Page last updated: 2024-08-18

xanthenes and ly 341495

xanthenes has been researched along with ly 341495 in 245 studies

Research

Studies (245)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's6 (2.45)18.2507
2000's127 (51.84)29.6817
2010's104 (42.45)24.3611
2020's8 (3.27)2.80

Authors

AuthorsStudies
Belagaje, R; Burnett, JP; Johnson, BG; Kingston, AE; Mayne, NG; Ornstein, PL; Schoepp, DD; Wright, RA; Wu, S1
Arnold, MB; Bleisch, TJ; Ornstein, PL; Schoepp, DD; Wheeler, WJ; Wright, RA1
Bortolotto, ZA; Collingridge, GL; Doherty, AJ; Fitzjohn, SM; Kingston, AE; Lodge, D; Ornstein, PL; Palmer, MJ; Schoepp, DD1
Chamberlain, M; Johnson, MP; Kelly, GM2
Arnold, MB; Johnson, BG; Ornstein, PL; Schoepp, DD; Wheeler, WJ; Wright, RA1
Bear, MF; Huber, KM; Roder, JC; Sawtell, NB1
Aghajanian, GK; Marek, GJ; Monn, JA; Schoepp, DD; Wright, RA1
Bear, MF; Huber, KM; Kayser, MS1
Adam, G; Kratzeisen, C; Lundstrom, K; Malherbe, P; Mutel, V; Ohresser, S; Schweitzer, C; Stadler, H; Wichmann, J; Woltering, T1
Cartmell, J; Monn, JA; Perry, KW; Salhoff, CR; Schoepp, DD1
Cartmell, J; Monn, JA; Schoepp, DD1
Gewirtz, JC; Marek, GJ1
Ducarre, JM; Kemp, JA; Kew, JN; Mutel, V; Pflimlin, MC1
Arnold, MB; Ornstein, PL; Schoepp, DD; Wheeler, WJ; Wright, RA2
Bradley, SR; Conn, PJ; Marino, MJ; Wittmann, M1
Cirone, J; Salt, TE1
Glitsch, MD; Jack, JJ1
Chamberlain, M; Johnson, MP; Kelly, G1
Abraini, JH; David, HN1
Bear, MF; Dong, X; Fallon, JR; Huber, KM; Philpot, BD; Snyder, EM1
Carlisle, HJ; O'Dell, TJ; Watabe, AM1
Cai, Z; Lin, S; Rhodes, PG1
Alonso, G; Bockaert, J; Chaumont, S; Manzoni, OJ; Robbe, D1
Cirone, J; Pothecary, CA; Salt, TE; Turner, JP1
Chen, AC; Duman, RC; Gewirtz, JC; Marek, GJ; Terwilliger, R1
Griffey, KI; Schoepp, DD; Tizzano, JP1
Frondaroli, A; Grassi, S; Pettorossi, VE2
Bleisch, TJ; Johnson, BG; Kingston, AE; Ornstein, PL; Schoepp, DD; Sørensen, US; Wright, RA1
George, CA; Johnson, MP; Nisenbaum, ES; Nisenbaum, LK; Zhai, J; Zhai, Y1
Arcella, A; Battaglia, G; Bruno, V; Calogero, A; D'Onofrio, M; Lombari, V; Ngomba, RT; Nicoletti, F; Ragona, G1
Laruelle, M; Mozley, PD; Schmidt, ME; Schoepp, DD; Sultana, A; Waterhouse, RN; Wheeler, WJ1
Bandrowski, AE; Huguenard, JR; Prince, DA1
Losonczy, A; Nusser, Z; Somogyi, P1
Howson, PA; Jane, DE1
Anderson, JJ; Baccei, CS; Bristow, LJ; Campbell, UC; Correa, LD; Lorrain, DS; Pinkerton, AB; Rodriguez, DE; Rowe, B; Schaffhauser, H; Varney, MA; Vernier, JM1
Battaglia, G; Biagioni, F; Bruno, V; Busceti, CL; Fornai, F; Nicoletti, F; Paparelli, A; Pontarelli, F; Ruggieri, S1
Keller, A; Sanabria, ER; Slusher, BS; Wozniak, KM1
Conway, MW; Heron-Maxwell, C; Monn, JA; O'Neill, MF; Ornstein, P1
Bain, G; Bristow, LJ; Chavez-Noriega, LE; Daggett, LP; Jachec, C; Morales, S; Pinkerton, AB; Rao, SP; Rowe, BA; Schaffhauser, H; Varney, MA; Vernier, JM; Yin, R1
Johnson, SW; Shen, KZ1
Hashimoto, K; Iyo, M; Koike, K; Koizumi, H; Komatsu, N; Kumakiri, C; Ohgake, S; Okamura, N; Shimizu, E1
Brotchie, JM; Brown, TM; Fitzjohn, SM1
Perry, KW; Schoepp, DD; Swanson, CJ1
Gregory, ML; Kalivas, PW; Owens, RW; Stech, NE1
Kalivas, PW; Tang, XC1
Rieke, F; Sampath, AP1
Anwyl, R; Rowan, MJ; Wu, J1
Irifune, M; Nishikawa, T; Ohnishi, Y; Sato, T; Tanaka, K; Teramoto, T1
Hsu, MA; Rasmussen, K; Vandergriff, J1
Gereau, RW; Yang, D1
Chen, HX; Roper, SN1
Adam, G; Ballard, TM; Higgins, GA; Kemp, JA; Kew, JN; Mutel, V; Nakanishi, S; Richards, JG; Woltering, T1
Capogna, M; Dalezios, Y; Ferraguti, F; Kogo, N; Shigemoto, R; Somogyi, P1
Capogna, M1
Irifune, M; Nishikawa, T; Ohnishi, Y; Sato, T; Tanaka, K1
DiGregorio, DA; Nielsen, TA; Silver, RA1
Duvoisin, RM; Grandes, P; Kushmerick, C; Price, GD; Puente, N; Renden, R; Taschenberger, H; von Gersdorff, H; Wadiche, JI1
Grajkowska, E; Hirasawa, S; Kozikowski, A; Neale, JH; Wroblewska, B; Wroblewski, J; Yamamoto, T; Zhou, J1
Freund, TF; Hájos, N; Pálhalmi, J; Paulsen, O1
Campbell, IG; Darchia, N; Feinberg, I; Hsieh, KC; Schoepp, DD1
Gebhardt, C; Heinemann, U; Iserhot, C; Schmitz, D1
Alagarsamy, S; Bough, KJ; Conn, PJ; Dingledine, R; Doherty, JJ; Mott, DD1
Neale, SA; Salt, TE; Thompson, H1
Bringmann, A; Klaus, C; Reichenbach, A; Rillich, K; Syková, E; Uckermann, O; Ulbricht, E; Vargová, L; Weick, M; Wiedemann, P1
Bickel, DJ; Burno, M; Chen, TB; Clements, MK; Conn, PJ; Duggan, ME; Jacobson, MA; Kinney, GG; Lemaire, W; Lindsley, CW; O'Brien, JA; Pettibone, DJ; Smith, S; Sur, C; Tiller, PR; Williams, DL; Wisnoski, DD1
Baez, M; Koester, A; Linden, AM; Schoepp, DD; Shannon, H; Yu, JL1
Druga, R; Folbergrová, J; Haugvicová, R; Kubová, H; Mares, P; Otáhal, J1
Alexander, GM; Godwin, DW2
Huber, KM; Nosyreva, ED1
Chaki, S; Karasawa, J; Kawashima, N; Nakazato, A; Okuyama, S; Shimazaki, T; Yasuhara, A1
Battaglia, G; Canudas, AM; Del Bianco, P; Matrisciano, F; Melchiorri, D; Molinaro, G; Ngomba, RT; Nicoletti, F; Panaccione, I; Riozzi, B; Scaccianoce, S; Tatarelli, R1
Abeniyi, OA; Conn, PJ; Poisik, O; Raju, DV; Rodriguez, A; Smith, Y; Verreault, M1
Capogna, M; Karayannis, T; Pál, BZ; Price, CJ1
Kalivas, PW; McFarland, K; Melendez, RI; Moran, MM; Seamans, JK1
Bergeron, M; Linden, AM; Schoepp, DD1
Battaglia, G; Biagioni, F; Bruno, V; Casciato, S; Ngomba, RT; Nicoletti, F; van Luijtelaar, EL; Willems-van Bree, E1
Arcella, A; Battaglia, G; Bruno, V; Carpinelli, G; Casolini, P; D'Onofrio, M; Giangaspero, F; Ngomba, RT; Nicoletti, F; Santoro, F1
Alger, BE; Jones, LM; Karnup, SV; Karson, MA; Reich, CG1
Ebinger, G; Hachimi-Idrissi, S; Michotte, Y; Sarre, S; Van Hemelrijck, A1
Daniel, WA; Kos, T; Kozela, E; Popik, P; Slusher, BS; Wojcikowski, J; Wozniak, KM; Wrobel, M1
Kitai, ST; Wang, L; Xiang, Z1
Bae, HB; Choi, Jl; Chung, SS; Chung, ST; Jeong, CY; Jeong, SW; Kim, SJ; Yoo, KY; Yoon, MH1
Ennis, M; Hayar, A; Heinbockel, T; Zhu, M1
Bzdega, T; Neale, JH; Olszewski, RT; Wegorzewska, IN; Wroblewska, B1
Daly, CA; Huber, KM; Volk, LJ1
Anwyl, R; Harney, SC; Rowan, M1
Chi, H; Jang, JK; Kim, JH; Vezina, P1
Anderson, H; Cottrell, DF; Fleetwood-Walker, SM; Garry, EM; Mitchell, R; Proudfoot, CJ; Robertson, DC; Rosie, R1
Marek, GJ; Zhang, C1
Chaki, S; Iijima, M; Ito, A; Shimazaki, T1
Liechti, ME; Markou, A1
Markou, A; Semenova, S1
Bespalov, A; Gross, G; Harich, S; Jongen-Rêlo, AL; Schoemaker, H; van Gaalen, M1
Lu, Y1
Battaglia, G; Beraudi, A; Biagioni, F; Bruno, V; Nicoletti, F; Poli, A; Rampello, L1
Griffey, KI; Johnson, BG; Knitowski, KM; McKinzie, DL; Monn, JA; Perry, KW; Rorick-Kehn, LM; Salhoff, CR; Schoepp, DD; Tizzano, JP; Witkin, JM1
Brady, AE; Conn, PJ; Da Costa, H; Hemstapat, K; Luo, Q; Niswender, CM; Nong, Y; Tamagnan, GD1
Mateo, Z; Porter, JT1
Chung, LY; Kim, U1
Girardi, P; Giusti, P; Gruber, SH; Iacovelli, L; Mathé, AA; Matrisciano, F; Nicoletti, F; Panaccione, I; Tatarelli, R; Zusso, M1
Baker, DA; Haroutunian, V; Kristiansen, LV; Madayag, A; Meador-Woodruff, JH; Raju, I1
Bédard, PJ; Bélanger, N; Calon, F; Di Paolo, T; Dridi, M; Grégoire, L; Hadj Tahar, A; Morissette, M; Samadi, P1
Ayala, JE; Conn, PJ; Johnson, KA; Kim, C; Luo, Q; Niswender, CM; Weaver, CD1
Ayala, JE; Banko, JL; Conn, PJ; Luo, Q; Niswender, CM1
Cleland, TA; Linster, C; Magidson, PD; McNamara, AM; Wilson, DA1
Anwyl, R; Harney, S; Rowan, MJ; Wu, J1
Kai, T; Shichida, Y; Terakita, A; Yamashita, T1
Carlton, SM; Du, J; Zhou, S2
Arcella, A; Battaglia, G; Carpinelli, G; Ciceroni, C; De Maria, R; Giangaspero, F; Mastrantoni, E; Melchiorri, D; Mosillo, P; Nicoletti, F; Oliva, MA; Pallini, R; Ricci-Vitiani, L; Sale, P; Santoro, F1
Conn, PJ; Sheffler, DJ1
Bespalov, AY; Gross, G; Mezler, M; Schoemaker, H; Sukhotina, IA; van Gaalen, MM; Wicke, K1
Steketee, JD; Xie, X1
Jang, JK; Kim, JH; Yoon, HS1
Abrahamsson, T; Gustafsson, B; Hanse, E1
Corsi, M; Corti, C; Ferraguti, F; Herdy, S; Hetzenauer, A; Singewald, N1
Martina, M; Mugnaini, E; Nunzi, MG; Russo, MJ; Yau, HJ1
Poo, MM; Xu, C; Zhang, XH; Zhao, MX1
Andreasen, M; Nedergaard, S; Skov, J1
Busceti, CL; Chiechio, S; Copani, A; Drago, F; Gereau, RW; Morales, ME; Nicoletti, F; Zammataro, M1
Calon, F; Di Paolo, T; Grégoire, L; Hornykiewicz, O; Rajput, A; Rajput, AH; Samadi, P1
Akiba, Y; Baker, H; Cave, JW; Estevez, AG; Huerta, PT; Sasaki, H1
Feng, Y; Li, H; Shi, J; Sun, ZS; Zhang, J; Zhang, T1
Battaglia, G; Bruno, V; Curto, M; Di Menna, L; Molinaro, G; Nicoletti, F; Pallottino, S; Riozzi, B; Traficante, A1
Gregg, RG; Heimel, JA; Kamermans, M; Nawy, S; Peachey, NS; Shen, Y1
Johnson, BG; Korpi, ER; Linden, AM; Schoepp, DD; Trokovic, N1
Kinouchi, H; Sugita, M; Yoshioka, H1
Dietrich, D; Wostrack, M1
Ashby, CR; Gardner, EL; Li, J; Peng, XQ; Slusher, BS; Thomas, A; Wozniak, K; Xi, ZX1
Belluardo, N; Bonomo, A; Di Liberto, V; Frinchi, M; Mudò, G1
Chen, WC; Mei, B; Sun, ZW; Zhang, L; Zhu, SJ1
Choi, S; Hong, I; Kim, J; Lee, S; Song, B1
Ehrlich, ME; Fraser, PE; Gandy, S; Kim, SH; St George-Hyslop, PH; Westaway, D1
Amitai, N; Markou, A1
Chaki, S; Kambe, D; Karasawa, J; Kotani, M1
Fujita, Y; Hashimoto, K; Slusher, BS; Takatsu, Y; Tsukamoto, T1
Battaglia, G; Britton, TC; Bruno, V; Cannella, M; Caraci, F; Copani, A; Drago, F; Giuffrida, ML; Heinz, BA; Merlo, S; Molinaro, G; Nicoletti, F; Nisenbaum, ES; Riozzi, B; Sortino, MA; Traficante, A; Wang, X1
Berridge, KC; Richard, JM1
Andreasen, M; Hablitz, JJ; Nedergaard, S; Skov, J1
Beveridge, TJ; Nader, MA; Porrino, LJ; Smith, HR1
Rushlow, WJ; Sutton, LP1
Coiret, G; Corsi, M; Corti, C; Gerber, U; Grewe, BF; Helmchen, F; Mateos, JM; Ster, J1
Bojang, P; Furukawa, T; Gregg, RG; Koike, C; Nawy, S; Pearring, JN; Shen, Y1
Chaban, V; Li, J; McDonald, JS; Micevych, P; Rapkin, A1
Ma, H; Yang, K1
Carlton, SM; Du, J; Govea, R; Zhou, S1
Chaki, S; Iijima, M; Koike, H3
Conn, PJ; Johnson, KA; Niswender, CM; Xiang, Z1
Gilley, JA; Kernie, SG1
Duman, RS; Dwyer, JM; Lepack, AE1
Brownell, AL; Kuruppu, D; Wang, JQ; Zhang, Z1
Dong, E; Sanford, LD; Wellman, LL; Yang, L1
Copeland, CS; Neale, SA; Salt, TE1
Bortolotto, ZA; Collingridge, GL; Lodge, D; Lucas, SJ1
Carroll, RC; Nawy, S; Rampino, MA; Shen, Y1
Kaffe, E; Markou, A; Pitsikas, N1
Raiteri, L; Raiteri, M; Romei, C1
Bojang, P; Furukawa, T; Goldberg, AF; Gregg, RG; Hirschtritt, ME; Koike, C; McCall, MA; Nawy, S; Nishina, PM; Peachey, NS; Pearring, JN; Ray, TA; Shen, Y; Sturgill-Short, G1
Bae, SA; Bischoff, F; Guo, N; Huang, Y; Hwang, DR; Laruelle, M; Lesage, AS; Narendran, R1
Breustedt, J; Kintscher, M; Miceli, S; Schmitz, D; Wozny, C1
Aston-Jones, G; Fallon, RV; Hensley-Simon, M; Kalivas, PW; LaLumiere, RT; Mahler, SV; Tahsili-Fahadan, P; Thomas, C1
Chaki, S; Fukumoto, K; Iijima, M; Koike, H1
Kaba, H; Murata, Y; Nakanishi, S; Okutani, F; Shinohara, Y; Taniguchi, M; Yokoi, M1
Arcella, A; Battaglia, G; Bonelli, M; Ciceroni, C; De Maria, R; Larocca, LM; Laurenza, M; Mastrantoni, E; Melchiorri, D; Niccolini, C; Nicoletti, F; Pallini, R; Ricci-Vitiani, L; Spinsanti, P; Traficante, A1
Bouwalerh, H; Maccari, S; Mairesse, J; Marrocco, J; Morley-Fletcher, S; Ngomba, RT; Nicoletti, F; Pittaluga, A; Silletti, V; Summa, M; Van Camp, G1
Bortolotto, ZA; Collett, VJ; Collingridge, GL; Fang, G; Jane, DE; Lodge, D; Mercier, MS; Nicolas, CS1
González-Maeso, J; Holloway, T; Moreno, JL; Rayannavar, V; Sealfon, SC1
Barone, Y; Battaglia, G; Caruso, A; Lionetto, L; Mathé, AA; Matrisciano, F; Nasca, C; Nicoletti, F; Pittaluga, A; Scaccianoce, S; Simmaco, M; Xenos, D1
Bannister, N; Bortolotto, ZA; Ceolin, L; Collingridge, GL; Fitzjohn, SM; Hanna, L; Jane, DE; Kritikos, M; Lodge, D; Lucas, SJ; Mercier, MS; Sherwood, JL; Tidball, P; Volianskis, A1
de Groat, WC; Mally, AD; Matsuta, Y; Roppolo, JR; Shen, B; Tai, C; Wang, J; Zhang, F1
Gao, WJ; Li, F; Li, YC; Snyder, MA; Wang, H; Wang, MJ1
Chaki, S; Hikichi, H; Kaku, A; Karasawa, J1
Carrillo, V; Dubisz, E; Gulzar, H; Mahajan, SS; Morgan, D; Yelskaya, Z1
Di Paolo, T; Gasparini, F; Gomez-Mancilla, B; Grégoire, L; Morin, N; Morissette, M1
Ahnaou, A; Andrés, JI; Atack, JR; Biesmans, I; Cid, JM; Dautzenberg, FM; Drinkenburg, W; Langlois, X; Lavreysen, H; Lütjens, R; Macdonald, G; Megens, A; Peeters, L; te Riele, P; Trabanco, AA; Van der Linden, I; Wintmolders, C1
Anwyl, R; Chang, L; Chen, X; Lin, R; Wang, C; Wang, Q; Wei, X; Xu, S; Zhang, J1
Caron, MG; Jacobsen, JP; Jørgensen, CV; Klein, AB; Knudsen, GM; Mikkelsen, JD1
Curry, RJ; Dinh, EH; Hamlet, WR; Liu, YW; Lu, Y; Shi, W; Tang, ZQ1
Chaki, S; Fukumoto, K; Iijima, M2
Shu, H; Song, Y; Wang, B; Yang, H; Zhang, C; Zhou, K; Zhou, W1
Chan, MH; Chen, HH; Chiang, CC; Chiu, HY; Lee, MY1
Fu, K; Furukawa-Hibi, Y; Iegaki, N; Ishikawa, Y; Miyamoto, Y; Muramatsu, S; Nabeshima, T; Nitta, A; Sato, K; Sumi, K; Uno, K1
DiRaddo, JO; Grajkowska, E; Hathaway, HA; Liotta, DC; Miller, EJ; Wolfe, BB; Wroblewska, B; Wroblewski, JT1
Ahnaou, A; Drinkenburg, WH; Ver Donck, L1
Chaki, S; Koike, H1
Callado, LF; Díez-Alarcia, R; González-Maeso, J; Meana, JJ; Miranda-Azpiazu, P; Morentin, B; Muguruza, C1
Borsotto, M; Bourcier-Lucas, C; Haddjeri, N; Heurteaux, C; Kanzari, A; Lucas, G; Moha ou Maati, H; Veyssiere, J1
Bai, G; Cao, DY; Ji, Y; Traub, RJ1
Kärkkäinen, O; Kautiainen, H; Kupila, J; Laukkanen, V; Storvik, M; Tiihonen, J1
Benn, A; Robinson, ES1
Karimi, SA; Komaki, A; Salehi, I; Sarihi, A; Shahidi, S1
Asseri, KA; MacLeod, BA; Puil, E; Schwarz, SK1
Battaglia, G; Cruccu, G; Di Stefano, G; Lattanzi, R; Nicoletti, F; Notartomaso, S; Pasquale, E; Piroso, S; Truini, A1
Kiritoshi, T; Neugebauer, V1
Ago, Y; Hasebe, S; Hashimoto, H; Matsuda, T; Nishiyama, S; Oka, S; Onaka, Y; Takuma, K1
An, B; Choi, S; Hong, I; Kim, J; Lee, S; Park, K; Park, S1
Besheer, J; Fisher, KR; Frisbee, S; Jaramillo, AA; Randall, PA1
Bollands, M; Jones, S; Morris, PG; Wild, AR1
Barker, JM; Chandler, LJ; Lench, DH1
Dean, B; Gibbons, A; Hopper, S; McOmish, CE; Pavey, G; Scarr, E; Udawela, M1
Carlsson, HA; Hesslow, G; Johansson, F; Rasmussen, A; Yeo, CH1
Call, CL; Hyson, RL1
Carter, G; Johnson, B; Li, X; Mitchell, SN; Monn, JA; Overshiner, C; Rasmussen, K; Rorick-Kehn, LM; Schoepp, DD; Witkin, JM1
Brański, P; Pałucha-Poniewiera, A; Pilc, A; Pochwat, B; Podkowa, K1
Bai, G; Cao, DY; Ji, Y; Karpowicz, JM; Traub, RJ1
Ahn, G; Bing, SJ; Cho, IH; Cho, J; Ha, D; Herath, KH; Jee, Y; Jo, SA; Kim, A; Kim, J; Yu, HS1
Ali, I; Amhaoul, H; Boets, S; Dedeurwaerdere, S; Janssens, P; Langlois, X; Van Eetveldt, A1
Lenda, T; Pałucha-Poniewiera, A; Pilc, A; Podkowa, A; Podkowa, K; Sałat, K1
Bang, E; Duman, RS; Dwyer, JM; Lee, B; Lepack, AE1
Cannella, LA; Gregg, RA; Hicks, C; Nayak, SU; Rawls, SM; Reitz, AB; Schena, GJ; Smith, GR; Tallarida, CS1
Chatton, JY; Rimmele, TS; Rocher, AB; Wellbourne-Wood, J1
Chen, W; Lai, M; Liu, H; Mei, D; Zhang, F; Zhou, W; Zhu, H1
Bermudez, I; García-Bea, A; Harrison, PJ; Lane, TA1
Grove, JCR; Koren, D; Wei, W1
Blaabjerg, M; Bogetofte, H; Dindler, A; Kamand, M; Meyer, M1
Andersson, M; Brandt, I; Karlsson, O; Pierozan, P1
Canella, R; Fesce, R; Martini, M; Rossi, ML; Rubbini, G1
Doornbos, MLJ; Heitman, LH; IJzerman, AP; Lavreysen, H; Tresadern, G; Vermond, SC1
Abe, M; Hiroshima, M; Murata, M; Sako, Y; Shichida, Y; Togashi, Y; Ueda, M; Yamashita, T; Yanagawa, M1
da Silva, EN; Dias, MB; Gargaglioni, LH; Horta-Júnior, JAC; Rodrigues, LTC1
Ago, Y; Goda, H; Mizuguchi, H; Morikawa, N; Sakurai, F; Tachibana, M1
Doornbos, MLJ; Heitman, LH1
Alexander, L; Cardinal, RN; Clarke, HF; Cockcroft, GJ; Dalley, JW; Quah, SKL; Roberts, AC; Santangelo, AM; Shiba, Y; Wallis, CU; Xia, J; Zeredo, JL1
Pałucha-Poniewiera, A; Pilc, A; Podkowa, K1
Georgiou, P; Gould, TD; Highland, JN; Zanos, P1
Kammermeier, PJ; McCullock, TW1
Eastwood, BJ; Gilmour, G; Hanley, N; Loomis, S; McCarthy, A; Paulissen, J; Wafford, KA1
Haddar, M; Hamatani, K; Muramatsu, SI; Nitta, A; Uno, K1
Mazzitelli, M; Neugebauer, V1
Fujiwara, T; Miyanishi, H; Miyazaki, T; Muramatsu, SI; Nitta, A; Sodeyama, K; Uno, K1
Choi, AJ; Hien, LT; Kim, SH; Lee, JG; Park, MK; Park, SW; Seo, MK; Seog, DH1
Du, H; Jiang, HD; Jiang, HJ; Ling, Y; Shen, HW; Wang, GZ; Wu, T; Xu, L; Yang, SY; Yu, ZP; Zhang, XQ; Zhang, ZY; Zhao, QQ1
Pałucha-Poniewiera, A; Podkowa, K; Rafało-Ulińska, A1
Jing, XY; Li, LF; Li, ZL; Liu, YJ; Wang, Y; Zou, HW1
Beck, J; Behringer, SP; Follo, M; Garrelfs, N; Goeldner, JM; Hannibal, L; Heiland, DH; Hofmann, UG; Joseph, K; Kueckelhaus, J; Maier, JP; Pfeifer, D; Ravi, VM; Schnell, O; Sun, N; von Ehr, J; Walch, AK; Will, P1
Cao, AM; Fatemi, F; Margeat, E; Pin, JP; Quast, RB; Rondard, P1
Guo, C; Huson, V; Macosko, EZ; Regehr, WG1
Jeong, S; Lee, JA; Lee, JG; Park, SW; Seo, MK; Seog, DH1

