y 27632 has been researched along with histamine in 16 studies
Studies (y 27632) | Trials (y 27632) | Recent Studies (post-2010) (y 27632) | Studies (histamine) | Trials (histamine) | Recent Studies (post-2010) (histamine) |
---|---|---|---|---|---|
1,924 | 3 | 891 | 37,718 | 1,372 | 3,457 |
Protein | Taxonomy | y 27632 (IC50) | histamine (IC50) |
---|---|---|---|
Histamine H1 receptor | Rattus norvegicus (Norway rat) | 0.1585 | |
Histamine H1 receptor | Homo sapiens (human) | 0.1585 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 10 (62.50) | 29.6817 |
2010's | 6 (37.50) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Brautigan, DL; Eto, M; Kitazawa, T; Woodsome, TP | 1 |
Hokazono, Y; Kobayashi, S; Kusuda, T; Miyake, T; Mizukami, Y; Mogami, K; Sato, M; Suzuki, S; Todoroki-Ikeda, N; Yamagata, H; Yamamoto, K | 1 |
Eichholtz, T; Potempa, S; Ridley, AJ; Wójciak-Stothard, B | 1 |
Brautigan, DL; Eto, M; Kitazawa, T; Mukai, H; Ono, Y; Yazawa, M | 1 |
Arakawa, H; Iizuka, K; Kato, M; Mochizuki, H; Morikawa, A; Nishimura, H; Saga, R; Tokuyama, K | 1 |
Hayashi, H; Honjo, H; Ito, S; Katoh, H; Kodama, I; Kume, H; Yamaki, K | 1 |
Fang, YI; Hashimoto, T; Momose, K; Nakano, Y; Ohata, H; Yamashita, M | 1 |
Glynos, K; Papapetropoulos, A; Pizurki, L; Roussos, C; Zhou, Z | 1 |
Meurs, H; Nelemans, SA; Schaafsma, D; Zaagsma, J; Zuidhof, AB | 1 |
Akça, T; Aydin, S; Büyükafşar, K; Nalan Tiftik, R; Sahan-Firat, S | 1 |
Joh, S; Kawaguchi, T; Kuji, A; Satoh, K | 1 |
Breslin, JW | 1 |
Calzetta, L; Cazzola, M; Kanabar, V; Lauro, D; Matera, MG; Novelli, L; Page, CP; Rogliani, P | 1 |
Butler, JP; Carman, CV; Fredberg, JJ; Hardin, C; Krishnan, R; Manomohan, G; Martinelli, R; Rajendran, K; Tambe, DT | 1 |
Adams, RH; Amornphimoltham, P; Ando, K; Chavakis, T; Fukuhara, S; Gutkind, JS; Masedunskas, A; Mikelis, CM; Mochizuki, N; Offermanns, S; Sakurai, A; Simaan, M; Weigert, R; Zheng, Y | 1 |
Beyerle, A; Bischoff, I; Fürst, R; Hornburger, MC; Mayer, BA; Wegener, J | 1 |
16 other study(ies) available for y 27632 and histamine
Article | Year |
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Agonists trigger G protein-mediated activation of the CPI-17 inhibitor phosphoprotein of myosin light chain phosphatase to enhance vascular smooth muscle contractility.
Topics: Amides; Animals; Cell Membrane Permeability; Enzyme Inhibitors; Femoral Artery; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Histamine; In Vitro Techniques; Indoles; Intracellular Signaling Peptides and Proteins; Maleimides; Muscle Contraction; Muscle Proteins; Muscle, Smooth, Vascular; Myosin-Light-Chain Phosphatase; Phenylephrine; Phosphoprotein Phosphatases; Phosphoproteins; Phosphorylation; Protein Kinase C; Protein Serine-Threonine Kinases; Pyridines; Rabbits; rho-Associated Kinases; Type C Phospholipases | 2000 |
Sphingosylphosphorylcholine induces Ca(2+)-sensitization of vascular smooth muscle contraction: possible involvement of rho-kinase.
