Page last updated: 2024-09-03

y 27632 and ag 1879

y 27632 has been researched along with ag 1879 in 11 studies

Compound Research Comparison

Studies
(y 27632)
Trials
(y 27632)
Recent Studies (post-2010)
(y 27632)
Studies
(ag 1879)
Trials
(ag 1879)
Recent Studies (post-2010) (ag 1879)
1,92438915750215

Protein Interaction Comparison

ProteinTaxonomyy 27632 (IC50)ag 1879 (IC50)
Chain A, Lck KinaseHomo sapiens (human)0.02
Chain A, Tyrosine-protein kinase LynMus musculus (house mouse)0.009
Chain A, Tyrosine-protein kinase LynMus musculus (house mouse)0.009
Receptor-interacting serine/threonine-protein kinase 2Homo sapiens (human)0.019
Proto-oncogene tyrosine-protein kinase SrcGallus gallus (chicken)0.036
Epidermal growth factor receptorHomo sapiens (human)0.48
Tyrosine-protein kinase LckHomo sapiens (human)0.004
Proto-oncogene tyrosine-protein kinase LCK Mus musculus (house mouse)0.031
Tyrosine-protein kinase FynHomo sapiens (human)0.0052
Tyrosine-protein kinase LynHomo sapiens (human)0.0005
Tyrosine-protein kinase HCKHomo sapiens (human)0.005
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)1.1814
Tyrosine-protein kinase CSKHomo sapiens (human)0.5
Casein kinase I isoform deltaHomo sapiens (human)0.041
Mitogen-activated protein kinase 14Homo sapiens (human)4.23

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's7 (63.64)29.6817
2010's4 (36.36)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Alessi, DR; Arthur, JS; Bain, J; Cohen, P; Elliott, M; Hastie, CJ; Klevernic, I; McLauchlan, H; Plater, L; Shpiro, N1
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M1
Cox, KJ; Gaj, A; Ghosh, I; Jester, BW; Shomin, CD1
Boettiger, D; Guvakova, MA; Lynch, L; Vodyanik, PI1
Shimoda, LA; Sylvester, JT; Weigand, L1
Berton, G; Cattaneo, M; Cavallini, C; Degan, M; Fumagalli, L; Gaino, S; Lecchi, A; Lechi Santonastaso, C; Minuz, P; Tommasoli, RM1
Lewis, SJ; Lewis, TH; Moore, JN; Noschka, E; Peroni, JF; Robertson, TP1
Giehl, K; Goppelt-Struebe, M; Graness, A1
Fu, X; Huang, J; Simoncini, T; Tan, Z; Wang, T; Xiang, Q; Zhang, Y; Zheng, S; Zhou, K1
Gahtan, V; Lawler, J; Maier, KG; Sadowitz, B; Seymour, KA; Stein, JJ1
Kunapuli, SP; Mao, Y1

Other Studies

11 other study(ies) available for y 27632 and ag 1879

ArticleYear
The selectivity of protein kinase inhibitors: a further update.
    The Biochemical journal, 2007, Dec-15, Volume: 408, Issue:3

    Topics: Amino Acid Sequence; Animals; Cell Line; Drug Design; Enzyme Activation; Humans; Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Recombinant Proteins; Spodoptera

2007
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
    Proceedings of the National Academy of Sciences of the United States of America, 2007, Dec-18, Volume: 104, Issue:51

    Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases

2007
Testing the promiscuity of commercial kinase inhibitors against the AGC kinase group using a split-luciferase screen.
    Journal of medicinal chemistry, 2012, Feb-23, Volume: 55, Issue:4

    Topics: Animals; Binding, Competitive; Catalytic Domain; Cell-Free System; Cyclic AMP-Dependent Protein Kinase Catalytic Subunits; Cyclic GMP-Dependent Protein Kinase Type I; Cyclic GMP-Dependent Protein Kinases; Databases, Factual; Genes, Reporter; Luciferases; Protein Kinase C; Protein Kinase Inhibitors; Rabbits; Recombinant Fusion Proteins; Structure-Activity Relationship

2012
Insulin-like growth factor I controls adhesion strength mediated by alpha5beta1 integrins in motile carcinoma cells.
    Molecular biology of the cell, 2005, Volume: 16, Issue:1

    Topics: Actins; Amides; Blotting, Western; Breast Neoplasms; Butadienes; Carcinoma; Catalysis; Cell Adhesion; Cell Line, Tumor; Cell Movement; Chromones; CSK Tyrosine-Protein Kinase; Culture Media, Serum-Free; Depsipeptides; Down-Regulation; Fibronectins; Flow Cytometry; Humans; Immunoprecipitation; Insulin-Like Growth Factor I; Integrin alpha5beta1; Intracellular Signaling Peptides and Proteins; MAP Kinase Signaling System; Microscopy, Phase-Contrast; Models, Biological; Morpholines; Nitriles; Phosphatidylinositol 3-Kinases; Phosphorylation; Protein Serine-Threonine Kinases; Protein Structure, Tertiary; Protein-Tyrosine Kinases; Pyridines; Pyrimidines; rho GTP-Binding Proteins; rho-Associated Kinases; Signal Transduction; src-Family Kinases; Time Factors