Other Studies

245 other study(ies) available for xanthenes and ly 341495

ArticleYear
LY341495 is a nanomolar potent and selective antagonist of group II metabotropic glutamate receptors.
    Neuropharmacology, 1998, Volume: 37, Issue:1

    Topics: Amino Acids; Animals; Cell Line; Colforsin; Cyclic AMP; Excitatory Amino Acid Antagonists; Humans; Prosencephalon; Rats; Receptors, Metabotropic Glutamate; Xanthenes

1998
[3H]LY341495, a highly potent, selective and novel radioligand for labeling Group II metabotropic glutamate receptors.
    Bioorganic & medicinal chemistry letters, 1998, Jul-21, Volume: 8, Issue:14

    Topics: Amino Acids; Animals; Excitatory Amino Acid Antagonists; Prosencephalon; Radioligand Assay; Rats; Receptors, Metabotropic Glutamate; Tritium; Xanthenes

1998
The potent mGlu receptor antagonist LY341495 identifies roles for both cloned and novel mGlu receptors in hippocampal synaptic plasticity.
    Neuropharmacology, 1998, Volume: 37, Issue:12

    Topics: Aging; Amino Acids; Animals; Binding, Competitive; Cell Line; CHO Cells; Cloning, Molecular; Cricetinae; Cycloleucine; Excitatory Amino Acid Antagonists; Glutamic Acid; Glycine; Hippocampus; Humans; In Vitro Techniques; Long-Term Potentiation; Neuronal Plasticity; Rats; Receptors, Metabotropic Glutamate; Recombinant Proteins; Resorcinols; Transfection; Xanthenes

1998
Phosphoinositide hydrolysis in vivo with group I metabotropic glutamate receptor agonists.
    Brain research, 1999, Mar-13, Volume: 821, Issue:2

    Topics: Amino Acids; Animals; Brain Chemistry; Cerebellum; Cycloleucine; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Glycine; Hippocampus; Hydrolysis; Injections, Intraventricular; Male; Neuroprotective Agents; Phenylacetates; Phosphatidylinositols; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Resorcinols; Tritium; Type C Phospholipases; Xanthenes

1999
[3H]-LY341495 as a novel antagonist radioligand for group II metabotropic glutamate (mGlu) receptors: characterization of binding to membranes of mGlu receptor subtype expressing cells.
    Neuropharmacology, 1999, Volume: 38, Issue:10

    Topics: Amino Acids; Animals; Binding, Competitive; Calcium; Cell Membrane; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Humans; Kinetics; Radioligand Assay; Receptors, Metabotropic Glutamate; Recombinant Proteins; Transfection; Tritium; Xanthenes

1999
Induction of NMDA receptor-dependent long-term depression in visual cortex does not require metabotropic glutamate receptors.
    Journal of neurophysiology, 1999, Volume: 82, Issue:6

    Topics: Amino Acids; Animals; Cycloleucine; Depression, Chemical; Excitatory Amino Acid Antagonists; Hydrolysis; In Vitro Techniques; Methoxyhydroxyphenylglycol; Mice; Mice, Knockout; Neuronal Plasticity; Phosphatidylinositols; Rats; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Synaptosomes; Visual Cortex; Xanthenes

1999
Physiological antagonism between 5-hydroxytryptamine(2A) and group II metabotropic glutamate receptors in prefrontal cortex.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 292, Issue:1

    Topics: Amino Acids; Animals; Autoradiography; Bridged Bicyclo Compounds; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Free Radical Scavengers; Glutamic Acid; Humans; In Vitro Techniques; Male; Membrane Potentials; Prefrontal Cortex; Protein Binding; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Receptors, Presynaptic; Serotonin; Xanthenes

2000
Blockade of pilocarpine-induced cerebellar phosphoinositide hydrolysis with metabotropic glutamate antagonists: evidence for an indirect control of granule cell glutamate release by muscarinic agonists.
    Neuroscience letters, 2000, May-05, Volume: 285, Issue:1

    Topics: Amino Acids; Animals; Cerebellum; Corpus Striatum; Frontal Lobe; Hippocampus; Hydrolysis; Lithium; Male; Muscarinic Agonists; Phosphatidylinositols; Pilocarpine; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M2; Receptors, Metabotropic Glutamate; Receptors, Muscarinic; Scopolamine; Xanthenes

2000
Role for rapid dendritic protein synthesis in hippocampal mGluR-dependent long-term depression.
    Science (New York, N.Y.), 2000, May-19, Volume: 288, Issue:5469

    Topics: Amino Acids; Animals; Anisomycin; Dendrites; Electric Stimulation; Excitatory Amino Acid Antagonists; Hippocampus; Methoxyhydroxyphenylglycol; Nerve Tissue Proteins; Neural Inhibition; Protein Biosynthesis; Protein Synthesis Inhibitors; Rats; Receptors, Metabotropic Glutamate; RNA, Messenger; Synaptic Transmission; Xanthenes

2000
Characterization of [(3)H]-LY354740 binding to rat mGlu2 and mGlu3 receptors expressed in CHO cells using semliki forest virus vectors.
    Neuropharmacology, 2000, Jul-24, Volume: 39, Issue:10

    Topics: Amino Acids; Animals; Binding, Competitive; Bridged Bicyclo Compounds; Cell Membrane; Chlorides; CHO Cells; Cricetinae; DNA, Recombinant; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Gene Expression; Genetic Vectors; Glutamic Acid; Guanosine 5'-O-(3-Thiotriphosphate); Kinetics; Rats; Receptors, Metabotropic Glutamate; Semliki forest virus; Tritium; Xanthenes; Zinc Compounds

2000
The potent, selective mGlu2/3 receptor agonist LY379268 increases extracellular levels of dopamine, 3,4-dihydroxyphenylacetic acid, homovanillic acid, and 5-hydroxyindole-3-acetic acid in the medial prefrontal cortex of the freely moving rat.
    Journal of neurochemistry, 2000, Volume: 75, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Amino Acids; Animals; Bridged Bicyclo Compounds, Heterocyclic; Clozapine; Dopamine; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Homovanillic Acid; Hydroxyindoleacetic Acid; Kinetics; Male; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Xanthenes

2000
The mGlu(2/3) receptor agonist LY379268 selectively blocks amphetamine ambulations and rearing.
    European journal of pharmacology, 2000, Jul-21, Volume: 400, Issue:2-3

    Topics: Amino Acids; Amphetamine; Animals; Bridged Bicyclo Compounds, Heterocyclic; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Male; Motor Activity; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Stereotyped Behavior; Xanthenes

2000
Behavioral evidence for interactions between a hallucinogenic drug and group II metabotropic glutamate receptors.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2000, Volume: 23, Issue:5

    Topics: Amino Acids; Amphetamines; Animals; Behavior, Animal; Bridged Bicyclo Compounds; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Hallucinogens; Male; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Metabotropic Glutamate; Receptors, Serotonin; Xanthenes

2000
Activity-dependent presynaptic autoinhibition by group II metabotropic glutamate receptors at the perforant path inputs to the dentate gyrus and CA1.
    Neuropharmacology, 2001, Volume: 40, Issue:1

    Topics: Amino Acids; Animals; Dentate Gyrus; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Hippocampus; In Vitro Techniques; Neural Pathways; Rats; Receptors, Metabotropic Glutamate; Xanthenes

2001
Binding of [3H](2S,1'S,2'S)-2-(9-xanthylmethyl)-2-(2'-carboxycyclopropyl) glycine ([3H]LY341495) to cell membranes expressing recombinant human group III metabotropic glutamate receptor subtypes.
    Naunyn-Schmiedeberg's archives of pharmacology, 2000, Volume: 362, Issue:6

    Topics: Amino Acids; Binding, Competitive; Cell Membrane; Excitatory Amino Acid Antagonists; Humans; Kinetics; Radioligand Assay; Receptors, Metabotropic Glutamate; Recombinant Proteins; Substrate Specificity; Tritium; Xanthenes

2000
Activation of group III mGluRs inhibits GABAergic and glutamatergic transmission in the substantia nigra pars reticulata.
    Journal of neurophysiology, 2001, Volume: 85, Issue:5

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Amino Acids; Aminobutyrates; Animals; Bicuculline; Drug Design; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Glycine; Kainic Acid; Nerve Tissue Proteins; Patch-Clamp Techniques; Phosphoserine; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, GABA-A; Receptors, Metabotropic Glutamate; Receptors, Presynaptic; Substantia Nigra; Xanthenes

2001
Group II and III metabotropic glutamate receptors contribute to different aspects of visual response processing in the rat superior colliculus.
    The Journal of physiology, 2001, Jul-01, Volume: 534, Issue:Pt 1

    Topics: Amino Acids; Animals; Bridged Bicyclo Compounds; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Habituation, Psychophysiologic; Rats; Rats, Inbred Strains; Receptors, Metabotropic Glutamate; Superior Colliculi; Visual Perception; Xanthenes

2001
[3H]LY341495 binding to group II metabotropic glutamate receptors in rat brain.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 298, Issue:2

    Topics: Amino Acids; Animals; Autoradiography; Binding, Competitive; Brain; Excitatory Amino Acid Antagonists; In Vitro Techniques; Kinetics; Male; Membranes; Protein Binding; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Xanthenes

2001
Evidence that glutamate acting on presynaptic type-II metabotropic glutamate receptors alone does not fully account for the phenomenon of depolarisation-induced suppression of inhibition in cerebellar Purkinje cells.
    Pflugers Archiv : European journal of physiology, 2001, Volume: 442, Issue:3

    Topics: Amino Acids; Animals; Excitatory Amino Acid Antagonists; Glutamic Acid; In Vitro Techniques; Neural Inhibition; Purkinje Cells; Rats; Receptors, Metabotropic Glutamate; Receptors, Presynaptic; Signal Transduction; Xanthenes

2001
Changes in rat serum corticosterone after treatment with metabotropic glutamate receptor agonists or antagonists.
    Journal of neuroendocrinology, 2001, Volume: 13, Issue:8

    Topics: Adrenalectomy; Adrenocorticotropic Hormone; Amino Acids; Animals; Benzoates; Bridged Bicyclo Compounds; Corticosterone; Cycloleucine; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Glycine; Male; Neuroprotective Agents; Paraventricular Hypothalamic Nucleus; Phenylacetates; Propionates; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols; Xanthenes

2001
Differential modulation of the D1-like- and D2-like dopamine receptor-induced locomotor responses by group II metabotropic glutamate receptors in the rat nucleus accumbens.
    Neuropharmacology, 2001, Volume: 41, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amino Acids; Animals; Dopamine Agonists; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Male; Motor Activity; Nucleus Accumbens; Proline; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Metabotropic Glutamate; Xanthenes

2001
Internalization of ionotropic glutamate receptors in response to mGluR activation.
    Nature neuroscience, 2001, Volume: 4, Issue:11

    Topics: Amino Acids; Animals; Cells, Cultured; Cycloheximide; Dendrites; Electrophysiology; Endocytosis; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glycine; Hippocampus; Immunohistochemistry; In Vitro Techniques; Methoxyhydroxyphenylglycol; Neurons; Protein Synthesis Inhibitors; Rats; Rats, Long-Evans; Receptors, AMPA; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Resorcinols; Synapses; Synapsins; Synaptic Transmission; Xanthenes

2001
Postsynaptic induction and presynaptic expression of group 1 mGluR-dependent LTD in the hippocampal CA1 region.
    Journal of neurophysiology, 2002, Volume: 87, Issue:3

    Topics: 4-Aminopyridine; Amino Acids; Animals; Calcium Signaling; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Hippocampus; Long-Term Potentiation; Male; Methoxyhydroxyphenylglycol; Mice; Mice, Inbred C57BL; Neural Inhibition; Organ Culture Techniques; Potassium Channel Blockers; Presynaptic Terminals; Receptors, Metabotropic Glutamate; Synaptic Transmission; Xanthenes

2002
Neuroprotective effects of N-acetylaspartylglutamate in a neonatal rat model of hypoxia-ischemia.
    European journal of pharmacology, 2002, Feb-22, Volume: 437, Issue:3

    Topics: Amino Acids; Animals; Animals, Newborn; Brain; Carboxypeptidases; Cyclic AMP; Cycloleucine; Dipeptides; Disease Models, Animal; Dose-Response Relationship, Drug; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Glutamate Carboxypeptidase II; Hippocampus; Hypoxia-Ischemia, Brain; Neurons; Neuroprotective Agents; Organophosphorus Compounds; Propionates; Rats; Rats, Sprague-Dawley; Xanthenes

2002
Role of p/q-Ca2+ channels in metabotropic glutamate receptor 2/3-dependent presynaptic long-term depression at nucleus accumbens synapses.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2002, Jun-01, Volume: 22, Issue:11

    Topics: Amino Acids; Animals; Bridged Bicyclo Compounds; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Channels, P-Type; Calcium Channels, Q-Type; Cyclic AMP-Dependent Protein Kinases; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Neural Inhibition; Neuronal Plasticity; Nucleus Accumbens; Patch-Clamp Techniques; Presynaptic Terminals; Receptors, Metabotropic Glutamate; Signal Transduction; Synapses; Synaptic Transmission; Xanthenes

2002
Group I metabotropic glutamate receptors (mGluRs) modulate visual responses in the superficial superior colliculus of the rat.
    The Journal of physiology, 2002, Jun-15, Volume: 541, Issue:Pt 3

    Topics: Amino Acids; Animals; Electric Stimulation; Electrodes; Excitatory Postsynaptic Potentials; GABA Antagonists; Habituation, Psychophysiologic; In Vitro Techniques; Iontophoresis; Membrane Potentials; Methoxyhydroxyphenylglycol; Photic Stimulation; Rats; Receptors, Metabotropic Glutamate; Superior Colliculi; Synapses; Vision, Ocular; Xanthenes

2002
Modulation of DOI-induced increases in cortical BDNF expression by group II mGlu receptors.
    Pharmacology, biochemistry, and behavior, 2002, Volume: 73, Issue:2

