Page last updated: 2024-08-16

xylazine and prazosin

xylazine has been researched along with prazosin in 38 studies

Research

Studies (38)

TimeframeStudies, this research(%)All Research%
pre-199023 (60.53)18.7374
1990's8 (21.05)18.2507
2000's4 (10.53)29.6817
2010's3 (7.89)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andrews, PR; Craik, DJ; Martin, JL1
Batink, H; de Jonge, A; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Sperlágh, B; Vizi, ES1
Hsu, WH; Ko, JC; Smith, BE1
Docherty, JR4
Hembrough, FB; Hsu, WH; Rong, YF1
Kawai, Y; Kobayashi, S; Ohhashi, T1
Hiley, CR; Nichols, AJ1
Maniwa, T; Morita, T; Satoh, K; Taira, N1
Livingston, A; Nolan, A; Waterman, A1
Allen, JM; McCarron, JG; McHale, NG; Thornbury, KD1
Emi, S; Hikasa, Y; Ogasawara, S; Takase, K1
Nyman, L; Virtanen, R1
Docherty, JR; Hyland, L2
Kobinger, W1
Harsing, LG; Kapocsi, J; Ludvig, N; Serfozo, P; Somogyi, GT; Vizi, ES; Woods, RJ1
Benson, GJ; Thurmon, JC; Tranquilli, WJ2
Maggi, CA; Manzini, S; Meli, A1
Ruckebusch, Y1
Hsu, WH; Hummel, SK1
Folly, G; Ludvig, N; Rónai, AZ; Vizi, ES1
Arrue, R; Cox, JF; Perez, R1
Day, TK; Muir, WW1
Bourin, M; Ganry, H1
Docherty, JR; Kearns, S; O'Rourke, M1
Blandizzi, C; Carignani, D; Colucci, R; Crema, F; Del Tacca, M; Lazzeri, G; Natale, G1
Katz, U; Nagel, W1
Bischoff, FP; Braeken, M; Kennis, LE; Leysen, JE; Love, CJ; Megens, AA; Mertens, CJ; Pieters, S; Van den Keybus, FA1
Chiba, S; Taguchi, Y; Yang, XP1
Muir, WW; Teng, B1
Gyires, K; Kató, E; Lipták, L; Mátyus, P; Rónai, AZ; Shujaa, N1
Hikasa, Y; Miki, Y; Murahata, Y1

Reviews

2 review(s) available for xylazine and prazosin

ArticleYear
Rudolf Buchheim lecture. Drugs as tools in research on adrenoceptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 332, Issue:2

    Topics: Angiotensin II; Animals; Azepines; Blood Pressure; Clonidine; Guanabenz; Guanfacine; Guanidines; Heart Rate; Humans; Imidazoles; Methoxamine; Oxymetazoline; Phenylacetates; Prazosin; Propanolamines; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Thiophenes; Xylazine; Yohimbine

1986
Pharmacology of reticulo-ruminal motor function.
    Journal of veterinary pharmacology and therapeutics, 1983, Volume: 6, Issue:4

    Topics: Adrenergic Agonists; Adrenergic alpha-Antagonists; Animals; Atropine; Behavior, Animal; Cattle; Central Nervous System; Gastrointestinal Motility; Goats; Naloxone; Narcotic Antagonists; Parasympathomimetics; Prazosin; Reticulum; Serotonin Antagonists; Sheep; Stomach, Ruminant; Xylazine

1983

Other Studies

36 other study(ies) available for xylazine and prazosin

ArticleYear
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Quantitative relationships between alpha-adrenergic activity and binding affinity of alpha-adrenoceptor agonists and antagonists.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Blood Pressure; Brain; Cell Membrane; Clonidine; Kinetics; Prazosin; Quinazolines; Rats; Receptors, Adrenergic, alpha; Structure-Activity Relationship; Vasoconstriction

1984
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Is the neuronal ATP release from guinea-pig vas deferens subject to alpha 2-adrenoceptor-mediated modulation?
    Neuroscience, 1992, Volume: 51, Issue:1

    Topics: Adenosine Triphosphate; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Berberine; Clonidine; Electric Stimulation; Guinea Pigs; Imidazoles; Male; Medetomidine; Muscle Contraction; Muscle, Smooth; Neurons; Norepinephrine; Oxymetazoline; Prazosin; Receptors, Adrenergic, alpha; Reserpine; Vas Deferens; Xylazine; Yohimbine

1992
Xylazine enhances porcine myometrial contractility in vitro: possible involvement of alpha 2-adrenoceptors and Ca2+ channels.
    Biology of reproduction, 1990, Volume: 43, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Calcium Channels; Carbachol; Dioxanes; Female; Idazoxan; Myometrium; Prazosin; Receptors, Adrenergic, alpha; Swine; Uterine Contraction; Verapamil; Xylazine; Yohimbine

