Page last updated: 2024-09-03

y 27632 and dinoprostone

y 27632 has been researched along with dinoprostone in 10 studies

Compound Research Comparison

Studies
(y 27632)
Trials
(y 27632)
Recent Studies (post-2010)
(y 27632)
Studies
(dinoprostone)
Trials
(dinoprostone)
Recent Studies (post-2010) (dinoprostone)
1,924389129,1051,3466,357

Protein Interaction Comparison

ProteinTaxonomyy 27632 (IC50)dinoprostone (IC50)
Prostaglandin E2 receptor EP1 subtypeHomo sapiens (human)0.0155
Prostaglandin E2 receptor EP4 subtypeHomo sapiens (human)0.0031
Prostaglandin E2 receptor EP4 subtypeRattus norvegicus (Norway rat)0.0021
Prostaglandin E2 receptor EP3 subtypeHomo sapiens (human)0.002
Prostaglandin E2 receptor EP2 subtypeHomo sapiens (human)0.0087
Prostacyclin receptorHomo sapiens (human)0.26
Prostaglandin E2 receptor EP2 subtypeRattus norvegicus (Norway rat)0.0052

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's6 (60.00)29.6817
2010's3 (30.00)24.3611
2020's1 (10.00)2.80

Authors

AuthorsStudies
Ito, S; Ito, Y; Kume, H; Yamaki, K1
Janssen, LJ; Miller, J; Tazzeo, T1
Wise, H1
Janssen, LJ; Liu, C; Tazzeo, T1
Friel, AM; Morrison, JJ; O'reilly, MW; Sexton, DJ; Smith, TJ1
Chakraborty, C; Chirpac, A; Lala, PK; Nicola, C1
Stamer, WD; Wang, JW; Woodward, DF1
Dzialowski, EM; Greyner, H1
Choi, YH; Kang, JL; Lee, YJ; Park, YM; Yoon, YS1
McNamara, LM; Schiavi, J; Simfia, I1

Other Studies

10 other study(ies) available for y 27632 and dinoprostone

ArticleYear
Role of lysophosphatidylcholine in the desensitization of beta-adrenergic receptors by Ca(2+) sensitization in tracheal smooth muscle.
    American journal of respiratory cell and molecular biology, 2001, Volume: 25, Issue:3

    Topics: Adenylate Cyclase Toxin; Adrenergic beta-Agonists; Amides; Animals; Bucladesine; Calcium; Cholera Toxin; Colforsin; Dinoprostone; Dose-Response Relationship, Drug; Enzyme Inhibitors; Guinea Pigs; In Vitro Techniques; Indoles; Isoproterenol; Lysophosphatidylcholines; Male; Maleimides; Methacholine Chloride; Muscarinic Agonists; Muscle Contraction; Muscle, Smooth; Pyridines; Receptors, Adrenergic, beta; rho GTP-Binding Proteins; Spectrometry, Fluorescence; Theophylline; Trachea; Virulence Factors, Bordetella

2001
Vasoconstrictor responses, and underlying mechanisms, to isoprostanes in human and porcine bronchial arterial smooth muscle.
    British journal of pharmacology, 2003, Volume: 140, Issue:4

    Topics: Alprostadil; Amides; Animals; Bronchial Arteries; Dinoprost; Dinoprostone; Dioxanes; Dose-Response Relationship, Drug; F2-Isoprostanes; Genistein; Humans; Isoprostanes; Muscle, Smooth, Vascular; Prostaglandins E; Prostaglandins F, Synthetic; Pyridines; Receptors, Thromboxane A2, Prostaglandin H2; Signal Transduction; Swine; Vasoconstriction; Vasoconstrictor Agents

2003
Lack of interaction between prostaglandin E2 receptor subtypes in regulating adenylyl cyclase activity in cultured rat dorsal root ganglion cells.
    European journal of pharmacology, 2006, Mar-27, Volume: 535, Issue:1-3

    Topics: Adenylyl Cyclases; Alprostadil; Amides; Animals; Cell Line; Cells, Cultured; Cyclic AMP; Dinoprostone; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Epoprostenol; Ganglia, Spinal; Humans; Intracellular Signaling Peptides and Proteins; Male; Methyl Ethers; Neurites; Prostaglandin D2; Protein Serine-Threonine Kinases; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP1 Subtype; Receptors, Prostaglandin E, EP2 Subtype; Receptors, Prostaglandin E, EP3 Subtype; Receptors, Prostaglandin E, EP4 Subtype; rho-Associated Kinases; Time Factors; Tritium