    Topics: Amino Acids; Amphetamines; Animals; Brain-Derived Neurotrophic Factor; Bridged Bicyclo Compounds; Cerebral Cortex; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; In Situ Hybridization; Male; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; RNA, Messenger; Xanthenes

2002
The anxiolytic action of mGlu2/3 receptor agonist, LY354740, in the fear-potentiated startle model in rats is mechanistically distinct from diazepam.
    Pharmacology, biochemistry, and behavior, 2002, Volume: 73, Issue:2

    Topics: Acoustic Stimulation; Amino Acids; Animals; Anti-Anxiety Agents; Bridged Bicyclo Compounds; Diazepam; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Fear; Flumazenil; GABA Modulators; Male; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Reflex, Startle; Xanthenes

2002
Different metabotropic glutamate receptors play opposite roles in synaptic plasticity of the rat medial vestibular nuclei.
    The Journal of physiology, 2002, Sep-15, Volume: 543, Issue:Pt 3

    Topics: Amino Acids; Animals; Chromones; Excitatory Amino Acid Antagonists; Glycine; Membrane Potentials; Neuronal Plasticity; Organ Culture Techniques; Phenylacetates; Pyridines; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols; Vestibular Nuclei; Xanthenes

2002
Synthesis and structure-activity relationship studies of novel 2-diarylethyl substituted (2-carboxycycloprop-1-yl)glycines as high-affinity group II metabotropic glutamate receptor ligands.
    Bioorganic & medicinal chemistry, 2003, Jan-17, Volume: 11, Issue:2

    Topics: Amino Acids; Benzene Derivatives; Cell Line; Cloning, Molecular; Excitatory Amino Acid Antagonists; Glycine; Humans; Inhibitory Concentration 50; Ligands; Receptors, Metabotropic Glutamate; Recombinant Proteins; Stereoisomerism; Structure-Activity Relationship; Tritium; Xanthenes

2003
Group II metabotropic glutamate receptor modulation of DOI-induced c-fos mRNA and excitatory responses in the cerebral cortex.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2003, Volume: 28, Issue:1

    Topics: Amino Acids; Amphetamines; Animals; Autoradiography; Bridged Bicyclo Compounds; Cerebral Cortex; DNA; Electrophysiology; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Agonists; Image Interpretation, Computer-Assisted; In Situ Hybridization; Male; Prefrontal Cortex; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; RNA, Messenger; Serotonin Receptor Agonists; Xanthenes

2003
Pharmacological blockade of mGlu2/3 metabotropic glutamate receptors reduces cell proliferation in cultured human glioma cells.
    Journal of neurochemistry, 2003, Volume: 84, Issue:6

    Topics: Amino Acids; Bridged Bicyclo Compounds, Heterocyclic; Cell Division; Cells, Cultured; Cyclin D1; Cyclin D2; Cyclins; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glioma; Humans; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Receptors, Metabotropic Glutamate; Thymidine; Tritium; Xanthenes

2003
Evaluation of [3H]LY341495 for labeling group II metabotropic glutamate receptors in vivo.
    Nuclear medicine and biology, 2003, Volume: 30, Issue:2

    Topics: Amino Acids; Animals; Brain; Male; Metabolic Clearance Rate; Radioligand Assay; Radionuclide Imaging; Radiopharmaceuticals; Rats; Receptors, Metabotropic Glutamate; Temperature; Tissue Distribution; Tritium; Xanthenes

2003
Baseline glutamate levels affect group I and II mGluRs in layer V pyramidal neurons of rat sensorimotor cortex.
    Journal of neurophysiology, 2003, Volume: 89, Issue:3

    Topics: Amino Acids; Anesthetics, Local; Animals; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; Glutamic Acid; Male; Membrane Potentials; Motor Cortex; Neural Inhibition; Organ Culture Techniques; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Somatosensory Cortex; Synaptic Transmission; Tetrodotoxin; Xanthenes

2003
Reduction of excitatory postsynaptic responses by persistently active metabotropic glutamate receptors in the hippocampus.
    Journal of neurophysiology, 2003, Volume: 89, Issue:4

    Topics: Amino Acids; Animals; Anticonvulsants; Cyclopropanes; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glycine; Hippocampus; Interneurons; Membrane Potentials; Mice; Mice, Inbred C57BL; Neuronal Plasticity; Presynaptic Terminals; Propionates; Receptors, Metabotropic Glutamate; Xanthenes

2003
Actions of LY341495 on metabotropic glutamate receptor-mediated responses in the neonatal rat spinal cord.
    British journal of pharmacology, 2003, Volume: 139, Issue:1

    Topics: Amino Acids; Aminobutyrates; Animals; Animals, Newborn; Cyclopentanes; In Vitro Techniques; Motor Neurons; Rats; Receptors, AMPA; Receptors, Kainic Acid; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Spinal Cord; Synaptic Transmission; Time Factors; Tricarboxylic Acids; Xanthenes

2003
Group II mGlu receptor activation suppresses norepinephrine release in the ventral hippocampus and locomotor responses to acute ketamine challenge.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2003, Volume: 28, Issue:9

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Amino Acids; Analysis of Variance; Animals; Area Under Curve; Binding Sites; Bridged Bicyclo Compounds, Heterocyclic; Chromatography, High Pressure Liquid; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Guanosine 5'-O-(3-Thiotriphosphate); Hippocampus; Humans; Hyperkinesis; In Vitro Techniques; Ketamine; Male; Microdialysis; Motor Activity; Norepinephrine; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Metabotropic Glutamate; Schizophrenia; Serotonin; Sulfur Isotopes; Time Factors; Trifluoroethanol; Xanthenes

2003
Protective role of group-II metabotropic glutamate receptors against nigro-striatal degeneration induced by 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine in mice.
    Neuropharmacology, 2003, Volume: 45, Issue:2

    Topics: Amino Acids; Animals; Bridged Bicyclo Compounds, Heterocyclic; Male; Mice; Mice, Inbred C57BL; MPTP Poisoning; Neuroprotective Agents; Receptors, AMPA; Xanthenes

2003
GCP II (NAALADase) inhibition suppresses mossy fiber-CA3 synaptic neurotransmission by a presynaptic mechanism.
    Journal of neurophysiology, 2004, Volume: 91, Issue:1

    Topics: Amino Acids; Analysis of Variance; Animals; Animals, Newborn; Calcium; Chemokine CXCL6; Chemokines, CXC; Dose-Response Relationship, Drug; Drug Interactions; Electric Conductivity; Electric Stimulation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutarates; In Vitro Techniques; Male; Mossy Fibers, Hippocampal; Neural Inhibition; Neurons; Patch-Clamp Techniques; Presynaptic Terminals; Probability; Rats; Sulfhydryl Compounds; Synaptic Transmission; Time Factors; Xanthenes

2004
Group II metabotropic glutamate receptor antagonists LY341495 and LY366457 increase locomotor activity in mice.
    Neuropharmacology, 2003, Volume: 45, Issue:5

    Topics: Amino Acids; Animals; Benzazepines; Dizocilpine Maleate; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Female; Fluorobenzenes; Haloperidol; Hyperkinesis; Mice; Motor Activity; Piperidines; Receptors, Metabotropic Glutamate; Serotonin Antagonists; Time Factors; Xanthenes

2003
Pharmacological characterization and identification of amino acids involved in the positive modulation of metabotropic glutamate receptor subtype 2.
    Molecular pharmacology, 2003, Volume: 64, Issue:4

    Topics: Allosteric Regulation; Amino Acid Sequence; Amino Acids; Animals; Binding Sites; Calcium; Cell Membrane; Cerebral Cortex; CHO Cells; Cricetinae; Cyclopropanes; Dentate Gyrus; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Guanosine 5'-O-(3-Thiotriphosphate); Hippocampus; Humans; Molecular Sequence Data; Perforant Pathway; Protein Structure, Tertiary; Pyridines; Rats; Receptors, Metabotropic Glutamate; Sequence Homology, Amino Acid; Sulfonamides; Tritium; Xanthenes

2003
Group II metabotropic glutamate receptor modulation of excitatory transmission in rat subthalamic nucleus.
    The Journal of physiology, 2003, Dec-01, Volume: 553, Issue:Pt 2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 2-Amino-5-phosphonovalerate; 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; 6-Cyano-7-nitroquinoxaline-2,3-dione; Adenylyl Cyclase Inhibitors; Amino Acids; Amino Acids, Dicarboxylic; Animals; Colforsin; Cyclopropanes; Electric Stimulation; Electrophysiology; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; Glycine; Imines; In Vitro Techniques; Isoquinolines; Male; Picrotoxin; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Subthalamic Nucleus; Sulfonamides; Synaptic Transmission; Tetradecanoylphorbol Acetate; Xanthenes

2003
Protective effect of LY379268, a selective group II metabotropic glutamate receptor agonist, on dizocilpine-induced neuropathological changes in rat retrosplenial cortex.
    Brain research, 2003, Nov-28, Volume: 992, Issue:1

    Topics: Acetylcholine; Amino Acids; Animals; Brain; Bridged Bicyclo Compounds, Heterocyclic; Chromatography, High Pressure Liquid; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Extracellular Fluid; Female; HSP70 Heat-Shock Proteins; Immunohistochemistry; Microdialysis; Neuroprotective Agents; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Xanthenes

2003
Cannabinoids decrease corticostriatal synaptic transmission via an effect on glutamate uptake.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2003, Dec-03, Volume: 23, Issue:35

    Topics: Amino Acids; Animals; Cannabinoids; Cerebral Cortex; Corpus Striatum; Dronabinol; Glutamic Acid; In Vitro Techniques; Male; Neural Inhibition; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Metabotropic Glutamate; Rimonabant; Synaptic Transmission; Xanthenes

2003
The mGlu2/3 receptor agonist, LY354740, blocks immobilization-induced increases in noradrenaline and dopamine release in the rat medial prefrontal cortex.
    Journal of neurochemistry, 2004, Volume: 88, Issue:1

    Topics: Amino Acids; Animals; Bridged Bicyclo Compounds; Catecholamines; Citalopram; Dopamine; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Extracellular Fluid; Male; Microdialysis; Norepinephrine; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Restraint, Physical; Selective Serotonin Reuptake Inhibitors; Stress, Physiological; Xanthenes

2004
Prefrontal group II metabotropic glutamate receptor activation decreases performance on a working memory task.
    Annals of the New York Academy of Sciences, 2003, Volume: 1003

    Topics: Amino Acids; Animals; Excitatory Amino Acid Antagonists; Extracellular Space; Feedback; Glutamates; Memory, Short-Term; Microinjections; Prefrontal Cortex; Proline; Psychomotor Performance; Rats; Receptors, AMPA; Xanthenes

2003
Bidirectional modulation of cystine/glutamate exchanger activity in cultured cortical astrocytes.
    Annals of the New York Academy of Sciences, 2003, Volume: 1003

    Topics: Amino Acids; Animals; Astrocytes; Carrier Proteins; Cells, Cultured; Cerebral Cortex; Cystine; Enzyme Activators; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Phosphotransferases; Proline; Rats; Receptors, Metabotropic Glutamate; Xanthenes

2003
Selective transmission of single photon responses by saturation at the rod-to-rod bipolar synapse.
    Neuron, 2004, Feb-05, Volume: 41, Issue:3

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Amino Acids; Aminobutyrates; Animals; Binding Sites; Darkness; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Light; Membrane Potentials; Mice; Mice, Inbred C57BL; Neurons; Patch-Clamp Techniques; Photons; Retina; Retinal Rod Photoreceptor Cells; Synapses; Synaptic Transmission; Valine; Xanthenes

2004
An NMDAR-independent LTP mediated by group II metabotropic glutamate receptors and p42/44 MAP kinase in the dentate gyrus in vitro.
    Neuropharmacology, 2004, Volume: 46, Issue:3

    Topics: Amino Acids; Animals; Cyclopropanes; Dentate Gyrus; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; Glycine; In Vitro Techniques; Long-Term Potentiation; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Xanthenes

2004
Inhibitory effects of group II mGluR-related drugs on memory performance in mice.
    Physiology & behavior, 2004, Volume: 80, Issue:5

    Topics: Amino Acids; Animals; Anticonvulsants; Avoidance Learning; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclopropanes; Dose-Response Relationship, Drug; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Glycine; Isoquinolines; Male; Memory; Mice; Reaction Time; Receptors, Metabotropic Glutamate; Rolipram; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Xanthenes

2004
The selective mGlu2/3 receptor antagonist LY341495 exacerbates behavioral signs of morphine withdrawal and morphine-withdrawal-induced activation of locus coeruleus neurons.
    Neuropharmacology, 2004, Volume: 46, Issue:5

    Topics: Action Potentials; Amino Acids; Animals; Excitatory Amino Acid Antagonists; Locus Coeruleus; Male; Morphine Dependence; Neurons; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Substance Withdrawal Syndrome; Xanthenes

2004
Group II metabotropic glutamate receptors inhibit cAMP-dependent protein kinase-mediated enhancemednt of tetrodotoxin-resistant sodium currents in mouse dorsal root ganglion neurons.
    Neuroscience letters, 2004, Mar-11, Volume: 357, Issue:3

    Topics: Amino Acids; Analysis of Variance; Animals; Animals, Newborn; Cells, Cultured; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Ganglia, Spinal; Membrane Potentials; Mice; NAV1.7 Voltage-Gated Sodium Channel; Neurons; Neuropeptides; Pyrrolidines; Receptors, Metabotropic Glutamate; Sodium Channels; Thiocarbamates; Time Factors; Xanthenes

2004
Tonic activity of metabotropic glutamate receptors is involved in developmental modification of short-term plasticity in the neocortex.
    Journal of neurophysiology, 2004, Volume: 92, Issue:2

    Topics: Aging; Amino Acids; Animals; Animals, Newborn; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; In Vitro Techniques; Neocortex; Neuronal Plasticity; Presynaptic Terminals; Rats; Receptors, Metabotropic Glutamate; Synapses; Time Factors; Xanthenes

2004
Pharmacological manipulation of mGlu2 receptors influences cognitive performance in the rodent.
    Neuropharmacology, 2004, Volume: 46, Issue:7

    Topics: Amino Acids; Animals; Bridged Bicyclo Compounds; Cognition; Dose-Response Relationship, Drug; Excitatory Postsynaptic Potentials; Male; Maze Learning; Mice; Mice, Inbred C57BL; Mice, Knockout; Psychomotor Performance; Rats; Reaction Time; Receptors, Metabotropic Glutamate; Xanthenes

2004
Depression of GABAergic input to identified hippocampal neurons by group III metabotropic glutamate receptors in the rat.
    The European journal of neuroscience, 2004, Volume: 19, Issue:10

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Animals, Newborn; Cell Count; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Hippocampus; Horseradish Peroxidase; Immunohistochemistry; In Vitro Techniques; Interneurons; Lysine; Membrane Potentials; Microscopy, Immunoelectron; Neural Inhibition; Patch-Clamp Techniques; Propionates; Pyramidal Cells; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Somatostatin; Statistics, Nonparametric; Synapses; Time Factors; Xanthenes

2004
Distinct properties of presynaptic group II and III metabotropic glutamate receptor-mediated inhibition of perforant pathway-CA1 EPSCs.
    The European journal of neuroscience, 2004, Volume: 19, Issue:10

    Topics: Amino Acids; Aminobutyrates; Animals; Bridged Bicyclo Compounds; Calcium Channel Blockers; Cyclic AMP; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Interactions; Elapid Venoms; Electric Stimulation; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; Hippocampus; In Vitro Techniques; Membrane Potentials; Neural Inhibition; omega-Conotoxin GVIA; Perforant Pathway; Phosphinic Acids; Propanolamines; Quinoxalines; Rats; Receptors, Metabotropic Glutamate; Statistics, Nonparametric; Synaptic Transmission; Thionucleotides; Time Factors; Xanthenes

2004
Effect of donepezil on group II mGlu receptor agonist- or antagonist-induced amnesia on passive avoidance in mice.
    Neural plasticity, 2003, Volume: 10, Issue:4

    Topics: Amino Acids; Amnesia; Animals; Avoidance Learning; Cholinesterase Inhibitors; Cyclopropanes; Donepezil; Excitatory Amino Acid Antagonists; Glycine; Indans; Male; Memory; Mice; Nootropic Agents; Piperidines; Receptors, Metabotropic Glutamate; Xanthenes

2003
Modulation of glutamate mobility reveals the mechanism underlying slow-rising AMPAR EPSCs and the diffusion coefficient in the synaptic cleft.
    Neuron, 2004, Jun-10, Volume: 42, Issue:5

    Topics: Amino Acids; Animals; Animals, Newborn; Benzylamines; Cerebellum; Computer Simulation; Dextrans; Diffusion; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; In Vitro Techniques; Membrane Potentials; Nerve Fibers; Neurons; Patch-Clamp Techniques; Phosphinic Acids; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, AMPA; Synapses; Synaptic Transmission; Time Factors; Xanthenes

2004
Retroinhibition of presynaptic Ca2+ currents by endocannabinoids released via postsynaptic mGluR activation at a calyx synapse.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2004, Jun-30, Volume: 24, Issue:26

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Amino Acids; Animals; Benzoxazines; Brain Stem; Calcium Signaling; Cannabinoid Receptor Modulators; Endocannabinoids; Evoked Potentials, Auditory, Brain Stem; Glycine; Ion Transport; Morpholines; Naphthalenes; Nerve Endings; Patch-Clamp Techniques; Picrotoxin; Piperidines; Pyrazoles; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Metabotropic Glutamate; Receptors, Presynaptic; Resorcinols; Scopolamine; Synaptic Transmission; Xanthenes

2004
Antinociceptive effects of N-acetylaspartylglutamate (NAAG) peptidase inhibitors ZJ-11, ZJ-17 and ZJ-43 in the rat formalin test and in the rat neuropathic pain model.
    The European journal of neuroscience, 2004, Volume: 20, Issue:2

    Topics: Amino Acids; Analgesics; Animals; Behavior, Animal; Cell Line; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Glutamate Carboxypeptidase II; Humans; Immunohistochemistry; Injections, Intravenous; Injections, Spinal; Nociceptors; Pain; Pain Measurement; Pain Threshold; Physical Stimulation; Protease Inhibitors; Proto-Oncogene Proteins c-fos; Rats; Reaction Time; Sciatic Neuropathy; Urea; Xanthenes

2004
Distinct properties of carbachol- and DHPG-induced network oscillations in hippocampal slices.
    Neuropharmacology, 2004, Volume: 47, Issue:3

    Topics: Action Potentials; Amino Acids; Animals; Animals, Newborn; Benzodiazepines; Bicuculline; Carbachol; Cholinergic Agonists; Diamines; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; Hippocampus; In Vitro Techniques; Male; Methoxyhydroxyphenylglycol; Muscarinic Antagonists; Pirenzepine; Pyridines; Rats; Receptors, Metabotropic Glutamate; Spectrum Analysis; Substance P; Xanthenes; Zolpidem

2004
The metabotropic glutamate (mGLU)2/3 receptor antagonist LY341495 [2S-2-amino-2-(1S,2S-2-carboxycyclopropyl-1-yl)-3-(xanth-9-yl)propanoic acid] stimulates waking and fast electroencephalogram power and blocks the effects of the mGLU2/3 receptor agonist ly
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 312, Issue:2

    Topics: Amino Acids; Animals; Arousal; Behavior, Animal; Bridged Bicyclo Compounds, Heterocyclic; Darkness; Electroencephalography; Excitatory Amino Acid Antagonists; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Metabotropic Glutamate; Sleep; Sleep Stages; Wakefulness; Xanthenes

2005
Glutamate transporters and metabotropic receptors regulate excitatory neurotransmission in the medial entorhinal cortex of the rat.
    Brain research, 2004, Nov-19, Volume: 1027, Issue:1-2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amino Acid Transport System X-AG; Amino Acids; Animals; Aspartic Acid; Dicarboxylic Acids; Drug Interactions; Entorhinal Cortex; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Glycine; In Vitro Techniques; N-Methylaspartate; Neurotransmitter Uptake Inhibitors; Patch-Clamp Techniques; Pyrrolidines; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Synaptic Transmission; Xanthenes

2004
Metabotropic glutamate receptors modulate feedback inhibition in a developmentally regulated manner in rat dentate gyrus.
    The Journal of physiology, 2004, Dec-01, Volume: 561, Issue:Pt 2

