Page last updated: 2024-09-03

y 27632 and ruboxistaurin

y 27632 has been researched along with ruboxistaurin in 2 studies

Compound Research Comparison

Studies
(y 27632)
Trials
(y 27632)
Recent Studies (post-2010)
(y 27632)
Studies
(ruboxistaurin)
Trials
(ruboxistaurin)
Recent Studies (post-2010) (ruboxistaurin)
1,92438912032956

Protein Interaction Comparison

ProteinTaxonomyy 27632 (IC50)ruboxistaurin (IC50)
3-phosphoinositide-dependent protein kinase 1Homo sapiens (human)0.6484
Protein kinase C gamma typeHomo sapiens (human)0.3
Protein kinase C alpha typeRattus norvegicus (Norway rat)0.32
Protein kinase C beta typeHomo sapiens (human)0.0054
Protein kinase C delta typeRattus norvegicus (Norway rat)0.32
Protein kinase C epsilon typeRattus norvegicus (Norway rat)0.32
Protein kinase C zeta typeRattus norvegicus (Norway rat)0.32
Serine/threonine-protein kinase pim-1Homo sapiens (human)0.2
Protein kinase C alpha typeHomo sapiens (human)0.36
Protein kinase C eta typeHomo sapiens (human)0.052
Protein kinase C gamma typeRattus norvegicus (Norway rat)0.32
Protein kinase C beta typeRattus norvegicus (Norway rat)0.32
Protein kinase C epsilon typeHomo sapiens (human)0.6
Protein kinase C delta typeHomo sapiens (human)0.25
Protein kinase C eta typeRattus norvegicus (Norway rat)0.32
Homeodomain-interacting protein kinase 1Homo sapiens (human)0.1
Homeodomain-interacting protein kinase 4Homo sapiens (human)0.1
Homeodomain-interacting protein kinase 2Homo sapiens (human)0.1
Homeodomain-interacting protein kinase 3Homo sapiens (human)0.1
Protein kinase C theta typeRattus norvegicus (Norway rat)0.32

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Alessi, DR; Arthur, JS; Bain, J; Cohen, P; Elliott, M; Hastie, CJ; Klevernic, I; McLauchlan, H; Plater, L; Shpiro, N1
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M1

Other Studies

2 other study(ies) available for y 27632 and ruboxistaurin

ArticleYear
The selectivity of protein kinase inhibitors: a further update.
    The Biochemical journal, 2007, Dec-15, Volume: 408, Issue:3

    Topics: Amino Acid Sequence; Animals; Cell Line; Drug Design; Enzyme Activation; Humans; Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Recombinant Proteins; Spodoptera

2007
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
    Proceedings of the National Academy of Sciences of the United States of America, 2007, Dec-18, Volume: 104, Issue:51

    Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases

2007