1990
An investigation of the effects of intravenous injection of the 5-hydroxytryptamine 2 receptor antagonists ketanserin and LY 53857 on blood pressure in anesthetized spontaneously hypertensive rats.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Anesthesia; Animals; Blood Pressure; Ergolines; Heart Rate; Hypertension; Ketanserin; Male; Prazosin; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha; Receptors, Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes; Xylazine

1989
The effects of jingsongling, a xylazine analog, on mean arterial blood pressure and heart rate in dogs--influences of yohimbine, tolazoline, prazosin, and atropine.
    Journal of veterinary pharmacology and therapeutics, 1989, Volume: 12, Issue:3

    Topics: Animals; Atropine; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Heart Rate; Male; Molecular Structure; Prazosin; Thiazines; Thiazoles; Tolazoline; Xylazine; Yohimbine

1989
Existence of two types of postjunctional alpha-adrenoceptors in the isolated canine internal carotid artery.
    Canadian journal of physiology and pharmacology, 1988, Volume: 66, Issue:5

    Topics: Animals; Carotid Artery, Internal; Dogs; Dose-Response Relationship, Drug; Female; Imidazoles; Male; Norepinephrine; Phentolamine; Phenylephrine; Prazosin; Receptors, Adrenergic, alpha; Xylazine; Yohimbine

1988
Identification of adrenoceptors and dopamine receptors mediating vascular responses in the superior mesenteric arterial bed of the rat.
    The Journal of pharmacy and pharmacology, 1985, Volume: 37, Issue:2

    Topics: Animals; Apomorphine; Blood Pressure; Dopamine; In Vitro Techniques; Male; Mesenteric Arteries; Norepinephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Dopamine; Xylazine

1985
Undifferentiated effects of calcium antagonists on pressor responses to selective alpha-1 and alpha-2 adrenoceptor agonists in anesthetized, spinal dogs.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 234, Issue:3

    Topics: Adrenergic alpha-Agonists; Anesthesia; Animals; Blood Pressure; Calcium Channel Blockers; Dogs; Female; Male; Methoxamine; Prazosin; Receptors, Adrenergic, alpha; Spinal Cord; Vasoconstriction; Xylazine; Yohimbine

1985
The effects of alpha 2 adrenoceptor agonists on airway pressure in anaesthetized sheep.
    Journal of veterinary pharmacology and therapeutics, 1986, Volume: 9, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Airway Resistance; Animals; Clonidine; Dioxanes; Female; Histamine; Idazoxan; Injections, Intravenous; Injections, Intraventricular; Methoxamine; Prazosin; Pyrilamine; Sheep; Tripelennamine; Xylazine

1986
Release of [3H]-noradrenaline from the sympathetic nerves to bovine mesenteric lymphatic vessels and its modification by alpha-agonists and antagonists.
    British journal of pharmacology, 1988, Volume: 94, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Calcium; Cattle; Clonidine; Cocaine; Electric Stimulation; Feedback; Lymphatic System; Mesentery; Norepinephrine; Phentolamine; Phenylephrine; Prazosin; Sympathetic Nervous System; Tetrodotoxin; Xylazine; Yohimbine

1988
Antagonistic effects of alpha-adrenoceptor blocking agents on reticuloruminal hypomotility induced by xylazine in cattle.
    Canadian journal of veterinary research = Revue canadienne de recherche veterinaire, 1988, Volume: 52, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Cattle; Domperidone; Female; Gastrointestinal Motility; Naloxone; Prazosin; Reticulum; Rumen; Thiazines; Tolazoline; Xylazine; Yohimbine

1988
Evaluation of the alpha 1- and alpha 2-adrenoceptor effects of detomidine, a novel veterinary sedative analgesic.
    European journal of pharmacology, 1985, Jan-22, Volume: 108, Issue:2

    Topics: Analgesics; Animals; Clonidine; Electric Stimulation; Female; Hypnotics and Sedatives; Imidazoles; In Vitro Techniques; Kinetics; Male; Membranes; Mice; Muscle Contraction; Muscle, Smooth; Prazosin; Rabbits; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Vas Deferens; Xylazine

1985
An investigation of age-related changes in pre- and postjunctional alpha-adrenoceptors in human saphenous vein.
    European journal of pharmacology, 1985, Aug-27, Volume: 114, Issue:3

    Topics: Adult; Age Factors; Aged; Electric Stimulation; Humans; In Vitro Techniques; Male; Middle Aged; Prazosin; Receptors, Adrenergic, alpha; Saphenous Vein; Tritium; Vasoconstriction; Xylazine; Yohimbine