Topics: Amides; Animals; Calcium; Coronary Vessels; Cytosol; Enzyme Inhibitors; Guanosine Triphosphate; Histamine; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Kinetics; Muscle Contraction; Muscle, Smooth, Vascular; Phosphorylcholine; Potassium; Protein Serine-Threonine Kinases; Pyridines; rho-Associated Kinases; Sphingosine; Swine | 2000 |
Rho and Rac but not Cdc42 regulate endothelial cell permeability.
Topics: Actins; Adherens Junctions; Amides; cdc42 GTP-Binding Protein; Cell Adhesion; Cell Membrane Permeability; Cells, Cultured; Cytoskeleton; Endothelium, Vascular; Enzyme Inhibitors; Histamine; Humans; Intracellular Signaling Peptides and Proteins; Protein Serine-Threonine Kinases; Pyridines; rac1 GTP-Binding Protein; rho-Associated Kinases; rhoA GTP-Binding Protein; Thrombin; Tight Junctions | 2001 |
Histamine-induced vasoconstriction involves phosphorylation of a specific inhibitor protein for myosin phosphatase by protein kinase C alpha and delta isoforms.
Topics: Amides; Amino Acid Sequence; Animals; Aorta; Carbazoles; Chromatography; Chromatography, Affinity; Chromatography, Ion Exchange; Durapatite; Enzyme Activation; Enzyme Inhibitors; Histamine; In Vitro Techniques; Indoles; Isoenzymes; Kinetics; Maleimides; Molecular Sequence Data; Muscle Contraction; Muscle Proteins; Muscle Relaxants, Central; Muscle, Smooth, Vascular; Myelin Basic Protein; Myosin-Light-Chain Phosphatase; Peptide Fragments; Phorbol 12,13-Dibutyrate; Phosphoprotein Phosphatases; Phosphoproteins; Phosphorylation; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-delta; Pyridines; Recombinant Proteins; Substrate Specificity; Swine; Vasoconstriction | 2001 |
Effects of Y-27632, a Rho/Rho kinase inhibitor, on leukotriene D(4)- and histamine-induced airflow obstruction and airway microvascular leakage in guinea pigs in vivo.
Topics: Airway Obstruction; Airway Resistance; Amides; Animals; Blood Pressure; Bronchoconstriction; Bronchodilator Agents; Capillary Permeability; Enzyme Inhibitors; Guinea Pigs; Histamine; Intracellular Signaling Peptides and Proteins; Leukotriene D4; Male; Procaterol; Protein Serine-Threonine Kinases; Pyridines; rho-Associated Kinases; Specific Pathogen-Free Organisms; Time Factors | 2002 |
Regulation of capacitative and noncapacitative receptor-operated Ca2+ entry by rho-kinase in tracheal smooth muscle.
Topics: Actins; Amides; Animals; Calcium Channel Blockers; Calcium Signaling; Cytoskeleton; Enzyme Inhibitors; Guinea Pigs; Histamine; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Male; Methacholine Chloride; Muscle Contraction; Muscle, Smooth; Protein Serine-Threonine Kinases; Pyridines; rho-Associated Kinases; rhoA GTP-Binding Protein; Sarcoplasmic Reticulum; Signal Transduction; Trachea | 2002 |
Role of Rho-associated protein kinase and histamine in lysophosphatidic acid-induced airway hyperresponsiveness in guinea pigs.
Topics: Acetylcholine; Amides; Animals; Bronchial Hyperreactivity; Enzyme Inhibitors; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine Release; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Ketotifen; Lung; Lysophospholipids; Male; Muscle Contraction; Muscle, Smooth; Protein Serine-Threonine Kinases; Pyridines; Pyrilamine; rho-Associated Kinases; Structure-Activity Relationship | 2002 |
Angiopoietin-1 inhibits endothelial permeability, neutrophil adherence and IL-8 production.
Topics: Amides; Angiopoietin-1; Animals; Bradykinin; Capillary Permeability; Cattle; Cell Adhesion; Cell Line; Cells, Cultured; Endothelium, Vascular; Histamine; Humans; Interleukin-8; Intracellular Signaling Peptides and Proteins; Lung; Neutrophils; Platelet Activating Factor; Protein Serine-Threonine Kinases; Pyridines; rho-Associated Kinases; Thrombin | 2003 |
Inhibition of Rho-kinase normalizes nonspecific hyperresponsiveness in passively sensitized airway smooth muscle preparations.
