Page last updated: 2024-09-03

y 27632 and dinoprost

y 27632 has been researched along with dinoprost in 6 studies

Compound Research Comparison

Studies
(y 27632)
Trials
(y 27632)
Recent Studies (post-2010)
(y 27632)
Studies
(dinoprost)
Trials
(dinoprost)
Recent Studies (post-2010) (dinoprost)
1,924389111,5549401,936

Protein Interaction Comparison

ProteinTaxonomyy 27632 (IC50)dinoprost (IC50)
Prostaglandin G/H synthase 1 Bos taurus (cattle)0.0025
Prostaglandin G/H synthase 2 Bos taurus (cattle)0.0713
Prostaglandin G/H synthase 1Homo sapiens (human)0.14
Prostaglandin E2 receptor EP1 subtypeHomo sapiens (human)0.3
Prostaglandin G/H synthase 2Homo sapiens (human)0.14
Prostaglandin E2 receptor EP4 subtypeHomo sapiens (human)4.2
Prostaglandin F2-alpha receptorBos taurus (cattle)0.14
Prostaglandin F2-alpha receptorHomo sapiens (human)0.0139
Prostaglandin E2 receptor EP3 subtypeHomo sapiens (human)0.216
Prostaglandin D2 receptorHomo sapiens (human)4.5
Solute carrier organic anion transporter family member 2B1Rattus norvegicus (Norway rat)0.287

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (83.33)29.6817
2010's1 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Janssen, LJ; Miller, J; Tazzeo, T1
Kawagishi, R; Morishige, K; Murata, Y; Sakata, M; Sawada, K; Tahara, M; Tasaka, K1
Friel, AM; Morrison, JJ; O'reilly, MW; Sexton, DJ; Smith, TJ1
Hashiba, Y; Imai, H; Saito, N; Sasaki, T; Shimizu, T; Tosaka, M1
Honjo, H; Ito, S; Kamiya, K; Kume, H; Makino, Y; Oguma, T; Shimokata, K; Shiraki, A1
Almeida-Reis, R; Charafeddine, HT; da Silva, PA; Leick-Maldonado, EA; Martins, MA; Perini, A; Possa, SS; Prado, CM; Righetti, RF; Saraiva-Romanholo, BM; Tibério, Ide F1

Other Studies

6 other study(ies) available for y 27632 and dinoprost

ArticleYear
Vasoconstrictor responses, and underlying mechanisms, to isoprostanes in human and porcine bronchial arterial smooth muscle.
    British journal of pharmacology, 2003, Volume: 140, Issue:4

    Topics: Alprostadil; Amides; Animals; Bronchial Arteries; Dinoprost; Dinoprostone; Dioxanes; Dose-Response Relationship, Drug; F2-Isoprostanes; Genistein; Humans; Isoprostanes; Muscle, Smooth, Vascular; Prostaglandins E; Prostaglandins F, Synthetic; Pyridines; Receptors, Thromboxane A2, Prostaglandin H2; Signal Transduction; Swine; Vasoconstriction; Vasoconstrictor Agents

2003
Tocolytic effect of a Rho-kinase inhibitor in a mouse model of lipopolysaccharide-induced preterm delivery.
    American journal of obstetrics and gynecology, 2005, Volume: 192, Issue:3

    Topics: Amides; Animals; Cells, Cultured; Dinoprost; Disease Models, Animal; Enzyme Inhibitors; Female; Intracellular Signaling Peptides and Proteins; Lipopolysaccharides; Mice; Mice, Inbred C3H; Obstetric Labor, Premature; Pregnancy; Protein Serine-Threonine Kinases; Pyridines; rho-Associated Kinases; Tocolytic Agents

2005
Rho A/Rho kinase: human umbilical artery mRNA expression in normal and pre eclamptic pregnancies and functional role in isoprostane-induced vasoconstriction.
    Reproduction (Cambridge, England), 2006, Volume: 132, Issue:1

    Topics: Acute-Phase Proteins; Amides; Analysis of Variance; Case-Control Studies; Dinoprost; Dinoprostone; Female; Humans; Intracellular Signaling Peptides and Proteins; Isoprostanes; Muscle, Smooth, Vascular; Pre-Eclampsia; Pregnancy; Protein Isoforms; Protein Serine-Threonine Kinases; Pyridines; Reverse Transcriptase Polymerase Chain Reaction; rho-Associated Kinases; RNA, Messenger; Tissue Culture Techniques; Umbilical Arteries; Vasoconstrictor Agents

2006
Vasorelaxing effect of the Rho-kinase inhibitor, Y-27632, in isolated canine basilar arteries.
    Neurological research, 2007, Volume: 29, Issue:5

    Topics: Amides; Animals; Basilar Artery; Calcium; Dinoprost; Dogs; Dose-Response Relationship, Drug; Enzyme Inhibitors; In Vitro Techniques; Myosin Light Chains; Phosphorylation; Phosphorylcholine; Pyridines; Sphingosine; Vasodilation

2007
Role of Ca2+ mobilization and Ca2+ sensitization in 8-iso-PGF 2 alpha-induced contraction in airway smooth muscle.
    Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology, 2009, Volume: 39, Issue:2

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Amides; Animals; Bridged-Ring Compounds; Calcium Channel Blockers; Calcium Signaling; Diltiazem; Dinoprost; Dioxanes; Enzyme Inhibitors; Estrenes; Guinea Pigs; Imidazoles; In Vitro Techniques; Indoles; Male; Maleimides; Muscle Contraction; Muscle, Smooth; Norbornanes; Pyridines; Pyrrolidinones; Receptors, Thromboxane A2, Prostaglandin H2; rho-Associated Kinases; Signal Transduction; Thiocarbamates; Thiones; Trachea; Type C Phospholipases; Vasoconstrictor Agents; Verapamil

2009
Rho-kinase inhibition attenuates airway responsiveness, inflammation, matrix remodeling, and oxidative stress activation induced by chronic inflammation.
    American journal of physiology. Lung cellular and molecular physiology, 2012, Dec-01, Volume: 303, Issue:11

    Topics: Airway Remodeling; Airway Resistance; Amides; Animals; Anti-Asthmatic Agents; Asthma; Collagen; Dinoprost; Drug Evaluation, Preclinical; Elastic Tissue; Elasticity; Eosinophils; Extracellular Matrix; Guinea Pigs; Inhalation; Interleukin-2; Lung; Male; Matrix Metalloproteinase 9; Nitric Oxide; Nitric Oxide Synthase Type II; Oxidative Stress; Pyridines; rho-Associated Kinases

2012