Page last updated: 2024-09-03

y 27632 and methacholine chloride

y 27632 has been researched along with methacholine chloride in 10 studies

Compound Research Comparison

Studies
(y 27632)
Trials
(y 27632)
Recent Studies (post-2010)
(y 27632)
Studies
(methacholine chloride)
Trials
(methacholine chloride)
Recent Studies (post-2010) (methacholine chloride)
1,92438915,443835824

Protein Interaction Comparison

ProteinTaxonomyy 27632 (IC50)methacholine chloride (IC50)
galanin receptor type 3Homo sapiens (human)7.365

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's10 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ishii, K; Moriuchi, H; Nakahara, T; Sakamato, K; Yunoki, M1
Hayashi, H; Honjo, H; Ito, S; Katoh, H; Kodama, I; Kume, H; Yamaki, K2
Ito, S; Ito, Y; Kume, H; Yamaki, K1
Boterman, M; de Jong, AM; Hovens, I; Meurs, H; Nelemans, SA; Penninks, JM; Schaafsma, D; Zaagsma, J1
Honjo, H; Ito, S; Kamiya, K; Kodama, I; Kume, H; Oguma, T; Shimokata, K; Takeda, N1
Meurs, H; Nelemans, SA; Schaafsma, D; Zaagsma, J; Zuidhof, AB1
Ito, S; Ito, Y; Kondo, M; Kume, H; Naruse, K; Oguma, T; Shimokata, K; Suki, B1
Ito, S; Ito, Y; Kojima, K; Kondo, M; Kume, H; Oguma, T; Shimokata, K; Shiraki, A1
Honjo, H; Ito, S; Kamiya, K; Kondo, M; Kume, H; Makino, Y; Oguma, T; Shimokata, K1

Other Studies

10 other study(ies) available for y 27632 and methacholine chloride

ArticleYear
Y-27632 potentiates relaxant effects of beta 2-adrenoceptor agonists in bovine tracheal smooth muscle.
    European journal of pharmacology, 2000, Feb-11, Volume: 389, Issue:1

    Topics: Adrenergic beta-Agonists; Albuterol; Amides; Animals; Bronchoconstrictor Agents; Bronchodilator Agents; Cattle; Intracellular Signaling Peptides and Proteins; Methacholine Chloride; Muscle Relaxants, Central; Muscle Relaxation; Muscle, Smooth; Protein Serine-Threonine Kinases; Pyridines; Receptors, Adrenergic, beta-2; rho-Associated Kinases; Terbutaline; Trachea

2000
Possible involvement of Rho kinase in Ca2+ sensitization and mobilization by MCh in tracheal smooth muscle.
    American journal of physiology. Lung cellular and molecular physiology, 2001, Volume: 280, Issue:6

    Topics: Amides; Animals; Bronchoconstriction; Bronchoconstrictor Agents; Calcium; Dose-Response Relationship, Drug; Enzyme Inhibitors; Fluorescent Dyes; Fura-2; Guinea Pigs; In Vitro Techniques; Indoles; Intracellular Fluid; Intracellular Signaling Peptides and Proteins; Isometric Contraction; Male; Maleimides; Methacholine Chloride; Muscle, Smooth; Protein Kinase C; Protein Serine-Threonine Kinases; Pyridines; rho-Associated Kinases; Spectrometry, Fluorescence; Trachea

2001
Role of lysophosphatidylcholine in the desensitization of beta-adrenergic receptors by Ca(2+) sensitization in tracheal smooth muscle.
    American journal of respiratory cell and molecular biology, 2001, Volume: 25, Issue:3

    Topics: Adenylate Cyclase Toxin; Adrenergic beta-Agonists; Amides; Animals; Bucladesine; Calcium; Cholera Toxin; Colforsin; Dinoprostone; Dose-Response Relationship, Drug; Enzyme Inhibitors; Guinea Pigs; In Vitro Techniques; Indoles; Isoproterenol; Lysophosphatidylcholines; Male; Maleimides; Methacholine Chloride; Muscarinic Agonists; Muscle Contraction; Muscle, Smooth; Pyridines; Receptors, Adrenergic, beta; rho GTP-Binding Proteins; Spectrometry, Fluorescence; Theophylline; Trachea; Virulence Factors, Bordetella

2001
Regulation of capacitative and noncapacitative receptor-operated Ca2+ entry by rho-kinase in tracheal smooth muscle.
    American journal of respiratory cell and molecular biology, 2002, Volume: 26, Issue:4

    Topics: Actins; Amides; Animals; Calcium Channel Blockers; Calcium Signaling; Cytoskeleton; Enzyme Inhibitors; Guinea Pigs; Histamine; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Male; Methacholine Chloride; Muscle Contraction; Muscle, Smooth; Protein Serine-Threonine Kinases; Pyridines; rho-Associated Kinases; rhoA GTP-Binding Protein; Sarcoplasmic Reticulum; Signal Transduction; Trachea

