y 27632 has been researched along with ag 1879 in 11 studies
Studies (y 27632) | Trials (y 27632) | Recent Studies (post-2010) (y 27632) | Studies (ag 1879) | Trials (ag 1879) | Recent Studies (post-2010) (ag 1879) |
---|---|---|---|---|---|
1,924 | 3 | 891 | 575 | 0 | 215 |
Protein | Taxonomy | y 27632 (IC50) | ag 1879 (IC50) |
---|---|---|---|
Chain A, Lck Kinase | Homo sapiens (human) | 0.02 | |
Chain A, Tyrosine-protein kinase Lyn | Mus musculus (house mouse) | 0.009 | |
Chain A, Tyrosine-protein kinase Lyn | Mus musculus (house mouse) | 0.009 | |
Receptor-interacting serine/threonine-protein kinase 2 | Homo sapiens (human) | 0.019 | |
Proto-oncogene tyrosine-protein kinase Src | Gallus gallus (chicken) | 0.036 | |
Epidermal growth factor receptor | Homo sapiens (human) | 0.48 | |
Tyrosine-protein kinase Lck | Homo sapiens (human) | 0.004 | |
Proto-oncogene tyrosine-protein kinase LCK | Mus musculus (house mouse) | 0.031 | |
Tyrosine-protein kinase Fyn | Homo sapiens (human) | 0.0052 | |
Tyrosine-protein kinase Lyn | Homo sapiens (human) | 0.0005 | |
Tyrosine-protein kinase HCK | Homo sapiens (human) | 0.005 | |
Proto-oncogene tyrosine-protein kinase Src | Homo sapiens (human) | 1.1814 | |
Tyrosine-protein kinase CSK | Homo sapiens (human) | 0.5 | |
Casein kinase I isoform delta | Homo sapiens (human) | 0.041 | |
Mitogen-activated protein kinase 14 | Homo sapiens (human) | 4.23 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 7 (63.64) | 29.6817 |
2010's | 4 (36.36) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Alessi, DR; Arthur, JS; Bain, J; Cohen, P; Elliott, M; Hastie, CJ; Klevernic, I; McLauchlan, H; Plater, L; Shpiro, N | 1 |
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M | 1 |
Cox, KJ; Gaj, A; Ghosh, I; Jester, BW; Shomin, CD | 1 |
Boettiger, D; Guvakova, MA; Lynch, L; Vodyanik, PI | 1 |
Shimoda, LA; Sylvester, JT; Weigand, L | 1 |
Berton, G; Cattaneo, M; Cavallini, C; Degan, M; Fumagalli, L; Gaino, S; Lecchi, A; Lechi Santonastaso, C; Minuz, P; Tommasoli, RM | 1 |
Lewis, SJ; Lewis, TH; Moore, JN; Noschka, E; Peroni, JF; Robertson, TP | 1 |
Giehl, K; Goppelt-Struebe, M; Graness, A | 1 |
Fu, X; Huang, J; Simoncini, T; Tan, Z; Wang, T; Xiang, Q; Zhang, Y; Zheng, S; Zhou, K | 1 |
Gahtan, V; Lawler, J; Maier, KG; Sadowitz, B; Seymour, KA; Stein, JJ | 1 |
Kunapuli, SP; Mao, Y | 1 |
11 other study(ies) available for y 27632 and ag 1879
Article | Year |
---|---|
The selectivity of protein kinase inhibitors: a further update.
Topics: Amino Acid Sequence; Animals; Cell Line; Drug Design; Enzyme Activation; Humans; Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Recombinant Proteins; Spodoptera | 2007 |
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases | 2007 |
Testing the promiscuity of commercial kinase inhibitors against the AGC kinase group using a split-luciferase screen.
Topics: Animals; Binding, Competitive; Catalytic Domain; Cell-Free System; Cyclic AMP-Dependent Protein Kinase Catalytic Subunits; Cyclic GMP-Dependent Protein Kinase Type I; Cyclic GMP-Dependent Protein Kinases; Databases, Factual; Genes, Reporter; Luciferases; Protein Kinase C; Protein Kinase Inhibitors; Rabbits; Recombinant Fusion Proteins; Structure-Activity Relationship | 2012 |
Insulin-like growth factor I controls adhesion strength mediated by alpha5beta1 integrins in motile carcinoma cells.