    Topics: Amino Acids; Animals; Dentate Gyrus; Excitatory Postsynaptic Potentials; Feedback, Physiological; Neural Inhibition; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Xanthenes

2004
Activation of Group II and Group III metabotropic glutamate receptors by endogenous ligand(s) and the modulation of synaptic transmission in the superficial superior colliculus.
    Neuropharmacology, 2004, Volume: 47, Issue:6

    Topics: Action Potentials; Amino Acids; Animals; Biotransformation; Dose-Response Relationship, Drug; Drug Synergism; Excitatory Postsynaptic Potentials; Extracellular Space; Glutamates; Ligands; Rats; Receptors, AMPA; Superior Colliculi; Synaptic Transmission; Xanthenes

2004
Glutamate-evoked alterations of glial and neuronal cell morphology in the guinea pig retina.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2004, Nov-10, Volume: 24, Issue:45

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Adenosine Triphosphate; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amino Acids; Animals; Aspartic Acid; Cell Size; Circadian Rhythm; Cytochalasin D; Cytoskeleton; Dicarboxylic Acids; Dopamine; Eye Proteins; Glutamic Acid; Guinea Pigs; Ischemia; Kainic Acid; N-Methylaspartate; Neuroglia; Neurons; Nocodazole; Potassium; Pyrrolidines; Receptors, AMPA; Receptors, Kainic Acid; Retina; Retinal Ganglion Cells; Synaptic Transmission; Xanthenes

2004
A novel selective positive allosteric modulator of metabotropic glutamate receptor subtype 5 has in vivo activity and antipsychotic-like effects in rat behavioral models.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 313, Issue:1

    Topics: Amino Acids; Amphetamine; Animals; Antipsychotic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Behavior, Animal; Benzamides; Cell Line; Central Nervous System Stimulants; CHO Cells; Cricetinae; Dogs; Excitatory Amino Acid Antagonists; Female; Haplorhini; Humans; Image Interpretation, Computer-Assisted; In Vitro Techniques; Microsomes, Liver; Models, Statistical; Motor Activity; Phthalimides; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Reflex, Startle; Xanthenes

2005
Anxiolytic-like activity of the mGLU2/3 receptor agonist LY354740 in the elevated plus maze test is disrupted in metabotropic glutamate receptor 2 and 3 knock-out mice.
    Psychopharmacology, 2005, Volume: 179, Issue:1

    Topics: Amino Acids; Amygdala; Animals; Anti-Anxiety Agents; Bridged Bicyclo Compounds; Excitatory Amino Acid Agonists; Female; Male; Maze Learning; Mice; Mice, Inbred C57BL; Mice, Inbred ICR; Mice, Knockout; Receptors, Metabotropic Glutamate; Xanthenes

2005
Seizures induced in immature rats by homocysteic acid and the associated brain damage are prevented by group II metabotropic glutamate receptor agonist (2R,4R)-4-aminopyrrolidine-2,4-dicarboxylate.
    Experimental neurology, 2005, Volume: 192, Issue:2

    Topics: Amino Acids; Animals; Animals, Newborn; Anticonvulsants; Behavior, Animal; Brain; Brain Chemistry; Brain Injuries; Dose-Response Relationship, Drug; Drug Interactions; Electroencephalography; Excitatory Amino Acid Antagonists; Fluoresceins; Fluorescent Dyes; Functional Laterality; Glucose; Glycogen; Homocysteine; Lactic Acid; Male; Nerve Degeneration; Organic Chemicals; Proline; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Seizures; Time Factors; Xanthenes

2005
Presynaptic inhibition of corticothalamic feedback by metabotropic glutamate receptors.
    Journal of neurophysiology, 2005, Volume: 94, Issue:1

    Topics: Amino Acids; Animals; Animals, Newborn; Bridged Bicyclo Compounds, Heterocyclic; Cyclopropanes; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Feedback; Ferrets; Geniculate Bodies; Glycine; In Vitro Techniques; Male; Neural Inhibition; Neural Pathways; Neurons; Presynaptic Terminals; Receptors, Metabotropic Glutamate; Synaptic Transmission; Time Factors; Xanthenes

2005
Developmental switch in synaptic mechanisms of hippocampal metabotropic glutamate receptor-dependent long-term depression.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Mar-16, Volume: 25, Issue:11

    Topics: Age Factors; Amino Acids; Animals; Animals, Newborn; Anisomycin; Benzoxazines; Cycloheximide; Dizocilpine Maleate; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Antagonists; Hippocampus; In Vitro Techniques; Long-Term Synaptic Depression; Methoxyhydroxyphenylglycol; Morpholines; Naphthalenes; Neurons; Protein Synthesis Inhibitors; Pyrazoles; Rats; Rats, Long-Evans; Reaction Time; Receptor, Cannabinoid, CB1; Receptors, Metabotropic Glutamate; Synapses; Xanthenes

2005
Neuropharmacological profiles of antagonists of group II metabotropic glutamate receptors.
    Neuroscience letters, 2005, Apr-22, Volume: 378, Issue:3

    Topics: Action Potentials; Amino Acids; Animals; Antidepressive Agents; Biogenic Monoamines; Bridged Bicyclo Compounds; Dicarboxylic Acids; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Extracellular Fluid; Locus Coeruleus; Male; Neurons; Prefrontal Cortex; Raphe Nuclei; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Serotonin; Xanthenes

2005
Metabotropic glutamate receptors and neuroadaptation to antidepressants: imipramine-induced down-regulation of beta-adrenergic receptors in mice treated with metabotropic glutamate 2/3 receptor ligands.
    Journal of neurochemistry, 2005, Volume: 93, Issue:5

    Topics: Adaptation, Physiological; Amino Acids; Animals; Antidepressive Agents, Tricyclic; Bridged Bicyclo Compounds, Heterocyclic; Down-Regulation; Excitatory Amino Acid Antagonists; Hippocampus; Imipramine; Ligands; Male; Mice; Mice, Inbred Strains; Nervous System Physiological Phenomena; Reaction Time; Receptors, Adrenergic, beta; Receptors, Metabotropic Glutamate; Xanthenes

2005
Metabotropic glutamate receptor 2 modulates excitatory synaptic transmission in the rat globus pallidus.
    Neuropharmacology, 2005, Volume: 49 Suppl 1

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Amino Acids; Aminobutyrates; Anesthetics, Local; Animals; Animals, Newborn; Cyclopropanes; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Globus Pallidus; Glycine; In Vitro Techniques; Lidocaine; Membrane Potentials; Methoxyhydroxyphenylglycol; Neurons; Patch-Clamp Techniques; Proline; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Sulfonamides; Synaptic Transmission; Xanthenes

2005
Group II and III mGluRs-mediated presynaptic inhibition of EPSCs recorded from hippocampal interneurons of CA1 stratum lacunosum moleculare.
    Neuropharmacology, 2005, Volume: 49 Suppl 1

    Topics: Amino Acids; Aminobutyrates; Analysis of Variance; Animals; Animals, Newborn; Bridged Bicyclo Compounds; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Hippocampus; In Vitro Techniques; Interneurons; Neural Inhibition; Perforant Pathway; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Strontium; Tetrodotoxin; Time Factors; Xanthenes

2005
Cystine/glutamate exchange regulates metabotropic glutamate receptor presynaptic inhibition of excitatory transmission and vulnerability to cocaine seeking.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Jul-06, Volume: 25, Issue:27

    Topics: Amino Acids; Animals; Biological Transport; Cocaine; Cocaine-Related Disorders; Consummatory Behavior; Cystine; Excitatory Amino Acid Antagonists; Extinction, Psychological; Glutamic Acid; Male; Neural Conduction; Nucleus Accumbens; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Receptors, Presynaptic; Self Administration; Xanthenes

2005
Comparison of c-Fos induction in the brain by the mGlu2/3 receptor antagonist LY341495 and agonist LY354740: evidence for widespread endogenous tone at brain mGlu2/3 receptors in vivo.
    Neuropharmacology, 2005, Volume: 49 Suppl 1

    Topics: Amino Acids; Analysis of Variance; Animals; Brain; Bridged Bicyclo Compounds; Cell Count; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Gene Expression Regulation; Immunohistochemistry; Male; Mice; Mice, Inbred ICR; Neurons; Proto-Oncogene Proteins c-fos; Xanthenes

2005
The preferential mGlu2/3 receptor antagonist, LY341495, reduces the frequency of spike-wave discharges in the WAG/Rij rat model of absence epilepsy.
    Neuropharmacology, 2005, Volume: 49 Suppl 1

    Topics: Age Factors; Amino Acids; Analysis of Variance; Animals; Baclofen; Behavior, Animal; Blotting, Western; Brain; Brain Mapping; Circadian Rhythm; Cyclic AMP; Disease Models, Animal; Electroencephalography; Epilepsy, Absence; Excitatory Amino Acid Antagonists; GABA Agonists; Glial Fibrillary Acidic Protein; Immunohistochemistry; Indoles; Male; Microdialysis; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Metabotropic Glutamate; Xanthenes

2005
Pharmacological blockade of group II metabotropic glutamate receptors reduces the growth of glioma cells in vivo.
    Neuro-oncology, 2005, Volume: 7, Issue:3

    Topics: Amino Acids; Animals; Blotting, Western; Brain Neoplasms; Cell Line, Tumor; Cell Proliferation; Cyclin D1; Cyclin D2; Cyclins; Enzyme Activation; Excitatory Amino Acid Antagonists; Glioma; Humans; Immunohistochemistry; Ki-67 Antigen; Magnetic Resonance Imaging; MAP Kinase Signaling System; Mice; Mice, Nude; Phosphatidylinositol 3-Kinases; Receptors, Metabotropic Glutamate; Reverse Transcriptase Polymerase Chain Reaction; Xanthenes

2005
Role of group II metabotropic glutamate receptors 2/3 and group I metabotropic glutamate receptor 5 in developing rat medial vestibular nuclei.
    Neuroreport, 2005, Aug-22, Volume: 16, Issue:12

    Topics: 2-Amino-5-phosphonovalerate; Age Factors; Amino Acids; Animals; Animals, Newborn; Dose-Response Relationship, Radiation; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; In Vitro Techniques; Long-Term Potentiation; Long-Term Synaptic Depression; Neural Inhibition; Phenylacetates; Rats; Rats, Wistar; Receptors, AMPA; Receptors, Kainic Acid; Synaptic Transmission; Vestibular Nuclei; Xanthenes

2005
Regulation of IPSP theta rhythm by muscarinic receptors and endocannabinoids in hippocampus.
    Journal of neurophysiology, 2005, Volume: 94, Issue:6

    Topics: Action Potentials; Amino Acids; Animals; Cannabinoid Receptor Modulators; Carbachol; Cholinergic Agonists; Endocannabinoids; Excitatory Amino Acid Antagonists; Hippocampus; In Vitro Techniques; Male; Methoxyhydroxyphenylglycol; Neural Inhibition; Piperidines; Pyrazoles; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Spectrum Analysis; Synapses; Theta Rhythm; Time Factors; Xanthenes

2005
Neuroprotective effect of N-acetyl-aspartyl-glutamate in combination with mild hypothermia in the endothelin-1 rat model of focal cerebral ischaemia.
    Journal of neurochemistry, 2005, Volume: 95, Issue:5

    Topics: Amino Acids; Animals; Blood-Brain Barrier; Brain Ischemia; Dipeptides; Disease Models, Animal; Drug Administration Schedule; Drug Therapy, Combination; Endothelin-1; Hypothermia; Male; Microdialysis; Neuroprotective Agents; Rats; Rats, Wistar; Time Factors; Xanthenes

2005
2-MPPA, a selective glutamate carboxypeptidase II inhibitor, attenuates morphine tolerance but not dependence in C57/Bl mice.
    Psychopharmacology, 2005, Volume: 183, Issue:3

    Topics: Amino Acids; Animals; Drug Tolerance; Enzyme Inhibitors; Glutamate Carboxypeptidase II; Male; Mice; Mice, Inbred C57BL; Morphine; Morphine Dependence; Naloxone; Organophosphorus Compounds; Receptors, Metabotropic Glutamate; Xanthenes

2005
Modulation of excitatory synaptic transmission by endogenous glutamate acting on presynaptic group II mGluRs in rat substantia nigra compacta.
    Journal of neuroscience research, 2005, Dec-15, Volume: 82, Issue:6

    Topics: Amino Acid Transport System X-AG; Amino Acids; Animals; Animals, Newborn; Aspartic Acid; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamates; In Vitro Techniques; Patch-Clamp Techniques; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Substantia Nigra; Synaptic Transmission; Xanthenes

2005
Antinociceptive effects and synergistic interaction with morphine of intrathecal metabotropic glutamate receptor 2/3 antagonist in the formalin test of rats.
    Neuroscience letters, 2006, Feb-20, Volume: 394, Issue:3

    Topics: Amino Acids; Analgesics; Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Drug Synergism; Excitatory Amino Acid Antagonists; Formaldehyde; Injections, Spinal; Male; Morphine; Pain Measurement; Proline; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Reflex; Xanthenes

2006
Olfactory nerve-evoked, metabotropic glutamate receptor-mediated synaptic responses in rat olfactory bulb mitral cells.
    Journal of neurophysiology, 2006, Volume: 95, Issue:4

    Topics: Amino Acids; Animals; Aspartic Acid; Benzoates; Dopamine D2 Receptor Antagonists; Electrophysiology; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; GABA-B Receptor Antagonists; Glutamic Acid; Glycine; In Vitro Techniques; Male; Neuronal Plasticity; Neurons, Afferent; Odorants; Olfactory Bulb; Olfactory Nerve; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, GABA-B; Receptors, Metabotropic Glutamate; Synapses; Tacrine; Xanthenes

2006
Differential negative coupling of type 3 metabotropic glutamate receptor to cyclic GMP levels in neurons and astrocytes.
    Journal of neurochemistry, 2006, Volume: 96, Issue:4

    Topics: Amino Acids; Animals; Animals, Newborn; Astrocytes; Cerebellum; Cyclic GMP; Dipeptides; Excitatory Amino Acid Antagonists; GTP-Binding Proteins; Neurons; Nitroprusside; Pertussis Toxin; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Xanthenes

2006
Differential roles for group 1 mGluR subtypes in induction and expression of chemically induced hippocampal long-term depression.
    Journal of neurophysiology, 2006, Volume: 95, Issue:4

    Topics: Action Potentials; Amino Acids; Animals; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Extracellular Signal-Regulated MAP Kinases; Hippocampus; Long-Term Synaptic Depression; Methoxyhydroxyphenylglycol; Mice; Mice, Knockout; Neuronal Plasticity; Neurons; Neurotransmitter Agents; Phosphorylation; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, AMPA; Receptors, Metabotropic Glutamate; Synapses; Xanthenes

2006
Long-term depression of NMDA receptor-mediated synaptic transmission is dependent on activation of metabotropic glutamate receptors and is altered to long-term potentiation by low intracellular calcium buffering.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2006, Jan-25, Volume: 26, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Amino Acids; Animals; Buffers; Calcium; Dentate Gyrus; Egtazic Acid; Electric Stimulation; Excitatory Amino Acid Antagonists; Long-Term Synaptic Depression; Male; Patch-Clamp Techniques; Perforant Pathway; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission; Xanthenes

2006
Unique presynaptic and postsynaptic roles of Group II metabotropic glutamate receptors in the modulation of thalamic network activity.
    Neuroscience, 2006, Aug-11, Volume: 141, Issue:1

    Topics: Amino Acids; Animals; Animals, Newborn; Bridged Bicyclo Compounds, Heterocyclic; Drug Interactions; Electric Stimulation; Excitatory Postsynaptic Potentials; Female; Ferrets; Gluconates; Guanosine Diphosphate; In Vitro Techniques; Male; Membrane Potentials; Nerve Net; Neurons; Organophosphorus Compounds; Patch-Clamp Techniques; Picrotoxin; Receptors, Metabotropic Glutamate; Synapses; Thalamus; Thionucleotides; Xanthenes

2006
Blockade of group II metabotropic glutamate receptors in the nucleus accumbens produces hyperlocomotion in rats previously exposed to amphetamine.
    Neuropharmacology, 2006, Volume: 51, Issue:5

    Topics: Amino Acids; Amphetamine; Analysis of Variance; Animals; Behavior, Animal; Bridged Bicyclo Compounds, Heterocyclic; Central Nervous System Stimulants; Drug Interactions; Hyperkinesis; Male; Motor Activity; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Xanthenes

2006
Analgesia mediated by the TRPM8 cold receptor in chronic neuropathic pain.
    Current biology : CB, 2006, Aug-22, Volume: 16, Issue:16

    Topics: Acrolein; Amino Acids; Analgesia; Analysis of Variance; Animals; Blotting, Western; Cold Temperature; Dose-Response Relationship, Drug; Electrophysiology; Immunohistochemistry; Male; Menthol; Neuralgia; Oligonucleotides, Antisense; Pyrimidinones; Rats; Rats, Wistar; Receptors, Glutamate; Reflex; TRPM Cation Channels; Xanthenes

2006
Group III metabotropic glutamate receptor agonists selectively suppress excitatory synaptic currents in the rat prefrontal cortex induced by 5-hydroxytryptamine2A receptor activation.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 320, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amino Acids; Animals; Bridged Bicyclo Compounds; Glycine; Male; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Metabotropic Glutamate; Serotonin; Synaptic Transmission; Xanthenes

2007
Effects of metabotropic glutamate 2/3 receptor antagonists in the stress-induced hyperthermia test in singly housed mice.
    Psychopharmacology, 2007, Volume: 190, Issue:2

    Topics: Amino Acids; Animals; Arousal; Autonomic Nervous System; Body Temperature Regulation; Bridged Bicyclo Compounds; Dicarboxylic Acids; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Male; Mice; Mice, Inbred ICR; Piperazines; Pyridines; Receptor, Serotonin, 5-HT1A; Receptors, Metabotropic Glutamate; Serotonin Antagonists; Social Isolation; Xanthenes

2007
Interactive effects of the mGlu5 receptor antagonist MPEP and the mGlu2/3 receptor antagonist LY341495 on nicotine self-administration and reward deficits associated with nicotine withdrawal in rats.
    European journal of pharmacology, 2007, Jan-12, Volume: 554, Issue:2-3

    Topics: Amino Acids; Animals; Dose-Response Relationship, Drug; Drug Interactions; Eating; Excitatory Amino Acid Antagonists; Ganglionic Stimulants; Infusions, Intravenous; Injections, Intraperitoneal; Male; Nicotine; Pyridines; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Reinforcement Schedule; Reward; Self Administration; Substance Withdrawal Syndrome; Time Factors; Xanthenes

2007
The effects of the mGluR5 antagonist MPEP and the mGluR2/3 antagonist LY341495 on rats' performance in the 5-choice serial reaction time task.
    Neuropharmacology, 2007, Volume: 52, Issue:3

    Topics: Amino Acids; Analysis of Variance; Animals; Behavior, Animal; Choice Behavior; Curare; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Male; Nicotinic Antagonists; Pyridines; Rats; Rats, Wistar; Reaction Time; Xanthenes

2007
Habituation deficits induced by metabotropic glutamate receptors 2/3 receptor blockade in mice: reversal by antipsychotic drugs.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 320, Issue:2

    Topics: Amino Acids; Animals; Antipsychotic Agents; Cognition Disorders; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Habituation, Psychophysiologic; Haloperidol; Male; Methamphetamine; Mice; Motor Activity; Nitriles; Receptors, Metabotropic Glutamate; Tetrahydroisoquinolines; Xanthenes

2007
Endogenous mGluR activity suppresses GABAergic transmission in avian cochlear nucleus magnocellularis neurons.
    Journal of neurophysiology, 2007, Volume: 97, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Chickens; Cochlear Nucleus; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Kinetics; Membrane Potentials; Models, Neurological; Neurons; Patch-Clamp Techniques; Receptors, GABA-B; Receptors, Metabotropic Glutamate; Resorcinols; Synapses; Synaptic Transmission; Xanthenes

2007
Pharmacological activation of mGlu2/3 metabotropic glutamate receptors protects retinal neurons against anoxic damage in the goldfish Carassius auratus.
    Experimental eye research, 2007, Volume: 84, Issue:3