2006
Isoprostane-induced airway hyperresponsiveness is dependent on internal Ca2+ handling and Rho/ROCK signaling.
    American journal of physiology. Lung cellular and molecular physiology, 2006, Volume: 291, Issue:6

    Topics: Amides; Animals; Bronchial Hyperreactivity; Calcium; Carbachol; Cattle; Dinoprostone; Enzyme Inhibitors; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Isoprostanes; Muscle, Smooth; Protein Serine-Threonine Kinases; Pyridines; Respiratory System; rho-Associated Kinases; Signal Transduction; Trachea

2006
Rho A/Rho kinase: human umbilical artery mRNA expression in normal and pre eclamptic pregnancies and functional role in isoprostane-induced vasoconstriction.
    Reproduction (Cambridge, England), 2006, Volume: 132, Issue:1

    Topics: Acute-Phase Proteins; Amides; Analysis of Variance; Case-Control Studies; Dinoprost; Dinoprostone; Female; Humans; Intracellular Signaling Peptides and Proteins; Isoprostanes; Muscle, Smooth, Vascular; Pre-Eclampsia; Pregnancy; Protein Isoforms; Protein Serine-Threonine Kinases; Pyridines; Reverse Transcriptase Polymerase Chain Reaction; rho-Associated Kinases; RNA, Messenger; Tissue Culture Techniques; Umbilical Arteries; Vasoconstrictor Agents

2006
Roles of Rho guanosine 5'-triphosphatase A, Rho kinases, and extracellular signal regulated kinase (1/2) in prostaglandin E2-mediated migration of first-trimester human extravillous trophoblast.
    Endocrinology, 2008, Volume: 149, Issue:3

    Topics: Amides; Butadienes; Cell Line; Cell Movement; Chorionic Villi; Dinoprostone; Enzyme Inhibitors; Female; Humans; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Nitriles; Pregnancy; Pregnancy Trimester, First; Pyridines; rho-Associated Kinases; rhoA GTP-Binding Protein; RNA, Small Interfering; Trophoblasts

2008
Differential effects of prostaglandin E2-sensitive receptors on contractility of human ocular cells that regulate conventional outflow.
    Investigative ophthalmology & visual science, 2013, Jul-16, Volume: 54, Issue:7

    Topics: Amides; Cells, Cultured; Dinoprostone; Elasticity; Enzyme Inhibitors; Humans; Polymerase Chain Reaction; Pyridines; Receptors, Prostaglandin; Trabecular Meshwork

2013
In vitro oxygen exposure promotes maturation of the oxygen sensitive contraction in pre-term chicken ductus arteriosus.
    Comparative biochemistry and physiology. Part A, Molecular & integrative physiology, 2015, Volume: 188

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amides; Animals; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Chick Embryo; Chickens; Dinoprostone; Dose-Response Relationship, Drug; Ductus Arteriosus; Enzyme Inhibitors; Nifedipine; Nitric Oxide; Oxygen; Pyridines; rho-Associated Kinases; Time Factors; Vasoconstriction

2015
Macrophages programmed by apoptotic cells inhibit epithelial-mesenchymal transition in lung alveolar epithelial cells via PGE2, PGD2, and HGF.
    Scientific reports, 2016, Feb-15, Volume: 6

    Topics: Alveolar Epithelial Cells; Amides; Animals; Apoptosis; Culture Media, Conditioned; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Dinoprostone; Epithelial-Mesenchymal Transition; Gene Expression Regulation; Hepatocyte Growth Factor; Macrophages; Mice; Nitrobenzenes; Prostaglandin D2; Pyridines; rho GTP-Binding Proteins; rhoA GTP-Binding Protein; Sulfonamides

2016
ROCK-II inhibition suppresses impaired mechanobiological responses in early estrogen deficient osteoblasts.
    Experimental cell research, 2020, 11-01, Volume: 396, Issue:1

    Topics: Actin Cytoskeleton; Alkaline Phosphatase; Amides; Animals; Cell Differentiation; Cell Line; Core Binding Factor Alpha 1 Subunit; Cyclooxygenase 2; Dinoprostone; Estradiol; Gene Expression Regulation; Mechanotransduction, Cellular; Mice; Osteoblasts; Osteogenesis; Osteopontin; Protein Kinase Inhibitors; Pyridines; Rheology; rho-Associated Kinases

2020