Page last updated: 2024-09-03

y 27632 and staurosporine aglycone

y 27632 has been researched along with staurosporine aglycone in 4 studies

Compound Research Comparison

Studies
(y 27632)
Trials
(y 27632)
Recent Studies (post-2010)
(y 27632)
Studies
(staurosporine aglycone)
Trials
(staurosporine aglycone)
Recent Studies (post-2010) (staurosporine aglycone)
1,92438917390175

Protein Interaction Comparison

ProteinTaxonomyy 27632 (IC50)staurosporine aglycone (IC50)
B2 bradykinin receptorCavia porcellus (domestic guinea pig)8
Serine/threonine-protein kinase D3Homo sapiens (human)2.45
cAMP-dependent protein kinase catalytic subunit alphaBos taurus (cattle)0.83
Beta-lactamaseEscherichia coli K-128
Protein kinase C gamma typeHomo sapiens (human)2.45
Protein kinase C beta typeHomo sapiens (human)2.45
Zinc finger protein GLI1Homo sapiens (human)1.8
Zinc finger protein GLI2Homo sapiens (human)2.7
Malate dehydrogenaseThermus thermophilus8
Cyclin-dependent kinase 4Homo sapiens (human)0.83
Protein kinase C alpha typeHomo sapiens (human)2.45
Chymotrypsinogen BHomo sapiens (human)10
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)8
G1/S-specific cyclin-D1Homo sapiens (human)0.83
Protein kinase C eta typeHomo sapiens (human)2.45
G1/S-specific cyclin-E1Homo sapiens (human)0.83
Cyclin-dependent kinase 2Homo sapiens (human)0.83
Protein kinase C iota typeHomo sapiens (human)2.45
Tyrosine-protein kinase JAK3Homo sapiens (human)0.061
Mitogen-activated protein kinase kinase kinase 9Homo sapiens (human)0.1083
Protein kinase C epsilon typeHomo sapiens (human)2.45
Mitogen-activated protein kinase kinase kinase 10Homo sapiens (human)0.0935
Protein kinase C theta typeHomo sapiens (human)2.45
Protein kinase C zeta typeHomo sapiens (human)2.45
Protein kinase C delta typeHomo sapiens (human)2.45
Calcium/calmodulin-dependent protein kinase type II subunit betaHomo sapiens (human)0.184
Calcium/calmodulin-dependent protein kinase type II subunit gammaHomo sapiens (human)0.184
Calcium/calmodulin-dependent protein kinase type II subunit deltaHomo sapiens (human)0.184
Serine/threonine-protein kinase D1Homo sapiens (human)2.45
Mitogen-activated protein kinase kinase kinase 11Homo sapiens (human)0.0787
Calcium/calmodulin-dependent protein kinase type II subunit alphaHomo sapiens (human)0.184

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (75.00)29.6817
2010's1 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Caivano, M; Cohen, P; Davies, SP; Reddy, H1
McGovern, SL; Shoichet, BK1
Doran, JD; Futer, O; Pazhanisamy, S; Raybuck, SA; Saadat, AR1
Kramer, B; Löwenheim, H; Müller, M; Tropitzsch, A1

Other Studies

4 other study(ies) available for y 27632 and staurosporine aglycone

ArticleYear
Specificity and mechanism of action of some commonly used protein kinase inhibitors.
    The Biochemical journal, 2000, Oct-01, Volume: 351, Issue:Pt 1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Alkaloids; Amides; Animals; Benzamides; Benzophenanthridines; Benzopyrans; Butadienes; Cell Line; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; Indoles; Inhibitory Concentration 50; Isoquinolines; Lithium; Magnesium; Nitriles; Phenanthridines; Phosphorylation; Potassium Chloride; Protein Kinase Inhibitors; Protein Kinases; Pyridines; Sirolimus; Substrate Specificity; Sulfonamides

2000
Kinase inhibitors: not just for kinases anymore.
    Journal of medicinal chemistry, 2003, Apr-10, Volume: 46, Issue:8

    Topics: beta-Lactamase Inhibitors; beta-Lactamases; Chymotrypsin; Enzyme Inhibitors; Kinetics; Light; Malate Dehydrogenase; Models, Biological; Phosphotransferases; Scattering, Radiation

2003
Phosphoryl transfer is not rate-limiting for the ROCK I-catalyzed kinase reaction.
    Biochemistry, 2006, Jun-27, Volume: 45, Issue:25

    Topics: Adenosine Triphosphatases; Amides; Carbazoles; Humans; Indole Alkaloids; Intracellular Signaling Peptides and Proteins; Kinetics; Phosphorylation; Protein Conformation; Protein Serine-Threonine Kinases; Pyridines; rho-Associated Kinases; Solvents; Substrate Specificity; Viscosity

2006
Myelin-induced inhibition in a spiral ganglion organ culture - Approaching a natural environment in vitro.
    Neuroscience, 2017, 08-15, Volume: 357

    Topics: Amides; Animals; Brain-Derived Neurotrophic Factor; Carbazoles; Flavones; Indole Alkaloids; Mice; Myelin Proteins; Myelin Sheath; Nerve Growth Factors; Neuronal Outgrowth; Protein Kinase Inhibitors; Pyridines; Receptor, trkB; Receptors, Nerve Growth Factor; rho-Associated Kinases; Spiral Ganglion; Tissue Culture Techniques

2017