    Topics: Amino Acids; Animals; Apoptosis; Blotting, Western; Bridged Bicyclo Compounds, Heterocyclic; Excitatory Amino Acid Antagonists; Glutamic Acid; Goldfish; Hypoxia; Hypoxia, Brain; Immunohistochemistry; In Situ Nick-End Labeling; Models, Animal; Receptors, Metabotropic Glutamate; Retina; Retinal Diseases; Telencephalon; Xanthenes

2007
In vivo pharmacological characterization of the structurally novel, potent, selective mGlu2/3 receptor agonist LY404039 in animal models of psychiatric disorders.
    Psychopharmacology, 2007, Volume: 193, Issue:1

    Topics: Amino Acids; Amphetamine; Animals; Behavior, Animal; Bridged Bicyclo Compounds, Heterocyclic; Cyclic S-Oxides; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Male; Mental Disorders; Mice; Molecular Structure; Motor Activity; Phencyclidine; Prefrontal Cortex; Rats; Rats, Inbred F344; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Xanthenes

2007
A novel family of potent negative allosteric modulators of group II metabotropic glutamate receptors.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 322, Issue:1

    Topics: Allosteric Regulation; Amino Acids; Animals; Binding Sites; CHO Cells; Cricetinae; Cricetulus; Humans; Male; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Structure-Activity Relationship; Sulfonamides; Xanthenes

2007
Group II metabotropic glutamate receptors inhibit glutamate release at thalamocortical synapses in the developing somatosensory cortex.
    Neuroscience, 2007, May-25, Volume: 146, Issue:3

    Topics: Amino Acids; Animals; Anticonvulsants; Cerebral Cortex; Cyclopropanes; Electrophysiology; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Glycine; Immunohistochemistry; In Vitro Techniques; Mice; Receptors, Metabotropic Glutamate; Receptors, Presynaptic; Somatosensory Cortex; Synapses; Thalamus; Xanthenes

2007
Dual GABAergic synaptic response of fast excitation and slow inhibition in the medial habenula of rat epithalamus.
    Journal of neurophysiology, 2007, Volume: 98, Issue:3

    Topics: Amino Acids; Animals; Animals, Newborn; Bicuculline; Electric Stimulation; Electrophysiology; Epithalamus; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Habenula; Neurons; Phosphinic Acids; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Synapses; Xanthenes

2007
Group-II metabotropic glutamate receptor ligands as adjunctive drugs in the treatment of depression: a new strategy to shorten the latency of antidepressant medication?
    Molecular psychiatry, 2007, Volume: 12, Issue:8

    Topics: Adjuvants, Pharmaceutic; Amino Acids; Animals; Antidepressive Agents, Tricyclic; Bridged Bicyclo Compounds, Heterocyclic; Depressive Disorder; Disease Models, Animal; Drug Interactions; Drug Therapy, Combination; Excitatory Amino Acid Agents; Hippocampus; Imipramine; In Vitro Techniques; Mice; Neurons; Rats; Rats, Inbred Strains; Receptor Cross-Talk; Receptors, Metabotropic Glutamate; Time Factors; Xanthenes

2007
Contribution of cystine-glutamate antiporters to the psychotomimetic effects of phencyclidine.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2008, Volume: 33, Issue:7

    Topics: Acetylcysteine; Aged; Aged, 80 and over; Amino Acids; Analysis of Variance; Animals; Behavior, Animal; Cell Line, Transformed; Disease Models, Animal; Dose-Response Relationship, Drug; Extracellular Fluid; Female; Free Radical Scavengers; Glutamic Acid; Glycine; Humans; Interpersonal Relations; Male; Maze Learning; Microdialysis; Phencyclidine; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Schizophrenia; Xanthenes

2008
Basal ganglia group II metabotropic glutamate receptors specific binding in non-human primate model of L-Dopa-induced dyskinesias.
    Neuropharmacology, 2008, Volume: 54, Issue:2

    Topics: Amino Acids; Animals; Antiparkinson Agents; Autoradiography; Basal Ganglia; Behavior, Animal; Cabergoline; Caudate Nucleus; Data Interpretation, Statistical; Dyskinesia, Drug-Induced; Ergolines; Excitatory Amino Acid Antagonists; Female; Levodopa; Macaca fascicularis; Ovariectomy; Putamen; Receptors, Metabotropic Glutamate; Xanthenes

2008
A novel assay of Gi/o-linked G protein-coupled receptor coupling to potassium channels provides new insights into the pharmacology of the group III metabotropic glutamate receptors.
    Molecular pharmacology, 2008, Volume: 73, Issue:4

    Topics: Adrenergic Agonists; Allosteric Regulation; Amino Acids; Animals; Biological Assay; Carbachol; Cell Line; Dose-Response Relationship, Drug; G Protein-Coupled Inwardly-Rectifying Potassium Channels; GTP-Binding Protein alpha Subunits, Gi-Go; Humans; Ion Channel Gating; Ligands; Muscarinic Agonists; Pertussis Toxin; Rats; Receptors, Metabotropic Glutamate; Receptors, Muscarinic; Reproducibility of Results; Thallium; Xanthenes

2008
Group III mGluR regulation of synaptic transmission at the SC-CA1 synapse is developmentally regulated.
    Neuropharmacology, 2008, Volume: 54, Issue:5

    Topics: Age Factors; Amino Acids; Aminobutyrates; Animals; Animals, Newborn; Cell Line, Transformed; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Hippocampus; Humans; In Vitro Techniques; Male; Neural Pathways; Neurons; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Synapses; Synaptic Transmission; Transfection; Xanthenes

2008
Distinct neural mechanisms mediate olfactory memory formation at different timescales.
    Learning & memory (Cold Spring Harbor, N.Y.), 2008, Volume: 15, Issue:3

    Topics: Amino Acids; Animals; Brain Mapping; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Habituation, Psychophysiologic; Injections; Male; Memory; Mice; Mice, Inbred Strains; Odorants; Olfactory Bulb; Olfactory Pathways; Smell; Time Factors; Xanthenes

2008
Involvement of group I mGluRs in LTP induced by strong high frequency stimulation in the dentate gyrus in vitro.
    Neuroscience letters, 2008, May-09, Volume: 436, Issue:2

    Topics: Amino Acids; Animals; Dentate Gyrus; Dose-Response Relationship, Radiation; Electric Stimulation; Excitatory Amino Acid Antagonists; In Vitro Techniques; Long-Term Potentiation; Patch-Clamp Techniques; Pyridines; Rats; Receptors, Metabotropic Glutamate; Ryanodine; Xanthenes

2008
Conformational change of the transmembrane helices II and IV of metabotropic glutamate receptor involved in G protein activation.
    Journal of neurochemistry, 2008, Volume: 106, Issue:2

    Topics: Amino Acids; Cell Line, Transformed; Dose-Response Relationship, Drug; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Models, Molecular; Mutagenesis, Site-Directed; Propionates; Protein Binding; Protein Conformation; Protein Structure, Secondary; Receptors, Metabotropic Glutamate; Structure-Activity Relationship; Transfection; Tritium; Xanthenes

2008
Group II metabotropic glutamate receptor activation attenuates peripheral sensitization in inflammatory states.
    Neuroscience, 2008, Jun-23, Volume: 154, Issue:2

    Topics: Amino Acids; Animals; Behavior, Animal; Cyclopentanes; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Hot Temperature; Inflammation; Male; Nerve Fibers; Nociceptors; Pain; Peripheral Nerves; Physical Stimulation; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Skin; Xanthenes

2008
Type-3 metabotropic glutamate receptors negatively modulate bone morphogenetic protein receptor signaling and support the tumourigenic potential of glioma-initiating cells.
    Neuropharmacology, 2008, Volume: 55, Issue:4

    Topics: Amino Acids; Animals; Bone Morphogenetic Protein Receptors; Brain Neoplasms; Bridged Bicyclo Compounds, Heterocyclic; Cell Differentiation; Cell Line, Tumor; Disease Models, Animal; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glioma; Humans; Magnetic Resonance Imaging; Mice; Mitogen-Activated Protein Kinases; Nerve Tissue Proteins; Phosphorylation; Receptors, Metabotropic Glutamate; Signal Transduction; Xanthenes

2008
Allosteric potentiators of metabotropic glutamate receptor subtype 1a differentially modulate independent signaling pathways in baby hamster kidney cells.
    Neuropharmacology, 2008, Volume: 55, Issue:4

    Topics: Allosteric Regulation; Amino Acids; Animals; Binding, Competitive; Calcium; Cell Line, Transformed; Cricetinae; Cyclic AMP; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Mitogen-Activated Protein Kinase 3; Pyrans; Quinolines; Radioligand Assay; Receptors, Metabotropic Glutamate; Signal Transduction; Time Factors; Transfection; Tritium; Xanthenes

2008
Behavioral characterization of the mGlu group II/III receptor antagonist, LY-341495, in animal models of anxiety and depression.
    European journal of pharmacology, 2008, Sep-11, Volume: 592, Issue:1-3

    Topics: Amino Acids; Amphetamine; Animals; Anti-Anxiety Agents; Antidepressive Agents, Second-Generation; Anxiety; Behavior, Animal; Central Nervous System Stimulants; Conditioning, Operant; Darkness; Depression; Diazepam; Fever; Fluoxetine; Light; Male; Mice; Paroxetine; Receptors, Metabotropic Glutamate; Reinforcement Schedule; Stress, Psychological; Xanthenes

2008
Repeated exposure to cocaine alters the modulation of mesocorticolimbic glutamate transmission by medial prefrontal cortex Group II metabotropic glutamate receptors.
    Journal of neurochemistry, 2008, Volume: 107, Issue:1

    Topics: Amino Acids; Animals; Cocaine; Cocaine-Related Disorders; Cystine; Disease Models, Animal; Dopamine Uptake Inhibitors; Drug Administration Schedule; Excitatory Amino Acid Antagonists; Glutamic Acid; Limbic System; Male; Neural Pathways; Prefrontal Cortex; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Synaptic Transmission; Synaptic Vesicles; Ventral Tegmental Area; Xanthenes

2008
Blockade of group II metabotropic glutamate receptors produces hyper-locomotion in cocaine pre-exposed rats by interactions with dopamine receptors.
    Neuropharmacology, 2008, Volume: 55, Issue:4

    Topics: Amino Acids; Animals; Behavior, Animal; Benzazepines; Cocaine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Hyperkinesis; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Metabotropic Glutamate; Salicylamides; Xanthenes

2008
AMPA silencing is a prerequisite for developmental long-term potentiation in the hippocampal CA1 region.
    Journal of neurophysiology, 2008, Volume: 100, Issue:5

    Topics: Aging; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amino Acids; Animals; Animals, Newborn; Colforsin; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Hippocampus; In Vitro Techniques; Long-Term Potentiation; Models, Biological; Rats; Valine; Xanthenes

2008
Individual contribution of metabotropic glutamate receptor (mGlu) 2 and 3 to c-Fos expression pattern evoked by mGlu2/3 antagonism.
    Psychopharmacology, 2008, Volume: 201, Issue:1

    Topics: Amino Acids; Amygdala; Animals; Excitatory Amino Acid Antagonists; Gene Expression; Genes, fos; Hippocampus; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurons; Prefrontal Cortex; Receptors, Metabotropic Glutamate; Septum of Brain; Xanthenes

2008
Dynamic metabotropic control of intrinsic firing in cerebellar unipolar brush cells.
    Journal of neurophysiology, 2008, Volume: 100, Issue:6

    Topics: Action Potentials; Amino Acids; Animals; Barium; Bee Venoms; Calbindin 2; Cerebellum; Cycloleucine; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; In Vitro Techniques; Interneurons; Male; Mice; Neural Inhibition; Potassium Channel Blockers; Receptors, Metabotropic Glutamate; S100 Calcium Binding Protein G; Xanthenes

2008
GABA(B) receptor activation mediates frequency-dependent plasticity of developing GABAergic synapses.
    Nature neuroscience, 2008, Volume: 11, Issue:12

    Topics: Age Factors; Amino Acids; Animals; Animals, Newborn; Bumetanide; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Dose-Response Relationship, Radiation; Electric Stimulation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; GABA Agents; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glycine; Hippocampus; In Vitro Techniques; Neuronal Plasticity; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Sodium Potassium Chloride Symporter Inhibitors; Sodium-Potassium-Chloride Symporters; Synapses; Synaptic Potentials; Xanthenes

2008
Group II metabotropic glutamate receptor activation on peripheral nociceptors modulates TRPV1 function.
    Brain research, 2009, Jan-12, Volume: 1248

    Topics: Amino Acids; Animals; Capsaicin; Colforsin; Electrophysiological Phenomena; Ganglia, Spinal; Hot Temperature; Hyperalgesia; Immunohistochemistry; Male; Nociceptors; Pain; Pain Measurement; Proline; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; TRPV Cation Channels; Xanthenes

2009
The slow Ca2+ -dependent K+ -current facilitates synchronization of hyperexcitable pyramidal neurons.
    Brain research, 2009, Feb-03, Volume: 1252

    Topics: Action Potentials; Amino Acids; Animals; Barium; Calcium; Carbachol; Cesium; Excitatory Amino Acid Antagonists; Hippocampus; In Vitro Techniques; Isoproterenol; Male; Membrane Potentials; Microelectrodes; Patch-Clamp Techniques; Potassium; Pyramidal Cells; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Xanthenes

2009
Epigenetic modulation of mGlu2 receptors by histone deacetylase inhibitors in the treatment of inflammatory pain.
    Molecular pharmacology, 2009, Volume: 75, Issue:5

    Topics: Amino Acids; Animals; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Enzyme Inhibitors; Epigenesis, Genetic; Histone Deacetylase Inhibitors; Hydroxamic Acids; Inflammation; Male; Mice; Pain; Pyridines; Receptors, Metabotropic Glutamate; Vorinostat; Xanthenes

2009
Metabotropic glutamate receptor II in the brains of Parkinsonian patients.
    Journal of neuropathology and experimental neurology, 2009, Volume: 68, Issue:4

    Topics: Aged; Aged, 80 and over; Amino Acids; Antiparkinson Agents; Brain; Cocaine; Dyskinesia, Drug-Induced; Excitatory Amino Acid Antagonists; Female; Humans; Iodine Radioisotopes; Levodopa; Male; Parkinsonian Disorders; Postmortem Changes; Radioligand Assay; Receptors, Metabotropic Glutamate; Tritium; Xanthenes

2009
gamma-Aminobutyric acid-mediated regulation of the activity-dependent olfactory bulb dopaminergic phenotype.
    Journal of neuroscience research, 2009, Aug-01, Volume: 87, Issue:10

    Topics: Agatoxins; Amino Acids; Animals; Animals, Newborn; Bicuculline; Calcium Channel Blockers; Dopamine; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Gene Expression; Green Fluorescent Proteins; Interneurons; Mice; Mice, Transgenic; Olfactory Bulb; Phosphinic Acids; Potassium Chloride; Prosencephalon; Spider Venoms; Tissue Culture Techniques; Tyrosine 3-Monooxygenase; Xanthenes

2009
Antinociceptive synergistic effect of spinal mGluR2/3 antagonist and glial cells inhibitor on peripheral inflammation-induced mechanical hypersensitivity.
    Brain research bulletin, 2009, May-29, Volume: 79, Issue:3-4

    Topics: Amino Acids; Analgesics; Animals; Citrates; Dose-Response Relationship, Drug; Freund's Adjuvant; Hyperesthesia; Inflammation; Male; Neuroglia; Pain; Proline; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Spinal Cord; Xanthenes

2009
Activation of mGlu2/3 metabotropic glutamate receptors negatively regulates the stimulation of inositol phospholipid hydrolysis mediated by 5-hydroxytryptamine2A serotonin receptors in the frontal cortex of living mice.
    Molecular pharmacology, 2009, Volume: 76, Issue:2

    Topics: Amino Acids; Amphetamines; Animals; Bridged Bicyclo Compounds, Heterocyclic; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Frontal Lobe; Hydrolysis; Male; Mice; Mice, Inbred Strains; Mice, Knockout; Phosphatidylinositols; Pyridines; Receptor, Serotonin, 5-HT2A; Receptors, Metabotropic Glutamate; Sulfonamides; Xanthenes

2009
A transient receptor potential-like channel mediates synaptic transmission in rod bipolar cells.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2009, May-13, Volume: 29, Issue:19

    Topics: Amino Acids; Anilides; Animals; Arachidonic Acids; Capsaicin; Cinnamates; Endocannabinoids; Excitatory Amino Acid Antagonists; Glutamic Acid; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Knockout; Polyunsaturated Alkamides; Propionates; Receptors, Metabotropic Glutamate; Retinal Bipolar Cells; Ruthenium Red; Synaptic Transmission; Transient Receptor Potential Channels; TRPM Cation Channels; TRPV Cation Channels; Xanthenes

2009
Use of MGLUR2 and MGLUR3 knockout mice to explore in vivo receptor specificity of the MGLUR2/3 selective antagonist LY341495.
    Neuropharmacology, 2009, Volume: 57, Issue:2

    Topics: Amino Acids; Analysis of Variance; Animals; Brain; Cell Count; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Habituation, Psychophysiologic; Immunohistochemistry; Locomotion; Male; Mice; Mice, Knockout; Photomicrography; Proto-Oncogene Proteins c-fos; Receptors, Metabotropic Glutamate; Xanthenes

2009
Neuroprotective effects of group II metabotropic glutamate receptor agonist DCG-IV on hippocampal neurons in transient forebrain ischemia.
    Neuroscience letters, 2009, Sep-25, Volume: 461, Issue:3

    Topics: Amino Acids; Animals; Carotid Stenosis; Cerebrovascular Circulation; Cyclopropanes; Extracellular Space; Glutamic Acid; Glycine; Hippocampus; Ischemic Attack, Transient; Male; Microdialysis; Neurons; Neuroprotective Agents; Prosencephalon; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Xanthenes

2009
Involvement of Group II mGluRs in mossy fiber LTD.
    Synapse (New York, N.Y.), 2009, Volume: 63, Issue:12

    Topics: Amino Acids; Amino Acids, Dicarboxylic; Animals; Cycloleucine; Cyclopropanes; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glycine; Hippocampus; In Vitro Techniques; Long-Term Synaptic Depression; Mice; Mice, Inbred C57BL; Neural Inhibition; Neurons; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Synaptic Transmission; Xanthenes

2009
Oral administration of the NAALADase inhibitor GPI-5693 attenuates cocaine-induced reinstatement of drug-seeking behavior in rats.
    European journal of pharmacology, 2010, Feb-10, Volume: 627, Issue:1-3

    Topics: Administration, Oral; Amino Acids; Animals; Behavior, Animal; Cocaine; Cocaine-Related Disorders; Dipeptides; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glutamate Carboxypeptidase II; Glutarates; Male; Rats; Receptors, Metabotropic Glutamate; Reward; Self Administration; Stereoisomerism; Sucrose; Sulfhydryl Compounds; Time Factors; Xanthenes

2010
Group II metabotropic glutamate receptor activation by agonist LY379268 treatment increases the expression of brain derived neurotrophic factor in the mouse brain.
    Neuroscience, 2010, Feb-03, Volume: 165, Issue:3

    Topics: Amino Acids; Animals; Brain; Brain-Derived Neurotrophic Factor; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Hippocampus; Male; Mice; Mice, Inbred C57BL; Neurons; Receptors, Metabotropic Glutamate; RNA, Messenger; Time Factors; Up-Regulation; Xanthenes

2010
Excitotoxicity effects of glutamate on human neuroblastoma SH-SY5Y cells via oxidative damage.
    Neuroscience bulletin, 2010, Volume: 26, Issue:1

    Topics: Abietanes; Amino Acids; Antioxidants; Calcium; Cell Line, Tumor; Cell Survival; Cytosol; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Extracellular Space; Glutamic Acid; Glutathione; Humans; Indoles; L-Lactate Dehydrogenase; Malondialdehyde; Oxidative Stress; Phenanthrenes; Superoxide Dismutase; Time Factors; Xanthenes

2010
Extinction of cued fear memory involves a distinct form of depotentiation at cortical input synapses onto the lateral amygdala.
    The European journal of neuroscience, 2009, Dec-03, Volume: 30, Issue:11

