xanthenes has been researched along with ly 341495 in 245 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 6 (2.45) | 18.2507 |
2000's | 127 (51.84) | 29.6817 |
2010's | 104 (42.45) | 24.3611 |
2020's | 8 (3.27) | 2.80 |
Authors | Studies |
---|---|
Belagaje, R; Burnett, JP; Johnson, BG; Kingston, AE; Mayne, NG; Ornstein, PL; Schoepp, DD; Wright, RA; Wu, S | 1 |
Arnold, MB; Bleisch, TJ; Ornstein, PL; Schoepp, DD; Wheeler, WJ; Wright, RA | 1 |
Bortolotto, ZA; Collingridge, GL; Doherty, AJ; Fitzjohn, SM; Kingston, AE; Lodge, D; Ornstein, PL; Palmer, MJ; Schoepp, DD | 1 |
Chamberlain, M; Johnson, MP; Kelly, GM | 2 |
Arnold, MB; Johnson, BG; Ornstein, PL; Schoepp, DD; Wheeler, WJ; Wright, RA | 1 |
Bear, MF; Huber, KM; Roder, JC; Sawtell, NB | 1 |
Aghajanian, GK; Marek, GJ; Monn, JA; Schoepp, DD; Wright, RA | 1 |
Bear, MF; Huber, KM; Kayser, MS | 1 |
Adam, G; Kratzeisen, C; Lundstrom, K; Malherbe, P; Mutel, V; Ohresser, S; Schweitzer, C; Stadler, H; Wichmann, J; Woltering, T | 1 |
Cartmell, J; Monn, JA; Perry, KW; Salhoff, CR; Schoepp, DD | 1 |
Cartmell, J; Monn, JA; Schoepp, DD | 1 |
Gewirtz, JC; Marek, GJ | 1 |
Ducarre, JM; Kemp, JA; Kew, JN; Mutel, V; Pflimlin, MC | 1 |
Arnold, MB; Ornstein, PL; Schoepp, DD; Wheeler, WJ; Wright, RA | 2 |
Bradley, SR; Conn, PJ; Marino, MJ; Wittmann, M | 1 |
Cirone, J; Salt, TE | 1 |
Glitsch, MD; Jack, JJ | 1 |
Chamberlain, M; Johnson, MP; Kelly, G | 1 |
Abraini, JH; David, HN | 1 |
Bear, MF; Dong, X; Fallon, JR; Huber, KM; Philpot, BD; Snyder, EM | 1 |
Carlisle, HJ; O'Dell, TJ; Watabe, AM | 1 |
Cai, Z; Lin, S; Rhodes, PG | 1 |
Alonso, G; Bockaert, J; Chaumont, S; Manzoni, OJ; Robbe, D | 1 |
Cirone, J; Pothecary, CA; Salt, TE; Turner, JP | 1 |
Chen, AC; Duman, RC; Gewirtz, JC; Marek, GJ; Terwilliger, R | 1 |
Griffey, KI; Schoepp, DD; Tizzano, JP | 1 |
Frondaroli, A; Grassi, S; Pettorossi, VE | 2 |
Bleisch, TJ; Johnson, BG; Kingston, AE; Ornstein, PL; Schoepp, DD; Sørensen, US; Wright, RA | 1 |
George, CA; Johnson, MP; Nisenbaum, ES; Nisenbaum, LK; Zhai, J; Zhai, Y | 1 |
Arcella, A; Battaglia, G; Bruno, V; Calogero, A; D'Onofrio, M; Lombari, V; Ngomba, RT; Nicoletti, F; Ragona, G | 1 |
Laruelle, M; Mozley, PD; Schmidt, ME; Schoepp, DD; Sultana, A; Waterhouse, RN; Wheeler, WJ | 1 |
Bandrowski, AE; Huguenard, JR; Prince, DA | 1 |
Losonczy, A; Nusser, Z; Somogyi, P | 1 |
Howson, PA; Jane, DE | 1 |
Anderson, JJ; Baccei, CS; Bristow, LJ; Campbell, UC; Correa, LD; Lorrain, DS; Pinkerton, AB; Rodriguez, DE; Rowe, B; Schaffhauser, H; Varney, MA; Vernier, JM | 1 |
Battaglia, G; Biagioni, F; Bruno, V; Busceti, CL; Fornai, F; Nicoletti, F; Paparelli, A; Pontarelli, F; Ruggieri, S | 1 |
Keller, A; Sanabria, ER; Slusher, BS; Wozniak, KM | 1 |
Conway, MW; Heron-Maxwell, C; Monn, JA; O'Neill, MF; Ornstein, P | 1 |
Bain, G; Bristow, LJ; Chavez-Noriega, LE; Daggett, LP; Jachec, C; Morales, S; Pinkerton, AB; Rao, SP; Rowe, BA; Schaffhauser, H; Varney, MA; Vernier, JM; Yin, R | 1 |
Johnson, SW; Shen, KZ | 1 |
Hashimoto, K; Iyo, M; Koike, K; Koizumi, H; Komatsu, N; Kumakiri, C; Ohgake, S; Okamura, N; Shimizu, E | 1 |
Brotchie, JM; Brown, TM; Fitzjohn, SM | 1 |
Perry, KW; Schoepp, DD; Swanson, CJ | 1 |
Gregory, ML; Kalivas, PW; Owens, RW; Stech, NE | 1 |
Kalivas, PW; Tang, XC | 1 |
Rieke, F; Sampath, AP | 1 |
Anwyl, R; Rowan, MJ; Wu, J | 1 |
Irifune, M; Nishikawa, T; Ohnishi, Y; Sato, T; Tanaka, K; Teramoto, T | 1 |
Hsu, MA; Rasmussen, K; Vandergriff, J | 1 |
Gereau, RW; Yang, D | 1 |
Chen, HX; Roper, SN | 1 |
Adam, G; Ballard, TM; Higgins, GA; Kemp, JA; Kew, JN; Mutel, V; Nakanishi, S; Richards, JG; Woltering, T | 1 |
Capogna, M; Dalezios, Y; Ferraguti, F; Kogo, N; Shigemoto, R; Somogyi, P | 1 |
Capogna, M | 1 |
Irifune, M; Nishikawa, T; Ohnishi, Y; Sato, T; Tanaka, K | 1 |
DiGregorio, DA; Nielsen, TA; Silver, RA | 1 |
Duvoisin, RM; Grandes, P; Kushmerick, C; Price, GD; Puente, N; Renden, R; Taschenberger, H; von Gersdorff, H; Wadiche, JI | 1 |
Grajkowska, E; Hirasawa, S; Kozikowski, A; Neale, JH; Wroblewska, B; Wroblewski, J; Yamamoto, T; Zhou, J | 1 |
Freund, TF; Hájos, N; Pálhalmi, J; Paulsen, O | 1 |
Campbell, IG; Darchia, N; Feinberg, I; Hsieh, KC; Schoepp, DD | 1 |
Gebhardt, C; Heinemann, U; Iserhot, C; Schmitz, D | 1 |
Alagarsamy, S; Bough, KJ; Conn, PJ; Dingledine, R; Doherty, JJ; Mott, DD | 1 |
Neale, SA; Salt, TE; Thompson, H | 1 |
Bringmann, A; Klaus, C; Reichenbach, A; Rillich, K; Syková, E; Uckermann, O; Ulbricht, E; Vargová, L; Weick, M; Wiedemann, P | 1 |
Bickel, DJ; Burno, M; Chen, TB; Clements, MK; Conn, PJ; Duggan, ME; Jacobson, MA; Kinney, GG; Lemaire, W; Lindsley, CW; O'Brien, JA; Pettibone, DJ; Smith, S; Sur, C; Tiller, PR; Williams, DL; Wisnoski, DD | 1 |
Baez, M; Koester, A; Linden, AM; Schoepp, DD; Shannon, H; Yu, JL | 1 |
Druga, R; Folbergrová, J; Haugvicová, R; Kubová, H; Mares, P; Otáhal, J | 1 |
Alexander, GM; Godwin, DW | 2 |
Huber, KM; Nosyreva, ED | 1 |
Chaki, S; Karasawa, J; Kawashima, N; Nakazato, A; Okuyama, S; Shimazaki, T; Yasuhara, A | 1 |
Battaglia, G; Canudas, AM; Del Bianco, P; Matrisciano, F; Melchiorri, D; Molinaro, G; Ngomba, RT; Nicoletti, F; Panaccione, I; Riozzi, B; Scaccianoce, S; Tatarelli, R | 1 |
Abeniyi, OA; Conn, PJ; Poisik, O; Raju, DV; Rodriguez, A; Smith, Y; Verreault, M | 1 |
Capogna, M; Karayannis, T; Pál, BZ; Price, CJ | 1 |
Kalivas, PW; McFarland, K; Melendez, RI; Moran, MM; Seamans, JK | 1 |
Bergeron, M; Linden, AM; Schoepp, DD | 1 |
Battaglia, G; Biagioni, F; Bruno, V; Casciato, S; Ngomba, RT; Nicoletti, F; van Luijtelaar, EL; Willems-van Bree, E | 1 |
Arcella, A; Battaglia, G; Bruno, V; Carpinelli, G; Casolini, P; D'Onofrio, M; Giangaspero, F; Ngomba, RT; Nicoletti, F; Santoro, F | 1 |
Alger, BE; Jones, LM; Karnup, SV; Karson, MA; Reich, CG | 1 |
Ebinger, G; Hachimi-Idrissi, S; Michotte, Y; Sarre, S; Van Hemelrijck, A | 1 |
Daniel, WA; Kos, T; Kozela, E; Popik, P; Slusher, BS; Wojcikowski, J; Wozniak, KM; Wrobel, M | 1 |
Kitai, ST; Wang, L; Xiang, Z | 1 |
Bae, HB; Choi, Jl; Chung, SS; Chung, ST; Jeong, CY; Jeong, SW; Kim, SJ; Yoo, KY; Yoon, MH | 1 |
Ennis, M; Hayar, A; Heinbockel, T; Zhu, M | 1 |
Bzdega, T; Neale, JH; Olszewski, RT; Wegorzewska, IN; Wroblewska, B | 1 |
Daly, CA; Huber, KM; Volk, LJ | 1 |
Anwyl, R; Harney, SC; Rowan, M | 1 |
Chi, H; Jang, JK; Kim, JH; Vezina, P | 1 |
Anderson, H; Cottrell, DF; Fleetwood-Walker, SM; Garry, EM; Mitchell, R; Proudfoot, CJ; Robertson, DC; Rosie, R | 1 |
Marek, GJ; Zhang, C | 1 |
Chaki, S; Iijima, M; Ito, A; Shimazaki, T | 1 |
Liechti, ME; Markou, A | 1 |
Markou, A; Semenova, S | 1 |
Bespalov, A; Gross, G; Harich, S; Jongen-Rêlo, AL; Schoemaker, H; van Gaalen, M | 1 |
Lu, Y | 1 |
Battaglia, G; Beraudi, A; Biagioni, F; Bruno, V; Nicoletti, F; Poli, A; Rampello, L | 1 |
Griffey, KI; Johnson, BG; Knitowski, KM; McKinzie, DL; Monn, JA; Perry, KW; Rorick-Kehn, LM; Salhoff, CR; Schoepp, DD; Tizzano, JP; Witkin, JM | 1 |
Brady, AE; Conn, PJ; Da Costa, H; Hemstapat, K; Luo, Q; Niswender, CM; Nong, Y; Tamagnan, GD | 1 |
Mateo, Z; Porter, JT | 1 |
Chung, LY; Kim, U | 1 |
Girardi, P; Giusti, P; Gruber, SH; Iacovelli, L; Mathé, AA; Matrisciano, F; Nicoletti, F; Panaccione, I; Tatarelli, R; Zusso, M | 1 |
Baker, DA; Haroutunian, V; Kristiansen, LV; Madayag, A; Meador-Woodruff, JH; Raju, I | 1 |
Bédard, PJ; Bélanger, N; Calon, F; Di Paolo, T; Dridi, M; Grégoire, L; Hadj Tahar, A; Morissette, M; Samadi, P | 1 |
Ayala, JE; Conn, PJ; Johnson, KA; Kim, C; Luo, Q; Niswender, CM; Weaver, CD | 1 |
Ayala, JE; Banko, JL; Conn, PJ; Luo, Q; Niswender, CM | 1 |
Cleland, TA; Linster, C; Magidson, PD; McNamara, AM; Wilson, DA | 1 |
Anwyl, R; Harney, S; Rowan, MJ; Wu, J | 1 |
Kai, T; Shichida, Y; Terakita, A; Yamashita, T | 1 |
Carlton, SM; Du, J; Zhou, S | 2 |
Arcella, A; Battaglia, G; Carpinelli, G; Ciceroni, C; De Maria, R; Giangaspero, F; Mastrantoni, E; Melchiorri, D; Mosillo, P; Nicoletti, F; Oliva, MA; Pallini, R; Ricci-Vitiani, L; Sale, P; Santoro, F | 1 |
Conn, PJ; Sheffler, DJ | 1 |
Bespalov, AY; Gross, G; Mezler, M; Schoemaker, H; Sukhotina, IA; van Gaalen, MM; Wicke, K | 1 |
Steketee, JD; Xie, X | 1 |
Jang, JK; Kim, JH; Yoon, HS | 1 |
Abrahamsson, T; Gustafsson, B; Hanse, E | 1 |
Corsi, M; Corti, C; Ferraguti, F; Herdy, S; Hetzenauer, A; Singewald, N | 1 |
Martina, M; Mugnaini, E; Nunzi, MG; Russo, MJ; Yau, HJ | 1 |
Poo, MM; Xu, C; Zhang, XH; Zhao, MX | 1 |
Andreasen, M; Nedergaard, S; Skov, J | 1 |
Busceti, CL; Chiechio, S; Copani, A; Drago, F; Gereau, RW; Morales, ME; Nicoletti, F; Zammataro, M | 1 |
Calon, F; Di Paolo, T; Grégoire, L; Hornykiewicz, O; Rajput, A; Rajput, AH; Samadi, P | 1 |
Akiba, Y; Baker, H; Cave, JW; Estevez, AG; Huerta, PT; Sasaki, H | 1 |
Feng, Y; Li, H; Shi, J; Sun, ZS; Zhang, J; Zhang, T | 1 |
Battaglia, G; Bruno, V; Curto, M; Di Menna, L; Molinaro, G; Nicoletti, F; Pallottino, S; Riozzi, B; Traficante, A | 1 |
Gregg, RG; Heimel, JA; Kamermans, M; Nawy, S; Peachey, NS; Shen, Y | 1 |
Johnson, BG; Korpi, ER; Linden, AM; Schoepp, DD; Trokovic, N | 1 |
Kinouchi, H; Sugita, M; Yoshioka, H | 1 |
Dietrich, D; Wostrack, M | 1 |
Ashby, CR; Gardner, EL; Li, J; Peng, XQ; Slusher, BS; Thomas, A; Wozniak, K; Xi, ZX | 1 |
Belluardo, N; Bonomo, A; Di Liberto, V; Frinchi, M; Mudò, G | 1 |
Chen, WC; Mei, B; Sun, ZW; Zhang, L; Zhu, SJ | 1 |
Choi, S; Hong, I; Kim, J; Lee, S; Song, B | 1 |
Ehrlich, ME; Fraser, PE; Gandy, S; Kim, SH; St George-Hyslop, PH; Westaway, D | 1 |
Amitai, N; Markou, A | 1 |
Chaki, S; Kambe, D; Karasawa, J; Kotani, M | 1 |
Fujita, Y; Hashimoto, K; Slusher, BS; Takatsu, Y; Tsukamoto, T | 1 |
Battaglia, G; Britton, TC; Bruno, V; Cannella, M; Caraci, F; Copani, A; Drago, F; Giuffrida, ML; Heinz, BA; Merlo, S; Molinaro, G; Nicoletti, F; Nisenbaum, ES; Riozzi, B; Sortino, MA; Traficante, A; Wang, X | 1 |
Berridge, KC; Richard, JM | 1 |
Andreasen, M; Hablitz, JJ; Nedergaard, S; Skov, J | 1 |
Beveridge, TJ; Nader, MA; Porrino, LJ; Smith, HR | 1 |
Rushlow, WJ; Sutton, LP | 1 |
Coiret, G; Corsi, M; Corti, C; Gerber, U; Grewe, BF; Helmchen, F; Mateos, JM; Ster, J | 1 |
Bojang, P; Furukawa, T; Gregg, RG; Koike, C; Nawy, S; Pearring, JN; Shen, Y | 1 |
Chaban, V; Li, J; McDonald, JS; Micevych, P; Rapkin, A | 1 |
Ma, H; Yang, K | 1 |
Carlton, SM; Du, J; Govea, R; Zhou, S | 1 |
Chaki, S; Iijima, M; Koike, H | 3 |
Conn, PJ; Johnson, KA; Niswender, CM; Xiang, Z | 1 |
Gilley, JA; Kernie, SG | 1 |
Duman, RS; Dwyer, JM; Lepack, AE | 1 |
Brownell, AL; Kuruppu, D; Wang, JQ; Zhang, Z | 1 |
Dong, E; Sanford, LD; Wellman, LL; Yang, L | 1 |
Copeland, CS; Neale, SA; Salt, TE | 1 |
Bortolotto, ZA; Collingridge, GL; Lodge, D; Lucas, SJ | 1 |
Carroll, RC; Nawy, S; Rampino, MA; Shen, Y | 1 |
Kaffe, E; Markou, A; Pitsikas, N | 1 |
Raiteri, L; Raiteri, M; Romei, C | 1 |
Bojang, P; Furukawa, T; Goldberg, AF; Gregg, RG; Hirschtritt, ME; Koike, C; McCall, MA; Nawy, S; Nishina, PM; Peachey, NS; Pearring, JN; Ray, TA; Shen, Y; Sturgill-Short, G | 1 |
Bae, SA; Bischoff, F; Guo, N; Huang, Y; Hwang, DR; Laruelle, M; Lesage, AS; Narendran, R | 1 |
Breustedt, J; Kintscher, M; Miceli, S; Schmitz, D; Wozny, C | 1 |
Aston-Jones, G; Fallon, RV; Hensley-Simon, M; Kalivas, PW; LaLumiere, RT; Mahler, SV; Tahsili-Fahadan, P; Thomas, C | 1 |
Chaki, S; Fukumoto, K; Iijima, M; Koike, H | 1 |
Kaba, H; Murata, Y; Nakanishi, S; Okutani, F; Shinohara, Y; Taniguchi, M; Yokoi, M | 1 |
Arcella, A; Battaglia, G; Bonelli, M; Ciceroni, C; De Maria, R; Larocca, LM; Laurenza, M; Mastrantoni, E; Melchiorri, D; Niccolini, C; Nicoletti, F; Pallini, R; Ricci-Vitiani, L; Spinsanti, P; Traficante, A | 1 |
Bouwalerh, H; Maccari, S; Mairesse, J; Marrocco, J; Morley-Fletcher, S; Ngomba, RT; Nicoletti, F; Pittaluga, A; Silletti, V; Summa, M; Van Camp, G | 1 |
Bortolotto, ZA; Collett, VJ; Collingridge, GL; Fang, G; Jane, DE; Lodge, D; Mercier, MS; Nicolas, CS | 1 |
González-Maeso, J; Holloway, T; Moreno, JL; Rayannavar, V; Sealfon, SC | 1 |
Barone, Y; Battaglia, G; Caruso, A; Lionetto, L; Mathé, AA; Matrisciano, F; Nasca, C; Nicoletti, F; Pittaluga, A; Scaccianoce, S; Simmaco, M; Xenos, D | 1 |
Bannister, N; Bortolotto, ZA; Ceolin, L; Collingridge, GL; Fitzjohn, SM; Hanna, L; Jane, DE; Kritikos, M; Lodge, D; Lucas, SJ; Mercier, MS; Sherwood, JL; Tidball, P; Volianskis, A | 1 |
de Groat, WC; Mally, AD; Matsuta, Y; Roppolo, JR; Shen, B; Tai, C; Wang, J; Zhang, F | 1 |
Gao, WJ; Li, F; Li, YC; Snyder, MA; Wang, H; Wang, MJ | 1 |
Chaki, S; Hikichi, H; Kaku, A; Karasawa, J | 1 |
Carrillo, V; Dubisz, E; Gulzar, H; Mahajan, SS; Morgan, D; Yelskaya, Z | 1 |
Di Paolo, T; Gasparini, F; Gomez-Mancilla, B; Grégoire, L; Morin, N; Morissette, M | 1 |
Ahnaou, A; Andrés, JI; Atack, JR; Biesmans, I; Cid, JM; Dautzenberg, FM; Drinkenburg, W; Langlois, X; Lavreysen, H; Lütjens, R; Macdonald, G; Megens, A; Peeters, L; te Riele, P; Trabanco, AA; Van der Linden, I; Wintmolders, C | 1 |