2005
Mechanisms of endothelin-1-induced contraction in pulmonary arteries from chronically hypoxic rats.
    American journal of physiology. Lung cellular and molecular physiology, 2006, Volume: 290, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Amides; Animals; Azepines; Endothelin-1; Enzyme Inhibitors; Genistein; Hypoxia; Indoles; Intracellular Signaling Peptides and Proteins; Isometric Contraction; Male; Maleimides; Myosin-Light-Chain Kinase; Potassium Chloride; Protein Kinase C; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Pulmonary Artery; Pyridines; Pyrimidines; Rats; Rats, Wistar; rho-Associated Kinases; src-Family Kinases; Staurosporine; Vasoconstriction

2006
Rapid stimulation of tyrosine phosphorylation signals downstream of G-protein-coupled receptors for thromboxane A2 in human platelets.
    The Biochemical journal, 2006, Nov-15, Volume: 400, Issue:1

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adult; Amides; Apyrase; Blood Platelets; Dose-Response Relationship, Drug; Epinephrine; Humans; Integrin alpha2; Intracellular Signaling Peptides and Proteins; Phosphorylation; Platelet Aggregation; Protein Serine-Threonine Kinases; Pyrazoles; Pyridines; Pyrimidines; Receptors, G-Protein-Coupled; Receptors, Purinergic P2; Receptors, Thromboxane A2, Prostaglandin H2; rho-Associated Kinases; Signal Transduction; Tyrosine

2006
Effects of Rho-kinase and Src protein tyrosine kinase inhibition on agonist-induced vasoconstriction of arteries and veins of the equine laminar dermis.
    American journal of veterinary research, 2007, Volume: 68, Issue:8

    Topics: Amides; Animals; Arteries; Calcium; Dose-Response Relationship, Drug; Endothelin-1; Foot; Intracellular Signaling Peptides and Proteins; Phenylephrine; Protein Serine-Threonine Kinases; Pyrazoles; Pyridines; Pyrimidines; rho-Associated Kinases; Serotonin; Signal Transduction; src-Family Kinases; Vasoconstriction; Vasoconstrictor Agents; Veins

2007
The small GTPase Rac-1 is a regulator of mesangial cell morphology and thrombospondin-1 expression.
    American journal of physiology. Renal physiology, 2008, Volume: 294, Issue:2

    Topics: Actins; Amides; Aminoquinolines; Animals; Cell Adhesion; Cell Shape; Cells, Cultured; Extracellular Signal-Regulated MAP Kinases; Flavonoids; Focal Adhesions; Gene Expression; Mesangial Cells; Microtubules; Nocodazole; Paxillin; Protein Kinase Inhibitors; Pyrazoles; Pyridines; Pyrimidines; rac1 GTP-Binding Protein; Rats; Rats, Sprague-Dawley; RNA, Small Interfering; Signal Transduction; src-Family Kinases; Thrombospondin 1

2008
Progesterone enhances vascular endothelial cell migration via activation of focal adhesion kinase.
    Journal of cellular and molecular medicine, 2012, Volume: 16, Issue:2

    Topics: Amides; Androstadienes; Cell Movement; Cells, Cultured; CSK Tyrosine-Protein Kinase; Endothelial Cells; Estrenes; Focal Adhesion Protein-Tyrosine Kinases; Focal Adhesions; Furans; Human Umbilical Vein Endothelial Cells; Humans; Phosphatidylinositol 3-Kinase; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Progesterone; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-akt; Pyridines; Pyrimidines; Receptors, Progesterone; rho-Associated Kinases; RNA Interference; RNA, Small Interfering; Signal Transduction; src-Family Kinases; Wortmannin

2012
Vascular smooth muscle cell migration induced by domains of thrombospondin-1 is differentially regulated.
    American journal of surgery, 2011, Volume: 202, Issue:5

    Topics: Amides; Cell Movement; Cells, Cultured; Chemotaxis; Chromones; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; Morpholines; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Organophosphonates; Protein Folding; Pyridines; Pyrimidines; Signal Transduction; Thrombospondin 1

2011
Trypsin causes platelet activation independently of known protease-activated receptors.
    Thrombosis and haemostasis, 2013, Volume: 110, Issue:6

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adaptor Proteins, Signal Transducing; Amides; Animals; Blood Platelets; Calcium; Cell Adhesion Molecules; Cell Adhesion Molecules, Neuron-Glia; Cell Cycle Proteins; Cell Shape; Cells, Cultured; Mice; Mice, Inbred Strains; Mice, Knockout; Myosin Light Chains; Peptides, Cyclic; Phosphorylation; Platelet Activation; Pyridines; Pyrimidines; Receptors, Thrombin; rho-Associated Kinases; rhoA GTP-Binding Protein; Signal Transduction; src-Family Kinases; Trypsin

2013