    Topics: Acoustic Stimulation; Amino Acids; Amygdala; Animals; Behavior, Animal; Cerebral Cortex; Conditioning, Classical; Cues; Electric Stimulation; Endocytosis; Excitatory Amino Acid Antagonists; Extinction, Psychological; Fear; In Vitro Techniques; Long-Term Synaptic Depression; Male; Memory; Methoxyhydroxyphenylglycol; Patch-Clamp Techniques; Peptides; Rats; Rats, Sprague-Dawley; Statistics, Nonparametric; Xanthenes

2009
Group II metabotropic glutamate receptor stimulation triggers production and release of Alzheimer's amyloid(beta)42 from isolated intact nerve terminals.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Mar-17, Volume: 30, Issue:11

    Topics: Alzheimer Disease; Amino Acids; Amyloid beta-Peptides; Amyloid beta-Protein Precursor; Amyloid Precursor Protein Secretases; Animals; Humans; Methoxyhydroxyphenylglycol; Mice; Mice, Transgenic; Nerve Endings; Peptide Fragments; Receptors, Metabotropic Glutamate; Signal Transduction; Xanthenes

2010
Effects of metabotropic glutamate receptor 2/3 agonism and antagonism on schizophrenia-like cognitive deficits induced by phencyclidine in rats.
    European journal of pharmacology, 2010, Aug-10, Volume: 639, Issue:1-3

    Topics: Amino Acids; Animals; Antipsychotic Agents; Bridged Bicyclo Compounds, Heterocyclic; Cognition; Excitatory Amino Acid Agents; Male; Phencyclidine; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Schizophrenia; Time Factors; Xanthenes

2010
AMPA receptor mediates mGlu 2/3 receptor antagonist-induced dopamine release in the rat nucleus accumbens shell.
    Neurochemistry international, 2010, Volume: 57, Issue:5

    Topics: Amino Acids; Animals; Dioxoles; Dopamine; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Male; Microdialysis; Nucleus Accumbens; Piperidines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Metabotropic Glutamate; Xanthenes

2010
Orally active glutamate carboxypeptidase II inhibitor 2-MPPA attenuates dizocilpine-induced prepulse inhibition deficits in mice.
    Brain research, 2011, Jan-31, Volume: 1371

    Topics: Administration, Oral; Amino Acids; Animals; Antipsychotic Agents; Bridged Bicyclo Compounds; Dipeptides; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Glutamate Carboxypeptidase II; Glutarates; Male; Mice; Neural Inhibition; Schizophrenia; Sensory Gating; Sulfhydryl Compounds; Xanthenes

2011
Targeting group II metabotropic glutamate (mGlu) receptors for the treatment of psychosis associated with Alzheimer's disease: selective activation of mGlu2 receptors amplifies beta-amyloid toxicity in cultured neurons, whereas dual activation of mGlu2 an
    Molecular pharmacology, 2011, Volume: 79, Issue:3

    Topics: Alzheimer Disease; Amino Acids; Amyloid beta-Peptides; Animals; Antipsychotic Agents; Astrocytes; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Mice; Mice, Knockout; Neurons; Neuroprotective Agents; Psychotic Disorders; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Reverse Transcriptase Polymerase Chain Reaction; Sulfonamides; Transforming Growth Factor beta1; Xanthenes

2011
Metabotropic glutamate receptor blockade in nucleus accumbens shell shifts affective valence towards fear and disgust.
    The European journal of neuroscience, 2011, Volume: 33, Issue:4

    Topics: Affect; Amino Acids; Analgesics, Non-Narcotic; Animals; Appetitive Behavior; Excitatory Amino Acid Antagonists; Fear; Male; Motivation; Nucleus Accumbens; Pleasure; Proto-Oncogene Proteins c-fos; Quinine; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Schizophrenia; Xanthenes

2011
Baclofen and adenosine inhibition of synaptic transmission at CA3-CA1 synapses display differential sensitivity to K+ channel blockade.
    Cellular and molecular neurobiology, 2011, Volume: 31, Issue:4

    Topics: 4-Aminopyridine; Adenosine; Adenosine A1 Receptor Antagonists; Amino Acids; Animals; Baclofen; Barium; Bee Venoms; CA1 Region, Hippocampal; CA3 Region, Hippocampal; Cesium; Excitatory Postsynaptic Potentials; In Vitro Techniques; Male; Potassium Channel Blockers; Rats; Rats, Wistar; Receptor, Adenosine A1; Receptors, Metabotropic Glutamate; Synapses; Synaptic Transmission; Theophylline; Xanthenes

2011
Group II metabotropic glutamate receptors in the striatum of non-human primates: dysregulation following chronic cocaine self-administration.
    Neuroscience letters, 2011, May-27, Volume: 496, Issue:1

    Topics: Amino Acids; Animals; Antimetabolites; Autoradiography; Carbon Isotopes; Cocaine; Conditioning, Operant; Corpus Striatum; Deoxyglucose; Dopamine Uptake Inhibitors; Excitatory Amino Acid Antagonists; Macaca mulatta; Male; Protein Binding; Receptors, AMPA; Receptors, Metabotropic Glutamate; Reinforcement Schedule; Self Administration; Tritium; Xanthenes

2011
Regulation of Akt and Wnt signaling by the group II metabotropic glutamate receptor antagonist LY341495 and agonist LY379268.
    Journal of neurochemistry, 2011, Volume: 117, Issue:6

    Topics: Amino Acids; Animals; Bridged Bicyclo Compounds, Heterocyclic; Corpus Striatum; Glycogen Synthase Kinase 3; Male; Motor Activity; Prefrontal Cortex; Proto-Oncogene Proteins c-akt; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Signal Transduction; Wnt Proteins; Xanthenes

2011
Enhancement of CA3 hippocampal network activity by activation of group II metabotropic glutamate receptors.
    Proceedings of the National Academy of Sciences of the United States of America, 2011, Jun-14, Volume: 108, Issue:24

    Topics: Action Potentials; Amino Acids; Animals; CA3 Region, Hippocampal; Cyclopropanes; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glycine; Interneurons; Mice; Mice, Knockout; Microscopy, Electron; Nerve Net; Patch-Clamp Techniques; Pyramidal Cells; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Theta Rhythm; Xanthenes

2011
A role for nyctalopin, a small leucine-rich repeat protein, in localizing the TRP melastatin 1 channel to retinal depolarizing bipolar cell dendrites.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Jul-06, Volume: 31, Issue:27

    Topics: Amino Acids; Animals; Bacterial Proteins; Biophysics; Cell Line, Transformed; Dendrites; Electric Stimulation; Excitatory Amino Acid Antagonists; Gene Expression Regulation, Developmental; Humans; In Vitro Techniques; Leucine-Rich Repeat Proteins; Luminescent Proteins; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Transgenic; Models, Biological; Patch-Clamp Techniques; Proteins; Proteoglycans; Retina; Retinal Bipolar Cells; Transfection; TRPM Cation Channels; Xanthenes

2011
Estradiol attenuates the adenosine triphosphate-induced increase of intracellular calcium through group II metabotropic glutamate receptors in rat dorsal root ganglion neurons.
    Journal of neuroscience research, 2011, Volume: 89, Issue:11

    Topics: Adenosine Triphosphate; Amino Acids; Animals; Calcium; Cells, Cultured; Estradiol; Estrogens; Female; Ganglia, Spinal; Neurons; Rats; Rats, Long-Evans; Receptors, Estrogen; Receptors, Metabotropic Glutamate; Xanthenes

2011
Blockade of GABA(B) receptors facilitates evoked neurotransmitter release at spinal dorsal horn synapse.
    Neuroscience, 2011, Oct-13, Volume: 193

    Topics: Amino Acids; Animals; Baclofen; Benzylamines; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Agonists; GABA-A Receptor Antagonists; In Vitro Techniques; Male; Neurotransmitter Agents; Nipecotic Acids; Patch-Clamp Techniques; Phosphinic Acids; Posterior Horn Cells; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Spinal Cord; Synapses; Synaptic Potentials; Tiagabine; Xanthenes

2011
Group II/III metabotropic glutamate receptors exert endogenous activity-dependent modulation of TRPV1 receptors on peripheral nociceptors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Sep-07, Volume: 31, Issue:36

    Topics: Amino Acids; Animals; Calcium; Capsaicin; Cells, Cultured; Cytosol; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Formaldehyde; Glutamic Acid; Hot Temperature; Male; Nociceptors; Pain; Pain Measurement; Peripheral Nervous System; Proline; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Skin; TRPV Cation Channels; Xanthenes

2011
Involvement of the mammalian target of rapamycin signaling in the antidepressant-like effect of group II metabotropic glutamate receptor antagonists.
    Neuropharmacology, 2011, Volume: 61, Issue:8

    Topics: Amino Acids; Analysis of Variance; Animals; Bridged Bicyclo Compounds; Depression; Dicarboxylic Acids; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Hindlimb Suspension; Ketamine; Male; Mice; Mice, Inbred ICR; Receptors, Metabotropic Glutamate; Sirolimus; Time Factors; TOR Serine-Threonine Kinases; Xanthenes

2011
Activation of group II metabotropic glutamate receptors induces long-term depression of excitatory synaptic transmission in the substantia nigra pars reticulata.
    Neuroscience letters, 2011, Oct-24, Volume: 504, Issue:2

    Topics: Amino Acids; Animals; Basal Ganglia; Bridged Bicyclo Compounds, Heterocyclic; Data Interpretation, Statistical; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; Mice; Mice, Knockout; Neuronal Plasticity; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Substantia Nigra; Synaptic Transmission; Xanthenes

2011
Excitatory amino acid transporter 2 and excitatory amino acid transporter 1 negatively regulate calcium-dependent proliferation of hippocampal neural progenitor cells and are persistently upregulated after injury.
    The European journal of neuroscience, 2011, Volume: 34, Issue:11

    Topics: Amino Acids; Animals; Calcium; Cell Proliferation; Cells, Cultured; Dentate Gyrus; Excitatory Amino Acid Antagonists; Excitatory Amino Acid Transporter 1; Excitatory Amino Acid Transporter 2; Mice; Mice, Transgenic; Neural Stem Cells; RNA, Small Interfering; Xanthenes

2011
mTOR activation is required for the antidepressant effects of mGluR₂/₃ blockade.
    The international journal of neuropsychopharmacology, 2012, Volume: 15, Issue:4

    Topics: Amino Acids; Animals; Disks Large Homolog 4 Protein; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Gene Expression Regulation; Intracellular Signaling Peptides and Proteins; Ketamine; Male; Membrane Proteins; Prefrontal Cortex; Rats; Receptors, Metabotropic Glutamate; Signal Transduction; Swimming; Synapsins; Synaptosomes; TOR Serine-Threonine Kinases; Xanthenes

2012
Radiosynthesis of PET radiotracer as a prodrug for imaging group II metabotropic glutamate receptors in vivo.
    Bioorganic & medicinal chemistry letters, 2012, Mar-01, Volume: 22, Issue:5

    Topics: Amino Acids; Animals; Brain; Corpus Striatum; Hippocampus; Male; Positron-Emission Tomography; Prodrugs; Protein Binding; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Xanthenes

2012
Effects of microinjections of Group II metabotropic glutamate agents into the amygdala on sleep.
    Brain research, 2012, May-03, Volume: 1452

    Topics: Amino Acids; Amygdala; Animals; Arousal; Bridged Bicyclo Compounds, Heterocyclic; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Male; Microinjections; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Sleep; Sleep, REM; Wakefulness; Xanthenes

2012
Actions of Xanthurenic acid, a putative endogenous Group II metabotropic glutamate receptor agonist, on sensory transmission in the thalamus.
    Neuropharmacology, 2013, Volume: 66

    Topics: Action Potentials; Administration, Intravenous; Afferent Pathways; Allosteric Regulation; Amino Acids; Animals; Bridged Bicyclo Compounds; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Iontophoresis; Male; Neural Inhibition; Neurons; Rats; Rats, Wistar; Ventral Thalamic Nuclei; Vibrissae; Xanthenes; Xanthurenates

2013
Selective activation of either mGlu2 or mGlu3 receptors can induce LTD in the amygdala.
    Neuropharmacology, 2013, Volume: 66

    Topics: Amino Acids; Amino Acids, Dicarboxylic; Amygdala; Animals; Bridged Bicyclo Compounds; Cyclopropanes; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Long-Term Synaptic Depression; Mice; Mice, Knockout; Rats; Rats, Mutant Strains; Rats, Wistar; Receptors, Metabotropic Glutamate; Xanthenes

2013
G-protein-mediated inhibition of the Trp channel TRPM1 requires the Gβγ dimer.
    Proceedings of the National Academy of Sciences of the United States of America, 2012, May-29, Volume: 109, Issue:22

    Topics: Amino Acids; Animals; Capsaicin; Cells, Cultured; Excitatory Amino Acid Antagonists; Glutamic Acid; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein beta Subunits; GTP-Binding Protein gamma Subunits; HEK293 Cells; Humans; Light; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Knockout; Protein Binding; Protein Multimerization; Receptors, Metabotropic Glutamate; Retinal Bipolar Cells; TRPM Cation Channels; Xanthenes

2012
The metabotropic glutamate 2/3 receptor antagonist LY341495 differentially affects recognition memory in rats.
    Behavioural brain research, 2012, May-01, Volume: 230, Issue:2

    Topics: Amino Acids; Animals; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Extinction, Psychological; Male; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Recognition, Psychology; Xanthenes

2012
Glycine release is regulated by metabotropic glutamate receptors sensitive to mGluR2/3 ligands and activated by N-acetylaspartylglutamate (NAAG).
    Neuropharmacology, 2013, Volume: 66

    Topics: Amino Acids; Animals; Bridged Bicyclo Compounds, Heterocyclic; Dipeptides; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Exocytosis; Glutamic Acid; Glycine; Male; Mice; Potassium Chloride; Receptors, Metabotropic Glutamate; Spinal Cord; Synaptosomes; Xanthenes

2013
Depolarizing bipolar cell dysfunction due to a Trpm1 point mutation.
    Journal of neurophysiology, 2012, Volume: 108, Issue:9

    Topics: Action Potentials; Amino Acid Sequence; Amino Acids; Animals; Capsaicin; Chromosome Mapping; Chromosomes, Mammalian; Dendrites; Disease Models, Animal; Exons; Eye Diseases, Hereditary; Genetic Diseases, X-Linked; Heterozygote; Mice; Mice, Transgenic; Molecular Sequence Data; Mutation, Missense; Myopia; Night Blindness; Point Mutation; Retina; Retinal Bipolar Cells; Sequence Analysis, DNA; Threonine; TRPM Cation Channels; Xanthenes

2012
Synthesis and characterization of two PET radioligands for the metabotropic glutamate 1 (mGlu1) receptor.
    Synapse (New York, N.Y.), 2012, Volume: 66, Issue:12

    Topics: Amino Acids; Animals; Brain; Carbon Radioisotopes; CHO Cells; Cricetinae; Cricetulus; Excitatory Amino Acid Antagonists; Fluorine Radioisotopes; Ligands; Male; Papio; Positron-Emission Tomography; Pyridines; Quinolines; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Metabotropic Glutamate; Tissue Distribution; Xanthenes

2012
Group II metabotropic glutamate receptors depress synaptic transmission onto subicular burst firing neurons.
    PloS one, 2012, Volume: 7, Issue:9

    Topics: Amino Acids; Amino Acids, Dicarboxylic; Animals; CA1 Region, Hippocampal; CA3 Region, Hippocampal; Cyclopropanes; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Female; Glutamic Acid; Glycine; Hippocampus; Male; Neurons; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Synaptic Transmission; Xanthenes

2012
Modafinil attenuates reinstatement of cocaine seeking: role for cystine-glutamate exchange and metabotropic glutamate receptors.
    Addiction biology, 2014, Volume: 19, Issue:1

    Topics: Amino Acid Transport System y+; Amino Acids; Analysis of Variance; Animals; Benzhydryl Compounds; Cocaine; Cocaine-Related Disorders; Disease Models, Animal; Dopamine Uptake Inhibitors; Drug-Seeking Behavior; Excitatory Amino Acid Antagonists; Extinction, Psychological; Glutamates; Male; Microdialysis; Microinjections; Modafinil; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Secondary Prevention; Self Administration; Wakefulness-Promoting Agents; Xanthenes

2014
Role of BDNF/TrkB signaling in antidepressant-like effects of a group II metabotropic glutamate receptor antagonist in animal models of depression.
    Behavioural brain research, 2013, Feb-01, Volume: 238

    Topics: Amino Acids; Animals; Antidepressive Agents; Behavior, Animal; Brain-Derived Neurotrophic Factor; Depressive Disorder; Disease Models, Animal; Excitatory Amino Acid Antagonists; Exploratory Behavior; Hindlimb Suspension; Male; Mice; Mice, Inbred C57BL; Mice, Inbred ICR; Receptor, trkB; Receptors, Metabotropic Glutamate; Signal Transduction; Xanthenes

2013
Regulation of synaptic currents by mGluR2 at reciprocal synapses in the mouse accessory olfactory bulb.
    The European journal of neuroscience, 2013, Volume: 37, Issue:3

    Topics: Action Potentials; Amino Acids; Animals; Anticonvulsants; Calcium Channels; Cyclopropanes; Dendrites; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glycine; Mice; Mice, Inbred BALB C; Mutation; Olfactory Bulb; Receptors, Metabotropic Glutamate; Synapses; Xanthenes

2013
Type-3 metabotropic glutamate receptors regulate chemoresistance in glioma stem cells, and their levels are inversely related to survival in patients with malignant gliomas.
    Cell death and differentiation, 2013, Volume: 20, Issue:3

    Topics: Amino Acids; Animals; Antineoplastic Agents, Alkylating; Chemotherapy, Adjuvant; Combined Modality Therapy; Dacarbazine; DNA Methylation; Drug Resistance, Neoplasm; Glioblastoma; Humans; Mice; Neoplastic Stem Cells; NF-kappa B; O(6)-Methylguanine-DNA Methyltransferase; Phosphatidylinositol 3-Kinases; Promoter Regions, Genetic; Receptors, Metabotropic Glutamate; RNA, Messenger; Signal Transduction; Survival Rate; Temozolomide; Transplantation, Heterologous; Tumor Cells, Cultured; Xanthenes

2013
Anxiety-like behavior of prenatally stressed rats is associated with a selective reduction of glutamate release in the ventral hippocampus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2012, Nov-28, Volume: 32, Issue:48

    Topics: Amino Acids; Animals; Anxiety; Behavior, Animal; Benzylamines; Excitatory Amino Acid Antagonists; Female; GABA-A Receptor Antagonists; Glutamic Acid; Hippocampus; Kainic Acid; Male; Munc18 Proteins; Phosphinic Acids; Pregnancy; Prenatal Exposure Delayed Effects; R-SNARE Proteins; rab3A GTP-Binding Protein; Rats; Rats, Sprague-Dawley; Seizures; Stress, Psychological; Synapsins; Synaptic Transmission; Synaptophysin; Syntaxin 1; Xanthenes

2012
Characterisation of an mGlu8 receptor-selective agonist and antagonist in the lateral and medial perforant path inputs to the dentate gyrus.
    Neuropharmacology, 2013, Volume: 67

    Topics: Amino Acids; Amino Acids, Dicarboxylic; Animals; Bridged Bicyclo Compounds; Dentate Gyrus; Female; Male; Mice; Mice, 129 Strain; Mice, Inbred C57BL; Mice, Knockout; Neural Pathways; Perforant Pathway; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Xanthenes

2013
Chronic treatment with LY341495 decreases 5-HT(2A) receptor binding and hallucinogenic effects of LSD in mice.
    Neuroscience letters, 2013, Mar-01, Volume: 536

    Topics: Amino Acids; Animals; Drug Antagonism; Early Growth Response Protein 1; Early Growth Response Protein 2; Hallucinogens; Lysergic Acid Diethylamide; Male; Mice; Mice, Knockout; Proto-Oncogene Proteins c-fos; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptors, Metabotropic Glutamate; Somatosensory Cortex; Stereotyped Behavior; Xanthenes

2013
L-acetylcarnitine causes rapid antidepressant effects through the epigenetic induction of mGlu2 receptors.
    Proceedings of the National Academy of Sciences of the United States of America, 2013, Mar-19, Volume: 110, Issue:12