Topics: Amides; Animals; Dose-Response Relationship, Drug; Enzyme Inhibitors; Guinea Pigs; Histamine; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Male; Methacholine Chloride; Muscle Contraction; Muscle, Smooth; Ovalbumin; Protein Serine-Threonine Kinases; Pyridines; rho-Associated Kinases; Time Factors; Trachea | 2006 |
Contribution of Rho-kinase in human gallbladder contractions.
Topics: Aged; Amides; Blotting, Western; Carbachol; Cholecystokinin; Dose-Response Relationship, Drug; Endothelin-1; Enzyme Inhibitors; Female; Gallbladder; Histamine; Humans; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Male; Middle Aged; Muscle Contraction; Neurokinin A; Peptide Fragments; Potassium Chloride; Protein Serine-Threonine Kinases; Pyridines; rho-Associated Kinases; Serotonin | 2006 |
Features of distinct contractions induced with a high and a low concentration of KCl, noradrenaline, and histamine in swine lingual artery.
Topics: Amides; Animals; Arteries; Boron Compounds; Calcium; Dose-Response Relationship, Drug; Endothelium, Vascular; Histamine; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Nitric Oxide Donors; Nitroprusside; Norepinephrine; Potassium Chloride; Pyridines; rho-Associated Kinases; Signal Transduction; Swine; Tongue; Vasoconstrictor Agents | 2010 |
ROCK and cAMP promote lymphatic endothelial cell barrier integrity and modulate histamine and thrombin-induced barrier dysfunction.
Topics: Adult; Amides; Azepines; Capillary Permeability; Cells, Cultured; Cyclic AMP; Endothelial Cells; Enzyme Inhibitors; Histamine; Humans; Myosin-Light-Chain Kinase; Naphthalenes; Pyridines; rho-Associated Kinases; Signal Transduction; Thrombin | 2011 |
High glucose enhances responsiveness of human airways smooth muscle via the Rho/ROCK pathway.
Topics: Acetylcholine; Amides; Bradykinin; Bronchi; Calcium Signaling; Cells, Cultured; Enzyme Activation; Female; Glucose; Histamine; Humans; Hyperglycemia; Imidazoles; In Vitro Techniques; Male; Mannitol; Middle Aged; Muscle Contraction; Muscle, Smooth; Myosin-Light-Chain Phosphatase; Osmolar Concentration; Oxadiazoles; Phosphorylation; Protein Processing, Post-Translational; Pyridines; rho GTP-Binding Proteins; rho-Associated Kinases | 2012 |
Glassy dynamics, cell mechanics, and endothelial permeability.
Topics: Amides; Cell Line; Cell Membrane Permeability; Cytoskeleton; Endothelial Cells; Fluorescent Dyes; Hepatocyte Growth Factor; Histamine; Humans; Hydrogen Peroxide; Lysophospholipids; Microscopy, Confocal; Phase Transition; Pyridines; Sphingosine; Thrombin | 2013 |
RhoA and ROCK mediate histamine-induced vascular leakage and anaphylactic shock.
Topics: Adherens Junctions; Amides; Anaphylaxis; Animals; Capillary Permeability; Endothelial Cells; Endothelium, Vascular; Female; Gene Expression Regulation; GTP-Binding Protein alpha Subunits, Gq-G11; Histamine; Humans; Male; Mice; Mice, Knockout; Phospholipase C beta; Protein Kinase Inhibitors; Pyridines; Receptors, Histamine H1; rho-Associated Kinases; rhoA GTP-Binding Protein; RNA, Small Interfering; Signal Transduction; Skin | 2015 |
Pitfalls in assessing microvascular endothelial barrier function: impedance-based devices versus the classic macromolecular tracer assay.
Topics: Amides; Biological Assay; Capillary Permeability; Cells, Cultured; Electric Impedance; Endothelial Cells; Endothelium, Vascular; Histamine; Humans; Pyridines | 2016 |