Anwyl, R; Chang, L; Chen, X; Lin, R; Wang, C; Wang, Q; Wei, X; Xu, S; Zhang, J | 1 |
Caron, MG; Jacobsen, JP; Jørgensen, CV; Klein, AB; Knudsen, GM; Mikkelsen, JD | 1 |
Curry, RJ; Dinh, EH; Hamlet, WR; Liu, YW; Lu, Y; Shi, W; Tang, ZQ | 1 |
Chaki, S; Fukumoto, K; Iijima, M | 2 |
Shu, H; Song, Y; Wang, B; Yang, H; Zhang, C; Zhou, K; Zhou, W | 1 |
Chan, MH; Chen, HH; Chiang, CC; Chiu, HY; Lee, MY | 1 |
Fu, K; Furukawa-Hibi, Y; Iegaki, N; Ishikawa, Y; Miyamoto, Y; Muramatsu, S; Nabeshima, T; Nitta, A; Sato, K; Sumi, K; Uno, K | 1 |
DiRaddo, JO; Grajkowska, E; Hathaway, HA; Liotta, DC; Miller, EJ; Wolfe, BB; Wroblewska, B; Wroblewski, JT | 1 |
Ahnaou, A; Drinkenburg, WH; Ver Donck, L | 1 |
Chaki, S; Koike, H | 1 |
Callado, LF; Díez-Alarcia, R; González-Maeso, J; Meana, JJ; Miranda-Azpiazu, P; Morentin, B; Muguruza, C | 1 |
Borsotto, M; Bourcier-Lucas, C; Haddjeri, N; Heurteaux, C; Kanzari, A; Lucas, G; Moha ou Maati, H; Veyssiere, J | 1 |
Bai, G; Cao, DY; Ji, Y; Traub, RJ | 1 |
Kärkkäinen, O; Kautiainen, H; Kupila, J; Laukkanen, V; Storvik, M; Tiihonen, J | 1 |
Benn, A; Robinson, ES | 1 |
Karimi, SA; Komaki, A; Salehi, I; Sarihi, A; Shahidi, S | 1 |
Asseri, KA; MacLeod, BA; Puil, E; Schwarz, SK | 1 |
Battaglia, G; Cruccu, G; Di Stefano, G; Lattanzi, R; Nicoletti, F; Notartomaso, S; Pasquale, E; Piroso, S; Truini, A | 1 |
Kiritoshi, T; Neugebauer, V | 1 |
Ago, Y; Hasebe, S; Hashimoto, H; Matsuda, T; Nishiyama, S; Oka, S; Onaka, Y; Takuma, K | 1 |
An, B; Choi, S; Hong, I; Kim, J; Lee, S; Park, K; Park, S | 1 |
Besheer, J; Fisher, KR; Frisbee, S; Jaramillo, AA; Randall, PA | 1 |
Bollands, M; Jones, S; Morris, PG; Wild, AR | 1 |
Barker, JM; Chandler, LJ; Lench, DH | 1 |
Dean, B; Gibbons, A; Hopper, S; McOmish, CE; Pavey, G; Scarr, E; Udawela, M | 1 |
Carlsson, HA; Hesslow, G; Johansson, F; Rasmussen, A; Yeo, CH | 1 |
Call, CL; Hyson, RL | 1 |
Carter, G; Johnson, B; Li, X; Mitchell, SN; Monn, JA; Overshiner, C; Rasmussen, K; Rorick-Kehn, LM; Schoepp, DD; Witkin, JM | 1 |
Brański, P; Pałucha-Poniewiera, A; Pilc, A; Pochwat, B; Podkowa, K | 1 |
Bai, G; Cao, DY; Ji, Y; Karpowicz, JM; Traub, RJ | 1 |
Ahn, G; Bing, SJ; Cho, IH; Cho, J; Ha, D; Herath, KH; Jee, Y; Jo, SA; Kim, A; Kim, J; Yu, HS | 1 |
Ali, I; Amhaoul, H; Boets, S; Dedeurwaerdere, S; Janssens, P; Langlois, X; Van Eetveldt, A | 1 |
Lenda, T; Pałucha-Poniewiera, A; Pilc, A; Podkowa, A; Podkowa, K; Sałat, K | 1 |
Bang, E; Duman, RS; Dwyer, JM; Lee, B; Lepack, AE | 1 |
Cannella, LA; Gregg, RA; Hicks, C; Nayak, SU; Rawls, SM; Reitz, AB; Schena, GJ; Smith, GR; Tallarida, CS | 1 |
Chatton, JY; Rimmele, TS; Rocher, AB; Wellbourne-Wood, J | 1 |
Chen, W; Lai, M; Liu, H; Mei, D; Zhang, F; Zhou, W; Zhu, H | 1 |
Bermudez, I; García-Bea, A; Harrison, PJ; Lane, TA | 1 |
Grove, JCR; Koren, D; Wei, W | 1 |
Blaabjerg, M; Bogetofte, H; Dindler, A; Kamand, M; Meyer, M | 1 |
Andersson, M; Brandt, I; Karlsson, O; Pierozan, P | 1 |
Canella, R; Fesce, R; Martini, M; Rossi, ML; Rubbini, G | 1 |
Doornbos, MLJ; Heitman, LH; IJzerman, AP; Lavreysen, H; Tresadern, G; Vermond, SC | 1 |
Abe, M; Hiroshima, M; Murata, M; Sako, Y; Shichida, Y; Togashi, Y; Ueda, M; Yamashita, T; Yanagawa, M | 1 |
da Silva, EN; Dias, MB; Gargaglioni, LH; Horta-Júnior, JAC; Rodrigues, LTC | 1 |
Ago, Y; Goda, H; Mizuguchi, H; Morikawa, N; Sakurai, F; Tachibana, M | 1 |
Doornbos, MLJ; Heitman, LH | 1 |
Alexander, L; Cardinal, RN; Clarke, HF; Cockcroft, GJ; Dalley, JW; Quah, SKL; Roberts, AC; Santangelo, AM; Shiba, Y; Wallis, CU; Xia, J; Zeredo, JL | 1 |
Pałucha-Poniewiera, A; Pilc, A; Podkowa, K | 1 |
Georgiou, P; Gould, TD; Highland, JN; Zanos, P | 1 |
Kammermeier, PJ; McCullock, TW | 1 |
Eastwood, BJ; Gilmour, G; Hanley, N; Loomis, S; McCarthy, A; Paulissen, J; Wafford, KA | 1 |
Haddar, M; Hamatani, K; Muramatsu, SI; Nitta, A; Uno, K | 1 |
Mazzitelli, M; Neugebauer, V | 1 |
Fujiwara, T; Miyanishi, H; Miyazaki, T; Muramatsu, SI; Nitta, A; Sodeyama, K; Uno, K | 1 |
Choi, AJ; Hien, LT; Kim, SH; Lee, JG; Park, MK; Park, SW; Seo, MK; Seog, DH | 1 |
Du, H; Jiang, HD; Jiang, HJ; Ling, Y; Shen, HW; Wang, GZ; Wu, T; Xu, L; Yang, SY; Yu, ZP; Zhang, XQ; Zhang, ZY; Zhao, QQ | 1 |
Pałucha-Poniewiera, A; Podkowa, K; Rafało-Ulińska, A | 1 |
Jing, XY; Li, LF; Li, ZL; Liu, YJ; Wang, Y; Zou, HW | 1 |
Beck, J; Behringer, SP; Follo, M; Garrelfs, N; Goeldner, JM; Hannibal, L; Heiland, DH; Hofmann, UG; Joseph, K; Kueckelhaus, J; Maier, JP; Pfeifer, D; Ravi, VM; Schnell, O; Sun, N; von Ehr, J; Walch, AK; Will, P | 1 |
Cao, AM; Fatemi, F; Margeat, E; Pin, JP; Quast, RB; Rondard, P | 1 |
Guo, C; Huson, V; Macosko, EZ; Regehr, WG | 1 |
Jeong, S; Lee, JA; Lee, JG; Park, SW; Seo, MK; Seog, DH | 1 |
245 other study(ies) available for xanthenes and ly 341495
Article | Year |
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LY341495 is a nanomolar potent and selective antagonist of group II metabotropic glutamate receptors.
Topics: Amino Acids; Animals; Cell Line; Colforsin; Cyclic AMP; Excitatory Amino Acid Antagonists; Humans; Prosencephalon; Rats; Receptors, Metabotropic Glutamate; Xanthenes | 1998 |
[3H]LY341495, a highly potent, selective and novel radioligand for labeling Group II metabotropic glutamate receptors.
Topics: Amino Acids; Animals; Excitatory Amino Acid Antagonists; Prosencephalon; Radioligand Assay; Rats; Receptors, Metabotropic Glutamate; Tritium; Xanthenes | 1998 |
The potent mGlu receptor antagonist LY341495 identifies roles for both cloned and novel mGlu receptors in hippocampal synaptic plasticity.
Topics: Aging; Amino Acids; Animals; Binding, Competitive; Cell Line; CHO Cells; Cloning, Molecular; Cricetinae; Cycloleucine; Excitatory Amino Acid Antagonists; Glutamic Acid; Glycine; Hippocampus; Humans; In Vitro Techniques; Long-Term Potentiation; Neuronal Plasticity; Rats; Receptors, Metabotropic Glutamate; Recombinant Proteins; Resorcinols; Transfection; Xanthenes | 1998 |
Phosphoinositide hydrolysis in vivo with group I metabotropic glutamate receptor agonists.
Topics: Amino Acids; Animals; Brain Chemistry; Cerebellum; Cycloleucine; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Glycine; Hippocampus; Hydrolysis; Injections, Intraventricular; Male; Neuroprotective Agents; Phenylacetates; Phosphatidylinositols; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Resorcinols; Tritium; Type C Phospholipases; Xanthenes | 1999 |
[3H]-LY341495 as a novel antagonist radioligand for group II metabotropic glutamate (mGlu) receptors: characterization of binding to membranes of mGlu receptor subtype expressing cells.
Topics: Amino Acids; Animals; Binding, Competitive; Calcium; Cell Membrane; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Humans; Kinetics; Radioligand Assay; Receptors, Metabotropic Glutamate; Recombinant Proteins; Transfection; Tritium; Xanthenes | 1999 |
Induction of NMDA receptor-dependent long-term depression in visual cortex does not require metabotropic glutamate receptors.
Topics: Amino Acids; Animals; Cycloleucine; Depression, Chemical; Excitatory Amino Acid Antagonists; Hydrolysis; In Vitro Techniques; Methoxyhydroxyphenylglycol; Mice; Mice, Knockout; Neuronal Plasticity; Phosphatidylinositols; Rats; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Synaptosomes; Visual Cortex; Xanthenes | 1999 |
Physiological antagonism between 5-hydroxytryptamine(2A) and group II metabotropic glutamate receptors in prefrontal cortex.
Topics: Amino Acids; Animals; Autoradiography; Bridged Bicyclo Compounds; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Free Radical Scavengers; Glutamic Acid; Humans; In Vitro Techniques; Male; Membrane Potentials; Prefrontal Cortex; Protein Binding; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Receptors, Presynaptic; Serotonin; Xanthenes | 2000 |
Blockade of pilocarpine-induced cerebellar phosphoinositide hydrolysis with metabotropic glutamate antagonists: evidence for an indirect control of granule cell glutamate release by muscarinic agonists.
Topics: Amino Acids; Animals; Cerebellum; Corpus Striatum; Frontal Lobe; Hippocampus; Hydrolysis; Lithium; Male; Muscarinic Agonists; Phosphatidylinositols; Pilocarpine; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M2; Receptors, Metabotropic Glutamate; Receptors, Muscarinic; Scopolamine; Xanthenes | 2000 |
Role for rapid dendritic protein synthesis in hippocampal mGluR-dependent long-term depression.
Topics: Amino Acids; Animals; Anisomycin; Dendrites; Electric Stimulation; Excitatory Amino Acid Antagonists; Hippocampus; Methoxyhydroxyphenylglycol; Nerve Tissue Proteins; Neural Inhibition; Protein Biosynthesis; Protein Synthesis Inhibitors; Rats; Receptors, Metabotropic Glutamate; RNA, Messenger; Synaptic Transmission; Xanthenes | 2000 |
Characterization of [(3)H]-LY354740 binding to rat mGlu2 and mGlu3 receptors expressed in CHO cells using semliki forest virus vectors.
Topics: Amino Acids; Animals; Binding, Competitive; Bridged Bicyclo Compounds; Cell Membrane; Chlorides; CHO Cells; Cricetinae; DNA, Recombinant; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Gene Expression; Genetic Vectors; Glutamic Acid; Guanosine 5'-O-(3-Thiotriphosphate); Kinetics; Rats; Receptors, Metabotropic Glutamate; Semliki forest virus; Tritium; Xanthenes; Zinc Compounds | 2000 |
The potent, selective mGlu2/3 receptor agonist LY379268 increases extracellular levels of dopamine, 3,4-dihydroxyphenylacetic acid, homovanillic acid, and 5-hydroxyindole-3-acetic acid in the medial prefrontal cortex of the freely moving rat.
Topics: 3,4-Dihydroxyphenylacetic Acid; Amino Acids; Animals; Bridged Bicyclo Compounds, Heterocyclic; Clozapine; Dopamine; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Homovanillic Acid; Hydroxyindoleacetic Acid; Kinetics; Male; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Xanthenes | 2000 |
The mGlu(2/3) receptor agonist LY379268 selectively blocks amphetamine ambulations and rearing.
Topics: Amino Acids; Amphetamine; Animals; Bridged Bicyclo Compounds, Heterocyclic; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Male; Motor Activity; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Stereotyped Behavior; Xanthenes | 2000 |
Behavioral evidence for interactions between a hallucinogenic drug and group II metabotropic glutamate receptors.
Topics: Amino Acids; Amphetamines; Animals; Behavior, Animal; Bridged Bicyclo Compounds; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Hallucinogens; Male; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Metabotropic Glutamate; Receptors, Serotonin; Xanthenes | 2000 |
Activity-dependent presynaptic autoinhibition by group II metabotropic glutamate receptors at the perforant path inputs to the dentate gyrus and CA1.
Topics: Amino Acids; Animals; Dentate Gyrus; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Hippocampus; In Vitro Techniques; Neural Pathways; Rats; Receptors, Metabotropic Glutamate; Xanthenes | 2001 |
Binding of [3H](2S,1'S,2'S)-2-(9-xanthylmethyl)-2-(2'-carboxycyclopropyl) glycine ([3H]LY341495) to cell membranes expressing recombinant human group III metabotropic glutamate receptor subtypes.
Topics: Amino Acids; Binding, Competitive; Cell Membrane; Excitatory Amino Acid Antagonists; Humans; Kinetics; Radioligand Assay; Receptors, Metabotropic Glutamate; Recombinant Proteins; Substrate Specificity; Tritium; Xanthenes | 2000 |
Activation of group III mGluRs inhibits GABAergic and glutamatergic transmission in the substantia nigra pars reticulata.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Amino Acids; Aminobutyrates; Animals; Bicuculline; Drug Design; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Glycine; Kainic Acid; Nerve Tissue Proteins; Patch-Clamp Techniques; Phosphoserine; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, GABA-A; Receptors, Metabotropic Glutamate; Receptors, Presynaptic; Substantia Nigra; Xanthenes | 2001 |
Group II and III metabotropic glutamate receptors contribute to different aspects of visual response processing in the rat superior colliculus.
Topics: Amino Acids; Animals; Bridged Bicyclo Compounds; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Habituation, Psychophysiologic; Rats; Rats, Inbred Strains; Receptors, Metabotropic Glutamate; Superior Colliculi; Visual Perception; Xanthenes | 2001 |
[3H]LY341495 binding to group II metabotropic glutamate receptors in rat brain.
Topics: Amino Acids; Animals; Autoradiography; Binding, Competitive; Brain; Excitatory Amino Acid Antagonists; In Vitro Techniques; Kinetics; Male; Membranes; Protein Binding; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Xanthenes | 2001 |
Evidence that glutamate acting on presynaptic type-II metabotropic glutamate receptors alone does not fully account for the phenomenon of depolarisation-induced suppression of inhibition in cerebellar Purkinje cells.
