Page last updated: 2024-09-03

y 27632 and cgp 57380

y 27632 has been researched along with cgp 57380 in 2 studies

Compound Research Comparison

Studies
(y 27632)
Trials
(y 27632)
Recent Studies (post-2010)
(y 27632)
Studies
(cgp 57380)
Trials
(cgp 57380)
Recent Studies (post-2010) (cgp 57380)
1,924389164044

Protein Interaction Comparison

ProteinTaxonomyy 27632 (IC50)cgp 57380 (IC50)
Serine/threonine-protein kinase Sgk1Homo sapiens (human)2.7
Dual specificity tyrosine-phosphorylation-regulated kinase 3Homo sapiens (human)3.2
Cytochrome P450 1A2Homo sapiens (human)1.6
Proto-oncogene tyrosine-protein kinase LCK Mus musculus (house mouse)2.5
Eukaryotic translation initiation factor 4EHomo sapiens (human)3
Cytochrome P450 2D6Homo sapiens (human)1.6
Interferon-induced, double-stranded RNA-activated protein kinaseHomo sapiens (human)5
Casein kinase I isoform deltaHomo sapiens (human)0.51
Serine/threonine-protein kinase BRSK2Homo sapiens (human)1.1
Aurora kinase BHomo sapiens (human)2.5
MAP kinase-interacting serine/threonine-protein kinase 1Homo sapiens (human)1.2182
MAP kinase-interacting serine/threonine-protein kinase 2Homo sapiens (human)2.06

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Alessi, DR; Arthur, JS; Bain, J; Cohen, P; Elliott, M; Hastie, CJ; Klevernic, I; McLauchlan, H; Plater, L; Shpiro, N1
Augustin, M; Davies, SP; Gao, Y; Harvey, KJ; Kovelman, R; Patel, UA; Woodward, A1

Other Studies

2 other study(ies) available for y 27632 and cgp 57380

ArticleYear
The selectivity of protein kinase inhibitors: a further update.
    The Biochemical journal, 2007, Dec-15, Volume: 408, Issue:3

    Topics: Amino Acid Sequence; Animals; Cell Line; Drug Design; Enzyme Activation; Humans; Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Recombinant Proteins; Spodoptera

2007
A broad activity screen in support of a chemogenomic map for kinase signalling research and drug discovery.
    The Biochemical journal, 2013, Apr-15, Volume: 451, Issue:2

    Topics: Aurora Kinases; Cluster Analysis; Drug Design; Drug Discovery; Drug Evaluation, Preclinical; ErbB Receptors; Humans; Intracellular Signaling Peptides and Proteins; MAP Kinase Kinase 4; p38 Mitogen-Activated Protein Kinases; Protein Kinase Inhibitors; Protein Kinases; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Receptors, Vascular Endothelial Growth Factor; Recombinant Proteins; Reproducibility of Results; Signal Transduction; Small Molecule Libraries; Structure-Activity Relationship; Syk Kinase

2013