    Topics: Acetylation; Acetylcarnitine; Amino Acids; Animals; Antidepressive Agents; Clomipramine; Epigenesis, Genetic; Excitatory Amino Acid Antagonists; Hippocampus; Histone Deacetylases; Histones; Humans; Male; Mice; Mice, Knockout; Nerve Tissue Proteins; NF-kappa B; Nootropic Agents; Prefrontal Cortex; Rats; Receptors, Metabotropic Glutamate; Selective Serotonin Reuptake Inhibitors; Stress, Psychological; Time Factors; Xanthenes

2013
Effect of an mGlu2/3 receptor antagonist on depressive behavior induced by withdrawal from chronic treatment with methamphetamine.
    Behavioural brain research, 2013, Jun-01, Volume: 246

    Topics: Amino Acids; Analysis of Variance; Animals; Central Nervous System Stimulants; Depression; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Delivery Systems; Drug Interactions; Excitatory Amino Acid Antagonists; Immobility Response, Tonic; Male; Methamphetamine; Motor Activity; Rats; Rats, Sprague-Dawley; Substance Withdrawal Syndrome; Swimming; Xanthenes

2013
Antagonists reversibly reverse chemical LTD induced by group I, group II and group III metabotropic glutamate receptors.
    Neuropharmacology, 2013, Volume: 74

    Topics: Amino Acids; Animals; Brain; Excitatory Amino Acid Antagonists; Glycine; Long-Term Synaptic Depression; Mice; Neural Pathways; Rats; Receptors, Metabotropic Glutamate; Xanthenes

2013
Contribution of opioid and metabotropic glutamate receptor mechanisms to inhibition of bladder overactivity by tibial nerve stimulation.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2013, Jul-15, Volume: 305, Issue:2

    Topics: Amino Acids; Animals; Cats; Electric Stimulation Therapy; Excitatory Amino Acid Antagonists; Female; Male; Naloxone; Narcotic Antagonists; Receptors, Metabotropic Glutamate; Receptors, Opioid; Tibial Nerve; Urinary Bladder; Urinary Bladder, Overactive; Xanthenes

2013
Effects of ketamine and LY341495 on the depressive-like behavior of repeated corticosterone-injected rats.
    Pharmacology, biochemistry, and behavior, 2013, Volume: 107

    Topics: Amino Acids; Animals; Corticosterone; Depressive Disorder, Treatment-Resistant; Disease Models, Animal; Drug Administration Schedule; Immobility Response, Tonic; Injections, Subcutaneous; Ketamine; Male; Rats; Receptors, Metabotropic Glutamate; Xanthenes

2013
Group II metabotropic glutamate receptor agonist LY379268 regulates AMPA receptor trafficking in prefrontal cortical neurons.
    PloS one, 2013, Volume: 8, Issue:4

    Topics: Amino Acids; Animals; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Cells, Cultured; Dactinomycin; Disks Large Homolog 4 Protein; Enzyme Activation; Extracellular Signal-Regulated MAP Kinases; Flavonoids; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Intracellular Signaling Peptides and Proteins; Intracellular Space; Membrane Proteins; Neurons; Prefrontal Cortex; Protein Kinase Inhibitors; Protein Subunits; Protein Transport; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Metabotropic Glutamate; Synapsins; Transcription, Genetic; Xanthenes

2013
Stimulation of metabotropic glutamate (mGlu) 2 receptor and blockade of mGlu1 receptor improve social memory impairment elicited by MK-801 in rats.
    Journal of pharmacological sciences, 2013, Volume: 122, Issue:1

    Topics: Amino Acids; Animals; Bridged Bicyclo Compounds, Heterocyclic; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Male; Memory Disorders; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Recognition, Psychology; Xanthenes

2013
Synergistic inhibition of survival, proliferation, and migration of U87 cells with a combination of LY341495 and Iressa.
    PloS one, 2013, Volume: 8, Issue:5

    Topics: Amino Acids; Antineoplastic Agents; Apoptosis; Cell Line, Tumor; Cell Movement; Cell Proliferation; Cell Survival; Dose-Response Relationship, Drug; Drug Synergism; Gefitinib; Glioblastoma; Glutamic Acid; Humans; Quinazolines; Riluzole; Xanthenes

2013
Chronic treatment with MPEP, an mGlu5 receptor antagonist, normalizes basal ganglia glutamate neurotransmission in L-DOPA-treated parkinsonian monkeys.
    Neuropharmacology, 2013, Volume: 73

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Basal Ganglia; Corpus Striatum; Dyskinesia, Drug-Induced; Female; Imidazoles; Levodopa; Macaca fascicularis; Oximes; Parkinsonian Disorders; Phenols; Piperidines; Pyridines; Quinazolines; Radioligand Assay; Receptor, Metabotropic Glutamate 5; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Tritium; Xanthenes

2013
Pharmacological characterization of JNJ-40068782, a new potent, selective, and systemically active positive allosteric modulator of the mGlu2 receptor and its radioligand [3H]JNJ-40068782.
    The Journal of pharmacology and experimental therapeutics, 2013, Volume: 346, Issue:3

    Topics: Amino Acids; Animals; Autoradiography; Binding, Competitive; Brain Chemistry; Calcium; Cell Membrane; Cerebral Cortex; CHO Cells; Cricetinae; Cricetulus; Cyclopropanes; Excitatory Amino Acid Agents; Excitatory Amino Acid Agonists; Glycine; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Isotope Labeling; Ligands; Male; Mice; Motor Activity; Piperidines; Pyridones; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Sleep; Tritium; Xanthenes

2013
Enhancement of long-term depression by soluble amyloid β protein in rat hippocampus is mediated by metabotropic glutamate receptor and involves activation of p38MAPK, STEP and caspase-3.
    Neuroscience, 2013, Dec-03, Volume: 253

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Amyloid beta-Peptides; Animals; Caspase 3; Electric Stimulation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Hippocampus; Immunosuppressive Agents; In Vitro Techniques; Long-Term Synaptic Depression; Male; Methoxyhydroxyphenylglycol; p38 Mitogen-Activated Protein Kinases; Patch-Clamp Techniques; Peptide Fragments; Protein Tyrosine Phosphatases, Non-Receptor; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Sirolimus; Xanthenes

2013
Cerebral 5-HT2A receptor binding, but not mGluR2, is increased in tryptophan hydroxylase 2 decrease-of-function mice.
    Neuroscience letters, 2013, Oct-25, Volume: 555

    Topics: Amino Acids; Animals; Brain; Gene Knock-In Techniques; Mice; Mice, Transgenic; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptors, Metabotropic Glutamate; Tryptophan Hydroxylase; Up-Regulation; Xanthenes

2013
Activation of synaptic group II metabotropic glutamate receptors induces long-term depression at GABAergic synapses in CNS neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2013, Oct-02, Volume: 33, Issue:40

    Topics: Amino Acids; Animals; Chick Embryo; Cochlear Nucleus; Cyclopropanes; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABAergic Neurons; Glycine; Inhibitory Postsynaptic Potentials; Long-Term Synaptic Depression; Neural Inhibition; Receptors, Metabotropic Glutamate; Synapses; Synaptic Transmission; Xanthenes

2013
Serotonin-1A receptor stimulation mediates effects of a metabotropic glutamate 2/3 receptor antagonist, 2S-2-amino-2-(1S,2S-2-carboxycycloprop-1-yl)-3-(xanth-9-yl)propanoic acid (LY341495), and an N-methyl-D-aspartate receptor antagonist, ketamine, in the
    Psychopharmacology, 2014, Volume: 231, Issue:11

    Topics: Amino Acids; Animals; Antidepressive Agents; Dioxoles; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Feeding Behavior; Fenclonine; Ketamine; Male; Mice, Inbred C57BL; Neuropsychological Tests; Piperazines; Piperidines; Pyridines; Quinoxalines; Receptors, AMPA; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Ritanserin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Tryptophan Hydroxylase; Xanthenes

2014
mGlu3 receptor blockade inhibits proliferation and promotes astrocytic phenotype in glioma stem cells.
    Cell biology international, 2014, Volume: 38, Issue:4

    Topics: AC133 Antigen; Amino Acids; Animals; Antigens, CD; Astrocytes; Bridged Bicyclo Compounds, Heterocyclic; Cell Differentiation; Cell Proliferation; Epidermal Growth Factor; Fibroblast Growth Factor 2; Glioma; Glycoproteins; Humans; Male; Mice; Mice, Inbred BALB C; Mice, Nude; Neoplastic Stem Cells; Peptides; Phenotype; Receptors, Metabotropic Glutamate; Recombinant Proteins; Transplantation, Heterologous; Xanthenes

2014
N-acetylcysteine modulates hallucinogenic 5-HT(2A) receptor agonist-mediated responses: behavioral, molecular, and electrophysiological studies.
    Neuropharmacology, 2014, Volume: 81

    Topics: Acetylcysteine; Action Potentials; Amino Acids; Amphetamines; Animals; Benzoates; Bicuculline; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Early Growth Response Protein 2; Excitatory Amino Acid Antagonists; Free Radical Scavengers; GABA-A Receptor Antagonists; Glycine; Hallucinations; Hallucinogens; Male; Mice; Proto-Oncogene Proteins c-fos; Receptors, Metabotropic Glutamate; Xanthenes

2014
Overexpression of Shati/Nat8l, an N-acetyltransferase, in the nucleus accumbens attenuates the response to methamphetamine via activation of group II mGluRs in mice.
    The international journal of neuropsychopharmacology, 2014, Volume: 17, Issue:8

    Topics: Acetyltransferases; Amino Acids; Animals; Aspartic Acid; Conditioning, Psychological; Corpus Striatum; Dipeptides; Dopamine; Male; Methamphetamine; Mice; Mice, Transgenic; Motor Activity; Nucleus Accumbens; Receptors, Metabotropic Glutamate; Xanthenes

2014
A real-time method for measuring cAMP production modulated by Gαi/o-coupled metabotropic glutamate receptors.
    The Journal of pharmacology and experimental therapeutics, 2014, Volume: 349, Issue:3

    Topics: Amino Acids; Animals; Biosensing Techniques; Buffers; Cell Culture Techniques; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Glutamic Acid; GTP-Binding Protein alpha Subunits, Gi-Go; Luciferases, Firefly; Radioligand Assay; Receptors, Metabotropic Glutamate; Reproducibility of Results; Sensitivity and Specificity; Transfection; Xanthenes

2014
Blockade of the metabotropic glutamate (mGluR2) modulates arousal through vigilance states transitions: evidence from sleep-wake EEG in rodents.
    Behavioural brain research, 2014, Aug-15, Volume: 270

    Topics: Amino Acids; Animals; Arousal; Body Temperature; Cerebral Cortex; Electroencephalography; Excitatory Amino Acid Antagonists; Locomotion; Male; Mice; Mice, Knockout; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Sleep; Wakefulness; Xanthenes

2014
Requirement of AMPA receptor stimulation for the sustained antidepressant activity of ketamine and LY341495 during the forced swim test in rats.
    Behavioural brain research, 2014, Sep-01, Volume: 271

    Topics: Adaptation, Psychological; Amino Acids; Animals; Antidepressive Agents; Depression; Disease Models, Animal; Excitatory Amino Acid Antagonists; Ketamine; Male; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Stress, Psychological; Swimming; Time Factors; Xanthenes

2014
Evaluation of 5-HT2A and mGlu2/3 receptors in postmortem prefrontal cortex of subjects with major depressive disorder: effect of antidepressant treatment.
    Neuropharmacology, 2014, Volume: 86

    Topics: Amino Acids; Animals; Antidepressive Agents; Citalopram; Depressive Disorder, Major; Down-Regulation; Female; Humans; Ketanserin; Male; Mianserin; Middle Aged; Mirtazapine; Morpholines; Prefrontal Cortex; Radioligand Assay; Rats, Sprague-Dawley; Reboxetine; Receptor, Serotonin, 5-HT2A; Receptors, Metabotropic Glutamate; RNA, Messenger; Tritium; Xanthenes

2014
The peptidic antidepressant spadin interacts with prefrontal 5-HT(4) and mGluR(2) receptors in the control of serotonergic function.
    Brain structure & function, 2016, Volume: 221, Issue:1

    Topics: Amino Acids; Aniline Compounds; Animals; Antidepressive Agents; Calcium; Dorsal Raphe Nucleus; Early Growth Response Protein 1; Excitatory Amino Acid Antagonists; Indoles; Male; Mice, Inbred C57BL; Mice, Knockout; Peptides; Piperazines; Piperidines; Potassium Channels, Tandem Pore Domain; Prefrontal Cortex; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Receptors, Serotonin, 5-HT4; Serotonergic Neurons; Serotonin 5-HT4 Receptor Agonists; Serotonin Receptor Agonists; Sulfonamides; Xanthenes

2016
Epigenetic upregulation of metabotropic glutamate receptor 2 in the spinal cord attenuates oestrogen-induced visceral hypersensitivity.
    Gut, 2015, Volume: 64, Issue:12

    Topics: Acetylation; Amino Acids; Animals; Disease Models, Animal; Epigenesis, Genetic; Estradiol; Estrogens; Female; Histone Deacetylase Inhibitors; Histones; Hydroxamic Acids; Nociception; Ovariectomy; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; RNA, Messenger; Spinal Cord; Up-Regulation; Viscera; Visceral Pain; Vorinostat; Xanthenes

2015
Increased metabotropic glutamate 2/3 receptor binding in the perigenual anterior cingulate cortex of Cloninger type 2 alcoholics: a whole-hemisphere autoradiography study.
    Alcohol and alcoholism (Oxford, Oxfordshire), 2015, Volume: 50, Issue:1

    Topics: Adolescent; Adult; Aged; Alcoholism; Amino Acids; Autoradiography; Brain; Case-Control Studies; Female; Gyrus Cinguli; Humans; Male; Middle Aged; Receptors, Metabotropic Glutamate; Xanthenes; Young Adult

2015
Investigating glutamatergic mechanism in attention and impulse control using rats in a modified 5-choice serial reaction time task.
    PloS one, 2014, Volume: 9, Issue:12

    Topics: Amino Acids; Animals; Attention; Disease Models, Animal; Dizocilpine Maleate; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Impulsive Behavior; Male; N-Methylaspartate; Prefrontal Cortex; Rats; Reaction Time; Xanthenes

2014
Role of group II metabotropic glutamate receptors (mGluR2/3) blockade on long-term potentiation in the dentate gyrus region of hippocampus in rats fed with high-fat diet.
    Neurochemical research, 2015, Volume: 40, Issue:4

    Topics: Amino Acids; Animals; Dentate Gyrus; Diet, High-Fat; Excitatory Amino Acid Antagonists; Long-Term Potentiation; Male; Microinjections; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Xanthenes

2015
Group II metabotropic glutamate receptor antagonism prevents the antiallodynic effects of R-isovaline.
    Neuroscience, 2015, May-07, Volume: 293

    Topics: Amino Acids; Analgesics; Animals; Dinoprostone; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Female; GABA-B Receptor Antagonists; Hyperalgesia; Mice; Pain Threshold; Receptors, GABA-B; Receptors, Metabotropic Glutamate; Valine; Xanthenes

2015
N-acetyl-cysteine, a drug that enhances the endogenous activation of group-II metabotropic glutamate receptors, inhibits nociceptive transmission in humans.
    Molecular pain, 2015, Mar-20, Volume: 11

    Topics: Acetylcysteine; Adult; Amino Acids; Analgesics; Dose-Response Relationship, Drug; Double-Blind Method; Female; Humans; Male; Middle Aged; Pain; Receptors, Metabotropic Glutamate; Treatment Outcome; Xanthenes; Young Adult

2015
Group II mGluRs modulate baseline and arthritis pain-related synaptic transmission in the rat medial prefrontal cortex.
    Neuropharmacology, 2015, Volume: 95

    Topics: Amino Acids; Animals; Arthritis, Experimental; Bridged Bicyclo Compounds, Heterocyclic; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Inhibitory Postsynaptic Potentials; Kaolin; Miniature Postsynaptic Potentials; Pain; Patch-Clamp Techniques; Prefrontal Cortex; Pyramidal Cells; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Synaptic Transmission; Tissue Culture Techniques; Xanthenes

2015
The Female Encounter Test: A Novel Method for Evaluating Reward-Seeking Behavior or Motivation in Mice.
    The international journal of neuropsychopharmacology, 2015, May-29, Volume: 18, Issue:11

    Topics: Amino Acids; Animals; Antidepressive Agents, Second-Generation; Castration; Choice Behavior; Corticosterone; Depressive Disorder; Disease Models, Animal; Equipment Design; Estrous Cycle; Excitatory Amino Acid Antagonists; Female; Fluvoxamine; Lipopolysaccharides; Male; Mice; Motivation; Nucleus Accumbens; Psychological Tests; Reward; Social Behavior; Social Isolation; Xanthenes

2015
mGluR2/3 in the Lateral Amygdala is Required for Fear Extinction: Cortical Input Synapses onto the Lateral Amygdala as a Target Site of the mGluR2/3 Action.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2015, Volume: 40, Issue:13

    Topics: Amino Acids; Amygdala; Animals; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Extinction, Psychological; Fear; Freezing Reaction, Cataleptic; Male; Patch-Clamp Techniques; Presynaptic Terminals; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Tissue Culture Techniques; Xanthenes

2015
Activation of mGluR2/3 following stress hormone exposure restores sensitivity to alcohol in rats.
    Alcohol (Fayetteville, N.Y.), 2015, Volume: 49, Issue:6

    Topics: Alcohol Drinking; Amino Acids; Animals; Bridged Bicyclo Compounds, Heterocyclic; Corticosterone; Discrimination Learning; Ethanol; Male; Rats; Rats, Long-Evans; Receptors, AMPA; Self Administration; Xanthenes

2015
The Antidepressant Effects of an mGlu2/3 Receptor Antagonist and Ketamine Require AMPA Receptor Stimulation in the mPFC and Subsequent Activation of the 5-HT Neurons in the DRN.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2016, Volume: 41, Issue:4

    Topics: Amino Acids; Animals; Antidepressive Agents; Depression; Dorsal Raphe Nucleus; Fenclonine; Ketamine; Male; Mice; Mice, Inbred C57BL; Neural Pathways; Prefrontal Cortex; Quinoxalines; Receptors, AMPA; Receptors, Metabotropic Glutamate; Serotonergic Neurons; Xanthenes

2016
Mechanisms regulating spill-over of synaptic glutamate to extrasynaptic NMDA receptors in mouse substantia nigra dopaminergic neurons.
    The European journal of neuroscience, 2015, Volume: 42, Issue:9

    Topics: Amino Acids; Animals; Aspartic Acid; Dizocilpine Maleate; Dopaminergic Neurons; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Male; Mice; Mice, Inbred C57BL; Receptors, N-Methyl-D-Aspartate; Substantia Nigra; Synapses; Xanthenes

2015
Reversal of alcohol dependence-induced deficits in cue-guided behavior via mGluR2/3 signaling in mice.
    Psychopharmacology, 2016, Volume: 233, Issue:2

    Topics: Adaptation, Psychological; Alcoholism; Amino Acids; Animals; Bridged Bicyclo Compounds, Heterocyclic; Conditioning, Operant; Consummatory Behavior; Cues; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Male; Mice; Mice, Inbred C57BL; Psychomotor Performance; Receptors, AMPA; Reward; Self Administration; Signal Transduction; Xanthenes

2016
Lower [3H]LY341495 binding to mGlu2/3 receptors in the anterior cingulate of subjects with major depressive disorder but not bipolar disorder or schizophrenia.
    Journal of affective disorders, 2016, Jan-15, Volume: 190

    Topics: Amino Acids; Animals; Antidepressive Agents; Bipolar Disorder; Brain; Depressive Disorder, Major; Excitatory Amino Acid Antagonists; Female; Fluoxetine; Gyrus Cinguli; Humans; Imipramine; Male; Middle Aged; Radioligand Assay; Radionuclide Imaging; Rats; Receptors, Metabotropic Glutamate; Schizophrenia; Tritium; Xanthenes

2016
Activation of a Temporal Memory in Purkinje Cells by the mGluR7 Receptor.
    Cell reports, 2015, Dec-01, Volume: 13, Issue:9