Topics: Amino Acids; Animals; Excitatory Amino Acid Antagonists; Glutamic Acid; In Vitro Techniques; Neural Inhibition; Purkinje Cells; Rats; Receptors, Metabotropic Glutamate; Receptors, Presynaptic; Signal Transduction; Xanthenes | 2001 |
Changes in rat serum corticosterone after treatment with metabotropic glutamate receptor agonists or antagonists.
Topics: Adrenalectomy; Adrenocorticotropic Hormone; Amino Acids; Animals; Benzoates; Bridged Bicyclo Compounds; Corticosterone; Cycloleucine; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Glycine; Male; Neuroprotective Agents; Paraventricular Hypothalamic Nucleus; Phenylacetates; Propionates; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols; Xanthenes | 2001 |
Differential modulation of the D1-like- and D2-like dopamine receptor-induced locomotor responses by group II metabotropic glutamate receptors in the rat nucleus accumbens.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amino Acids; Animals; Dopamine Agonists; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Male; Motor Activity; Nucleus Accumbens; Proline; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Metabotropic Glutamate; Xanthenes | 2001 |
Internalization of ionotropic glutamate receptors in response to mGluR activation.
Topics: Amino Acids; Animals; Cells, Cultured; Cycloheximide; Dendrites; Electrophysiology; Endocytosis; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glycine; Hippocampus; Immunohistochemistry; In Vitro Techniques; Methoxyhydroxyphenylglycol; Neurons; Protein Synthesis Inhibitors; Rats; Rats, Long-Evans; Receptors, AMPA; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Resorcinols; Synapses; Synapsins; Synaptic Transmission; Xanthenes | 2001 |
Postsynaptic induction and presynaptic expression of group 1 mGluR-dependent LTD in the hippocampal CA1 region.
Topics: 4-Aminopyridine; Amino Acids; Animals; Calcium Signaling; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Hippocampus; Long-Term Potentiation; Male; Methoxyhydroxyphenylglycol; Mice; Mice, Inbred C57BL; Neural Inhibition; Organ Culture Techniques; Potassium Channel Blockers; Presynaptic Terminals; Receptors, Metabotropic Glutamate; Synaptic Transmission; Xanthenes | 2002 |
Neuroprotective effects of N-acetylaspartylglutamate in a neonatal rat model of hypoxia-ischemia.
Topics: Amino Acids; Animals; Animals, Newborn; Brain; Carboxypeptidases; Cyclic AMP; Cycloleucine; Dipeptides; Disease Models, Animal; Dose-Response Relationship, Drug; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Glutamate Carboxypeptidase II; Hippocampus; Hypoxia-Ischemia, Brain; Neurons; Neuroprotective Agents; Organophosphorus Compounds; Propionates; Rats; Rats, Sprague-Dawley; Xanthenes | 2002 |
Role of p/q-Ca2+ channels in metabotropic glutamate receptor 2/3-dependent presynaptic long-term depression at nucleus accumbens synapses.
Topics: Amino Acids; Animals; Bridged Bicyclo Compounds; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Channels, P-Type; Calcium Channels, Q-Type; Cyclic AMP-Dependent Protein Kinases; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Neural Inhibition; Neuronal Plasticity; Nucleus Accumbens; Patch-Clamp Techniques; Presynaptic Terminals; Receptors, Metabotropic Glutamate; Signal Transduction; Synapses; Synaptic Transmission; Xanthenes | 2002 |
Group I metabotropic glutamate receptors (mGluRs) modulate visual responses in the superficial superior colliculus of the rat.
Topics: Amino Acids; Animals; Electric Stimulation; Electrodes; Excitatory Postsynaptic Potentials; GABA Antagonists; Habituation, Psychophysiologic; In Vitro Techniques; Iontophoresis; Membrane Potentials; Methoxyhydroxyphenylglycol; Photic Stimulation; Rats; Receptors, Metabotropic Glutamate; Superior Colliculi; Synapses; Vision, Ocular; Xanthenes | 2002 |
Modulation of DOI-induced increases in cortical BDNF expression by group II mGlu receptors.
Topics: Amino Acids; Amphetamines; Animals; Brain-Derived Neurotrophic Factor; Bridged Bicyclo Compounds; Cerebral Cortex; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; In Situ Hybridization; Male; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; RNA, Messenger; Xanthenes | 2002 |
The anxiolytic action of mGlu2/3 receptor agonist, LY354740, in the fear-potentiated startle model in rats is mechanistically distinct from diazepam.
Topics: Acoustic Stimulation; Amino Acids; Animals; Anti-Anxiety Agents; Bridged Bicyclo Compounds; Diazepam; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Fear; Flumazenil; GABA Modulators; Male; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Reflex, Startle; Xanthenes | 2002 |
Different metabotropic glutamate receptors play opposite roles in synaptic plasticity of the rat medial vestibular nuclei.
Topics: Amino Acids; Animals; Chromones; Excitatory Amino Acid Antagonists; Glycine; Membrane Potentials; Neuronal Plasticity; Organ Culture Techniques; Phenylacetates; Pyridines; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols; Vestibular Nuclei; Xanthenes | 2002 |
Synthesis and structure-activity relationship studies of novel 2-diarylethyl substituted (2-carboxycycloprop-1-yl)glycines as high-affinity group II metabotropic glutamate receptor ligands.
Topics: Amino Acids; Benzene Derivatives; Cell Line; Cloning, Molecular; Excitatory Amino Acid Antagonists; Glycine; Humans; Inhibitory Concentration 50; Ligands; Receptors, Metabotropic Glutamate; Recombinant Proteins; Stereoisomerism; Structure-Activity Relationship; Tritium; Xanthenes | 2003 |
Group II metabotropic glutamate receptor modulation of DOI-induced c-fos mRNA and excitatory responses in the cerebral cortex.
Topics: Amino Acids; Amphetamines; Animals; Autoradiography; Bridged Bicyclo Compounds; Cerebral Cortex; DNA; Electrophysiology; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Agonists; Image Interpretation, Computer-Assisted; In Situ Hybridization; Male; Prefrontal Cortex; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; RNA, Messenger; Serotonin Receptor Agonists; Xanthenes | 2003 |
Pharmacological blockade of mGlu2/3 metabotropic glutamate receptors reduces cell proliferation in cultured human glioma cells.
Topics: Amino Acids; Bridged Bicyclo Compounds, Heterocyclic; Cell Division; Cells, Cultured; Cyclin D1; Cyclin D2; Cyclins; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glioma; Humans; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Receptors, Metabotropic Glutamate; Thymidine; Tritium; Xanthenes | 2003 |
Evaluation of [3H]LY341495 for labeling group II metabotropic glutamate receptors in vivo.
Topics: Amino Acids; Animals; Brain; Male; Metabolic Clearance Rate; Radioligand Assay; Radionuclide Imaging; Radiopharmaceuticals; Rats; Receptors, Metabotropic Glutamate; Temperature; Tissue Distribution; Tritium; Xanthenes | 2003 |
Baseline glutamate levels affect group I and II mGluRs in layer V pyramidal neurons of rat sensorimotor cortex.
Topics: Amino Acids; Anesthetics, Local; Animals; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; Glutamic Acid; Male; Membrane Potentials; Motor Cortex; Neural Inhibition; Organ Culture Techniques; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Somatosensory Cortex; Synaptic Transmission; Tetrodotoxin; Xanthenes | 2003 |
Reduction of excitatory postsynaptic responses by persistently active metabotropic glutamate receptors in the hippocampus.
Topics: Amino Acids; Animals; Anticonvulsants; Cyclopropanes; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glycine; Hippocampus; Interneurons; Membrane Potentials; Mice; Mice, Inbred C57BL; Neuronal Plasticity; Presynaptic Terminals; Propionates; Receptors, Metabotropic Glutamate; Xanthenes | 2003 |
Actions of LY341495 on metabotropic glutamate receptor-mediated responses in the neonatal rat spinal cord.
Topics: Amino Acids; Aminobutyrates; Animals; Animals, Newborn; Cyclopentanes; In Vitro Techniques; Motor Neurons; Rats; Receptors, AMPA; Receptors, Kainic Acid; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Spinal Cord; Synaptic Transmission; Time Factors; Tricarboxylic Acids; Xanthenes | 2003 |
Group II mGlu receptor activation suppresses norepinephrine release in the ventral hippocampus and locomotor responses to acute ketamine challenge.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Amino Acids; Analysis of Variance; Animals; Area Under Curve; Binding Sites; Bridged Bicyclo Compounds, Heterocyclic; Chromatography, High Pressure Liquid; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Guanosine 5'-O-(3-Thiotriphosphate); Hippocampus; Humans; Hyperkinesis; In Vitro Techniques; Ketamine; Male; Microdialysis; Motor Activity; Norepinephrine; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Metabotropic Glutamate; Schizophrenia; Serotonin; Sulfur Isotopes; Time Factors; Trifluoroethanol; Xanthenes | 2003 |
Protective role of group-II metabotropic glutamate receptors against nigro-striatal degeneration induced by 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine in mice.
Topics: Amino Acids; Animals; Bridged Bicyclo Compounds, Heterocyclic; Male; Mice; Mice, Inbred C57BL; MPTP Poisoning; Neuroprotective Agents; Receptors, AMPA; Xanthenes | 2003 |
GCP II (NAALADase) inhibition suppresses mossy fiber-CA3 synaptic neurotransmission by a presynaptic mechanism.
Topics: Amino Acids; Analysis of Variance; Animals; Animals, Newborn; Calcium; Chemokine CXCL6; Chemokines, CXC; Dose-Response Relationship, Drug; Drug Interactions; Electric Conductivity; Electric Stimulation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutarates; In Vitro Techniques; Male; Mossy Fibers, Hippocampal; Neural Inhibition; Neurons; Patch-Clamp Techniques; Presynaptic Terminals; Probability; Rats; Sulfhydryl Compounds; Synaptic Transmission; Time Factors; Xanthenes | 2004 |
Group II metabotropic glutamate receptor antagonists LY341495 and LY366457 increase locomotor activity in mice.
Topics: Amino Acids; Animals; Benzazepines; Dizocilpine Maleate; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Female; Fluorobenzenes; Haloperidol; Hyperkinesis; Mice; Motor Activity; Piperidines; Receptors, Metabotropic Glutamate; Serotonin Antagonists; Time Factors; Xanthenes | 2003 |
Pharmacological characterization and identification of amino acids involved in the positive modulation of metabotropic glutamate receptor subtype 2.
Topics: Allosteric Regulation; Amino Acid Sequence; Amino Acids; Animals; Binding Sites; Calcium; Cell Membrane; Cerebral Cortex; CHO Cells; Cricetinae; Cyclopropanes; Dentate Gyrus; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Guanosine 5'-O-(3-Thiotriphosphate); Hippocampus; Humans; Molecular Sequence Data; Perforant Pathway; Protein Structure, Tertiary; Pyridines; Rats; Receptors, Metabotropic Glutamate; Sequence Homology, Amino Acid; Sulfonamides; Tritium; Xanthenes | 2003 |
Group II metabotropic glutamate receptor modulation of excitatory transmission in rat subthalamic nucleus.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 2-Amino-5-phosphonovalerate; 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; 6-Cyano-7-nitroquinoxaline-2,3-dione; Adenylyl Cyclase Inhibitors; Amino Acids; Amino Acids, Dicarboxylic; Animals; Colforsin; Cyclopropanes; Electric Stimulation; Electrophysiology; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; Glycine; Imines; In Vitro Techniques; Isoquinolines; Male; Picrotoxin; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Subthalamic Nucleus; Sulfonamides; Synaptic Transmission; Tetradecanoylphorbol Acetate; Xanthenes | 2003 |
Protective effect of LY379268, a selective group II metabotropic glutamate receptor agonist, on dizocilpine-induced neuropathological changes in rat retrosplenial cortex.
Topics: Acetylcholine; Amino Acids; Animals; Brain; Bridged Bicyclo Compounds, Heterocyclic; Chromatography, High Pressure Liquid; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Extracellular Fluid; Female; HSP70 Heat-Shock Proteins; Immunohistochemistry; Microdialysis; Neuroprotective Agents; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Xanthenes | 2003 |
Cannabinoids decrease corticostriatal synaptic transmission via an effect on glutamate uptake.
Topics: Amino Acids; Animals; Cannabinoids; Cerebral Cortex; Corpus Striatum; Dronabinol; Glutamic Acid; In Vitro Techniques; Male; Neural Inhibition; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Metabotropic Glutamate; Rimonabant; Synaptic Transmission; Xanthenes | 2003 |
The mGlu2/3 receptor agonist, LY354740, blocks immobilization-induced increases in noradrenaline and dopamine release in the rat medial prefrontal cortex.
Topics: Amino Acids; Animals; Bridged Bicyclo Compounds; Catecholamines; Citalopram; Dopamine; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Extracellular Fluid; Male; Microdialysis; Norepinephrine; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Restraint, Physical; Selective Serotonin Reuptake Inhibitors; Stress, Physiological; Xanthenes | 2004 |
Prefrontal group II metabotropic glutamate receptor activation decreases performance on a working memory task.
Topics: Amino Acids; Animals; Excitatory Amino Acid Antagonists; Extracellular Space; Feedback; Glutamates; Memory, Short-Term; Microinjections; Prefrontal Cortex; Proline; Psychomotor Performance; Rats; Receptors, AMPA; Xanthenes | 2003 |
Bidirectional modulation of cystine/glutamate exchanger activity in cultured cortical astrocytes.
Topics: Amino Acids; Animals; Astrocytes; Carrier Proteins; Cells, Cultured; Cerebral Cortex; Cystine; Enzyme Activators; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Phosphotransferases; Proline; Rats; Receptors, Metabotropic Glutamate; Xanthenes | 2003 |
Selective transmission of single photon responses by saturation at the rod-to-rod bipolar synapse.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Amino Acids; Aminobutyrates; Animals; Binding Sites; Darkness; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Light; Membrane Potentials; Mice; Mice, Inbred C57BL; Neurons; Patch-Clamp Techniques; Photons; Retina; Retinal Rod Photoreceptor Cells; Synapses; Synaptic Transmission; Valine; Xanthenes | 2004 |
An NMDAR-independent LTP mediated by group II metabotropic glutamate receptors and p42/44 MAP kinase in the dentate gyrus in vitro.
Topics: Amino Acids; Animals; Cyclopropanes; Dentate Gyrus; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; Glycine; In Vitro Techniques; Long-Term Potentiation; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Xanthenes | 2004 |
Inhibitory effects of group II mGluR-related drugs on memory performance in mice.
Topics: Amino Acids; Animals; Anticonvulsants; Avoidance Learning; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclopropanes; Dose-Response Relationship, Drug; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Glycine; Isoquinolines; Male; Memory; Mice; Reaction Time; Receptors, Metabotropic Glutamate; Rolipram; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Xanthenes | 2004 |
The selective mGlu2/3 receptor antagonist LY341495 exacerbates behavioral signs of morphine withdrawal and morphine-withdrawal-induced activation of locus coeruleus neurons.
Topics: Action Potentials; Amino Acids; Animals; Excitatory Amino Acid Antagonists; Locus Coeruleus; Male; Morphine Dependence; Neurons; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Substance Withdrawal Syndrome; Xanthenes | 2004 |
Group II metabotropic glutamate receptors inhibit cAMP-dependent protein kinase-mediated enhancemednt of tetrodotoxin-resistant sodium currents in mouse dorsal root ganglion neurons.
Topics: Amino Acids; Analysis of Variance; Animals; Animals, Newborn; Cells, Cultured; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Ganglia, Spinal; Membrane Potentials; Mice; NAV1.7 Voltage-Gated Sodium Channel; Neurons; Neuropeptides; Pyrrolidines; Receptors, Metabotropic Glutamate; Sodium Channels; Thiocarbamates; Time Factors; Xanthenes | 2004 |
Tonic activity of metabotropic glutamate receptors is involved in developmental modification of short-term plasticity in the neocortex.
Topics: Aging; Amino Acids; Animals; Animals, Newborn; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; In Vitro Techniques; Neocortex; Neuronal Plasticity; Presynaptic Terminals; Rats; Receptors, Metabotropic Glutamate; Synapses; Time Factors; Xanthenes | 2004 |
Pharmacological manipulation of mGlu2 receptors influences cognitive performance in the rodent.
Topics: Amino Acids; Animals; Bridged Bicyclo Compounds; Cognition; Dose-Response Relationship, Drug; Excitatory Postsynaptic Potentials; Male; Maze Learning; Mice; Mice, Inbred C57BL; Mice, Knockout; Psychomotor Performance; Rats; Reaction Time; Receptors, Metabotropic Glutamate; Xanthenes | 2004 |
Depression of GABAergic input to identified hippocampal neurons by group III metabotropic glutamate receptors in the rat.
Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Animals, Newborn; Cell Count; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Hippocampus; Horseradish Peroxidase; Immunohistochemistry; In Vitro Techniques; Interneurons; Lysine; Membrane Potentials; Microscopy, Immunoelectron; Neural Inhibition; Patch-Clamp Techniques; Propionates; Pyramidal Cells; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Somatostatin; Statistics, Nonparametric; Synapses; Time Factors; Xanthenes | 2004 |
Distinct properties of presynaptic group II and III metabotropic glutamate receptor-mediated inhibition of perforant pathway-CA1 EPSCs.
Topics: Amino Acids; Aminobutyrates; Animals; Bridged Bicyclo Compounds; Calcium Channel Blockers; Cyclic AMP; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Interactions; Elapid Venoms; Electric Stimulation; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; Hippocampus; In Vitro Techniques; Membrane Potentials; Neural Inhibition; omega-Conotoxin GVIA; Perforant Pathway; Phosphinic Acids; Propanolamines; Quinoxalines; Rats; Receptors, Metabotropic Glutamate; Statistics, Nonparametric; Synaptic Transmission; Thionucleotides; Time Factors; Xanthenes | 2004 |
Effect of donepezil on group II mGlu receptor agonist- or antagonist-induced amnesia on passive avoidance in mice.
Topics: Amino Acids; Amnesia; Animals; Avoidance Learning; Cholinesterase Inhibitors; Cyclopropanes; Donepezil; Excitatory Amino Acid Antagonists; Glycine; Indans; Male; Memory; Mice; Nootropic Agents; Piperidines; Receptors, Metabotropic Glutamate; Xanthenes | 2003 |
Modulation of glutamate mobility reveals the mechanism underlying slow-rising AMPAR EPSCs and the diffusion coefficient in the synaptic cleft.
Topics: Amino Acids; Animals; Animals, Newborn; Benzylamines; Cerebellum; Computer Simulation; Dextrans; Diffusion; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; In Vitro Techniques; Membrane Potentials; Nerve Fibers; Neurons; Patch-Clamp Techniques; Phosphinic Acids; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, AMPA; Synapses; Synaptic Transmission; Time Factors; Xanthenes | 2004 |
Retroinhibition of presynaptic Ca2+ currents by endocannabinoids released via postsynaptic mGluR activation at a calyx synapse.
Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Amino Acids; Animals; Benzoxazines; Brain Stem; Calcium Signaling; Cannabinoid Receptor Modulators; Endocannabinoids; Evoked Potentials, Auditory, Brain Stem; Glycine; Ion Transport; Morpholines; Naphthalenes; Nerve Endings; Patch-Clamp Techniques; Picrotoxin; Piperidines; Pyrazoles; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Metabotropic Glutamate; Receptors, Presynaptic; Resorcinols; Scopolamine; Synaptic Transmission; Xanthenes | 2004 |
Antinociceptive effects of N-acetylaspartylglutamate (NAAG) peptidase inhibitors ZJ-11, ZJ-17 and ZJ-43 in the rat formalin test and in the rat neuropathic pain model.
Topics: Amino Acids; Analgesics; Animals; Behavior, Animal; Cell Line; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Glutamate Carboxypeptidase II; Humans; Immunohistochemistry; Injections, Intravenous; Injections, Spinal; Nociceptors; Pain; Pain Measurement; Pain Threshold; Physical Stimulation; Protease Inhibitors; Proto-Oncogene Proteins c-fos; Rats; Reaction Time; Sciatic Neuropathy; Urea; Xanthenes | 2004 |
Distinct properties of carbachol- and DHPG-induced network oscillations in hippocampal slices.
Topics: Action Potentials; Amino Acids; Animals; Animals, Newborn; Benzodiazepines; Bicuculline; Carbachol; Cholinergic Agonists; Diamines; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; Hippocampus; In Vitro Techniques; Male; Methoxyhydroxyphenylglycol; Muscarinic Antagonists; Pirenzepine; Pyridines; Rats; Receptors, Metabotropic Glutamate; Spectrum Analysis; Substance P; Xanthenes; Zolpidem | 2004 |
The metabotropic glutamate (mGLU)2/3 receptor antagonist LY341495 [2S-2-amino-2-(1S,2S-2-carboxycyclopropyl-1-yl)-3-(xanth-9-yl)propanoic acid] stimulates waking and fast electroencephalogram power and blocks the effects of the mGLU2/3 receptor agonist ly
Topics: Amino Acids; Animals; Arousal; Behavior, Animal; Bridged Bicyclo Compounds, Heterocyclic; Darkness; Electroencephalography; Excitatory Amino Acid Antagonists; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Metabotropic Glutamate; Sleep; Sleep Stages; Wakefulness; Xanthenes | 2005 |
Glutamate transporters and metabotropic receptors regulate excitatory neurotransmission in the medial entorhinal cortex of the rat.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amino Acid Transport System X-AG; Amino Acids; Animals; Aspartic Acid; Dicarboxylic Acids; Drug Interactions; Entorhinal Cortex; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Glycine; In Vitro Techniques; N-Methylaspartate; Neurotransmitter Uptake Inhibitors; Patch-Clamp Techniques; Pyrrolidines; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Synaptic Transmission; Xanthenes | 2004 |
Metabotropic glutamate receptors modulate feedback inhibition in a developmentally regulated manner in rat dentate gyrus.
Topics: Amino Acids; Animals; Dentate Gyrus; Excitatory Postsynaptic Potentials; Feedback, Physiological; Neural Inhibition; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Xanthenes | 2004 |
Activation of Group II and Group III metabotropic glutamate receptors by endogenous ligand(s) and the modulation of synaptic transmission in the superficial superior colliculus.
Topics: Action Potentials; Amino Acids; Animals; Biotransformation; Dose-Response Relationship, Drug; Drug Synergism; Excitatory Postsynaptic Potentials; Extracellular Space; Glutamates; Ligands; Rats; Receptors, AMPA; Superior Colliculi; Synaptic Transmission; Xanthenes | 2004 |
Glutamate-evoked alterations of glial and neuronal cell morphology in the guinea pig retina.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Adenosine Triphosphate; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amino Acids; Animals; Aspartic Acid; Cell Size; Circadian Rhythm; Cytochalasin D; Cytoskeleton; Dicarboxylic Acids; Dopamine; Eye Proteins; Glutamic Acid; Guinea Pigs; Ischemia; Kainic Acid; N-Methylaspartate; Neuroglia; Neurons; Nocodazole; Potassium; Pyrrolidines; Receptors, AMPA; Receptors, Kainic Acid; Retina; Retinal Ganglion Cells; Synaptic Transmission; Xanthenes | 2004 |
A novel selective positive allosteric modulator of metabotropic glutamate receptor subtype 5 has in vivo activity and antipsychotic-like effects in rat behavioral models.
Topics: Amino Acids; Amphetamine; Animals; Antipsychotic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Behavior, Animal; Benzamides; Cell Line; Central Nervous System Stimulants; CHO Cells; Cricetinae; Dogs; Excitatory Amino Acid Antagonists; Female; Haplorhini; Humans; Image Interpretation, Computer-Assisted; In Vitro Techniques; Microsomes, Liver; Models, Statistical; Motor Activity; Phthalimides; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Reflex, Startle; Xanthenes | 2005 |
Anxiolytic-like activity of the mGLU2/3 receptor agonist LY354740 in the elevated plus maze test is disrupted in metabotropic glutamate receptor 2 and 3 knock-out mice.
Topics: Amino Acids; Amygdala; Animals; Anti-Anxiety Agents; Bridged Bicyclo Compounds; Excitatory Amino Acid Agonists; Female; Male; Maze Learning; Mice; Mice, Inbred C57BL; Mice, Inbred ICR; Mice, Knockout; Receptors, Metabotropic Glutamate; Xanthenes | 2005 |
Seizures induced in immature rats by homocysteic acid and the associated brain damage are prevented by group II metabotropic glutamate receptor agonist (2R,4R)-4-aminopyrrolidine-2,4-dicarboxylate.
Topics: Amino Acids; Animals; Animals, Newborn; Anticonvulsants; Behavior, Animal; Brain; Brain Chemistry; Brain Injuries; Dose-Response Relationship, Drug; Drug Interactions; Electroencephalography; Excitatory Amino Acid Antagonists; Fluoresceins; Fluorescent Dyes; Functional Laterality; Glucose; Glycogen; Homocysteine; Lactic Acid; Male; Nerve Degeneration; Organic Chemicals; Proline; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Seizures; Time Factors; Xanthenes | 2005 |
Presynaptic inhibition of corticothalamic feedback by metabotropic glutamate receptors.
Topics: Amino Acids; Animals; Animals, Newborn; Bridged Bicyclo Compounds, Heterocyclic; Cyclopropanes; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Feedback; Ferrets; Geniculate Bodies; Glycine; In Vitro Techniques; Male; Neural Inhibition; Neural Pathways; Neurons; Presynaptic Terminals; Receptors, Metabotropic Glutamate; Synaptic Transmission; Time Factors; Xanthenes | 2005 |
Developmental switch in synaptic mechanisms of hippocampal metabotropic glutamate receptor-dependent long-term depression.
Topics: Age Factors; Amino Acids; Animals; Animals, Newborn; Anisomycin; Benzoxazines; Cycloheximide; Dizocilpine Maleate; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Antagonists; Hippocampus; In Vitro Techniques; Long-Term Synaptic Depression; Methoxyhydroxyphenylglycol; Morpholines; Naphthalenes; Neurons; Protein Synthesis Inhibitors; Pyrazoles; Rats; Rats, Long-Evans; Reaction Time; Receptor, Cannabinoid, CB1; Receptors, Metabotropic Glutamate; Synapses; Xanthenes | 2005 |
Neuropharmacological profiles of antagonists of group II metabotropic glutamate receptors.
Topics: Action Potentials; Amino Acids; Animals; Antidepressive Agents; Biogenic Monoamines; Bridged Bicyclo Compounds; Dicarboxylic Acids; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Extracellular Fluid; Locus Coeruleus; Male; Neurons; Prefrontal Cortex; Raphe Nuclei; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Serotonin; Xanthenes | 2005 |
Metabotropic glutamate receptors and neuroadaptation to antidepressants: imipramine-induced down-regulation of beta-adrenergic receptors in mice treated with metabotropic glutamate 2/3 receptor ligands.
Topics: Adaptation, Physiological; Amino Acids; Animals; Antidepressive Agents, Tricyclic; Bridged Bicyclo Compounds, Heterocyclic; Down-Regulation; Excitatory Amino Acid Antagonists; Hippocampus; Imipramine; Ligands; Male; Mice; Mice, Inbred Strains; Nervous System Physiological Phenomena; Reaction Time; Receptors, Adrenergic, beta; Receptors, Metabotropic Glutamate; Xanthenes | 2005 |
Metabotropic glutamate receptor 2 modulates excitatory synaptic transmission in the rat globus pallidus.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Amino Acids; Aminobutyrates; Anesthetics, Local; Animals; Animals, Newborn; Cyclopropanes; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Globus Pallidus; Glycine; In Vitro Techniques; Lidocaine; Membrane Potentials; Methoxyhydroxyphenylglycol; Neurons; Patch-Clamp Techniques; Proline; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Sulfonamides; Synaptic Transmission; Xanthenes | 2005 |
Group II and III mGluRs-mediated presynaptic inhibition of EPSCs recorded from hippocampal interneurons of CA1 stratum lacunosum moleculare.
Topics: Amino Acids; Aminobutyrates; Analysis of Variance; Animals; Animals, Newborn; Bridged Bicyclo Compounds; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Hippocampus; In Vitro Techniques; Interneurons; Neural Inhibition; Perforant Pathway; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Strontium; Tetrodotoxin; Time Factors; Xanthenes | 2005 |
Cystine/glutamate exchange regulates metabotropic glutamate receptor presynaptic inhibition of excitatory transmission and vulnerability to cocaine seeking.
Topics: Amino Acids; Animals; Biological Transport; Cocaine; Cocaine-Related Disorders; Consummatory Behavior; Cystine; Excitatory Amino Acid Antagonists; Extinction, Psychological; Glutamic Acid; Male; Neural Conduction; Nucleus Accumbens; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Receptors, Presynaptic; Self Administration; Xanthenes | 2005 |
Comparison of c-Fos induction in the brain by the mGlu2/3 receptor antagonist LY341495 and agonist LY354740: evidence for widespread endogenous tone at brain mGlu2/3 receptors in vivo.
Topics: Amino Acids; Analysis of Variance; Animals; Brain; Bridged Bicyclo Compounds; Cell Count; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Gene Expression Regulation; Immunohistochemistry; Male; Mice; Mice, Inbred ICR; Neurons; Proto-Oncogene Proteins c-fos; Xanthenes | 2005 |
The preferential mGlu2/3 receptor antagonist, LY341495, reduces the frequency of spike-wave discharges in the WAG/Rij rat model of absence epilepsy.
Topics: Age Factors; Amino Acids; Analysis of Variance; Animals; Baclofen; Behavior, Animal; Blotting, Western; Brain; Brain Mapping; Circadian Rhythm; Cyclic AMP; Disease Models, Animal; Electroencephalography; Epilepsy, Absence; Excitatory Amino Acid Antagonists; GABA Agonists; Glial Fibrillary Acidic Protein; Immunohistochemistry; Indoles; Male; Microdialysis; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Metabotropic Glutamate; Xanthenes | 2005 |
Pharmacological blockade of group II metabotropic glutamate receptors reduces the growth of glioma cells in vivo.
Topics: Amino Acids; Animals; Blotting, Western; Brain Neoplasms; Cell Line, Tumor; Cell Proliferation; Cyclin D1; Cyclin D2; Cyclins; Enzyme Activation; Excitatory Amino Acid Antagonists; Glioma; Humans; Immunohistochemistry; Ki-67 Antigen; Magnetic Resonance Imaging; MAP Kinase Signaling System; Mice; Mice, Nude; Phosphatidylinositol 3-Kinases; Receptors, Metabotropic Glutamate; Reverse Transcriptase Polymerase Chain Reaction; Xanthenes | 2005 |
Role of group II metabotropic glutamate receptors 2/3 and group I metabotropic glutamate receptor 5 in developing rat medial vestibular nuclei.
Topics: 2-Amino-5-phosphonovalerate; Age Factors; Amino Acids; Animals; Animals, Newborn; Dose-Response Relationship, Radiation; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; In Vitro Techniques; Long-Term Potentiation; Long-Term Synaptic Depression; Neural Inhibition; Phenylacetates; Rats; Rats, Wistar; Receptors, AMPA; Receptors, Kainic Acid; Synaptic Transmission; Vestibular Nuclei; Xanthenes | 2005 |
Regulation of IPSP theta rhythm by muscarinic receptors and endocannabinoids in hippocampus.
Topics: Action Potentials; Amino Acids; Animals; Cannabinoid Receptor Modulators; Carbachol; Cholinergic Agonists; Endocannabinoids; Excitatory Amino Acid Antagonists; Hippocampus; In Vitro Techniques; Male; Methoxyhydroxyphenylglycol; Neural Inhibition; Piperidines; Pyrazoles; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Spectrum Analysis; Synapses; Theta Rhythm; Time Factors; Xanthenes | 2005 |
Neuroprotective effect of N-acetyl-aspartyl-glutamate in combination with mild hypothermia in the endothelin-1 rat model of focal cerebral ischaemia.
Topics: Amino Acids; Animals; Blood-Brain Barrier; Brain Ischemia; Dipeptides; Disease Models, Animal; Drug Administration Schedule; Drug Therapy, Combination; Endothelin-1; Hypothermia; Male; Microdialysis; Neuroprotective Agents; Rats; Rats, Wistar; Time Factors; Xanthenes | 2005 |
2-MPPA, a selective glutamate carboxypeptidase II inhibitor, attenuates morphine tolerance but not dependence in C57/Bl mice.
Topics: Amino Acids; Animals; Drug Tolerance; Enzyme Inhibitors; Glutamate Carboxypeptidase II; Male; Mice; Mice, Inbred C57BL; Morphine; Morphine Dependence; Naloxone; Organophosphorus Compounds; Receptors, Metabotropic Glutamate; Xanthenes | 2005 |
Modulation of excitatory synaptic transmission by endogenous glutamate acting on presynaptic group II mGluRs in rat substantia nigra compacta.
Topics: Amino Acid Transport System X-AG; Amino Acids; Animals; Animals, Newborn; Aspartic Acid; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamates; In Vitro Techniques; Patch-Clamp Techniques; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Substantia Nigra; Synaptic Transmission; Xanthenes | 2005 |
Antinociceptive effects and synergistic interaction with morphine of intrathecal metabotropic glutamate receptor 2/3 antagonist in the formalin test of rats.
Topics: Amino Acids; Analgesics; Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Drug Synergism; Excitatory Amino Acid Antagonists; Formaldehyde; Injections, Spinal; Male; Morphine; Pain Measurement; Proline; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Reflex; Xanthenes | 2006 |
Olfactory nerve-evoked, metabotropic glutamate receptor-mediated synaptic responses in rat olfactory bulb mitral cells.
Topics: Amino Acids; Animals; Aspartic Acid; Benzoates; Dopamine D2 Receptor Antagonists; Electrophysiology; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; GABA-B Receptor Antagonists; Glutamic Acid; Glycine; In Vitro Techniques; Male; Neuronal Plasticity; Neurons, Afferent; Odorants; Olfactory Bulb; Olfactory Nerve; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, GABA-B; Receptors, Metabotropic Glutamate; Synapses; Tacrine; Xanthenes | 2006 |
Differential negative coupling of type 3 metabotropic glutamate receptor to cyclic GMP levels in neurons and astrocytes.
Topics: Amino Acids; Animals; Animals, Newborn; Astrocytes; Cerebellum; Cyclic GMP; Dipeptides; Excitatory Amino Acid Antagonists; GTP-Binding Proteins; Neurons; Nitroprusside; Pertussis Toxin; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Xanthenes | 2006 |
Differential roles for group 1 mGluR subtypes in induction and expression of chemically induced hippocampal long-term depression.
Topics: Action Potentials; Amino Acids; Animals; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Extracellular Signal-Regulated MAP Kinases; Hippocampus; Long-Term Synaptic Depression; Methoxyhydroxyphenylglycol; Mice; Mice, Knockout; Neuronal Plasticity; Neurons; Neurotransmitter Agents; Phosphorylation; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, AMPA; Receptors, Metabotropic Glutamate; Synapses; Xanthenes | 2006 |
Long-term depression of NMDA receptor-mediated synaptic transmission is dependent on activation of metabotropic glutamate receptors and is altered to long-term potentiation by low intracellular calcium buffering.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Amino Acids; Animals; Buffers; Calcium; Dentate Gyrus; Egtazic Acid; Electric Stimulation; Excitatory Amino Acid Antagonists; Long-Term Synaptic Depression; Male; Patch-Clamp Techniques; Perforant Pathway; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission; Xanthenes | 2006 |
Unique presynaptic and postsynaptic roles of Group II metabotropic glutamate receptors in the modulation of thalamic network activity.
Topics: Amino Acids; Animals; Animals, Newborn; Bridged Bicyclo Compounds, Heterocyclic; Drug Interactions; Electric Stimulation; Excitatory Postsynaptic Potentials; Female; Ferrets; Gluconates; Guanosine Diphosphate; In Vitro Techniques; Male; Membrane Potentials; Nerve Net; Neurons; Organophosphorus Compounds; Patch-Clamp Techniques; Picrotoxin; Receptors, Metabotropic Glutamate; Synapses; Thalamus; Thionucleotides; Xanthenes | 2006 |
Blockade of group II metabotropic glutamate receptors in the nucleus accumbens produces hyperlocomotion in rats previously exposed to amphetamine.
Topics: Amino Acids; Amphetamine; Analysis of Variance; Animals; Behavior, Animal; Bridged Bicyclo Compounds, Heterocyclic; Central Nervous System Stimulants; Drug Interactions; Hyperkinesis; Male; Motor Activity; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Xanthenes | 2006 |
Analgesia mediated by the TRPM8 cold receptor in chronic neuropathic pain.
Topics: Acrolein; Amino Acids; Analgesia; Analysis of Variance; Animals; Blotting, Western; Cold Temperature; Dose-Response Relationship, Drug; Electrophysiology; Immunohistochemistry; Male; Menthol; Neuralgia; Oligonucleotides, Antisense; Pyrimidinones; Rats; Rats, Wistar; Receptors, Glutamate; Reflex; TRPM Cation Channels; Xanthenes | 2006 |
Group III metabotropic glutamate receptor agonists selectively suppress excitatory synaptic currents in the rat prefrontal cortex induced by 5-hydroxytryptamine2A receptor activation.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amino Acids; Animals; Bridged Bicyclo Compounds; Glycine; Male; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Metabotropic Glutamate; Serotonin; Synaptic Transmission; Xanthenes | 2007 |
Effects of metabotropic glutamate 2/3 receptor antagonists in the stress-induced hyperthermia test in singly housed mice.