1985
Alpha-adrenoceptor responsiveness in the aged rat.
    European journal of pharmacology, 1986, Jul-15, Volume: 126, Issue:1-2

    Topics: Aging; Anesthesia; Animals; Blood Pressure; Cocaine; Decerebrate State; Ethanolamines; Heart Rate; Male; Norepinephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Xylazine

1986
Neurochemical evidence for two types of presynaptic alpha 2-adrenoceptors.
    Neurochemical research, 1987, Volume: 12, Issue:2

    Topics: Adrenergic Fibers; Animals; Cholinergic Fibers; Guinea Pigs; Male; Muscle, Smooth; Myenteric Plexus; Norepinephrine; Prazosin; Rats; Receptors, Adrenergic, alpha; Vas Deferens; Xylazine

1987
Halothane-catecholamine arrhythmias in swine (Sus scrofa).
    American journal of veterinary research, 1986, Volume: 47, Issue:10

    Topics: Anesthesia; Animals; Arrhythmias, Cardiac; Blood Pressure; Epinephrine; Female; Halothane; Heart Rate; Male; Metoprolol; Prazosin; Swine; Xylazine

1986
Alterations in the arrhythmogenic dose of epinephrine after adrenergic receptor blockade with prazosin, metoprolol, or yohimbine in halothane-xylazine-anesthetized dogs.
    American journal of veterinary research, 1986, Volume: 47, Issue:1

    Topics: Anesthesia; Animals; Arrhythmias, Cardiac; Dogs; Dose-Response Relationship, Drug; Epinephrine; Female; Halothane; Male; Metoprolol; Prazosin; Receptors, Adrenergic; Xylazine; Yohimbine

1986
Alpha-adrenoceptor subtypes and Ca2+ mobilization in the rabbit ear artery.
    The Journal of pharmacy and pharmacology, 1983, Volume: 35, Issue:9

    Topics: Animals; Calcium; Drug Interactions; Hydroxydopamines; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Norepinephrine; Oxidopamine; Phenylephrine; Prazosin; Rabbits; Receptors, Adrenergic, alpha; Vasoconstriction; Xylazine; Yohimbine

1983
An investigation of presynaptic alpha-adrenoceptor subtypes in the pithed rat heart and in the rat isolated vas deferens.
    British journal of pharmacology, 1984, Volume: 82, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Blood Pressure; Electric Stimulation; Ethanolamines; Heart Rate; Imidazoles; In Vitro Techniques; Isometric Contraction; Male; Muscle Contraction; Muscle, Smooth; Myocardial Contraction; Myocardium; Nifedipine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Synapses; Vas Deferens; Xylazine; Yohimbine

1984
Xylazine-induced hyperglycemia in cattle: a possible involvement of alpha 2-adrenergic receptors regulating insulin release.
    Endocrinology, 1981, Volume: 109, Issue:3

    Topics: Animals; Blood Glucose; Cattle; Female; Hyperglycemia; Insulin; Insulin Secretion; Phentolamine; Prazosin; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Thiazines; Xylazine; Yohimbine

1981
An investigation of presynaptic alpha-adrenoceptor subtypes in the pithed rat heart.
    British journal of pharmacology, 1983, Volume: 78, Issue:4

    Topics: Animals; Imidazoles; Male; Myocardium; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Synapses; Xylazine; Yohimbine

1983
Dissociation of presynaptic alpha 2-adrenoceptors following prazosin administration: presynaptic effect of prazosin.
    European journal of pharmacology, 1983, Nov-25, Volume: 95, Issue:3-4

    Topics: Animals; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Prazosin; Propranolol; Quinazolines; Rats; Receptors, Adrenergic, alpha; Synapses; Vas Deferens; Xylazine; Yohimbine

1983
Probable post-synaptic alpha 2 adrenergic mediated effect of xylazine on goat uterine motility.
    Journal of veterinary pharmacology and therapeutics, 1994, Volume: 17, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Dose-Response Relationship, Drug; Electrophysiology; Estrus; Female; Goats; Muscle, Smooth; Myometrium; Prazosin; Receptors, Adrenergic, alpha-2; Reserpine; Uterine Contraction; Xylazine; Yohimbine

1994
Alpha 2-adrenergic receptor agonist effects on supraventricular and ventricular automaticity in dogs with complete atrioventricular block.
    American journal of veterinary research, 1993, Volume: 54, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Dog Diseases; Dogs; Formaldehyde; Glycopyrrolate; Heart Block; Heart Rate; Imidazoles; Medetomidine; Prazosin; Ventricular Function; Xylazine

