; Neurons; Occipital Lobe; Organ Culture Techniques; Pyridines; Rats; Rats, Sprague-Dawley; rhoA GTP-Binding Protein; Signal Transduction; Sodium Channel Blockers; Tetrodotoxin

2008
Myosin light chain phosphatase activation is involved in the hydrogen sulfide-induced relaxation in mouse gastric fundus.
    European journal of pharmacology, 2009, Mar-15, Volume: 606, Issue:1-3

    Topics: Adenine; Amides; Animals; Enzyme Activation; Gastric Fundus; Glyburide; Hydrogen Sulfide; In Vitro Techniques; Male; Marine Toxins; Mice; Muscle Relaxation; Myosin-Light-Chain Phosphatase; NG-Nitroarginine Methyl Ester; omega-Conotoxins; Oxazoles; Pyridines; rho-Associated Kinases; rhoA GTP-Binding Protein; Signal Transduction; Tetrodotoxin

2009