Topics: Amino Acids; Animals; Arousal; Autonomic Nervous System; Body Temperature Regulation; Bridged Bicyclo Compounds; Dicarboxylic Acids; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Male; Mice; Mice, Inbred ICR; Piperazines; Pyridines; Receptor, Serotonin, 5-HT1A; Receptors, Metabotropic Glutamate; Serotonin Antagonists; Social Isolation; Xanthenes | 2007 |
Interactive effects of the mGlu5 receptor antagonist MPEP and the mGlu2/3 receptor antagonist LY341495 on nicotine self-administration and reward deficits associated with nicotine withdrawal in rats.
Topics: Amino Acids; Animals; Dose-Response Relationship, Drug; Drug Interactions; Eating; Excitatory Amino Acid Antagonists; Ganglionic Stimulants; Infusions, Intravenous; Injections, Intraperitoneal; Male; Nicotine; Pyridines; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Reinforcement Schedule; Reward; Self Administration; Substance Withdrawal Syndrome; Time Factors; Xanthenes | 2007 |
The effects of the mGluR5 antagonist MPEP and the mGluR2/3 antagonist LY341495 on rats' performance in the 5-choice serial reaction time task.
Topics: Amino Acids; Analysis of Variance; Animals; Behavior, Animal; Choice Behavior; Curare; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Male; Nicotinic Antagonists; Pyridines; Rats; Rats, Wistar; Reaction Time; Xanthenes | 2007 |
Habituation deficits induced by metabotropic glutamate receptors 2/3 receptor blockade in mice: reversal by antipsychotic drugs.
Topics: Amino Acids; Animals; Antipsychotic Agents; Cognition Disorders; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Habituation, Psychophysiologic; Haloperidol; Male; Methamphetamine; Mice; Motor Activity; Nitriles; Receptors, Metabotropic Glutamate; Tetrahydroisoquinolines; Xanthenes | 2007 |
Endogenous mGluR activity suppresses GABAergic transmission in avian cochlear nucleus magnocellularis neurons.
Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Chickens; Cochlear Nucleus; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Kinetics; Membrane Potentials; Models, Neurological; Neurons; Patch-Clamp Techniques; Receptors, GABA-B; Receptors, Metabotropic Glutamate; Resorcinols; Synapses; Synaptic Transmission; Xanthenes | 2007 |
Pharmacological activation of mGlu2/3 metabotropic glutamate receptors protects retinal neurons against anoxic damage in the goldfish Carassius auratus.
Topics: Amino Acids; Animals; Apoptosis; Blotting, Western; Bridged Bicyclo Compounds, Heterocyclic; Excitatory Amino Acid Antagonists; Glutamic Acid; Goldfish; Hypoxia; Hypoxia, Brain; Immunohistochemistry; In Situ Nick-End Labeling; Models, Animal; Receptors, Metabotropic Glutamate; Retina; Retinal Diseases; Telencephalon; Xanthenes | 2007 |
In vivo pharmacological characterization of the structurally novel, potent, selective mGlu2/3 receptor agonist LY404039 in animal models of psychiatric disorders.
Topics: Amino Acids; Amphetamine; Animals; Behavior, Animal; Bridged Bicyclo Compounds, Heterocyclic; Cyclic S-Oxides; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Male; Mental Disorders; Mice; Molecular Structure; Motor Activity; Phencyclidine; Prefrontal Cortex; Rats; Rats, Inbred F344; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Xanthenes | 2007 |
A novel family of potent negative allosteric modulators of group II metabotropic glutamate receptors.
Topics: Allosteric Regulation; Amino Acids; Animals; Binding Sites; CHO Cells; Cricetinae; Cricetulus; Humans; Male; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Structure-Activity Relationship; Sulfonamides; Xanthenes | 2007 |
Group II metabotropic glutamate receptors inhibit glutamate release at thalamocortical synapses in the developing somatosensory cortex.
Topics: Amino Acids; Animals; Anticonvulsants; Cerebral Cortex; Cyclopropanes; Electrophysiology; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Glycine; Immunohistochemistry; In Vitro Techniques; Mice; Receptors, Metabotropic Glutamate; Receptors, Presynaptic; Somatosensory Cortex; Synapses; Thalamus; Xanthenes | 2007 |
Dual GABAergic synaptic response of fast excitation and slow inhibition in the medial habenula of rat epithalamus.
Topics: Amino Acids; Animals; Animals, Newborn; Bicuculline; Electric Stimulation; Electrophysiology; Epithalamus; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Habenula; Neurons; Phosphinic Acids; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Synapses; Xanthenes | 2007 |
Group-II metabotropic glutamate receptor ligands as adjunctive drugs in the treatment of depression: a new strategy to shorten the latency of antidepressant medication?
Topics: Adjuvants, Pharmaceutic; Amino Acids; Animals; Antidepressive Agents, Tricyclic; Bridged Bicyclo Compounds, Heterocyclic; Depressive Disorder; Disease Models, Animal; Drug Interactions; Drug Therapy, Combination; Excitatory Amino Acid Agents; Hippocampus; Imipramine; In Vitro Techniques; Mice; Neurons; Rats; Rats, Inbred Strains; Receptor Cross-Talk; Receptors, Metabotropic Glutamate; Time Factors; Xanthenes | 2007 |
Contribution of cystine-glutamate antiporters to the psychotomimetic effects of phencyclidine.
Topics: Acetylcysteine; Aged; Aged, 80 and over; Amino Acids; Analysis of Variance; Animals; Behavior, Animal; Cell Line, Transformed; Disease Models, Animal; Dose-Response Relationship, Drug; Extracellular Fluid; Female; Free Radical Scavengers; Glutamic Acid; Glycine; Humans; Interpersonal Relations; Male; Maze Learning; Microdialysis; Phencyclidine; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Schizophrenia; Xanthenes | 2008 |
Basal ganglia group II metabotropic glutamate receptors specific binding in non-human primate model of L-Dopa-induced dyskinesias.
Topics: Amino Acids; Animals; Antiparkinson Agents; Autoradiography; Basal Ganglia; Behavior, Animal; Cabergoline; Caudate Nucleus; Data Interpretation, Statistical; Dyskinesia, Drug-Induced; Ergolines; Excitatory Amino Acid Antagonists; Female; Levodopa; Macaca fascicularis; Ovariectomy; Putamen; Receptors, Metabotropic Glutamate; Xanthenes | 2008 |
A novel assay of Gi/o-linked G protein-coupled receptor coupling to potassium channels provides new insights into the pharmacology of the group III metabotropic glutamate receptors.
Topics: Adrenergic Agonists; Allosteric Regulation; Amino Acids; Animals; Biological Assay; Carbachol; Cell Line; Dose-Response Relationship, Drug; G Protein-Coupled Inwardly-Rectifying Potassium Channels; GTP-Binding Protein alpha Subunits, Gi-Go; Humans; Ion Channel Gating; Ligands; Muscarinic Agonists; Pertussis Toxin; Rats; Receptors, Metabotropic Glutamate; Receptors, Muscarinic; Reproducibility of Results; Thallium; Xanthenes | 2008 |
Group III mGluR regulation of synaptic transmission at the SC-CA1 synapse is developmentally regulated.
Topics: Age Factors; Amino Acids; Aminobutyrates; Animals; Animals, Newborn; Cell Line, Transformed; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Hippocampus; Humans; In Vitro Techniques; Male; Neural Pathways; Neurons; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Synapses; Synaptic Transmission; Transfection; Xanthenes | 2008 |
Distinct neural mechanisms mediate olfactory memory formation at different timescales.
Topics: Amino Acids; Animals; Brain Mapping; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Habituation, Psychophysiologic; Injections; Male; Memory; Mice; Mice, Inbred Strains; Odorants; Olfactory Bulb; Olfactory Pathways; Smell; Time Factors; Xanthenes | 2008 |
Involvement of group I mGluRs in LTP induced by strong high frequency stimulation in the dentate gyrus in vitro.
Topics: Amino Acids; Animals; Dentate Gyrus; Dose-Response Relationship, Radiation; Electric Stimulation; Excitatory Amino Acid Antagonists; In Vitro Techniques; Long-Term Potentiation; Patch-Clamp Techniques; Pyridines; Rats; Receptors, Metabotropic Glutamate; Ryanodine; Xanthenes | 2008 |
Conformational change of the transmembrane helices II and IV of metabotropic glutamate receptor involved in G protein activation.
Topics: Amino Acids; Cell Line, Transformed; Dose-Response Relationship, Drug; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Models, Molecular; Mutagenesis, Site-Directed; Propionates; Protein Binding; Protein Conformation; Protein Structure, Secondary; Receptors, Metabotropic Glutamate; Structure-Activity Relationship; Transfection; Tritium; Xanthenes | 2008 |
Group II metabotropic glutamate receptor activation attenuates peripheral sensitization in inflammatory states.
Topics: Amino Acids; Animals; Behavior, Animal; Cyclopentanes; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Hot Temperature; Inflammation; Male; Nerve Fibers; Nociceptors; Pain; Peripheral Nerves; Physical Stimulation; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Skin; Xanthenes | 2008 |
Type-3 metabotropic glutamate receptors negatively modulate bone morphogenetic protein receptor signaling and support the tumourigenic potential of glioma-initiating cells.
Topics: Amino Acids; Animals; Bone Morphogenetic Protein Receptors; Brain Neoplasms; Bridged Bicyclo Compounds, Heterocyclic; Cell Differentiation; Cell Line, Tumor; Disease Models, Animal; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glioma; Humans; Magnetic Resonance Imaging; Mice; Mitogen-Activated Protein Kinases; Nerve Tissue Proteins; Phosphorylation; Receptors, Metabotropic Glutamate; Signal Transduction; Xanthenes | 2008 |
Allosteric potentiators of metabotropic glutamate receptor subtype 1a differentially modulate independent signaling pathways in baby hamster kidney cells.
Topics: Allosteric Regulation; Amino Acids; Animals; Binding, Competitive; Calcium; Cell Line, Transformed; Cricetinae; Cyclic AMP; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Mitogen-Activated Protein Kinase 3; Pyrans; Quinolines; Radioligand Assay; Receptors, Metabotropic Glutamate; Signal Transduction; Time Factors; Transfection; Tritium; Xanthenes | 2008 |
Behavioral characterization of the mGlu group II/III receptor antagonist, LY-341495, in animal models of anxiety and depression.
Topics: Amino Acids; Amphetamine; Animals; Anti-Anxiety Agents; Antidepressive Agents, Second-Generation; Anxiety; Behavior, Animal; Central Nervous System Stimulants; Conditioning, Operant; Darkness; Depression; Diazepam; Fever; Fluoxetine; Light; Male; Mice; Paroxetine; Receptors, Metabotropic Glutamate; Reinforcement Schedule; Stress, Psychological; Xanthenes | 2008 |
Repeated exposure to cocaine alters the modulation of mesocorticolimbic glutamate transmission by medial prefrontal cortex Group II metabotropic glutamate receptors.
Topics: Amino Acids; Animals; Cocaine; Cocaine-Related Disorders; Cystine; Disease Models, Animal; Dopamine Uptake Inhibitors; Drug Administration Schedule; Excitatory Amino Acid Antagonists; Glutamic Acid; Limbic System; Male; Neural Pathways; Prefrontal Cortex; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Synaptic Transmission; Synaptic Vesicles; Ventral Tegmental Area; Xanthenes | 2008 |
Blockade of group II metabotropic glutamate receptors produces hyper-locomotion in cocaine pre-exposed rats by interactions with dopamine receptors.
Topics: Amino Acids; Animals; Behavior, Animal; Benzazepines; Cocaine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Hyperkinesis; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Metabotropic Glutamate; Salicylamides; Xanthenes | 2008 |
AMPA silencing is a prerequisite for developmental long-term potentiation in the hippocampal CA1 region.
Topics: Aging; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amino Acids; Animals; Animals, Newborn; Colforsin; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Hippocampus; In Vitro Techniques; Long-Term Potentiation; Models, Biological; Rats; Valine; Xanthenes | 2008 |
Individual contribution of metabotropic glutamate receptor (mGlu) 2 and 3 to c-Fos expression pattern evoked by mGlu2/3 antagonism.
Topics: Amino Acids; Amygdala; Animals; Excitatory Amino Acid Antagonists; Gene Expression; Genes, fos; Hippocampus; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurons; Prefrontal Cortex; Receptors, Metabotropic Glutamate; Septum of Brain; Xanthenes | 2008 |
Dynamic metabotropic control of intrinsic firing in cerebellar unipolar brush cells.
Topics: Action Potentials; Amino Acids; Animals; Barium; Bee Venoms; Calbindin 2; Cerebellum; Cycloleucine; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; In Vitro Techniques; Interneurons; Male; Mice; Neural Inhibition; Potassium Channel Blockers; Receptors, Metabotropic Glutamate; S100 Calcium Binding Protein G; Xanthenes | 2008 |
GABA(B) receptor activation mediates frequency-dependent plasticity of developing GABAergic synapses.
Topics: Age Factors; Amino Acids; Animals; Animals, Newborn; Bumetanide; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Dose-Response Relationship, Radiation; Electric Stimulation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; GABA Agents; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glycine; Hippocampus; In Vitro Techniques; Neuronal Plasticity; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Sodium Potassium Chloride Symporter Inhibitors; Sodium-Potassium-Chloride Symporters; Synapses; Synaptic Potentials; Xanthenes | 2008 |
Group II metabotropic glutamate receptor activation on peripheral nociceptors modulates TRPV1 function.
Topics: Amino Acids; Animals; Capsaicin; Colforsin; Electrophysiological Phenomena; Ganglia, Spinal; Hot Temperature; Hyperalgesia; Immunohistochemistry; Male; Nociceptors; Pain; Pain Measurement; Proline; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; TRPV Cation Channels; Xanthenes | 2009 |
The slow Ca2+ -dependent K+ -current facilitates synchronization of hyperexcitable pyramidal neurons.
Topics: Action Potentials; Amino Acids; Animals; Barium; Calcium; Carbachol; Cesium; Excitatory Amino Acid Antagonists; Hippocampus; In Vitro Techniques; Isoproterenol; Male; Membrane Potentials; Microelectrodes; Patch-Clamp Techniques; Potassium; Pyramidal Cells; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Xanthenes | 2009 |
Epigenetic modulation of mGlu2 receptors by histone deacetylase inhibitors in the treatment of inflammatory pain.
Topics: Amino Acids; Animals; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Enzyme Inhibitors; Epigenesis, Genetic; Histone Deacetylase Inhibitors; Hydroxamic Acids; Inflammation; Male; Mice; Pain; Pyridines; Receptors, Metabotropic Glutamate; Vorinostat; Xanthenes | 2009 |
Metabotropic glutamate receptor II in the brains of Parkinsonian patients.
Topics: Aged; Aged, 80 and over; Amino Acids; Antiparkinson Agents; Brain; Cocaine; Dyskinesia, Drug-Induced; Excitatory Amino Acid Antagonists; Female; Humans; Iodine Radioisotopes; Levodopa; Male; Parkinsonian Disorders; Postmortem Changes; Radioligand Assay; Receptors, Metabotropic Glutamate; Tritium; Xanthenes | 2009 |
gamma-Aminobutyric acid-mediated regulation of the activity-dependent olfactory bulb dopaminergic phenotype.
Topics: Agatoxins; Amino Acids; Animals; Animals, Newborn; Bicuculline; Calcium Channel Blockers; Dopamine; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Gene Expression; Green Fluorescent Proteins; Interneurons; Mice; Mice, Transgenic; Olfactory Bulb; Phosphinic Acids; Potassium Chloride; Prosencephalon; Spider Venoms; Tissue Culture Techniques; Tyrosine 3-Monooxygenase; Xanthenes | 2009 |
Antinociceptive synergistic effect of spinal mGluR2/3 antagonist and glial cells inhibitor on peripheral inflammation-induced mechanical hypersensitivity.
Topics: Amino Acids; Analgesics; Animals; Citrates; Dose-Response Relationship, Drug; Freund's Adjuvant; Hyperesthesia; Inflammation; Male; Neuroglia; Pain; Proline; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Spinal Cord; Xanthenes | 2009 |
Activation of mGlu2/3 metabotropic glutamate receptors negatively regulates the stimulation of inositol phospholipid hydrolysis mediated by 5-hydroxytryptamine2A serotonin receptors in the frontal cortex of living mice.
Topics: Amino Acids; Amphetamines; Animals; Bridged Bicyclo Compounds, Heterocyclic; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Frontal Lobe; Hydrolysis; Male; Mice; Mice, Inbred Strains; Mice, Knockout; Phosphatidylinositols; Pyridines; Receptor, Serotonin, 5-HT2A; Receptors, Metabotropic Glutamate; Sulfonamides; Xanthenes | 2009 |
A transient receptor potential-like channel mediates synaptic transmission in rod bipolar cells.
Topics: Amino Acids; Anilides; Animals; Arachidonic Acids; Capsaicin; Cinnamates; Endocannabinoids; Excitatory Amino Acid Antagonists; Glutamic Acid; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Knockout; Polyunsaturated Alkamides; Propionates; Receptors, Metabotropic Glutamate; Retinal Bipolar Cells; Ruthenium Red; Synaptic Transmission; Transient Receptor Potential Channels; TRPM Cation Channels; TRPV Cation Channels; Xanthenes | 2009 |
Use of MGLUR2 and MGLUR3 knockout mice to explore in vivo receptor specificity of the MGLUR2/3 selective antagonist LY341495.
Topics: Amino Acids; Analysis of Variance; Animals; Brain; Cell Count; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Habituation, Psychophysiologic; Immunohistochemistry; Locomotion; Male; Mice; Mice, Knockout; Photomicrography; Proto-Oncogene Proteins c-fos; Receptors, Metabotropic Glutamate; Xanthenes | 2009 |
Neuroprotective effects of group II metabotropic glutamate receptor agonist DCG-IV on hippocampal neurons in transient forebrain ischemia.
Topics: Amino Acids; Animals; Carotid Stenosis; Cerebrovascular Circulation; Cyclopropanes; Extracellular Space; Glutamic Acid; Glycine; Hippocampus; Ischemic Attack, Transient; Male; Microdialysis; Neurons; Neuroprotective Agents; Prosencephalon; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Xanthenes | 2009 |
Involvement of Group II mGluRs in mossy fiber LTD.