    Topics: Amino Acids; Animals; Electric Stimulation; Excitatory Amino Acid Antagonists; Ferrets; gamma-Aminobutyric Acid; Glutamic Acid; Male; Patch-Clamp Techniques; Purkinje Cells; Pyridones; Quinoxalines; Receptors, AMPA; Receptors, Metabotropic Glutamate; Xanthenes

2015
Activity-dependent regulation of calcium and ribosomes in the chick cochlear nucleus.
    Neuroscience, 2016, Mar-01, Volume: 316

    Topics: Amino Acids; Analysis of Variance; Animals; Calcium; Chick Embryo; Cochlear Nucleus; Electric Stimulation; Evoked Potentials, Auditory; Excitatory Amino Acid Antagonists; Gene Expression Regulation; In Vitro Techniques; Indans; Optical Imaging; Ribosomes; Time Factors; Xanthenes

2016
The Rapidly Acting Antidepressant Ketamine and the mGlu2/3 Receptor Antagonist LY341495 Rapidly Engage Dopaminergic Mood Circuits.
    The Journal of pharmacology and experimental therapeutics, 2016, Volume: 358, Issue:1

    Topics: Action Potentials; Amino Acids; Animals; Antidepressive Agents; Dopamine; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Ketamine; Male; Mice, Inbred BALB C; Microdialysis; Motor Activity; Neurons; Nucleus Accumbens; Prefrontal Cortex; Quinoxalines; Rats, Wistar; Receptors, AMPA; Receptors, Metabotropic Glutamate; Ventral Tegmental Area; Xanthenes

2016
Group II mGlu receptor antagonist LY341495 enhances the antidepressant-like effects of ketamine in the forced swim test in rats.
    Psychopharmacology, 2016, Volume: 233, Issue:15-16

    Topics: Amino Acids; Animals; Antidepressive Agents; Behavior, Animal; Blotting, Western; Depression; Drug Synergism; Excitatory Amino Acid Antagonists; Ketamine; Male; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Signal Transduction; Swimming; TOR Serine-Threonine Kinases; Xanthenes

2016
EXPRESS: Histone hyperacetylation modulates spinal type II metabotropic glutamate receptor alleviating stress-induced visceral hypersensitivity in female rats.
    Molecular pain, 2016, Volume: 12

    Topics: Acetylation; Amino Acids; Animals; Chromatin Immunoprecipitation; Female; Histone Deacetylase Inhibitors; Histones; Hydroxamic Acids; Hyperalgesia; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; RNA, Messenger; Spinal Cord; Stress, Psychological; Viscera; Vorinostat; Xanthenes

2016
Blocking glutamate carboxypeptidase II inhibits glutamate excitotoxicity and regulates immune responses in experimental autoimmune encephalomyelitis.
    The FEBS journal, 2016, Volume: 283, Issue:18

    Topics: Amino Acids; Animals; Astrocytes; Disease Progression; Encephalomyelitis, Autoimmune, Experimental; Excitatory Amino Acid Antagonists; Female; Glutamate Carboxypeptidase II; Glutamic Acid; Humans; Immunohistochemistry; Mice; Mice, Inbred C57BL; Organophosphorus Compounds; Protease Inhibitors; Rats, Inbred Lew; Receptors, Metabotropic Glutamate; Spinal Cord; Th1 Cells; Xanthenes

2016
Metabotropic glutamate receptor 2/3 density and its relation to the hippocampal neuropathology in a model of temporal lobe epilepsy in rats.
    Epilepsy research, 2016, Volume: 127

    Topics: Acute Disease; Amino Acids; Animals; Autoradiography; Chronic Disease; Cross-Sectional Studies; Disease Models, Animal; Disease Progression; Epilepsy, Temporal Lobe; Excitatory Amino Acid Antagonists; Hippocampus; Kainic Acid; Male; Parietal Lobe; Radiopharmaceuticals; Rats, Wistar; Receptors, Metabotropic Glutamate; Thalamus; Time Factors; Tritium; Xanthenes

2016
Antidepressant-like effects of scopolamine in mice are enhanced by the group II mGlu receptor antagonist LY341495.
    Neuropharmacology, 2016, Volume: 111

    Topics: Amino Acids; Animals; Antidepressive Agents; Depressive Disorder; Excitatory Amino Acid Antagonists; Male; Maze Learning; Mice; Mice, Inbred C57BL; Motor Activity; Prefrontal Cortex; Quinoxalines; Receptors, AMPA; Receptors, Metabotropic Glutamate; Scopolamine; Serotonin; Xanthenes

2016
Fast-acting antidepressants rapidly stimulate ERK signaling and BDNF release in primary neuronal cultures.
    Neuropharmacology, 2016, Volume: 111

    Topics: Amino Acids; Animals; Antidepressive Agents; Brain-Derived Neurotrophic Factor; Cells, Cultured; Cerebral Cortex; Dendrites; GABAergic Neurons; Ketamine; MAP Kinase Signaling System; Oligopeptides; Primary Cell Culture; Rats; Receptor, trkB; Receptors, AMPA; Xanthenes

2016
Glutamate carboxypeptidase II (GCPII) inhibitor 2-PMPA reduces rewarding effects of the synthetic cathinone MDPV in rats: a role for N-acetylaspartylglutamate (NAAG).
    Psychopharmacology, 2017, Volume: 234, Issue:11

    Topics: Alkaloids; Amino Acids; Animals; Benzodioxoles; Conditioning, Psychological; Dipeptides; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Glutamate Carboxypeptidase II; Male; Organophosphorus Compounds; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Reward; Synthetic Cathinone; Xanthenes

2017
Control of Glutamate Transport by Extracellular Potassium: Basis for a Negative Feedback on Synaptic Transmission.
    Cerebral cortex (New York, N.Y. : 1991), 2017, 06-01, Volume: 27, Issue:6

    Topics: 2-Amino-5-phosphonovalerate; Amino Acid Transport System X-AG; Amino Acids; Animals; Animals, Newborn; Aspartic Acid; Astrocytes; Cerebral Cortex; Excitatory Amino Acid Antagonists; Extracellular Fluid; GABA-A Receptor Antagonists; Glutamic Acid; HEK293 Cells; Humans; Membrane Potentials; Mice; Mice, Inbred C57BL; Neural Inhibition; Neurons; Potassium; Synaptic Transmission; Xanthenes

2017
N-acetylaspartylglutamate Inhibits Heroin Self-Administration and Heroin-Seeking Behaviors Induced by Cue or Priming in Rats.
    Neuroscience bulletin, 2017, Volume: 33, Issue:4

    Topics: Amino Acids; Analysis of Variance; Animals; Conditioning, Operant; Cues; Dipeptides; Dose-Response Relationship, Drug; Drug-Seeking Behavior; Excitatory Amino Acid Antagonists; Heroin; Male; Motivation; Neuroprotective Agents; Rats; Rats, Sprague-Dawley; Reinforcement Schedule; Self Administration; Time Factors; Xanthenes

2017
A group II metabotropic glutamate receptor 3 (mGlu3, GRM3) isoform implicated in schizophrenia interacts with canonical mGlu3 and reduces ligand binding.
    Journal of psychopharmacology (Oxford, England), 2017, Volume: 31, Issue:12

    Topics: Amino Acids; Cell Membrane; HEK293 Cells; Humans; Ligands; Protein Isoforms; Radioligand Assay; Receptors, Metabotropic Glutamate; Schizophrenia; Transfection; Tritium; Xanthenes

2017
Cross-compartmental Modulation of Dendritic Signals for Retinal Direction Selectivity.
    Neuron, 2017, Aug-16, Volume: 95, Issue:4

    Topics: Action Potentials; Amacrine Cells; Amino Acids; Animals; Animals, Newborn; Cadmium Chloride; Calcium Channel Blockers; Dendrites; Excitatory Amino Acid Antagonists; Female; Inhibitory Postsynaptic Potentials; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Motion Perception; omega-Conotoxin GVIA; Photic Stimulation; Receptors, AMPA; Retina; Signal Transduction; Synapses; Xanthenes

2017
Activation of Group II Metabotropic Glutamate Receptors Increases Proliferation but does not Influence Neuronal Differentiation of a Human Neural Stem Cell Line.
    Basic & clinical pharmacology & toxicology, 2018, Volume: 122, Issue:4

    Topics: Amino Acids; Cell Differentiation; Cell Line; Cell Proliferation; Cell Survival; Cyclopropanes; Glutamic Acid; Glycine; Humans; Neural Stem Cells; Neurons; Receptors, Metabotropic Glutamate; Xanthenes

2018
The environmental neurotoxin β-N-methylamino-L-alanine inhibits melatonin synthesis in primary pinealocytes and a rat model.
    Journal of pineal research, 2018, Volume: 65, Issue:1

    Topics: Amino Acids; Amino Acids, Diamino; Animals; Cyanobacteria Toxins; Female; Male; Melatonin; Oxidative Stress; Phorbol Esters; Pineal Gland; Protein Kinase C; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Xanthenes

2018
Pre- and Postsynaptic Effects of Glutamate in the Frog Labyrinth.
    Neuroscience, 2018, 08-10, Volume: 385

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Amino Acids; Animals; Anura; Aspartic Acid; Ear, Inner; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Hair Cells, Auditory; Patch-Clamp Techniques; Receptors, Ionotropic Glutamate; Receptors, Metabotropic Glutamate; Synapses; Xanthenes

2018
Impact of allosteric modulation: Exploring the binding kinetics of glutamate and other orthosteric ligands of the metabotropic glutamate receptor 2.
    Biochemical pharmacology, 2018, Volume: 155

    Topics: Allosteric Regulation; Amino Acids; Animals; Binding Sites; Bridged Bicyclo Compounds; CHO Cells; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Ligands; Receptors, Metabotropic Glutamate; Xanthenes

2018
Single-molecule diffusion-based estimation of ligand effects on G protein-coupled receptors.
    Science signaling, 2018, 09-18, Volume: 11, Issue:548

    Topics: Amino Acids; GTP-Binding Proteins; HEK293 Cells; Humans; Ligands; Microscopy, Fluorescence; Pertussis Toxin; Protein Binding; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Metabotropic Glutamate; Signal Transduction; Xanthenes

2018
Glutamate metabotropic receptors in the lateral hypothalamus/perifornical area reduce the CO
    Respiratory physiology & neurobiology, 2019, Volume: 260

    Topics: Amino Acids; Animals; Carbon Dioxide; Electroencephalography; Electromyography; Excitatory Amino Acid Antagonists; Glycine; Hypothalamic Area, Lateral; Male; Microdialysis; Microinjections; Pulmonary Ventilation; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Sleep; Tidal Volume; Ventilation; Wakefulness; Xanthenes

2019
LY341495, an mGluR2/3 Antagonist, Regulates the Immunosuppressive Function of Myeloid-Derived Suppressor Cells and Inhibits Melanoma Tumor Growth.
    Biological & pharmaceutical bulletin, 2018, Volume: 41, Issue:12

    Topics: Amino Acids; Animals; Cell Proliferation; Cells, Cultured; Glutamic Acid; Glutamine; Melanoma, Experimental; Mice, Inbred C57BL; Myeloid-Derived Suppressor Cells; Receptors, Metabotropic Glutamate; Xanthenes

2018
Label-free impedance-based whole cell assay to study GPCR pharmacology.
    Methods in cell biology, 2019, Volume: 149

    Topics: Amino Acids; Animals; Biological Assay; Biosensing Techniques; Bridged Bicyclo Compounds; Cell Count; CHO Cells; Cricetinae; Cricetulus; Electric Impedance; Humans; Ligands; Receptors, G-Protein-Coupled; Receptors, Metabotropic Glutamate; Signal Transduction; Staining and Labeling; Xanthenes

2019
Glutamate Within the Marmoset Anterior Hippocampus Interacts with Area 25 to Regulate the Behavioral and Cardiovascular Correlates of High-Trait Anxiety.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2019, 04-17, Volume: 39, Issue:16

    Topics: Amino Acids; Animals; Anxiety; Behavior, Animal; Benzylamines; Callithrix; Excitatory Amino Acid Antagonists; Female; GABA-A Receptor Antagonists; Glutamic Acid; Heart Rate; Hippocampus; Male; Phosphinic Acids; Xanthenes

2019
Role of AMPA receptor stimulation and TrkB signaling in the antidepressant-like effect of ketamine co-administered with a group II mGlu receptor antagonist, LY341495, in the forced swim test in rats.
    Behavioural pharmacology, 2019, Volume: 30, Issue:6

    Topics: Amino Acids; Animals; Antidepressive Agents; Azepines; Benzamides; Depression; Depressive Disorder; Excitatory Amino Acid Antagonists; Ketamine; Male; Prefrontal Cortex; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptor, trkB; Receptors, AMPA; Receptors, Metabotropic Glutamate; Signal Transduction; Xanthenes

2019
Group II metabotropic glutamate receptor blockade promotes stress resilience in mice.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2019, Volume: 44, Issue:10

    Topics: Amino Acids; Anhedonia; Animals; Behavior, Animal; Corticosterone; Electroshock; Escape Reaction; Excitatory Amino Acid Antagonists; Mice; Mice, Knockout; Receptors, Metabotropic Glutamate; Resilience, Psychological; Stress, Psychological; Xanthenes

2019
Target validation: Weak selectivity of LY341495 for mGluR2 over mGluR4 makes glutamate a less selective agonist.
    Pharmacology research & perspectives, 2019, Volume: 7, Issue:3

    Topics: Amino Acids; Animals; Dose-Response Relationship, Drug; Down-Regulation; Ganglia, Sympathetic; Gene Expression Regulation; Male; Rats; Receptors, Metabotropic Glutamate; Signal Transduction; Superior Cervical Ganglion; Xanthenes

2019
Pharmacological Modulation of Sleep Homeostasis in Rat: Novel Effects of an mGluR2/3 Antagonist.
    Sleep, 2019, 09-06, Volume: 42, Issue:9

    Topics: Amino Acids; Animals; Caffeine; Central Nervous System Stimulants; Cyclohexanes; Dextroamphetamine; Electroencephalography; Excitatory Amino Acid Antagonists; Homeostasis; Male; Rats; Rats, Wistar; Reaction Time; Receptors, Metabotropic Glutamate; Sleep; Sleep Deprivation; Sleep, REM; Wakefulness; Xanthenes

2019
Regulatory system of mGluR group II in the nucleus accumbens for methamphetamine-induced dopamine increase by the medial prefrontal cortex.
    Neuropsychopharmacology reports, 2019, Volume: 39, Issue:3

    Topics: Acetyltransferases; Amino Acids; Animals; Dopamine; Dopamine Agents; Dopamine and cAMP-Regulated Phosphoprotein 32; Excitatory Amino Acid Antagonists; Glutamic Acid; Male; Methamphetamine; Mice; Mice, Inbred C57BL; Nucleus Accumbens; Prefrontal Cortex; Receptors, Metabotropic Glutamate; Xanthenes

2019
Amygdala group II mGluRs mediate the inhibitory effects of systemic group II mGluR activation on behavior and spinal neurons in a rat model of arthritis pain.
    Neuropharmacology, 2019, 11-01, Volume: 158

    Topics: Amino Acids; Amygdala; Animals; Arthralgia; Arthritis, Experimental; Behavior, Animal; Bridged Bicyclo Compounds, Heterocyclic; Carrageenan; Central Amygdaloid Nucleus; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Kaolin; Nociception; Pain; Posterior Horn Cells; Rats; Receptors, Metabotropic Glutamate; Spinal Cord; Vocalization, Animal; Xanthenes

2019
Vulnerability to depressive behavior induced by overexpression of striatal Shati/Nat8l via the serotonergic neuronal pathway in mice.
    Behavioural brain research, 2019, 12-30, Volume: 376

    Topics: Acetyltransferases; Amino Acids; Animals; Brain; Causality; Corpus Striatum; Depression; Fluvoxamine; Male; Mice; Mice, Inbred C57BL; Serotonergic Neurons; Stress, Psychological; Xanthenes

2019
AMPA receptor-mTORC1 signaling activation is required for neuroplastic effects of LY341495 in rat hippocampal neurons.
    Scientific reports, 2020, 01-22, Volume: 10, Issue:1

    Topics: Amino Acids; Animals; Excitatory Amino Acid Antagonists; Hippocampus; Mechanistic Target of Rapamycin Complex 1; Neuronal Plasticity; Neurons; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Metabotropic Glutamate; Signal Transduction; Xanthenes

2020
The metabotropic glutamate receptor 2/3 antagonist LY341495 improves working memory in adult mice following juvenile social isolation.
    Neuropharmacology, 2020, 10-15, Volume: 177

    Topics: Age Factors; Amino Acids; Animals; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Male; Maze Learning; Memory, Short-Term; Mice; Mice, Inbred C57BL; Receptors, Metabotropic Glutamate; Social Isolation; Xanthenes

2020
The group II mGlu receptor antagonist LY341495 induces a rapid antidepressant-like effect and enhances the effect of ketamine in the chronic unpredictable mild stress model of depression in C57BL/6J mice.
    Progress in neuro-psychopharmacology & biological psychiatry, 2021, 07-13, Volume: 109

    Topics: Amino Acids; Animals; Antidepressive Agents; Depression; Disease Models, Animal; Excitatory Amino Acid Antagonists; Hippocampus; Ketamine; Male; Mice; Mice, Inbred C57BL; Motor Skills; Prefrontal Cortex; Receptors, Metabotropic Glutamate; Synaptosomes; Xanthenes

2021
mGlu2/3 receptor in the prelimbic cortex is implicated in stress resilience and vulnerability in mice.
    European journal of pharmacology, 2021, Sep-05, Volume: 906

    Topics: Amino Acids; Animals; Depression; Disease Models, Animal; Humans; Male; Mice; Prefrontal Cortex; Receptors, Metabotropic Glutamate; Resilience, Psychological; Social Defeat; Stress, Psychological; Xanthenes

2021
Inhibition of metabotropic glutamate receptor III facilitates sensitization to alkylating chemotherapeutics in glioblastoma.
    Cell death & disease, 2021, 07-21, Volume: 12, Issue:8

    Topics: Amino Acids; Antineoplastic Agents, Alkylating; Cell Death; Cell Line, Tumor; Cell Survival; Drug Resistance, Neoplasm; Gene Expression Regulation, Neoplastic; Glioblastoma; Glutamic Acid; Humans; Kinetics; Neoadjuvant Therapy; Receptors, Metabotropic Glutamate; Temozolomide; Tumor Microenvironment; Xanthenes

2021
Allosteric modulators enhance agonist efficacy by increasing the residence time of a GPCR in the active state.
    Nature communications, 2021, 09-14, Volume: 12, Issue:1

    Topics: Allosteric Regulation; Allosteric Site; Amino Acids; Biphenyl Compounds; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Catalytic Domain; Cell Membrane; Cholesterol Esters; Diosgenin; Disaccharides; Fluorescence Resonance Energy Transfer; Gene Expression; Glucosides; Glutamic Acid; Glycolipids; HEK293 Cells; Humans; Indans; Micelles; Octoxynol; Protein Binding; Protein Conformation; Protein Multimerization; Receptors, Metabotropic Glutamate; Recombinant Proteins; Single Molecule Imaging; Xanthenes

2021
Graded heterogeneity of metabotropic signaling underlies a continuum of cell-intrinsic temporal responses in unipolar brush cells.
    Nature communications, 2021, 10-07, Volume: 12, Issue:1

    Topics: Action Potentials; Amino Acids; Animals; Cerebellar Cortex; Electric Stimulation; Excitatory Amino Acid Antagonists; Female; Male; Mice, Inbred C57BL; Nerve Fibers; Neurons; Patch-Clamp Techniques; Receptors, Metabotropic Glutamate; Synaptic Transmission; Time Factors; Xanthenes

2021
Effects of Chronic LY341495 on Hippocampal mTORC1 Signaling in Mice with Chronic Unpredictable Stress-Induced Depression.
    International journal of molecular sciences, 2022, Jun-08, Volume: 23, Issue:12

    Topics: Amino Acids; Animals; Antidepressive Agents; Depression; Hippocampus; Mechanistic Target of Rapamycin Complex 1; Mice; Stress, Psychological; Xanthenes

2022