Topics: Actins; Amides; Blotting, Western; Breast Neoplasms; Butadienes; Carcinoma; Catalysis; Cell Adhesion; Cell Line, Tumor; Cell Movement; Chromones; CSK Tyrosine-Protein Kinase; Culture Media, Serum-Free; Depsipeptides; Down-Regulation; Fibronectins; Flow Cytometry; Humans; Immunoprecipitation; Insulin-Like Growth Factor I; Integrin alpha5beta1; Intracellular Signaling Peptides and Proteins; MAP Kinase Signaling System; Microscopy, Phase-Contrast; Models, Biological; Morpholines; Nitriles; Phosphatidylinositol 3-Kinases; Phosphorylation; Protein Serine-Threonine Kinases; Protein Structure, Tertiary; Protein-Tyrosine Kinases; Pyridines; Pyrimidines; rho GTP-Binding Proteins; rho-Associated Kinases; Signal Transduction; src-Family Kinases; Time Factors | 2005 |
Mechanisms of endothelin-1-induced contraction in pulmonary arteries from chronically hypoxic rats.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Amides; Animals; Azepines; Endothelin-1; Enzyme Inhibitors; Genistein; Hypoxia; Indoles; Intracellular Signaling Peptides and Proteins; Isometric Contraction; Male; Maleimides; Myosin-Light-Chain Kinase; Potassium Chloride; Protein Kinase C; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Pulmonary Artery; Pyridines; Pyrimidines; Rats; Rats, Wistar; rho-Associated Kinases; src-Family Kinases; Staurosporine; Vasoconstriction | 2006 |
Rapid stimulation of tyrosine phosphorylation signals downstream of G-protein-coupled receptors for thromboxane A2 in human platelets.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adult; Amides; Apyrase; Blood Platelets; Dose-Response Relationship, Drug; Epinephrine; Humans; Integrin alpha2; Intracellular Signaling Peptides and Proteins; Phosphorylation; Platelet Aggregation; Protein Serine-Threonine Kinases; Pyrazoles; Pyridines; Pyrimidines; Receptors, G-Protein-Coupled; Receptors, Purinergic P2; Receptors, Thromboxane A2, Prostaglandin H2; rho-Associated Kinases; Signal Transduction; Tyrosine | 2006 |
Effects of Rho-kinase and Src protein tyrosine kinase inhibition on agonist-induced vasoconstriction of arteries and veins of the equine laminar dermis.
Topics: Amides; Animals; Arteries; Calcium; Dose-Response Relationship, Drug; Endothelin-1; Foot; Intracellular Signaling Peptides and Proteins; Phenylephrine; Protein Serine-Threonine Kinases; Pyrazoles; Pyridines; Pyrimidines; rho-Associated Kinases; Serotonin; Signal Transduction; src-Family Kinases; Vasoconstriction; Vasoconstrictor Agents; Veins | 2007 |
The small GTPase Rac-1 is a regulator of mesangial cell morphology and thrombospondin-1 expression.
Topics: Actins; Amides; Aminoquinolines; Animals; Cell Adhesion; Cell Shape; Cells, Cultured; Extracellular Signal-Regulated MAP Kinases; Flavonoids; Focal Adhesions; Gene Expression; Mesangial Cells; Microtubules; Nocodazole; Paxillin; Protein Kinase Inhibitors; Pyrazoles; Pyridines; Pyrimidines; rac1 GTP-Binding Protein; Rats; Rats, Sprague-Dawley; RNA, Small Interfering; Signal Transduction; src-Family Kinases; Thrombospondin 1 | 2008 |
Progesterone enhances vascular endothelial cell migration via activation of focal adhesion kinase.
Topics: Amides; Androstadienes; Cell Movement; Cells, Cultured; CSK Tyrosine-Protein Kinase; Endothelial Cells; Estrenes; Focal Adhesion Protein-Tyrosine Kinases; Focal Adhesions; Furans; Human Umbilical Vein Endothelial Cells; Humans; Phosphatidylinositol 3-Kinase; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Progesterone; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-akt; Pyridines; Pyrimidines; Receptors, Progesterone; rho-Associated Kinases; RNA Interference; RNA, Small Interfering; Signal Transduction; src-Family Kinases; Wortmannin | 2012 |
Vascular smooth muscle cell migration induced by domains of thrombospondin-1 is differentially regulated.
Topics: Amides; Cell Movement; Cells, Cultured; Chemotaxis; Chromones; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; Morpholines; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Organophosphonates; Protein Folding; Pyridines; Pyrimidines; Signal Transduction; Thrombospondin 1 | 2011 |
Trypsin causes platelet activation independently of known protease-activated receptors.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adaptor Proteins, Signal Transducing; Amides; Animals; Blood Platelets; Calcium; Cell Adhesion Molecules; Cell Adhesion Molecules, Neuron-Glia; Cell Cycle Proteins; Cell Shape; Cells, Cultured; Mice; Mice, Inbred Strains; Mice, Knockout; Myosin Light Chains; Peptides, Cyclic; Phosphorylation; Platelet Activation; Pyridines; Pyrimidines; Receptors, Thrombin; rho-Associated Kinases; rhoA GTP-Binding Protein; Signal Transduction; src-Family Kinases; Trypsin | 2013 |