Topics: Amino Acids; Amino Acids, Dicarboxylic; Animals; Cycloleucine; Cyclopropanes; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glycine; Hippocampus; In Vitro Techniques; Long-Term Synaptic Depression; Mice; Mice, Inbred C57BL; Neural Inhibition; Neurons; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Synaptic Transmission; Xanthenes | 2009 |
Oral administration of the NAALADase inhibitor GPI-5693 attenuates cocaine-induced reinstatement of drug-seeking behavior in rats.
Topics: Administration, Oral; Amino Acids; Animals; Behavior, Animal; Cocaine; Cocaine-Related Disorders; Dipeptides; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glutamate Carboxypeptidase II; Glutarates; Male; Rats; Receptors, Metabotropic Glutamate; Reward; Self Administration; Stereoisomerism; Sucrose; Sulfhydryl Compounds; Time Factors; Xanthenes | 2010 |
Group II metabotropic glutamate receptor activation by agonist LY379268 treatment increases the expression of brain derived neurotrophic factor in the mouse brain.
Topics: Amino Acids; Animals; Brain; Brain-Derived Neurotrophic Factor; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Hippocampus; Male; Mice; Mice, Inbred C57BL; Neurons; Receptors, Metabotropic Glutamate; RNA, Messenger; Time Factors; Up-Regulation; Xanthenes | 2010 |
Excitotoxicity effects of glutamate on human neuroblastoma SH-SY5Y cells via oxidative damage.
Topics: Abietanes; Amino Acids; Antioxidants; Calcium; Cell Line, Tumor; Cell Survival; Cytosol; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Extracellular Space; Glutamic Acid; Glutathione; Humans; Indoles; L-Lactate Dehydrogenase; Malondialdehyde; Oxidative Stress; Phenanthrenes; Superoxide Dismutase; Time Factors; Xanthenes | 2010 |
Extinction of cued fear memory involves a distinct form of depotentiation at cortical input synapses onto the lateral amygdala.
Topics: Acoustic Stimulation; Amino Acids; Amygdala; Animals; Behavior, Animal; Cerebral Cortex; Conditioning, Classical; Cues; Electric Stimulation; Endocytosis; Excitatory Amino Acid Antagonists; Extinction, Psychological; Fear; In Vitro Techniques; Long-Term Synaptic Depression; Male; Memory; Methoxyhydroxyphenylglycol; Patch-Clamp Techniques; Peptides; Rats; Rats, Sprague-Dawley; Statistics, Nonparametric; Xanthenes | 2009 |
Group II metabotropic glutamate receptor stimulation triggers production and release of Alzheimer's amyloid(beta)42 from isolated intact nerve terminals.
Topics: Alzheimer Disease; Amino Acids; Amyloid beta-Peptides; Amyloid beta-Protein Precursor; Amyloid Precursor Protein Secretases; Animals; Humans; Methoxyhydroxyphenylglycol; Mice; Mice, Transgenic; Nerve Endings; Peptide Fragments; Receptors, Metabotropic Glutamate; Signal Transduction; Xanthenes | 2010 |
Effects of metabotropic glutamate receptor 2/3 agonism and antagonism on schizophrenia-like cognitive deficits induced by phencyclidine in rats.
Topics: Amino Acids; Animals; Antipsychotic Agents; Bridged Bicyclo Compounds, Heterocyclic; Cognition; Excitatory Amino Acid Agents; Male; Phencyclidine; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Schizophrenia; Time Factors; Xanthenes | 2010 |
AMPA receptor mediates mGlu 2/3 receptor antagonist-induced dopamine release in the rat nucleus accumbens shell.
Topics: Amino Acids; Animals; Dioxoles; Dopamine; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Male; Microdialysis; Nucleus Accumbens; Piperidines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Metabotropic Glutamate; Xanthenes | 2010 |
Orally active glutamate carboxypeptidase II inhibitor 2-MPPA attenuates dizocilpine-induced prepulse inhibition deficits in mice.
Topics: Administration, Oral; Amino Acids; Animals; Antipsychotic Agents; Bridged Bicyclo Compounds; Dipeptides; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Glutamate Carboxypeptidase II; Glutarates; Male; Mice; Neural Inhibition; Schizophrenia; Sensory Gating; Sulfhydryl Compounds; Xanthenes | 2011 |
Targeting group II metabotropic glutamate (mGlu) receptors for the treatment of psychosis associated with Alzheimer's disease: selective activation of mGlu2 receptors amplifies beta-amyloid toxicity in cultured neurons, whereas dual activation of mGlu2 an
Topics: Alzheimer Disease; Amino Acids; Amyloid beta-Peptides; Animals; Antipsychotic Agents; Astrocytes; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Mice; Mice, Knockout; Neurons; Neuroprotective Agents; Psychotic Disorders; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Reverse Transcriptase Polymerase Chain Reaction; Sulfonamides; Transforming Growth Factor beta1; Xanthenes | 2011 |
Metabotropic glutamate receptor blockade in nucleus accumbens shell shifts affective valence towards fear and disgust.
Topics: Affect; Amino Acids; Analgesics, Non-Narcotic; Animals; Appetitive Behavior; Excitatory Amino Acid Antagonists; Fear; Male; Motivation; Nucleus Accumbens; Pleasure; Proto-Oncogene Proteins c-fos; Quinine; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Schizophrenia; Xanthenes | 2011 |
Baclofen and adenosine inhibition of synaptic transmission at CA3-CA1 synapses display differential sensitivity to K+ channel blockade.
Topics: 4-Aminopyridine; Adenosine; Adenosine A1 Receptor Antagonists; Amino Acids; Animals; Baclofen; Barium; Bee Venoms; CA1 Region, Hippocampal; CA3 Region, Hippocampal; Cesium; Excitatory Postsynaptic Potentials; In Vitro Techniques; Male; Potassium Channel Blockers; Rats; Rats, Wistar; Receptor, Adenosine A1; Receptors, Metabotropic Glutamate; Synapses; Synaptic Transmission; Theophylline; Xanthenes | 2011 |
Group II metabotropic glutamate receptors in the striatum of non-human primates: dysregulation following chronic cocaine self-administration.
Topics: Amino Acids; Animals; Antimetabolites; Autoradiography; Carbon Isotopes; Cocaine; Conditioning, Operant; Corpus Striatum; Deoxyglucose; Dopamine Uptake Inhibitors; Excitatory Amino Acid Antagonists; Macaca mulatta; Male; Protein Binding; Receptors, AMPA; Receptors, Metabotropic Glutamate; Reinforcement Schedule; Self Administration; Tritium; Xanthenes | 2011 |
Regulation of Akt and Wnt signaling by the group II metabotropic glutamate receptor antagonist LY341495 and agonist LY379268.
Topics: Amino Acids; Animals; Bridged Bicyclo Compounds, Heterocyclic; Corpus Striatum; Glycogen Synthase Kinase 3; Male; Motor Activity; Prefrontal Cortex; Proto-Oncogene Proteins c-akt; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Signal Transduction; Wnt Proteins; Xanthenes | 2011 |
Enhancement of CA3 hippocampal network activity by activation of group II metabotropic glutamate receptors.
Topics: Action Potentials; Amino Acids; Animals; CA3 Region, Hippocampal; Cyclopropanes; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glycine; Interneurons; Mice; Mice, Knockout; Microscopy, Electron; Nerve Net; Patch-Clamp Techniques; Pyramidal Cells; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Theta Rhythm; Xanthenes | 2011 |
A role for nyctalopin, a small leucine-rich repeat protein, in localizing the TRP melastatin 1 channel to retinal depolarizing bipolar cell dendrites.
Topics: Amino Acids; Animals; Bacterial Proteins; Biophysics; Cell Line, Transformed; Dendrites; Electric Stimulation; Excitatory Amino Acid Antagonists; Gene Expression Regulation, Developmental; Humans; In Vitro Techniques; Leucine-Rich Repeat Proteins; Luminescent Proteins; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Transgenic; Models, Biological; Patch-Clamp Techniques; Proteins; Proteoglycans; Retina; Retinal Bipolar Cells; Transfection; TRPM Cation Channels; Xanthenes | 2011 |
Estradiol attenuates the adenosine triphosphate-induced increase of intracellular calcium through group II metabotropic glutamate receptors in rat dorsal root ganglion neurons.
Topics: Adenosine Triphosphate; Amino Acids; Animals; Calcium; Cells, Cultured; Estradiol; Estrogens; Female; Ganglia, Spinal; Neurons; Rats; Rats, Long-Evans; Receptors, Estrogen; Receptors, Metabotropic Glutamate; Xanthenes | 2011 |
Blockade of GABA(B) receptors facilitates evoked neurotransmitter release at spinal dorsal horn synapse.
Topics: Amino Acids; Animals; Baclofen; Benzylamines; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Agonists; GABA-A Receptor Antagonists; In Vitro Techniques; Male; Neurotransmitter Agents; Nipecotic Acids; Patch-Clamp Techniques; Phosphinic Acids; Posterior Horn Cells; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Spinal Cord; Synapses; Synaptic Potentials; Tiagabine; Xanthenes | 2011 |
Group II/III metabotropic glutamate receptors exert endogenous activity-dependent modulation of TRPV1 receptors on peripheral nociceptors.
Topics: Amino Acids; Animals; Calcium; Capsaicin; Cells, Cultured; Cytosol; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Formaldehyde; Glutamic Acid; Hot Temperature; Male; Nociceptors; Pain; Pain Measurement; Peripheral Nervous System; Proline; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Skin; TRPV Cation Channels; Xanthenes | 2011 |
Involvement of the mammalian target of rapamycin signaling in the antidepressant-like effect of group II metabotropic glutamate receptor antagonists.
Topics: Amino Acids; Analysis of Variance; Animals; Bridged Bicyclo Compounds; Depression; Dicarboxylic Acids; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Hindlimb Suspension; Ketamine; Male; Mice; Mice, Inbred ICR; Receptors, Metabotropic Glutamate; Sirolimus; Time Factors; TOR Serine-Threonine Kinases; Xanthenes | 2011 |
Activation of group II metabotropic glutamate receptors induces long-term depression of excitatory synaptic transmission in the substantia nigra pars reticulata.
Topics: Amino Acids; Animals; Basal Ganglia; Bridged Bicyclo Compounds, Heterocyclic; Data Interpretation, Statistical; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; Mice; Mice, Knockout; Neuronal Plasticity; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Substantia Nigra; Synaptic Transmission; Xanthenes | 2011 |
Excitatory amino acid transporter 2 and excitatory amino acid transporter 1 negatively regulate calcium-dependent proliferation of hippocampal neural progenitor cells and are persistently upregulated after injury.
Topics: Amino Acids; Animals; Calcium; Cell Proliferation; Cells, Cultured; Dentate Gyrus; Excitatory Amino Acid Antagonists; Excitatory Amino Acid Transporter 1; Excitatory Amino Acid Transporter 2; Mice; Mice, Transgenic; Neural Stem Cells; RNA, Small Interfering; Xanthenes | 2011 |
mTOR activation is required for the antidepressant effects of mGluR₂/₃ blockade.
Topics: Amino Acids; Animals; Disks Large Homolog 4 Protein; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Gene Expression Regulation; Intracellular Signaling Peptides and Proteins; Ketamine; Male; Membrane Proteins; Prefrontal Cortex; Rats; Receptors, Metabotropic Glutamate; Signal Transduction; Swimming; Synapsins; Synaptosomes; TOR Serine-Threonine Kinases; Xanthenes | 2012 |
Radiosynthesis of PET radiotracer as a prodrug for imaging group II metabotropic glutamate receptors in vivo.
Topics: Amino Acids; Animals; Brain; Corpus Striatum; Hippocampus; Male; Positron-Emission Tomography; Prodrugs; Protein Binding; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Xanthenes | 2012 |
Effects of microinjections of Group II metabotropic glutamate agents into the amygdala on sleep.
Topics: Amino Acids; Amygdala; Animals; Arousal; Bridged Bicyclo Compounds, Heterocyclic; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Male; Microinjections; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Sleep; Sleep, REM; Wakefulness; Xanthenes | 2012 |
Actions of Xanthurenic acid, a putative endogenous Group II metabotropic glutamate receptor agonist, on sensory transmission in the thalamus.
Topics: Action Potentials; Administration, Intravenous; Afferent Pathways; Allosteric Regulation; Amino Acids; Animals; Bridged Bicyclo Compounds; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Iontophoresis; Male; Neural Inhibition; Neurons; Rats; Rats, Wistar; Ventral Thalamic Nuclei; Vibrissae; Xanthenes; Xanthurenates | 2013 |
Selective activation of either mGlu2 or mGlu3 receptors can induce LTD in the amygdala.
Topics: Amino Acids; Amino Acids, Dicarboxylic; Amygdala; Animals; Bridged Bicyclo Compounds; Cyclopropanes; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Long-Term Synaptic Depression; Mice; Mice, Knockout; Rats; Rats, Mutant Strains; Rats, Wistar; Receptors, Metabotropic Glutamate; Xanthenes | 2013 |
G-protein-mediated inhibition of the Trp channel TRPM1 requires the Gβγ dimer.
Topics: Amino Acids; Animals; Capsaicin; Cells, Cultured; Excitatory Amino Acid Antagonists; Glutamic Acid; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein beta Subunits; GTP-Binding Protein gamma Subunits; HEK293 Cells; Humans; Light; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Knockout; Protein Binding; Protein Multimerization; Receptors, Metabotropic Glutamate; Retinal Bipolar Cells; TRPM Cation Channels; Xanthenes | 2012 |
The metabotropic glutamate 2/3 receptor antagonist LY341495 differentially affects recognition memory in rats.
Topics: Amino Acids; Animals; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Extinction, Psychological; Male; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Recognition, Psychology; Xanthenes | 2012 |
Glycine release is regulated by metabotropic glutamate receptors sensitive to mGluR2/3 ligands and activated by N-acetylaspartylglutamate (NAAG).
Topics: Amino Acids; Animals; Bridged Bicyclo Compounds, Heterocyclic; Dipeptides; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Exocytosis; Glutamic Acid; Glycine; Male; Mice; Potassium Chloride; Receptors, Metabotropic Glutamate; Spinal Cord; Synaptosomes; Xanthenes | 2013 |
Depolarizing bipolar cell dysfunction due to a Trpm1 point mutation.
Topics: Action Potentials; Amino Acid Sequence; Amino Acids; Animals; Capsaicin; Chromosome Mapping; Chromosomes, Mammalian; Dendrites; Disease Models, Animal; Exons; Eye Diseases, Hereditary; Genetic Diseases, X-Linked; Heterozygote; Mice; Mice, Transgenic; Molecular Sequence Data; Mutation, Missense; Myopia; Night Blindness; Point Mutation; Retina; Retinal Bipolar Cells; Sequence Analysis, DNA; Threonine; TRPM Cation Channels; Xanthenes | 2012 |
Synthesis and characterization of two PET radioligands for the metabotropic glutamate 1 (mGlu1) receptor.
Topics: Amino Acids; Animals; Brain; Carbon Radioisotopes; CHO Cells; Cricetinae; Cricetulus; Excitatory Amino Acid Antagonists; Fluorine Radioisotopes; Ligands; Male; Papio; Positron-Emission Tomography; Pyridines; Quinolines; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Metabotropic Glutamate; Tissue Distribution; Xanthenes | 2012 |
Group II metabotropic glutamate receptors depress synaptic transmission onto subicular burst firing neurons.
Topics: Amino Acids; Amino Acids, Dicarboxylic; Animals; CA1 Region, Hippocampal; CA3 Region, Hippocampal; Cyclopropanes; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Female; Glutamic Acid; Glycine; Hippocampus; Male; Neurons; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Synaptic Transmission; Xanthenes | 2012 |
Modafinil attenuates reinstatement of cocaine seeking: role for cystine-glutamate exchange and metabotropic glutamate receptors.
Topics: Amino Acid Transport System y+; Amino Acids; Analysis of Variance; Animals; Benzhydryl Compounds; Cocaine; Cocaine-Related Disorders; Disease Models, Animal; Dopamine Uptake Inhibitors; Drug-Seeking Behavior; Excitatory Amino Acid Antagonists; Extinction, Psychological; Glutamates; Male; Microdialysis; Microinjections; Modafinil; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Secondary Prevention; Self Administration; Wakefulness-Promoting Agents; Xanthenes | 2014 |
Role of BDNF/TrkB signaling in antidepressant-like effects of a group II metabotropic glutamate receptor antagonist in animal models of depression.
Topics: Amino Acids; Animals; Antidepressive Agents; Behavior, Animal; Brain-Derived Neurotrophic Factor; Depressive Disorder; Disease Models, Animal; Excitatory Amino Acid Antagonists; Exploratory Behavior; Hindlimb Suspension; Male; Mice; Mice, Inbred C57BL; Mice, Inbred ICR; Receptor, trkB; Receptors, Metabotropic Glutamate; Signal Transduction; Xanthenes | 2013 |
Regulation of synaptic currents by mGluR2 at reciprocal synapses in the mouse accessory olfactory bulb.
Topics: Action Potentials; Amino Acids; Animals; Anticonvulsants; Calcium Channels; Cyclopropanes; Dendrites; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glycine; Mice; Mice, Inbred BALB C; Mutation; Olfactory Bulb; Receptors, Metabotropic Glutamate; Synapses; Xanthenes | 2013 |
Type-3 metabotropic glutamate receptors regulate chemoresistance in glioma stem cells, and their levels are inversely related to survival in patients with malignant gliomas.
Topics: Amino Acids; Animals; Antineoplastic Agents, Alkylating; Chemotherapy, Adjuvant; Combined Modality Therapy; Dacarbazine; DNA Methylation; Drug Resistance, Neoplasm; Glioblastoma; Humans; Mice; Neoplastic Stem Cells; NF-kappa B; O(6)-Methylguanine-DNA Methyltransferase; Phosphatidylinositol 3-Kinases; Promoter Regions, Genetic; Receptors, Metabotropic Glutamate; RNA, Messenger; Signal Transduction; Survival Rate; Temozolomide; Transplantation, Heterologous; Tumor Cells, Cultured; Xanthenes | 2013 |
Anxiety-like behavior of prenatally stressed rats is associated with a selective reduction of glutamate release in the ventral hippocampus.