1993
Has iprindole an alpha adrenergic activity?
    Progress in neuro-psychopharmacology & biological psychiatry, 1993, Volume: 17, Issue:3

    Topics: Adrenergic alpha-Agonists; Animals; Exophthalmos; Iprindole; Lethal Dose 50; Male; Mice; Motor Activity; Norepinephrine; Oxotremorine; Postural Balance; Prazosin; Receptors, Adrenergic, alpha; Swimming; Xylazine

1993
Investigation of the actions of chloroethylclonidine in rat aorta.
    British journal of pharmacology, 1995, Volume: 115, Issue:8

    Topics: Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Aorta; Clonidine; Cystamine; Dioxanes; Dose-Response Relationship, Drug; Drug Synergism; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxathiins; Phenoxybenzamine; Phentolamine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Spiperone; Xylazine; Yohimbine

1995
Determination on functional basis of presynaptic alpha 2-adrenoceptor subtypes in guinea-pig duodenum.
    Neuroscience letters, 1996, May-24, Volume: 210, Issue:1

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Cholinergic Fibers; Duodenum; Electric Stimulation; Gastrointestinal Motility; Guinea Pigs; Idazoxan; Imidazoles; Indoles; Isoindoles; Isoquinolines; Male; Medetomidine; Muscle Contraction; Nordefrin; Norepinephrine; Oxymetazoline; Piperazines; Prazosin; Receptors, Adrenergic, alpha-2; Synaptic Membranes; Vasoconstrictor Agents; Xylazine; Yohimbine

1996
alpha1-adrenoceptors antagonize activated chloride conductance of amphibian skin epithelium.
    Pflugers Archiv : European journal of physiology, 1998, Volume: 436, Issue:6

    Topics: 1-Methyl-3-isobutylxanthine; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Animals; Bufonidae; Calcium; Chloride Channels; Chlorides; Electric Conductivity; Epinephrine; Epithelium; Isoproterenol; Phenylephrine; Prazosin; Rana esculenta; Receptors, Adrenergic, alpha-1; Skin; Xylazine

1998
New 2-substituted 1,2,3,4-tetrahydrobenzofuro[3,2-c]pyridine having highly active and potent central alpha 2-antagonistic activity as potential antidepressants.
    Bioorganic & medicinal chemistry letters, 2000, Jan-03, Volume: 10, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antidepressive Agents; CHO Cells; Clonidine; Cricetinae; Humans; Male; Prazosin; Pyridines; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-2; Xylazine; Yohimbine

2000
Existence of alpha(1A)- and alpha(1B)-adrenoceptor subtypes in canine mandibular alveolar arteries.
    Clinical and experimental pharmacology & physiology, 2001, Volume: 28, Issue:9

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Alveolar Process; Animals; Arteries; Clonidine; Dioxanes; Dogs; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Male; Mandible; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Vasoconstriction; Xylazine; Yohimbine

2001
Effects of xylazine on canine coronary artery vascular rings.
    American journal of veterinary research, 2004, Volume: 65, Issue:4

    Topics: Analysis of Variance; Animals; Coronary Vessels; Dogs; Dose-Response Relationship, Drug; Imidazoles; Muscle Tonus; Prazosin; Vasoconstriction; Xylazine

2004
alpha2B-adrenoceptor agonist ST-91 antagonizes beta2-adrenoceptor-mediated relaxation in rat mesenteric artery rings.
    European journal of pharmacology, 2008, Feb-12, Volume: 580, Issue:3

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic beta-2 Receptor Antagonists; Analysis of Variance; Animals; Aorta; Clonidine; Dose-Response Relationship, Drug; In Vitro Techniques; Isoproterenol; Male; Mesenteric Arteries; Phenylephrine; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta-2; Terbutaline; Vas Deferens; Vasodilation; Xylazine; Yohimbine

2008
Yohimbine antagonises α1A- and α1D-adrenoceptor mediated components in addition to the α2A-adrenoceptor component to pressor responses in the pithed rat.
    European journal of pharmacology, 2012, Mar-15, Volume: 679, Issue:1-3

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Dose-Response Relationship, Drug; Drug Interactions; Ethanolamines; Idazoxan; Male; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Thymine; Vasoconstriction; Xylazine; Yohimbine

2012
Antagonistic effects of atipamezole, yohimbine, and prazosin on xylazine-induced diuresis in clinically normal cats.
    Canadian journal of veterinary research = Revue canadienne de recherche veterinaire, 2014, Volume: 78, Issue:4

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Area Under Curve; Arginine Vasopressin; Cats; Creatinine; Diuresis; Female; Imidazoles; Male; Osmolar Concentration; Prazosin; Random Allocation; Specific Gravity; Xylazine; Yohimbine

2014