2002
Differential Rho-kinase dependency of full and partial muscarinic receptor agonists in airway smooth muscle contraction.
    British journal of pharmacology, 2006, Volume: 147, Issue:7

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Alkylation; Amides; Animals; Bronchoconstrictor Agents; Calcium; Cattle; Enzyme Inhibitors; Intracellular Signaling Peptides and Proteins; Isometric Contraction; Methacholine Chloride; Muscarinic Agonists; Muscle Contraction; Muscle, Smooth; Organ Culture Techniques; Pilocarpine; Protein Serine-Threonine Kinases; Pyridines; Receptors, Muscarinic; rho-Associated Kinases; Trachea

2006
Involvement of reduced sensitivity to Ca in beta-adrenergic action on airway smooth muscle.
    Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology, 2006, Volume: 36, Issue:2

    Topics: Adrenergic beta-Agonists; Amides; Animals; Asthma; Bucladesine; Calcium; Calcium Channel Blockers; Colforsin; Cyclic AMP Receptor Protein; Cyclic AMP-Dependent Protein Kinases; Depression, Chemical; Fura-2; Guinea Pigs; Imidazoles; In Vitro Techniques; Indoles; Intracellular Signaling Peptides and Proteins; Isoproterenol; Male; Maleimides; Marine Toxins; Methacholine Chloride; Muscle Contraction; Muscle, Smooth; Myosin-Light-Chain Phosphatase; Oxazoles; Protein Kinase C; Protein Serine-Threonine Kinases; Pyridines; rho-Associated Kinases; Trachea

2006
Inhibition of Rho-kinase normalizes nonspecific hyperresponsiveness in passively sensitized airway smooth muscle preparations.
    European journal of pharmacology, 2006, Feb-15, Volume: 531, Issue:1-3

    Topics: Amides; Animals; Dose-Response Relationship, Drug; Enzyme Inhibitors; Guinea Pigs; Histamine; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Male; Methacholine Chloride; Muscle Contraction; Muscle, Smooth; Ovalbumin; Protein Serine-Threonine Kinases; Pyridines; rho-Associated Kinases; Time Factors; Trachea

2006
Roles of stretch-activated cation channel and Rho-kinase in the spontaneous contraction of airway smooth muscle.
    European journal of pharmacology, 2006, Dec-15, Volume: 552, Issue:1-3

    Topics: Amides; Animals; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Cations; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Gadolinium; Guinea Pigs; Imidazoles; In Vitro Techniques; Indomethacin; Intracellular Signaling Peptides and Proteins; Ion Channels; Male; Methacholine Chloride; Muscle Contraction; Muscle, Smooth; Nifedipine; Nitrobenzenes; Protein Serine-Threonine Kinases; Pyrazoles; Pyridines; rho-Associated Kinases; Simvastatin; Stress, Mechanical; Sulfonamides; Trachea

2006
Direct effects of hydrogen peroxide on airway smooth muscle tone: roles of Ca2+ influx and Rho-kinase.
    European journal of pharmacology, 2007, Feb-05, Volume: 556, Issue:1-3

    Topics: Amides; Animals; Bronchoconstrictor Agents; Calcium; Calcium Channel Blockers; Epithelium; Guinea Pigs; Hydrogen Peroxide; Imidazoles; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Isometric Contraction; Male; Methacholine Chloride; Muscle Tonus; Muscle, Smooth; Oxidative Stress; Protein Serine-Threonine Kinases; Pyridines; rho-Associated Kinases; Signal Transduction; Trachea; Verapamil

2007
Roles of P2X receptors and Ca2+ sensitization in extracellular adenosine triphosphate-induced hyperresponsiveness in airway smooth muscle.
    Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology, 2007, Volume: 37, Issue:6

    Topics: Adenosine Triphosphate; Amides; Animals; Bronchi; Bronchial Hyperreactivity; Bronchoconstrictor Agents; Calcium; Calcium Signaling; Cells, Cultured; Drug Synergism; Enzyme Inhibitors; Guinea Pigs; Intracellular Signaling Peptides and Proteins; Isometric Contraction; Male; Methacholine Chloride; Myocytes, Smooth Muscle; Organ Culture Techniques; Phosphoprotein Phosphatases; Protein Serine-Threonine Kinases; Pulmonary Disease, Chronic Obstructive; Purinergic P2 Receptor Agonists; Pyridines; Receptors, Purinergic P2; Receptors, Purinergic P2X; Respiratory Mucosa; rho-Associated Kinases; src-Family Kinases; Time Factors

2007