Topics: Amino Acids; Animals; Anxiety; Behavior, Animal; Benzylamines; Excitatory Amino Acid Antagonists; Female; GABA-A Receptor Antagonists; Glutamic Acid; Hippocampus; Kainic Acid; Male; Munc18 Proteins; Phosphinic Acids; Pregnancy; Prenatal Exposure Delayed Effects; R-SNARE Proteins; rab3A GTP-Binding Protein; Rats; Rats, Sprague-Dawley; Seizures; Stress, Psychological; Synapsins; Synaptic Transmission; Synaptophysin; Syntaxin 1; Xanthenes | 2012 |
Characterisation of an mGlu8 receptor-selective agonist and antagonist in the lateral and medial perforant path inputs to the dentate gyrus.
Topics: Amino Acids; Amino Acids, Dicarboxylic; Animals; Bridged Bicyclo Compounds; Dentate Gyrus; Female; Male; Mice; Mice, 129 Strain; Mice, Inbred C57BL; Mice, Knockout; Neural Pathways; Perforant Pathway; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Xanthenes | 2013 |
Chronic treatment with LY341495 decreases 5-HT(2A) receptor binding and hallucinogenic effects of LSD in mice.
Topics: Amino Acids; Animals; Drug Antagonism; Early Growth Response Protein 1; Early Growth Response Protein 2; Hallucinogens; Lysergic Acid Diethylamide; Male; Mice; Mice, Knockout; Proto-Oncogene Proteins c-fos; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptors, Metabotropic Glutamate; Somatosensory Cortex; Stereotyped Behavior; Xanthenes | 2013 |
L-acetylcarnitine causes rapid antidepressant effects through the epigenetic induction of mGlu2 receptors.
Topics: Acetylation; Acetylcarnitine; Amino Acids; Animals; Antidepressive Agents; Clomipramine; Epigenesis, Genetic; Excitatory Amino Acid Antagonists; Hippocampus; Histone Deacetylases; Histones; Humans; Male; Mice; Mice, Knockout; Nerve Tissue Proteins; NF-kappa B; Nootropic Agents; Prefrontal Cortex; Rats; Receptors, Metabotropic Glutamate; Selective Serotonin Reuptake Inhibitors; Stress, Psychological; Time Factors; Xanthenes | 2013 |
Effect of an mGlu2/3 receptor antagonist on depressive behavior induced by withdrawal from chronic treatment with methamphetamine.
Topics: Amino Acids; Analysis of Variance; Animals; Central Nervous System Stimulants; Depression; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Delivery Systems; Drug Interactions; Excitatory Amino Acid Antagonists; Immobility Response, Tonic; Male; Methamphetamine; Motor Activity; Rats; Rats, Sprague-Dawley; Substance Withdrawal Syndrome; Swimming; Xanthenes | 2013 |
Antagonists reversibly reverse chemical LTD induced by group I, group II and group III metabotropic glutamate receptors.
Topics: Amino Acids; Animals; Brain; Excitatory Amino Acid Antagonists; Glycine; Long-Term Synaptic Depression; Mice; Neural Pathways; Rats; Receptors, Metabotropic Glutamate; Xanthenes | 2013 |
Contribution of opioid and metabotropic glutamate receptor mechanisms to inhibition of bladder overactivity by tibial nerve stimulation.
Topics: Amino Acids; Animals; Cats; Electric Stimulation Therapy; Excitatory Amino Acid Antagonists; Female; Male; Naloxone; Narcotic Antagonists; Receptors, Metabotropic Glutamate; Receptors, Opioid; Tibial Nerve; Urinary Bladder; Urinary Bladder, Overactive; Xanthenes | 2013 |
Effects of ketamine and LY341495 on the depressive-like behavior of repeated corticosterone-injected rats.
Topics: Amino Acids; Animals; Corticosterone; Depressive Disorder, Treatment-Resistant; Disease Models, Animal; Drug Administration Schedule; Immobility Response, Tonic; Injections, Subcutaneous; Ketamine; Male; Rats; Receptors, Metabotropic Glutamate; Xanthenes | 2013 |
Group II metabotropic glutamate receptor agonist LY379268 regulates AMPA receptor trafficking in prefrontal cortical neurons.
Topics: Amino Acids; Animals; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Cells, Cultured; Dactinomycin; Disks Large Homolog 4 Protein; Enzyme Activation; Extracellular Signal-Regulated MAP Kinases; Flavonoids; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Intracellular Signaling Peptides and Proteins; Intracellular Space; Membrane Proteins; Neurons; Prefrontal Cortex; Protein Kinase Inhibitors; Protein Subunits; Protein Transport; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Metabotropic Glutamate; Synapsins; Transcription, Genetic; Xanthenes | 2013 |
Stimulation of metabotropic glutamate (mGlu) 2 receptor and blockade of mGlu1 receptor improve social memory impairment elicited by MK-801 in rats.
Topics: Amino Acids; Animals; Bridged Bicyclo Compounds, Heterocyclic; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Male; Memory Disorders; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Recognition, Psychology; Xanthenes | 2013 |
Synergistic inhibition of survival, proliferation, and migration of U87 cells with a combination of LY341495 and Iressa.
Topics: Amino Acids; Antineoplastic Agents; Apoptosis; Cell Line, Tumor; Cell Movement; Cell Proliferation; Cell Survival; Dose-Response Relationship, Drug; Drug Synergism; Gefitinib; Glioblastoma; Glutamic Acid; Humans; Quinazolines; Riluzole; Xanthenes | 2013 |
Chronic treatment with MPEP, an mGlu5 receptor antagonist, normalizes basal ganglia glutamate neurotransmission in L-DOPA-treated parkinsonian monkeys.
Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Basal Ganglia; Corpus Striatum; Dyskinesia, Drug-Induced; Female; Imidazoles; Levodopa; Macaca fascicularis; Oximes; Parkinsonian Disorders; Phenols; Piperidines; Pyridines; Quinazolines; Radioligand Assay; Receptor, Metabotropic Glutamate 5; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Tritium; Xanthenes | 2013 |
Pharmacological characterization of JNJ-40068782, a new potent, selective, and systemically active positive allosteric modulator of the mGlu2 receptor and its radioligand [3H]JNJ-40068782.
Topics: Amino Acids; Animals; Autoradiography; Binding, Competitive; Brain Chemistry; Calcium; Cell Membrane; Cerebral Cortex; CHO Cells; Cricetinae; Cricetulus; Cyclopropanes; Excitatory Amino Acid Agents; Excitatory Amino Acid Agonists; Glycine; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Isotope Labeling; Ligands; Male; Mice; Motor Activity; Piperidines; Pyridones; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Sleep; Tritium; Xanthenes | 2013 |
Enhancement of long-term depression by soluble amyloid β protein in rat hippocampus is mediated by metabotropic glutamate receptor and involves activation of p38MAPK, STEP and caspase-3.
Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Amyloid beta-Peptides; Animals; Caspase 3; Electric Stimulation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Hippocampus; Immunosuppressive Agents; In Vitro Techniques; Long-Term Synaptic Depression; Male; Methoxyhydroxyphenylglycol; p38 Mitogen-Activated Protein Kinases; Patch-Clamp Techniques; Peptide Fragments; Protein Tyrosine Phosphatases, Non-Receptor; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Sirolimus; Xanthenes | 2013 |
Cerebral 5-HT2A receptor binding, but not mGluR2, is increased in tryptophan hydroxylase 2 decrease-of-function mice.
Topics: Amino Acids; Animals; Brain; Gene Knock-In Techniques; Mice; Mice, Transgenic; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptors, Metabotropic Glutamate; Tryptophan Hydroxylase; Up-Regulation; Xanthenes | 2013 |
Activation of synaptic group II metabotropic glutamate receptors induces long-term depression at GABAergic synapses in CNS neurons.
Topics: Amino Acids; Animals; Chick Embryo; Cochlear Nucleus; Cyclopropanes; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABAergic Neurons; Glycine; Inhibitory Postsynaptic Potentials; Long-Term Synaptic Depression; Neural Inhibition; Receptors, Metabotropic Glutamate; Synapses; Synaptic Transmission; Xanthenes | 2013 |
Serotonin-1A receptor stimulation mediates effects of a metabotropic glutamate 2/3 receptor antagonist, 2S-2-amino-2-(1S,2S-2-carboxycycloprop-1-yl)-3-(xanth-9-yl)propanoic acid (LY341495), and an N-methyl-D-aspartate receptor antagonist, ketamine, in the
Topics: Amino Acids; Animals; Antidepressive Agents; Dioxoles; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Feeding Behavior; Fenclonine; Ketamine; Male; Mice, Inbred C57BL; Neuropsychological Tests; Piperazines; Piperidines; Pyridines; Quinoxalines; Receptors, AMPA; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Ritanserin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Tryptophan Hydroxylase; Xanthenes | 2014 |
mGlu3 receptor blockade inhibits proliferation and promotes astrocytic phenotype in glioma stem cells.
Topics: AC133 Antigen; Amino Acids; Animals; Antigens, CD; Astrocytes; Bridged Bicyclo Compounds, Heterocyclic; Cell Differentiation; Cell Proliferation; Epidermal Growth Factor; Fibroblast Growth Factor 2; Glioma; Glycoproteins; Humans; Male; Mice; Mice, Inbred BALB C; Mice, Nude; Neoplastic Stem Cells; Peptides; Phenotype; Receptors, Metabotropic Glutamate; Recombinant Proteins; Transplantation, Heterologous; Xanthenes | 2014 |
N-acetylcysteine modulates hallucinogenic 5-HT(2A) receptor agonist-mediated responses: behavioral, molecular, and electrophysiological studies.
Topics: Acetylcysteine; Action Potentials; Amino Acids; Amphetamines; Animals; Benzoates; Bicuculline; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Early Growth Response Protein 2; Excitatory Amino Acid Antagonists; Free Radical Scavengers; GABA-A Receptor Antagonists; Glycine; Hallucinations; Hallucinogens; Male; Mice; Proto-Oncogene Proteins c-fos; Receptors, Metabotropic Glutamate; Xanthenes | 2014 |
Overexpression of Shati/Nat8l, an N-acetyltransferase, in the nucleus accumbens attenuates the response to methamphetamine via activation of group II mGluRs in mice.
Topics: Acetyltransferases; Amino Acids; Animals; Aspartic Acid; Conditioning, Psychological; Corpus Striatum; Dipeptides; Dopamine; Male; Methamphetamine; Mice; Mice, Transgenic; Motor Activity; Nucleus Accumbens; Receptors, Metabotropic Glutamate; Xanthenes | 2014 |
A real-time method for measuring cAMP production modulated by Gαi/o-coupled metabotropic glutamate receptors.
Topics: Amino Acids; Animals; Biosensing Techniques; Buffers; Cell Culture Techniques; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Glutamic Acid; GTP-Binding Protein alpha Subunits, Gi-Go; Luciferases, Firefly; Radioligand Assay; Receptors, Metabotropic Glutamate; Reproducibility of Results; Sensitivity and Specificity; Transfection; Xanthenes | 2014 |
Blockade of the metabotropic glutamate (mGluR2) modulates arousal through vigilance states transitions: evidence from sleep-wake EEG in rodents.
Topics: Amino Acids; Animals; Arousal; Body Temperature; Cerebral Cortex; Electroencephalography; Excitatory Amino Acid Antagonists; Locomotion; Male; Mice; Mice, Knockout; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Sleep; Wakefulness; Xanthenes | 2014 |
Requirement of AMPA receptor stimulation for the sustained antidepressant activity of ketamine and LY341495 during the forced swim test in rats.
Topics: Adaptation, Psychological; Amino Acids; Animals; Antidepressive Agents; Depression; Disease Models, Animal; Excitatory Amino Acid Antagonists; Ketamine; Male; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Stress, Psychological; Swimming; Time Factors; Xanthenes | 2014 |
Evaluation of 5-HT2A and mGlu2/3 receptors in postmortem prefrontal cortex of subjects with major depressive disorder: effect of antidepressant treatment.
Topics: Amino Acids; Animals; Antidepressive Agents; Citalopram; Depressive Disorder, Major; Down-Regulation; Female; Humans; Ketanserin; Male; Mianserin; Middle Aged; Mirtazapine; Morpholines; Prefrontal Cortex; Radioligand Assay; Rats, Sprague-Dawley; Reboxetine; Receptor, Serotonin, 5-HT2A; Receptors, Metabotropic Glutamate; RNA, Messenger; Tritium; Xanthenes | 2014 |
The peptidic antidepressant spadin interacts with prefrontal 5-HT(4) and mGluR(2) receptors in the control of serotonergic function.
Topics: Amino Acids; Aniline Compounds; Animals; Antidepressive Agents; Calcium; Dorsal Raphe Nucleus; Early Growth Response Protein 1; Excitatory Amino Acid Antagonists; Indoles; Male; Mice, Inbred C57BL; Mice, Knockout; Peptides; Piperazines; Piperidines; Potassium Channels, Tandem Pore Domain; Prefrontal Cortex; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Receptors, Serotonin, 5-HT4; Serotonergic Neurons; Serotonin 5-HT4 Receptor Agonists; Serotonin Receptor Agonists; Sulfonamides; Xanthenes | 2016 |
Epigenetic upregulation of metabotropic glutamate receptor 2 in the spinal cord attenuates oestrogen-induced visceral hypersensitivity.
Topics: Acetylation; Amino Acids; Animals; Disease Models, Animal; Epigenesis, Genetic; Estradiol; Estrogens; Female; Histone Deacetylase Inhibitors; Histones; Hydroxamic Acids; Nociception; Ovariectomy; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; RNA, Messenger; Spinal Cord; Up-Regulation; Viscera; Visceral Pain; Vorinostat; Xanthenes | 2015 |
Increased metabotropic glutamate 2/3 receptor binding in the perigenual anterior cingulate cortex of Cloninger type 2 alcoholics: a whole-hemisphere autoradiography study.
Topics: Adolescent; Adult; Aged; Alcoholism; Amino Acids; Autoradiography; Brain; Case-Control Studies; Female; Gyrus Cinguli; Humans; Male; Middle Aged; Receptors, Metabotropic Glutamate; Xanthenes; Young Adult | 2015 |
Investigating glutamatergic mechanism in attention and impulse control using rats in a modified 5-choice serial reaction time task.
Topics: Amino Acids; Animals; Attention; Disease Models, Animal; Dizocilpine Maleate; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Impulsive Behavior; Male; N-Methylaspartate; Prefrontal Cortex; Rats; Reaction Time; Xanthenes | 2014 |
Role of group II metabotropic glutamate receptors (mGluR2/3) blockade on long-term potentiation in the dentate gyrus region of hippocampus in rats fed with high-fat diet.
Topics: Amino Acids; Animals; Dentate Gyrus; Diet, High-Fat; Excitatory Amino Acid Antagonists; Long-Term Potentiation; Male; Microinjections; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Xanthenes | 2015 |
Group II metabotropic glutamate receptor antagonism prevents the antiallodynic effects of R-isovaline.
Topics: Amino Acids; Analgesics; Animals; Dinoprostone; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Female; GABA-B Receptor Antagonists; Hyperalgesia; Mice; Pain Threshold; Receptors, GABA-B; Receptors, Metabotropic Glutamate; Valine; Xanthenes | 2015 |
N-acetyl-cysteine, a drug that enhances the endogenous activation of group-II metabotropic glutamate receptors, inhibits nociceptive transmission in humans.
Topics: Acetylcysteine; Adult; Amino Acids; Analgesics; Dose-Response Relationship, Drug; Double-Blind Method; Female; Humans; Male; Middle Aged; Pain; Receptors, Metabotropic Glutamate; Treatment Outcome; Xanthenes; Young Adult | 2015 |
Group II mGluRs modulate baseline and arthritis pain-related synaptic transmission in the rat medial prefrontal cortex.
Topics: Amino Acids; Animals; Arthritis, Experimental; Bridged Bicyclo Compounds, Heterocyclic; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Inhibitory Postsynaptic Potentials; Kaolin; Miniature Postsynaptic Potentials; Pain; Patch-Clamp Techniques; Prefrontal Cortex; Pyramidal Cells; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Synaptic Transmission; Tissue Culture Techniques; Xanthenes | 2015 |
The Female Encounter Test: A Novel Method for Evaluating Reward-Seeking Behavior or Motivation in Mice.
Topics: Amino Acids; Animals; Antidepressive Agents, Second-Generation; Castration; Choice Behavior; Corticosterone; Depressive Disorder; Disease Models, Animal; Equipment Design; Estrous Cycle; Excitatory Amino Acid Antagonists; Female; Fluvoxamine; Lipopolysaccharides; Male; Mice; Motivation; Nucleus Accumbens; Psychological Tests; Reward; Social Behavior; Social Isolation; Xanthenes | 2015 |
mGluR2/3 in the Lateral Amygdala is Required for Fear Extinction: Cortical Input Synapses onto the Lateral Amygdala as a Target Site of the mGluR2/3 Action.
Topics: Amino Acids; Amygdala; Animals; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Extinction, Psychological; Fear; Freezing Reaction, Cataleptic; Male; Patch-Clamp Techniques; Presynaptic Terminals; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Tissue Culture Techniques; Xanthenes | 2015 |
Activation of mGluR2/3 following stress hormone exposure restores sensitivity to alcohol in rats.
Topics: Alcohol Drinking; Amino Acids; Animals; Bridged Bicyclo Compounds, Heterocyclic; Corticosterone; Discrimination Learning; Ethanol; Male; Rats; Rats, Long-Evans; Receptors, AMPA; Self Administration; Xanthenes | 2015 |
The Antidepressant Effects of an mGlu2/3 Receptor Antagonist and Ketamine Require AMPA Receptor Stimulation in the mPFC and Subsequent Activation of the 5-HT Neurons in the DRN.
Topics: Amino Acids; Animals; Antidepressive Agents; Depression; Dorsal Raphe Nucleus; Fenclonine; Ketamine; Male; Mice; Mice, Inbred C57BL; Neural Pathways; Prefrontal Cortex; Quinoxalines; Receptors, AMPA; Receptors, Metabotropic Glutamate; Serotonergic Neurons; Xanthenes | 2016 |
Mechanisms regulating spill-over of synaptic glutamate to extrasynaptic NMDA receptors in mouse substantia nigra dopaminergic neurons.
Topics: Amino Acids; Animals; Aspartic Acid; Dizocilpine Maleate; Dopaminergic Neurons; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Male; Mice; Mice, Inbred C57BL; Receptors, N-Methyl-D-Aspartate; Substantia Nigra; Synapses; Xanthenes | 2015 |
Reversal of alcohol dependence-induced deficits in cue-guided behavior via mGluR2/3 signaling in mice.
Topics: Adaptation, Psychological; Alcoholism; Amino Acids; Animals; Bridged Bicyclo Compounds, Heterocyclic; Conditioning, Operant; Consummatory Behavior; Cues; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Male; Mice; Mice, Inbred C57BL; Psychomotor Performance; Receptors, AMPA; Reward; Self Administration; Signal Transduction; Xanthenes | 2016 |
Lower [3H]LY341495 binding to mGlu2/3 receptors in the anterior cingulate of subjects with major depressive disorder but not bipolar disorder or schizophrenia.
