Page last updated: 2024-09-03

y 27632 and ex 527

y 27632 has been researched along with ex 527 in 2 studies

Compound Research Comparison

Studies
(y 27632)
Trials
(y 27632)
Recent Studies (post-2010)
(y 27632)
Studies
(ex 527)
Trials
(ex 527)
Recent Studies (post-2010) (ex 527)
1,92438912252209

Protein Interaction Comparison

ProteinTaxonomyy 27632 (IC50)ex 527 (IC50)
NAD-dependent protein deacetylase sirtuin-2Homo sapiens (human)2.725
NAD-dependent protein deacetylase sirtuin-1Homo sapiens (human)0.3666
NAD-dependent protein deacetylase sirtuin-3, mitochondrialHomo sapiens (human)6.4

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ1
Fu, C; Hao, S; Jin, W; Li, S; Liu, Z; Lu, H; Wang, L; Xu, X; Zhou, J1

Other Studies

2 other study(ies) available for y 27632 and ex 527

ArticleYear
Identification of potent Yes1 kinase inhibitors using a library screening approach.
    Bioorganic & medicinal chemistry letters, 2013, Aug-01, Volume: 23, Issue:15

    Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship

2013
Activation of SIRT1 ameliorates LPS-induced lung injury in mice via decreasing endothelial tight junction permeability.
    Acta pharmacologica Sinica, 2019, Volume: 40, Issue:5

    Topics: Acute Lung Injury; Administration, Inhalation; Amides; Animals; Carbazoles; Cell Membrane Permeability; Endothelial Cells; Enzyme Activators; Enzyme Inhibitors; Female; Heterocyclic Compounds, 4 or More Rings; Humans; Lipopolysaccharides; Lung; Male; Mice, Inbred BALB C; Pyridines; Signal Transduction; Sirtuin 1; Tight Junction Proteins; Tight Junctions

2019