Page last updated: 2024-09-03

y 27632 and ketotifen

y 27632 has been researched along with ketotifen in 3 studies

Compound Research Comparison

Studies
(y 27632)
Trials
(y 27632)
Recent Studies (post-2010)
(y 27632)
Studies
(ketotifen)
Trials
(ketotifen)
Recent Studies (post-2010) (ketotifen)
1,92438911,212275151

Protein Interaction Comparison

ProteinTaxonomyy 27632 (IC50)ketotifen (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.16
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.838
Muscarinic acetylcholine receptor M4Homo sapiens (human)1.009
Muscarinic acetylcholine receptor M5Homo sapiens (human)0.374
Alpha-2A adrenergic receptorHomo sapiens (human)2.187
Muscarinic acetylcholine receptor M1Homo sapiens (human)1.112
Alpha-2B adrenergic receptorHomo sapiens (human)0.71
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)2.537
Muscarinic acetylcholine receptor M3Homo sapiens (human)2.209
D(1A) dopamine receptorHomo sapiens (human)0.872
Histamine H2 receptorHomo sapiens (human)4.129
Alpha-1D adrenergic receptorHomo sapiens (human)3.727
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.031
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.16
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)2.537
Histamine H1 receptorHomo sapiens (human)0.0011
D(3) dopamine receptorHomo sapiens (human)1.963
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.046
5-hydroxytryptamine receptor 6Homo sapiens (human)1.141

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fang, YI; Hashimoto, T; Momose, K; Nakano, Y; Ohata, H; Yamashita, M1
Hashimoto, T; Momose, K; Ohata, H1
Han, ES; Kim, H; Kim, HJ; Kim, JJ; Kim, KM; Koh, JY; Lee, CH; Noh, MS; Park, SM1

Other Studies

3 other study(ies) available for y 27632 and ketotifen

ArticleYear
Role of Rho-associated protein kinase and histamine in lysophosphatidic acid-induced airway hyperresponsiveness in guinea pigs.
    Japanese journal of pharmacology, 2002, Volume: 88, Issue:3

    Topics: Acetylcholine; Amides; Animals; Bronchial Hyperreactivity; Enzyme Inhibitors; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine Release; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Ketotifen; Lung; Lysophospholipids; Male; Muscle Contraction; Muscle, Smooth; Protein Serine-Threonine Kinases; Pyridines; Pyrilamine; rho-Associated Kinases; Structure-Activity Relationship

2002
Itch-scratch responses induced by lysophosphatidic acid in mice.
    Pharmacology, 2004, Volume: 72, Issue:1

    Topics: Amides; Animals; Antipruritics; Capsaicin; Injections, Intradermal; Intracellular Signaling Peptides and Proteins; Ketotifen; Lysophospholipids; Mice; Mice, Inbred ICR; Protein Serine-Threonine Kinases; Pruritus; Pyridines; Rats; rho-Associated Kinases

2004
Characterizations of sphingosylphosphorylcholine-induced scratching responses in ICR mice using naltrexon, capsaicin, ketotifen and Y-27632.
    European journal of pharmacology, 2008, Mar-31, Volume: 583, Issue:1

    Topics: Amides; Animals; Antipruritics; Behavior, Animal; Capsaicin; Dose-Response Relationship, Drug; Injections, Intradermal; Ketotifen; Male; Mice; Mice, Inbred ICR; Muscle Relaxants, Central; Naltrexone; Narcotic Antagonists; Phosphorylcholine; Pruritus; Pyridines; rho-Associated Kinases; Sphingosine

2008