Topics: Amino Acids; Animals; Antidepressive Agents; Bipolar Disorder; Brain; Depressive Disorder, Major; Excitatory Amino Acid Antagonists; Female; Fluoxetine; Gyrus Cinguli; Humans; Imipramine; Male; Middle Aged; Radioligand Assay; Radionuclide Imaging; Rats; Receptors, Metabotropic Glutamate; Schizophrenia; Tritium; Xanthenes | 2016 |
Activation of a Temporal Memory in Purkinje Cells by the mGluR7 Receptor.
Topics: Amino Acids; Animals; Electric Stimulation; Excitatory Amino Acid Antagonists; Ferrets; gamma-Aminobutyric Acid; Glutamic Acid; Male; Patch-Clamp Techniques; Purkinje Cells; Pyridones; Quinoxalines; Receptors, AMPA; Receptors, Metabotropic Glutamate; Xanthenes | 2015 |
Activity-dependent regulation of calcium and ribosomes in the chick cochlear nucleus.
Topics: Amino Acids; Analysis of Variance; Animals; Calcium; Chick Embryo; Cochlear Nucleus; Electric Stimulation; Evoked Potentials, Auditory; Excitatory Amino Acid Antagonists; Gene Expression Regulation; In Vitro Techniques; Indans; Optical Imaging; Ribosomes; Time Factors; Xanthenes | 2016 |
The Rapidly Acting Antidepressant Ketamine and the mGlu2/3 Receptor Antagonist LY341495 Rapidly Engage Dopaminergic Mood Circuits.
Topics: Action Potentials; Amino Acids; Animals; Antidepressive Agents; Dopamine; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Ketamine; Male; Mice, Inbred BALB C; Microdialysis; Motor Activity; Neurons; Nucleus Accumbens; Prefrontal Cortex; Quinoxalines; Rats, Wistar; Receptors, AMPA; Receptors, Metabotropic Glutamate; Ventral Tegmental Area; Xanthenes | 2016 |
Group II mGlu receptor antagonist LY341495 enhances the antidepressant-like effects of ketamine in the forced swim test in rats.
Topics: Amino Acids; Animals; Antidepressive Agents; Behavior, Animal; Blotting, Western; Depression; Drug Synergism; Excitatory Amino Acid Antagonists; Ketamine; Male; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Signal Transduction; Swimming; TOR Serine-Threonine Kinases; Xanthenes | 2016 |
EXPRESS: Histone hyperacetylation modulates spinal type II metabotropic glutamate receptor alleviating stress-induced visceral hypersensitivity in female rats.
Topics: Acetylation; Amino Acids; Animals; Chromatin Immunoprecipitation; Female; Histone Deacetylase Inhibitors; Histones; Hydroxamic Acids; Hyperalgesia; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; RNA, Messenger; Spinal Cord; Stress, Psychological; Viscera; Vorinostat; Xanthenes | 2016 |
Blocking glutamate carboxypeptidase II inhibits glutamate excitotoxicity and regulates immune responses in experimental autoimmune encephalomyelitis.
Topics: Amino Acids; Animals; Astrocytes; Disease Progression; Encephalomyelitis, Autoimmune, Experimental; Excitatory Amino Acid Antagonists; Female; Glutamate Carboxypeptidase II; Glutamic Acid; Humans; Immunohistochemistry; Mice; Mice, Inbred C57BL; Organophosphorus Compounds; Protease Inhibitors; Rats, Inbred Lew; Receptors, Metabotropic Glutamate; Spinal Cord; Th1 Cells; Xanthenes | 2016 |
Metabotropic glutamate receptor 2/3 density and its relation to the hippocampal neuropathology in a model of temporal lobe epilepsy in rats.
Topics: Acute Disease; Amino Acids; Animals; Autoradiography; Chronic Disease; Cross-Sectional Studies; Disease Models, Animal; Disease Progression; Epilepsy, Temporal Lobe; Excitatory Amino Acid Antagonists; Hippocampus; Kainic Acid; Male; Parietal Lobe; Radiopharmaceuticals; Rats, Wistar; Receptors, Metabotropic Glutamate; Thalamus; Time Factors; Tritium; Xanthenes | 2016 |
Antidepressant-like effects of scopolamine in mice are enhanced by the group II mGlu receptor antagonist LY341495.
Topics: Amino Acids; Animals; Antidepressive Agents; Depressive Disorder; Excitatory Amino Acid Antagonists; Male; Maze Learning; Mice; Mice, Inbred C57BL; Motor Activity; Prefrontal Cortex; Quinoxalines; Receptors, AMPA; Receptors, Metabotropic Glutamate; Scopolamine; Serotonin; Xanthenes | 2016 |
Fast-acting antidepressants rapidly stimulate ERK signaling and BDNF release in primary neuronal cultures.
Topics: Amino Acids; Animals; Antidepressive Agents; Brain-Derived Neurotrophic Factor; Cells, Cultured; Cerebral Cortex; Dendrites; GABAergic Neurons; Ketamine; MAP Kinase Signaling System; Oligopeptides; Primary Cell Culture; Rats; Receptor, trkB; Receptors, AMPA; Xanthenes | 2016 |
Glutamate carboxypeptidase II (GCPII) inhibitor 2-PMPA reduces rewarding effects of the synthetic cathinone MDPV in rats: a role for N-acetylaspartylglutamate (NAAG).
Topics: Alkaloids; Amino Acids; Animals; Benzodioxoles; Conditioning, Psychological; Dipeptides; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Glutamate Carboxypeptidase II; Male; Organophosphorus Compounds; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Reward; Synthetic Cathinone; Xanthenes | 2017 |
Control of Glutamate Transport by Extracellular Potassium: Basis for a Negative Feedback on Synaptic Transmission.
Topics: 2-Amino-5-phosphonovalerate; Amino Acid Transport System X-AG; Amino Acids; Animals; Animals, Newborn; Aspartic Acid; Astrocytes; Cerebral Cortex; Excitatory Amino Acid Antagonists; Extracellular Fluid; GABA-A Receptor Antagonists; Glutamic Acid; HEK293 Cells; Humans; Membrane Potentials; Mice; Mice, Inbred C57BL; Neural Inhibition; Neurons; Potassium; Synaptic Transmission; Xanthenes | 2017 |
N-acetylaspartylglutamate Inhibits Heroin Self-Administration and Heroin-Seeking Behaviors Induced by Cue or Priming in Rats.
Topics: Amino Acids; Analysis of Variance; Animals; Conditioning, Operant; Cues; Dipeptides; Dose-Response Relationship, Drug; Drug-Seeking Behavior; Excitatory Amino Acid Antagonists; Heroin; Male; Motivation; Neuroprotective Agents; Rats; Rats, Sprague-Dawley; Reinforcement Schedule; Self Administration; Time Factors; Xanthenes | 2017 |
A group II metabotropic glutamate receptor 3 (mGlu3, GRM3) isoform implicated in schizophrenia interacts with canonical mGlu3 and reduces ligand binding.
Topics: Amino Acids; Cell Membrane; HEK293 Cells; Humans; Ligands; Protein Isoforms; Radioligand Assay; Receptors, Metabotropic Glutamate; Schizophrenia; Transfection; Tritium; Xanthenes | 2017 |
Cross-compartmental Modulation of Dendritic Signals for Retinal Direction Selectivity.
Topics: Action Potentials; Amacrine Cells; Amino Acids; Animals; Animals, Newborn; Cadmium Chloride; Calcium Channel Blockers; Dendrites; Excitatory Amino Acid Antagonists; Female; Inhibitory Postsynaptic Potentials; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Motion Perception; omega-Conotoxin GVIA; Photic Stimulation; Receptors, AMPA; Retina; Signal Transduction; Synapses; Xanthenes | 2017 |
Activation of Group II Metabotropic Glutamate Receptors Increases Proliferation but does not Influence Neuronal Differentiation of a Human Neural Stem Cell Line.
Topics: Amino Acids; Cell Differentiation; Cell Line; Cell Proliferation; Cell Survival; Cyclopropanes; Glutamic Acid; Glycine; Humans; Neural Stem Cells; Neurons; Receptors, Metabotropic Glutamate; Xanthenes | 2018 |
The environmental neurotoxin β-N-methylamino-L-alanine inhibits melatonin synthesis in primary pinealocytes and a rat model.
Topics: Amino Acids; Amino Acids, Diamino; Animals; Cyanobacteria Toxins; Female; Male; Melatonin; Oxidative Stress; Phorbol Esters; Pineal Gland; Protein Kinase C; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Xanthenes | 2018 |
Pre- and Postsynaptic Effects of Glutamate in the Frog Labyrinth.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Amino Acids; Animals; Anura; Aspartic Acid; Ear, Inner; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Hair Cells, Auditory; Patch-Clamp Techniques; Receptors, Ionotropic Glutamate; Receptors, Metabotropic Glutamate; Synapses; Xanthenes | 2018 |
Impact of allosteric modulation: Exploring the binding kinetics of glutamate and other orthosteric ligands of the metabotropic glutamate receptor 2.
Topics: Allosteric Regulation; Amino Acids; Animals; Binding Sites; Bridged Bicyclo Compounds; CHO Cells; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Ligands; Receptors, Metabotropic Glutamate; Xanthenes | 2018 |
Single-molecule diffusion-based estimation of ligand effects on G protein-coupled receptors.
Topics: Amino Acids; GTP-Binding Proteins; HEK293 Cells; Humans; Ligands; Microscopy, Fluorescence; Pertussis Toxin; Protein Binding; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Metabotropic Glutamate; Signal Transduction; Xanthenes | 2018 |
Glutamate metabotropic receptors in the lateral hypothalamus/perifornical area reduce the CO
Topics: Amino Acids; Animals; Carbon Dioxide; Electroencephalography; Electromyography; Excitatory Amino Acid Antagonists; Glycine; Hypothalamic Area, Lateral; Male; Microdialysis; Microinjections; Pulmonary Ventilation; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Sleep; Tidal Volume; Ventilation; Wakefulness; Xanthenes | 2019 |
LY341495, an mGluR2/3 Antagonist, Regulates the Immunosuppressive Function of Myeloid-Derived Suppressor Cells and Inhibits Melanoma Tumor Growth.
Topics: Amino Acids; Animals; Cell Proliferation; Cells, Cultured; Glutamic Acid; Glutamine; Melanoma, Experimental; Mice, Inbred C57BL; Myeloid-Derived Suppressor Cells; Receptors, Metabotropic Glutamate; Xanthenes | 2018 |
Label-free impedance-based whole cell assay to study GPCR pharmacology.
Topics: Amino Acids; Animals; Biological Assay; Biosensing Techniques; Bridged Bicyclo Compounds; Cell Count; CHO Cells; Cricetinae; Cricetulus; Electric Impedance; Humans; Ligands; Receptors, G-Protein-Coupled; Receptors, Metabotropic Glutamate; Signal Transduction; Staining and Labeling; Xanthenes | 2019 |
Glutamate Within the Marmoset Anterior Hippocampus Interacts with Area 25 to Regulate the Behavioral and Cardiovascular Correlates of High-Trait Anxiety.
Topics: Amino Acids; Animals; Anxiety; Behavior, Animal; Benzylamines; Callithrix; Excitatory Amino Acid Antagonists; Female; GABA-A Receptor Antagonists; Glutamic Acid; Heart Rate; Hippocampus; Male; Phosphinic Acids; Xanthenes | 2019 |
Role of AMPA receptor stimulation and TrkB signaling in the antidepressant-like effect of ketamine co-administered with a group II mGlu receptor antagonist, LY341495, in the forced swim test in rats.
Topics: Amino Acids; Animals; Antidepressive Agents; Azepines; Benzamides; Depression; Depressive Disorder; Excitatory Amino Acid Antagonists; Ketamine; Male; Prefrontal Cortex; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptor, trkB; Receptors, AMPA; Receptors, Metabotropic Glutamate; Signal Transduction; Xanthenes | 2019 |
Group II metabotropic glutamate receptor blockade promotes stress resilience in mice.
Topics: Amino Acids; Anhedonia; Animals; Behavior, Animal; Corticosterone; Electroshock; Escape Reaction; Excitatory Amino Acid Antagonists; Mice; Mice, Knockout; Receptors, Metabotropic Glutamate; Resilience, Psychological; Stress, Psychological; Xanthenes | 2019 |
Target validation: Weak selectivity of LY341495 for mGluR2 over mGluR4 makes glutamate a less selective agonist.
Topics: Amino Acids; Animals; Dose-Response Relationship, Drug; Down-Regulation; Ganglia, Sympathetic; Gene Expression Regulation; Male; Rats; Receptors, Metabotropic Glutamate; Signal Transduction; Superior Cervical Ganglion; Xanthenes | 2019 |
Pharmacological Modulation of Sleep Homeostasis in Rat: Novel Effects of an mGluR2/3 Antagonist.
Topics: Amino Acids; Animals; Caffeine; Central Nervous System Stimulants; Cyclohexanes; Dextroamphetamine; Electroencephalography; Excitatory Amino Acid Antagonists; Homeostasis; Male; Rats; Rats, Wistar; Reaction Time; Receptors, Metabotropic Glutamate; Sleep; Sleep Deprivation; Sleep, REM; Wakefulness; Xanthenes | 2019 |
Regulatory system of mGluR group II in the nucleus accumbens for methamphetamine-induced dopamine increase by the medial prefrontal cortex.
Topics: Acetyltransferases; Amino Acids; Animals; Dopamine; Dopamine Agents; Dopamine and cAMP-Regulated Phosphoprotein 32; Excitatory Amino Acid Antagonists; Glutamic Acid; Male; Methamphetamine; Mice; Mice, Inbred C57BL; Nucleus Accumbens; Prefrontal Cortex; Receptors, Metabotropic Glutamate; Xanthenes | 2019 |
Amygdala group II mGluRs mediate the inhibitory effects of systemic group II mGluR activation on behavior and spinal neurons in a rat model of arthritis pain.
Topics: Amino Acids; Amygdala; Animals; Arthralgia; Arthritis, Experimental; Behavior, Animal; Bridged Bicyclo Compounds, Heterocyclic; Carrageenan; Central Amygdaloid Nucleus; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Kaolin; Nociception; Pain; Posterior Horn Cells; Rats; Receptors, Metabotropic Glutamate; Spinal Cord; Vocalization, Animal; Xanthenes | 2019 |
Vulnerability to depressive behavior induced by overexpression of striatal Shati/Nat8l via the serotonergic neuronal pathway in mice.
Topics: Acetyltransferases; Amino Acids; Animals; Brain; Causality; Corpus Striatum; Depression; Fluvoxamine; Male; Mice; Mice, Inbred C57BL; Serotonergic Neurons; Stress, Psychological; Xanthenes | 2019 |
AMPA receptor-mTORC1 signaling activation is required for neuroplastic effects of LY341495 in rat hippocampal neurons.
Topics: Amino Acids; Animals; Excitatory Amino Acid Antagonists; Hippocampus; Mechanistic Target of Rapamycin Complex 1; Neuronal Plasticity; Neurons; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Metabotropic Glutamate; Signal Transduction; Xanthenes | 2020 |
The metabotropic glutamate receptor 2/3 antagonist LY341495 improves working memory in adult mice following juvenile social isolation.
Topics: Age Factors; Amino Acids; Animals; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Male; Maze Learning; Memory, Short-Term; Mice; Mice, Inbred C57BL; Receptors, Metabotropic Glutamate; Social Isolation; Xanthenes | 2020 |
The group II mGlu receptor antagonist LY341495 induces a rapid antidepressant-like effect and enhances the effect of ketamine in the chronic unpredictable mild stress model of depression in C57BL/6J mice.
Topics: Amino Acids; Animals; Antidepressive Agents; Depression; Disease Models, Animal; Excitatory Amino Acid Antagonists; Hippocampus; Ketamine; Male; Mice; Mice, Inbred C57BL; Motor Skills; Prefrontal Cortex; Receptors, Metabotropic Glutamate; Synaptosomes; Xanthenes | 2021 |
mGlu2/3 receptor in the prelimbic cortex is implicated in stress resilience and vulnerability in mice.
Topics: Amino Acids; Animals; Depression; Disease Models, Animal; Humans; Male; Mice; Prefrontal Cortex; Receptors, Metabotropic Glutamate; Resilience, Psychological; Social Defeat; Stress, Psychological; Xanthenes | 2021 |
Inhibition of metabotropic glutamate receptor III facilitates sensitization to alkylating chemotherapeutics in glioblastoma.
Topics: Amino Acids; Antineoplastic Agents, Alkylating; Cell Death; Cell Line, Tumor; Cell Survival; Drug Resistance, Neoplasm; Gene Expression Regulation, Neoplastic; Glioblastoma; Glutamic Acid; Humans; Kinetics; Neoadjuvant Therapy; Receptors, Metabotropic Glutamate; Temozolomide; Tumor Microenvironment; Xanthenes | 2021 |
Allosteric modulators enhance agonist efficacy by increasing the residence time of a GPCR in the active state.
Topics: Allosteric Regulation; Allosteric Site; Amino Acids; Biphenyl Compounds; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Catalytic Domain; Cell Membrane; Cholesterol Esters; Diosgenin; Disaccharides; Fluorescence Resonance Energy Transfer; Gene Expression; Glucosides; Glutamic Acid; Glycolipids; HEK293 Cells; Humans; Indans; Micelles; Octoxynol; Protein Binding; Protein Conformation; Protein Multimerization; Receptors, Metabotropic Glutamate; Recombinant Proteins; Single Molecule Imaging; Xanthenes | 2021 |
Graded heterogeneity of metabotropic signaling underlies a continuum of cell-intrinsic temporal responses in unipolar brush cells.
Topics: Action Potentials; Amino Acids; Animals; Cerebellar Cortex; Electric Stimulation; Excitatory Amino Acid Antagonists; Female; Male; Mice, Inbred C57BL; Nerve Fibers; Neurons; Patch-Clamp Techniques; Receptors, Metabotropic Glutamate; Synaptic Transmission; Time Factors; Xanthenes | 2021 |
Effects of Chronic LY341495 on Hippocampal mTORC1 Signaling in Mice with Chronic Unpredictable Stress-Induced Depression.
Topics: Amino Acids; Animals; Antidepressive Agents; Depression; Hippocampus; Mechanistic Target of Rapamycin Complex 1; Mice; Stress, Psychological; Xanthenes | 2022 |