Page last updated: 2024-09-03

y 27632 and rottlerin

y 27632 has been researched along with rottlerin in 6 studies

Compound Research Comparison

Studies
(y 27632)
Trials
(y 27632)
Recent Studies (post-2010)
(y 27632)
Studies
(rottlerin)
Trials
(rottlerin)
Recent Studies (post-2010) (rottlerin)
1,92438915561202

Protein Interaction Comparison

ProteinTaxonomyy 27632 (IC50)rottlerin (IC50)
Eukaryotic elongation factor 2 kinaseHomo sapiens (human)5.3
B2 bradykinin receptorCavia porcellus (domestic guinea pig)1.2
Ubiquitin carboxyl-terminal hydrolase 1Homo sapiens (human)8
Beta-lactamaseEscherichia coli K-121.5
Malate dehydrogenaseThermus thermophilus0.7
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)1.2
MAP kinase-activated protein kinase 2Homo sapiens (human)5.4
Protein kinase C delta typeHomo sapiens (human)3
MAP kinase-activated protein kinase 5Homo sapiens (human)1.9
WD repeat-containing protein 48Homo sapiens (human)8
RuvB-like 1Homo sapiens (human)10

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (66.67)29.6817
2010's2 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Caivano, M; Cohen, P; Davies, SP; Reddy, H1
McGovern, SL; Shoichet, BK1
Alessi, DR; Arthur, JS; Bain, J; Cohen, P; Elliott, M; Hastie, CJ; Klevernic, I; McLauchlan, H; Plater, L; Shpiro, N1
Gimona, M; Hahne, P; Hai, CM; Harrington, EO1
Ishimaru, Y; Narahara, S; Sakamoto, A; Sugiuchi, H; Yamaguchi, R; Yamaguchi, Y; Yamamoto, T1
Kim, BJ; Kim, JN1

Other Studies

6 other study(ies) available for y 27632 and rottlerin

ArticleYear
Specificity and mechanism of action of some commonly used protein kinase inhibitors.
    The Biochemical journal, 2000, Oct-01, Volume: 351, Issue:Pt 1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Alkaloids; Amides; Animals; Benzamides; Benzophenanthridines; Benzopyrans; Butadienes; Cell Line; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; Indoles; Inhibitory Concentration 50; Isoquinolines; Lithium; Magnesium; Nitriles; Phenanthridines; Phosphorylation; Potassium Chloride; Protein Kinase Inhibitors; Protein Kinases; Pyridines; Sirolimus; Substrate Specificity; Sulfonamides

2000
Kinase inhibitors: not just for kinases anymore.
    Journal of medicinal chemistry, 2003, Apr-10, Volume: 46, Issue:8

    Topics: beta-Lactamase Inhibitors; beta-Lactamases; Chymotrypsin; Enzyme Inhibitors; Kinetics; Light; Malate Dehydrogenase; Models, Biological; Phosphotransferases; Scattering, Radiation

2003
The selectivity of protein kinase inhibitors: a further update.
    The Biochemical journal, 2007, Dec-15, Volume: 408, Issue:3

    Topics: Amino Acid Sequence; Animals; Cell Line; Drug Design; Enzyme Activation; Humans; Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Recombinant Proteins; Spodoptera

2007
Conventional protein kinase C mediates phorbol-dibutyrate-induced cytoskeletal remodeling in a7r5 smooth muscle cells.
    Experimental cell research, 2002, Oct-15, Volume: 280, Issue:1

    Topics: Acetophenones; Actinin; Actins; Amides; Animals; Benzopyrans; Carbazoles; Cells, Cultured; Cytoskeleton; Enzyme Inhibitors; Green Fluorescent Proteins; Indoles; Isoenzymes; Luminescent Proteins; Muscle, Smooth, Vascular; Phorbol 12,13-Dibutyrate; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-delta; Protein Transport; Pyridines; Rats; Recombinant Fusion Proteins; Transfection; Vinculin

2002
Substance P enhances tissue factor release from granulocyte-macrophage colony-stimulating factor-dependent macrophages via the p22phox/β-arrestin 2/Rho A signaling pathway.
    Blood cells, molecules & diseases, 2016, Volume: 57

    Topics: Acetophenones; Adipocytes; Amides; Aprepitant; Arrestins; Benzopyrans; beta-Arrestin 2; beta-Arrestins; Dynamins; Free Radical Scavengers; Gene Expression Regulation; Granulocyte-Macrophage Colony-Stimulating Factor; Humans; Macrophage Activation; Macrophages; Morpholines; NADPH Oxidases; Neurokinin-1 Receptor Antagonists; Phosphorylcholine; Primary Cell Culture; Protein Kinase Inhibitors; Pyridines; Pyrrolidines; rho-Associated Kinases; RNA, Small Interfering; Signal Transduction; Substance P; Thiocarbamates; Thromboplastin

2016
The Mechanism of Action of Ghrelin and Motilin in the Pacemaker Potentials of Interstitial Cells of Cajal from the Murine Small Intestine.
    Molecules and cells, 2019, Jun-30, Volume: 42, Issue:6

    Topics: Acetophenones; Amides; Animals; Benzopyrans; Boron Compounds; Calcium; Carbazoles; Gastrointestinal Motility; Ghrelin; Inositol 1,4,5-Trisphosphate Receptors; Interstitial Cells of Cajal; Intestine, Small; Macrocyclic Compounds; Membrane Potentials; Mice; Mice, Inbred ICR; Motilin; Oligopeptides; Oxazoles; Protein Kinase C; Pyridines; Receptors, Ghrelin; rho-Associated Kinases; Signal Transduction; Staurosporine; Thapsigargin

2019